G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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MRGPRX1 agonist 1
CAS:2377379-39-8
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
Formula:
C23H21N3O4S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
435.5
Ref: TM-T12104
| 1mg | 87.00 € | ||
| 5mg | 206.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 228.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BIBO3304 TFA
CAS:191868-14-1
BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).
Formula:
C31H36F3N7O5
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
643.66
Ref: TM-T10539
| 1mg | 95.00 € | ||
| 2mg | 143.00 € | ||
| 5mg | 218.00 € | ||
| 10mg | 385.00 € | ||
| 25mg | 640.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,226.00 € | ||
| 1mL*10mM (DMSO) | 329.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
L-DOPA
CAS:59-92-7
L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is …
Formula:
C9H11NO4
Purity:
99.16% - 99.99%
Color and Shape:
Colorless To White Crystals Or Crystalline Powder; Needles From Water Solid
Molecular weight:
197.19
Ref: TM-T0848
| 200mg | 54.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
JNJ-18038683
CAS:851376-05-1
JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for …
Formula:
C26H28ClN3O7
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
529.97
Ref: TM-T11720
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 373.00 € | ||
| 200mg | 530.00 € | ||
| 1mL*10mM (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dexchlorpheniramine Maleate
CAS:2438-32-6
Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active …
Formula:
C20H23ClN2O4
Purity:
98.49%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
390.86
Ref: TM-T0785
| 100mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Quetiapine hemifumarate
CAS:111974-72-2
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, …
Formula:
C46H54N6O8S2
Purity:
100% - 97.63%
Color and Shape:
White Crystalline Solid
Molecular weight:
883.09
Ref: TM-T6241
| 1g | 53.00 € | ||
| 200mg | 40.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Promethazine hydrochloride
CAS:58-33-3
Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
Formula:
C17H20N2S·HCl
Purity:
95.36%
Color and Shape:
Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
Molecular weight:
320.88
Ref: TM-T0445L
| 1g | 34.00 € | ||
| 5g | 47.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fezolinetant
CAS:1629229-37-3
Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective …
Formula:
C16H15FN6OS
Purity:
98.62% - 99.70%
Color and Shape:
Solid
Molecular weight:
358.39
Ref: TM-T15278
| 1mg | 79.00 € | ||
| 5mg | 146.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 453.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 1,095.00 € | ||
| 1mL*10mM (DMSO) | 161.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pemirolast potassium
CAS:100299-08-9
Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.
Formula:
C10H7KN6O
Purity:
98.91% - 99.63%
Color and Shape:
Crystals From Dimethylformamide Crystalline Solid
Molecular weight:
266.31
Ref: TM-T1425
| 5mg | 35.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 162.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Labetalol
CAS:36894-69-6
Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.
Formula:
C19H24N2O3
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
328.41
Ref: TM-T20570
| 10mg | 42.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 210.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Meptazinol hydrochloride
CAS:59263-76-2
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic …
Formula:
C15H23NO·HCl
Purity:
99.83%
Color and Shape:
White Solid
Molecular weight:
269.81
Ref: TM-T0201
| 5mg | 48.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 166.00 € | ||
| 200mg | 222.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
JNJ-39758979
CAS:1046447-90-8
JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).
Formula:
C11H19N5
Purity:
98.00% - 98.3%
Color and Shape:
Solid
Molecular weight:
221.3
Ref: TM-T11723L
| 1mg | 74.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 247.00 € | ||
| 25mg | 419.00 € | ||
| 50mg | 608.00 € | ||
| 100mg | 894.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sodium butanoate
CAS:156-54-7
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity.
Formula:
C4H7NaO2
Purity:
98.02% - 99.44%
Color and Shape:
White Powder
Molecular weight:
110.09
Ref: TM-T1393
| 1g | 52.00 € | ||
| 5g | 93.00 € | ||
| 10g | 139.00 € | ||
| 500mg | 38.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LIT-001
CAS:2245072-21-1
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin …
Formula:
C30H34F3N7O4S
Purity:
96.88% - 98.25%
Color and Shape:
Solid
Molecular weight:
645.7
Ref: TM-T11857
| 1mg | 71.00 € | ||
| 5mg | 154.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 917.00 € | ||
| 500mg | 1,789.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ziprasidone
CAS:146939-27-7
Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects …
Formula:
C21H21ClN4OS
Purity:
100% - 99.53%
Color and Shape:
Tan Solid
Molecular weight:
412.94
Ref: TM-T0031L2
| 10mg | 70.00 € | ||
| 25mg | 98.00 € | ||
| 50mg | 158.00 € | ||
| 100mg | 199.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ticagrelor
CAS:274693-27-5
Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.
Formula:
C23H28F2N6O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
522.57
Ref: TM-T0179
| 1g | 356.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 65.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 107.00 € | ||
| 200mg | 151.00 € | ||
| 500mg | 240.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bromperidol
CAS:10457-90-6
Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
Formula:
C21H23BrFNO2
Purity:
99.89%
Color and Shape:
Tan Solid
Molecular weight:
420.32
Ref: TM-T14830
| 10mg | 43.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(±) Clopidogrel hydrogen sulfate
CAS:135046-48-9
(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, …
Formula:
C16H16ClNO2S·H2SO4
Purity:
98.67% - 99.04%
Color and Shape:
Colorless To Light Yellow Liquid
Molecular weight:
419.9
Ref: TM-T0182L2
| 100mg | 55.00 € | ||
| 200mg | 82.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fipexide
CAS:34161-24-5
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy …
Formula:
C20H21ClN2O4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
388.84
Ref: TM-T0322
| 25mg | 36.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GR 103691
CAS:162408-66-4
GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
Formula:
C30H35N3O3
Purity:
98.94% - 99.29%
Color and Shape:
Solid
Molecular weight:
485.62
Ref: TM-T11463
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 193.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 493.00 € | ||
| 500mg | 1,095.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
