PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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PIK-108
CAS:901398-68-3
PIK-108 is an allosteric inhibitor of phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunits β and δ (PI3Kβ/δ).
Formula:
C22H24N2O3
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
364.44
Ref: TM-T28416
| 1mg | 39.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 491.00 € | ||
| 200mg | 674.00 € | ||
| 1mL*10mM (DMSO) | 102.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LY294002
CAS:154447-36-6
LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 …
Formula:
C19H17NO3
Purity:
98% - 99.96%
Color and Shape:
Pale Yellow Solid
Molecular weight:
307.34
Ref: TM-T2008
| 5mg | 39.00 € | ||
| 10mg | 50.00 € | ||
| 50mg | 71.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 121.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dihydrocapsaicin
CAS:19408-84-5
Dihydrocapsaicin, similar to capsaicin, is an irritant found in Capsicum, used in "pure" capsaicin products …
Formula:
C18H29NO3
Purity:
99.61% - ≥95%
Color and Shape:
White Crystal
Molecular weight:
307.43
Ref: TM-T2163
| 10mg | 58.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 221.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Copanlisib
CAS:1032568-63-0
Copanlisib (BAY 80-6946), a PI3K inhibitor, may block tumor growth and improve cancer treatment efficacy.
Formula:
C23H28N8O4
Purity:
99.02% - 99.88%
Color and Shape:
Solid
Molecular weight:
480.52
Ref: TM-T6322
| 2mg | 38.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 348.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Bimiralisib
CAS:1225037-39-7
Bimiralisib (PI3K-IN-2) is an orally bioavailable pan inhibitor of PI3K and inhibitor of the mTOR, …
Formula:
C17H20F3N7O2
Purity:
97.58% - 99.88%
Color and Shape:
Solid
Molecular weight:
411.38
Ref: TM-T2265
| 1mg | 35.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 530.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sapanisertib
CAS:1224844-38-5
Sapanisertib (INK 128) is an oral raptor-mTOR and rictor-mTOR inhibitor with potential cancer-fighting properties.
Formula:
C15H15N7O
Purity:
100% - 99.34%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T1838
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 344.00 € | ||
| 500mg | 824.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Idelalisib
CAS:870281-82-6
Idelalisib (GS-1101) is a small molecule inhibitor of the PI3K catalytic subunit p110δ (IC50: 2.5 …
Formula:
C22H18FN7O
Purity:
98% - 99.94%
Color and Shape:
Solid
Molecular weight:
415.42
Ref: TM-T1894
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 107.00 € | ||
| 200mg | 138.00 € | ||
| 500mg | 221.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Hederacolchiside A1
CAS:106577-39-3
Hederacolchiside A1 exhibits anti-leishmanial and anticancer activities by disrupting cell membranes and inducing apoptosis via …
Formula:
C47H76O16
Purity:
99.54% - 99.92%
Color and Shape:
Solid
Molecular weight:
897.1
Ref: TM-T2P2806
| 1mg | 47.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 166.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ZSTK474
CAS:475110-96-4
PI3K Inhibitor ZSTK474 is an orally available, s-triazine derivative, ATP-competitive phosphatidylinositol 3-kinase (PI3K) inhibitor with …
Formula:
C19H21F2N7O2
Purity:
98.29% - 99.76%
Color and Shape:
White Powder
Molecular weight:
417.41
Ref: TM-T6168
| 5mg | 38.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 139.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Omipalisib
CAS:1086062-66-9
Omipalisib (GSK2126458) is a small-molecule pyridylsulfonamide inhibitor of phosphatidylinositol 3-kinase (PI3K) with potential antineoplastic activity.
Formula:
C25H17F2N5O3S
Purity:
98% - 99.8%
Color and Shape:
Solid
Molecular weight:
505.5
Ref: TM-T1861
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 417.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Rigosertib
CAS:592542-59-1
Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by …
Formula:
C21H25NO8S
Purity:
97.33%
Color and Shape:
Solid
Molecular weight:
451.49
Ref: TM-T16750
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 94.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
YS-49
CAS:132836-42-1
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
Formula:
C20H20BrNO2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
386.28
Ref: TM-T13376
| 1mg | 48.00 € | ||
| 2mg | 61.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 401.00 € | ||
| 100mg | 581.00 € | ||
| 500mg | 1,196.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GNE-317
CAS:1394076-92-6
GNE-317, a PI3K/mTOR inhibitor, can pass through the blood-brain barrier (BBB).
Formula:
C19H22N6O3S
Purity:
99.08% - 99.42%
Color and Shape:
Solid
Molecular weight:
414.48
Ref: TM-T6845
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 342.00 € | ||
| 100mg | 426.00 € | ||
| 200mg | 623.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TGX-221
CAS:663619-89-4
TGX-221, an effective, specific, and cell membrane permeable inhibitor of the PI3K p110β catalytic subunit, …
Formula:
C21H24N4O2
Purity:
100% - 99.8%
Color and Shape:
Solid
Molecular weight:
364.44
Ref: TM-T2661
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 351.00 € | ||
| 100mg | 551.00 € | ||
| 500mg | 1,177.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LX2343
CAS:333745-53-2
LX2343 inhibits BACE1 (IC50: 11.43 μM) and PI3K non-competitively (IC50: 15.99 μM), and enhances autophagy …
Formula:
C22H19ClN2O6S
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
474.91
Ref: TM-T4398
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 221.00 € | ||
| 100mg | 328.00 € | ||
| 200mg | 456.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BQR-695
CAS:1513879-21-4
BQR-695 (NVP-BQR695) is a PI4K inhibitor with IC50s of 80 and 3.5 nM for human …
Formula:
C19H20N4O3
Purity:
100% - 97.16%
Color and Shape:
Solid
Molecular weight:
352.39
Ref: TM-T4220
| 5mg | 70.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 427.00 € | ||
| 500mg | 917.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PI-3065
CAS:955977-50-1
PI-3065 is a novel potent and selective PI3K p110δ inhibitor.
Formula:
C27H31FN6OS
Purity:
98.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
506.64
Ref: TM-T2083
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 540.00 € | ||
| 500mg | 1,107.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Fimepinostat
CAS:1339928-25-4
Fimepinostat (CUDC 907) is an orally bioavailable inhibitor of both PI3K class I and pan-HDAC …
Formula:
C23H24N8O4S
Purity:
97.13% - 99.87%
Color and Shape:
Solid
Molecular weight:
508.55
Ref: TM-T2078
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 500.00 € | ||
| 500mg | 1,068.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TASP0415914
CAS:1292300-75-4
TASP0415914 is an orally potent inhibitor of phosphoinositide 3-kinase γ (PI3Kγ). T
Formula:
C13H17N5O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
323.37
Ref: TM-T7879
| 1mg | 53.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 181.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 433.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 805.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Flavanomarein
CAS:577-38-8
Flavanomarein: Antioxidant with radical scavenging, lipid peroxidation inhibition, and lipid-lowering in HepG2 cells.
Formula:
C21H22O11
Purity:
97.53% - 98.63%
Color and Shape:
Solid
Molecular weight:
450.39
Ref: TM-TN1644
| 1mg | 47.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
