PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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(E)-Akt inhibitor-IV
CAS:959841-49-7
(E)-Akt inhibitor-IV ((E)-AKTIV) ((E)-AKTIV) is an inhibitor of PI3K-Akt.
Formula:
C31H29IN4S
Purity:
99.01% - 99.74%
Color and Shape:
Solid
Molecular weight:
616.56
Ref: TM-T9393
| 1mg | 53.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 630.00 € | ||
| 200mg | 890.00 € | ||
| 1mL*10mM (DMSO) | 151.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
iMDK
CAS:881970-80-5
iMDK quarterhydrate, a PI3K inhibitor, blocks MDK growth factor and enhances NSCLC treatment with MEK …
Formula:
C21H13FN2O2S
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
376.4
Ref: TM-T9460
| 1mg | 58.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 628.00 € | ||
| 100mg | 888.00 € | ||
| 500mg | 1,790.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Vps34-PIK-III
CAS:1383716-40-2
Vps34-PIK-III (VPS34-IN2), a selective inhibitor of VPS34 enzymatic activity, inhibits autophagy and results in the …
Formula:
C17H17N7
Purity:
98.39% - 98.43%
Color and Shape:
Solid
Molecular weight:
319.36
Ref: TM-T6945
| 1mg | 51.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 443.00 € | ||
| 50mg | 651.00 € | ||
| 100mg | 922.00 € | ||
| 500mg | 1,848.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
GNE-477
CAS:1032754-81-6
GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor.
Formula:
C21H28N8O3S2
Purity:
98.88% - 99.55%
Color and Shape:
Solid
Molecular weight:
504.63
Ref: TM-T3692
| 1mg | 70.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 617.00 € | ||
| 100mg | 862.00 € | ||
| 1mL*10mM (DMSO) | 151.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
TG 100713
CAS:925705-73-3
TG 100713 is a pan-PI3K inhibitor against PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of …
Formula:
C12H10N6O
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
254.25
Ref: TM-T6704
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 271.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
BEBT-908
CAS:1235449-52-1
BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor (IC50 <0.1 μM). BEBT-908 also inhibits …
Formula:
C23H25N9O3S
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
507.57
Ref: TM-T16529
| 1mg | 121.00 € | ||
| 2mg | 170.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 377.00 € | ||
| 25mg | 629.00 € | ||
| 50mg | 897.00 € | ||
| 100mg | 1,214.00 € | ||
| 500mg | 2,401.00 € | ||
| 1mL*10mM (DMSO) | 278.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
PI3K-IN-1
CAS:1349796-36-6
PI3K-IN-1 (Voxtalisib Analogue) is a dual inhibitor of mTOR/PI3K, mostly for p110γ , also inhibits …
Formula:
C31H29N5O6S
Purity:
97.03% - 98%
Color and Shape:
Solid
Molecular weight:
599.66
Ref: TM-T1826
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 496.00 € | ||
| 500mg | 1,096.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
1,3-Dicaffeoylquinic acid
CAS:19870-46-3
1,3-Dicaffeoylquinic acid (CYNARIN) is a natural product. It shows antioxidant and choleretic properties and is …
Formula:
C25H24O12
Purity:
98% - 98.68%
Color and Shape:
Solid
Molecular weight:
516.45
Ref: TM-T5736
| 20mg | 135.00 € | ||
| 1mL*10mM (DMSO) | 108.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Euscaphic acid
CAS:53155-25-2
Euscaphic acid has anti-diabetic and anti-inflammatory effects, blocking IKK/MAPKs and NF-κB activation by disrupting TRAF6/IRAK1/TAK1 …
Formula:
C30H48O5
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
488.7
Ref: TM-TN1134
| 1mg | 79.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 219.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
PI3Kδ-IN-15
CAS:1146702-54-6
CAL-101 (Idelalisib) is a selective inhibitor of p110δ; shown to have 40- to 300-fold greater …
Formula:
C21H16FN7O
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
401.4
Ref: TM-T8651
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 123.00 € | ||
| 200mg | 180.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
AS-605240
CAS:648450-29-7
AS-605240 is an effective and specific inhibitor of PI3Kγ (IC50/Ki: 87.8 nM).
Formula:
C12H7N3O2S
Purity:
97% - 99.91%
Color and Shape:
Solid
Molecular weight:
257.27
Ref: TM-T2248
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 165.00 € | ||
| 100mg | 229.00 € | ||
| 200mg | 341.00 € | ||
| 500mg | 552.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
ETP-46321
CAS:1252594-99-2
ETP-46321 is an effective and orally bioavailable PI3Kα/PI3Kδ inhibitor (Ki: 2.3/14.2 nM).
Formula:
C20H27N9O3S
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
473.55
Ref: TM-TQ0229
| 1mg | 50.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 309.00 € | ||
| 50mg | 432.00 € | ||
| 100mg | 593.00 € | ||
| 200mg | 803.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Esculetin
CAS:305-01-1
Esculetin: a coumarin from plants with anti-edema, anti-inflammatory, anti-tumor properties; inhibits LOs.
Formula:
C9H6O4
Purity:
98.43% - 99.76%
Color and Shape:
Yellow Crystalline Powder
Molecular weight:
178.14
Ref: TM-T2798
| 100mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Alpelisib
CAS:1217486-61-7
Alpelisib (BYL-719) is a PI3Kα inhibitor (IC50=5 nM) with selective, potent, and oral activity.
Formula:
C19H22F3N5O2S
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
441.47
Ref: TM-T1921
| 1g | 642.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 261.00 € | ||
| 500mg | 438.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
GSK1059615
CAS:958852-01-2
GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, …
Formula:
C18H11N3O2S
Purity:
≥95% - ≥95%
Color and Shape:
Solid
Molecular weight:
333.36
Ref: TM-T2357
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 191.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 498.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Wortmannin
CAS:19545-26-7
Wortmannin (SL-2052) is a PI3K inhibitor (IC50=3 nM) that is covalent and irreversible.
Formula:
C23H24O8
Purity:
95.84% - 99.76%
Color and Shape:
White Solid
Molecular weight:
428.43
Ref: TM-T6283
| 1mg | 38.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 190.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
3-Methyladenine
CAS:5142-23-4
3-Methyladenine (3-MA) is a PI3K inhibitor that selectively inhibits class IB PI3Kγ (IC50=60 μM) and …
Formula:
C6H7N5
Purity:
98.02% - 99.51%
Color and Shape:
Solid
Molecular weight:
149.15
Ref: TM-T1879
| 25mg | 41.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 135.00 € | ||
| 500mg | 247.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
PI-103
CAS:371935-74-9
PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for …
Formula:
C19H16N4O3
Purity:
96.59% - 99.3%
Color and Shape:
Solid
Molecular weight:
348.36
Ref: TM-T6143
| 5mg | 58.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 197.00 € | ||
| 100mg | 363.00 € | ||
| 200mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Erucic acid
CAS:112-86-7
Increased levels of erucic acid (22:1n9) have been found in the red blood cell membranes …
Formula:
C22H42O2
Purity:
97.85%
Color and Shape:
Needles From Alcohol Liquid Othersolid
Molecular weight:
338.57
Ref: TM-T4867
| 100mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
Brevianamide F
CAS:38136-70-8
Brevianamide F (Cyclo(L-Pro-L-Trp)), also known as cyclo-(L-Trp-L-Pro), belongs to a class of naturally occurring 2,5-diketopiperazines.
Formula:
C16H17N3O2
Purity:
97.30% - 98.82%
Color and Shape:
Solid
Molecular weight:
283.33
Ref: TM-T3208
| 1mg | 44.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 418.00 € | ||
| 100mg | 611.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 23 Dec 2024
