PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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(E)-Akt inhibitor-IV
CAS:959841-49-7
(E)-Akt inhibitor-IV ((E)-AKTIV) ((E)-AKTIV) is an inhibitor of PI3K-Akt.
Formula:
C31H29IN4S
Purity:
99.01% - 99.74%
Color and Shape:
Solid
Molecular weight:
616.56
Ref: TM-T9393
| 1mg | 55.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 469.00 € | ||
| 100mg | 655.00 € | ||
| 200mg | 924.00 € | ||
| 1mL*10mM (DMSO) | 157.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
iMDK
CAS:881970-80-5
iMDK quarterhydrate, a PI3K inhibitor, blocks MDK growth factor and enhances NSCLC treatment with MEK …
Formula:
C21H13FN2O2S
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
376.4
Ref: TM-T9460
| 1mg | 59.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 908.00 € | ||
| 500mg | 1,825.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Vps34-PIK-III
CAS:1383716-40-2
Vps34-PIK-III (VPS34-IN2), a selective inhibitor of VPS34 enzymatic activity, inhibits autophagy and results in the …
Formula:
C17H17N7
Purity:
98.39% - 98.43%
Color and Shape:
Solid
Molecular weight:
319.36
Ref: TM-T6945
| 1mg | 51.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 454.00 € | ||
| 50mg | 663.00 € | ||
| 100mg | 944.00 € | ||
| 500mg | 1,890.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
GNE-477
CAS:1032754-81-6
GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor.
Formula:
C21H28N8O3S2
Purity:
98.88% - 99.55%
Color and Shape:
Solid
Molecular weight:
504.63
Ref: TM-T3692
| 1mg | 70.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 873.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
TG 100713
CAS:925705-73-3
TG 100713 is a pan-PI3K inhibitor against PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of …
Formula:
C12H10N6O
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
254.25
Ref: TM-T6704
| 5mg | 39.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 192.00 € | ||
| 100mg | 281.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
BEBT-908
CAS:1235449-52-1
BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor (IC50 <0.1 μM). BEBT-908 also inhibits …
Formula:
C23H25N9O3S
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
507.57
Ref: TM-T16529
| 1mg | 120.00 € | ||
| 2mg | 167.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 630.00 € | ||
| 50mg | 898.00 € | ||
| 100mg | 1,216.00 € | ||
| 500mg | 2,442.00 € | ||
| 1mL*10mM (DMSO) | 279.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
PI3K-IN-1
CAS:1349796-36-6
PI3K-IN-1 (Voxtalisib Analogue) is a dual inhibitor of mTOR/PI3K, mostly for p110γ , also inhibits …
Formula:
C31H29N5O6S
Purity:
97.03% - 98%
Color and Shape:
Solid
Molecular weight:
599.66
Ref: TM-T1826
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,121.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
1,3-Dicaffeoylquinic acid
CAS:19870-46-3
1,3-Dicaffeoylquinic acid (CYNARIN) is a natural product. It shows antioxidant and choleretic properties and is …
Formula:
C25H24O12
Purity:
98% - 98.81%
Color and Shape:
Solid
Molecular weight:
516.45
Ref: TM-T5736
| 20mg | 138.00 € | ||
| 1mL*10mM (DMSO) | 108.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Euscaphic acid
CAS:53155-25-2
Euscaphic acid has anti-diabetic and anti-inflammatory effects, blocking IKK/MAPKs and NF-κB activation by disrupting TRAF6/IRAK1/TAK1 …
Formula:
C30H48O5
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
488.7
Ref: TM-TN1134
| 1mg | 80.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
PI3Kδ-IN-15
CAS:1146702-54-6
CAL-101 (Idelalisib) is a selective inhibitor of p110δ; shown to have 40- to 300-fold greater …
Formula:
C21H16FN7O
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
401.4
Ref: TM-T8651
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 77.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 183.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
AS-605240
CAS:648450-29-7
AS-605240 is an effective and specific inhibitor of PI3Kγ (IC50/Ki: 87.8 nM).
Formula:
C12H7N3O2S
Purity:
97% - 99.91%
Color and Shape:
Solid
Molecular weight:
257.27
Ref: TM-T2248
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 349.00 € | ||
| 500mg | 565.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
HS-173
CAS:1276110-06-5
HS-173 is an effective PI3Kα inhibitor (IC50: 0.8 nM).
Formula:
C21H18N4O4S
Purity:
99.33% - 99.64%
Color and Shape:
Solid
Molecular weight:
422.46
Ref: TM-T2308
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Serabelisib
CAS:1268454-23-4
Serabelisib (INK1117) is a p110α/β/γ/δ inhibitor (IC50: 15/4.5/1.9/13.39 μM).
Formula:
C19H17N5O3
Purity:
98.41% - 99.5%
Color and Shape:
Solid
Molecular weight:
363.37
Ref: TM-T3153
| 1mg | 44.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 520.00 € | ||
| 500mg | 1,111.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
TG100-115
CAS:677297-51-7
TG100-115 is a PI3Kγ/δ inhibitor (IC50: 83/235 nM), with fewer effects on PI3Kα/β.
Formula:
C18H14N6O2
Purity:
100% - 98.95%
Color and Shape:
Solid
Molecular weight:
346.34
Ref: TM-T2672
| 1mg | 43.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 588.00 € | ||
| 500mg | 1,216.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Sophocarpine
CAS:6483-15-4
Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.
Formula:
C15H22N2O
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
246.35
Ref: TM-T6677
| 5mg | 49.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 205.00 € | ||
| 100mg | 305.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Quercetin Dihydrate
CAS:6151-25-3
Quercetin Dihydrate (Sophoretin) is a flavonoid natural product that activates or inhibits the activity of …
Formula:
C15H10O7·2H2O
Purity:
97.03% - 97.77%
Color and Shape:
Yellow Solid
Molecular weight:
338.27
Ref: TM-T6630
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
25(R,S)-Ruscogenin
CAS:874485-32-2
25(R,S)-Ruscogenin is able to regulate the PI3K/Akt/mTOR signalling pathway, and hinder the metastasis of hepatocellular …
Formula:
C27H42O4
Purity:
99.32% - 99.89%
Color and Shape:
Solid
Molecular weight:
430.62
Ref: TM-T5740
| 1mg | 52.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Buparlisib
CAS:944396-07-0
Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: …
Formula:
C18H21F3N6O2
Purity:
95.32% - 98.45%
Color and Shape:
Solid
Molecular weight:
410.39
Ref: TM-T1827
| 5mg | 63.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 115.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 235.00 € | ||
| 500mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Autophinib
CAS:1644443-47-9
Autophinib is a potent autophagy inhibitor with a novel chemotype with IC50 values of 90 …
Formula:
C14H11ClN6O3
Purity:
99.25% - 99.41%
Color and Shape:
Solid
Molecular weight:
346.73
Ref: TM-T4219
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 427.00 € | ||
| 500mg | 938.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Esculetin
CAS:305-01-1
Esculetin: a coumarin from plants with anti-edema, anti-inflammatory, anti-tumor properties; inhibits LOs.
Formula:
C9H6O4
Purity:
98.03% - 99.76%
Color and Shape:
Yellow Crystalline Powder
Molecular weight:
178.14
Ref: TM-T2798
| 100mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
