PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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P110δ-IN-1
CAS:1595129-71-7
P110δ-IN-1 (PWT-143) is an effective and selective inhibitor of P110δ (IC50: 8.4 nM).
Formula:
C31H40N8O3S
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
604.77
Ref: TM-T16422
| 1mg | 48.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 535.00 € | ||
| 100mg | 753.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Recilisib
CAS:334969-03-8
Recilisib (ON 01210) is a radioprotectant,can activate AKT, PI3K activities in cells.
Formula:
C16H13ClO4S
Purity:
98.85% - 98.96%
Color and Shape:
Solid
Molecular weight:
336.79
Ref: TM-T13862
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 528.00 € | ||
| 500mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Inavolisib
CAS:2060571-02-8
Inavolisib (GDC-0077) is an orally available selective PI3Kα inhibitor with an IC50 value of 0.038 …
Formula:
C18H19F2N5O4
Purity:
97.36% - 99.83%
Color and Shape:
Solid
Molecular weight:
407.37
Ref: TM-T15375
| 1mg | 88.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 373.00 € | ||
| 25mg | 635.00 € | ||
| 50mg | 1,035.00 € | ||
| 100mg | 1,795.00 € | ||
| 1mL*10mM (DMSO) | 404.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
IPI-3063
CAS:1425043-73-7
IPI-3063 is an effective and selective inhibitor of PI3K p110δ (IC50: 2.5 ± 1.2 nM).
Formula:
C25H25N7O2
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
455.51
Ref: TM-T15592
| 1mg | 47.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 340.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 645.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
NSC781406
CAS:1676893-24-5
NSC781406 is a highly effective inhibitor of PI3K and mTOR (IC50: 2 nM for PI3Kα).
Formula:
C29H27F2N5O5S2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
627.68
Ref: TM-T16355
| 2mg | 42.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 375.00 € | ||
| 200mg | 533.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Isoprenaline hydrochloride
CAS:51-30-9
Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac …
Formula:
C11H18ClNO3
Purity:
98% - 99.25%
Color and Shape:
Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
Molecular weight:
247.719
Ref: TM-T1056
| 1g | 39.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Copanlisib dihydrochloride
CAS:1402152-13-9
Copanlisib dihydrochloride: ATP-competitive PI3K inhibitor, potent for PI3Kα/δ/β/γ, antitumor, 2000x selectivity over other kinases except …
Formula:
C23H30Cl2N8O4
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
553.44
Ref: TM-T14998
| 5mg | 51.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 354.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
PI4KIIIbeta-IN-9
CAS:1429624-84-9
PI4KIIIbeta-IN-9 is a potent inhibitor of PI4KIIIβ(IC50 of 7 nM). .
Formula:
C23H25N3O5S2
Purity:
97.18%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T12469
| 1mg | 80.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 512.00 € | ||
| 50mg | 715.00 € | ||
| 100mg | 938.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Parsaclisib
CAS:1426698-88-5
Parsaclisib (INCB050465) is a potent and selective inhibitor of PI3Kδ(IC50 of 1 nM at 1 …
Formula:
C20H22ClFN6O2
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
432.88
Ref: TM-T12367
| 1mg | 145.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 805.00 € | ||
| 50mg | 1,111.00 € | ||
| 100mg | 1,501.00 € | ||
| 1mL*10mM (DMSO) | 335.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
CGS 15943
CAS:104615-18-1
CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
Formula:
C13H8ClN5O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
285.69
Ref: TM-T14944
| 1mg | 47.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 316.00 € | ||
| 100mg | 474.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Thioridazine hydrochloride
CAS:130-61-0
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and …
Formula:
C21H27ClN2S2
Purity:
99.55% - 99.55%
Color and Shape:
White To Off-White Solid
Molecular weight:
407.04
Ref: TM-T0365
| 50mg | 43.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Tenalisib
CAS:1639417-53-0
Tenalisib (RP6530) (RP6530) is a potent and selective inhibitor of PI3Kδ and PI3Kγ(IC50 values of …
Formula:
C23H18FN5O2
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
415.42
Ref: TM-T13119
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 457.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Sophocarpine monohydrate
CAS:145572-44-7
Sophocarpine monohydrate, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.
Formula:
C15H22N2O
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
246.35
Ref: TM-T2746
| 50mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
BAY1082439
CAS:1375469-38-7
BAY1082439, an orally bioavailable, selective inhibitor of PI3Kα/β/δ, demonstrates high efficacy in inhibiting the growth …
Formula:
C25H30N6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
494.54
Ref: TM-T14511
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
Pictilisib dimethanesulfonate
CAS:957054-33-0
Pictilisib dimethanesulfonate (GDC-0941 2 MeSO3H salt) is a potent inhibitor of PI3Kα/δ with IC50 of …
Formula:
C25H35N7O9S4
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
705.85
Ref: TM-T11381
| 10mg | 35.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
PI4KIIIbeta-IN-10
CAS:1881233-39-1
PI4KIIIbeta-IN-10 is a potent inhibitor of PI4KIIIβ (IC50 of 3.6 nM).
Formula:
C22H25N3O5S2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
475.58
Ref: TM-T12468
| 1mg | 80.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 420.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 792.00 € | ||
| 200mg | 1,064.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Wednesday 30 Apr 2025
PI3Kα-IN-12
PI3Kα-IN-12 (compound 13), a potent and selective PI3Kα inhibitor (IC50: 1.2 nM), effectively suppresses HCT-116 …
Formula:
C28H36F2N10O5S3
Color and Shape:
Liquid
Molecular weight:
726.84
Ref: TM-T78804
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 2 May 2025
PI3Kδ-IN-18
Se15, a selective PI3Kδ inhibitor, exhibits potency with an IC50 value of less than 0.1nM …
Purity:
98%
Color and Shape:
Odour Solid
Ref: TM-T81467
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 2 May 2025
WYE-687
CAS:1062161-90-3
WYE-687 is a selective mTOR inhibitor (IC50: 7 nM), over 100x more selective for mTOR …
Formula:
C28H32N8O3
Purity:
98.98%
Color and Shape:
Solid
Molecular weight:
528.61
Ref: TM-T6732
| 5mg | 39.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 2 May 2025
ARUK2001607
ARUK2001607 selectively inhibits PI5P4Kγ (Kd=7.1 nM) with high selectivity over 150+ kinases.
Formula:
C14H13N3O2S2
Purity:
99.86%
Color and Shape:
Soild
Molecular weight:
319.40
Ref: TM-T67845
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 113.00 € | ||
| 1mL*10mM (DMSO) | 48.00 € |
Estimated delivery in United States, on Friday 2 May 2025
