G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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p-MPPI hydrochloride
CAS:220643-77-6
p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.
Formula:
C25H28ClIN4O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
578.87
Ref: TM-T16421
| 1ml | 89.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 366.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
LY2510924 acetate(1088715-84-7 free base)
Ly2510924 acetate is an potent and selective CXCR4 antagonist. It prevents the binding of SDF-1 …
Formula:
C64H91N13O13
Purity:
97.32%
Color and Shape:
Solid
Molecular weight:
1250.49
Ref: TM-T15805L
| 1mg | 156.00 € | ||
| 1ml | 725.00 € | ||
| 5mg | 300.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 735.00 € | ||
| 50mg | 1,006.00 € | ||
| 100mg | 1,389.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Tizanidine hydrochloride
CAS:64461-82-1
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Formula:
C9H9Cl2N5S
Purity:
99.87%
Color and Shape:
Solid White
Molecular weight:
290.17
Ref: TM-T0290
| 1ml | 47.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 131.00 € | ||
| 500mg | 209.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Linaclotide
CAS:851199-59-2
Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.
Formula:
C59H79N15O21S6
Purity:
97.93% - 98.71%
Color and Shape:
Solid
Molecular weight:
1526.74
Ref: TM-T11852
| 1mg | 65.00 € | ||
| 1ml | 268.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 480.00 € | ||
| 100mg | 684.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
NE 52-QQ57
CAS:1401728-56-0
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …
Formula:
C24H28N6O
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T11461
| 1mg | 73.00 € | ||
| 1ml | 168.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 231.00 € | ||
| 25mg | 386.00 € | ||
| 50mg | 573.00 € | ||
| 100mg | 821.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Rupatadine Fumarate
CAS:182349-12-8
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 …
Formula:
C26H26ClN3·C4H4O4
Purity:
99.64%
Color and Shape:
White Or Almost-White Powder
Molecular weight:
532.03
Ref: TM-T6242
| 1g | 180.00 € | ||
| 1ml | 55.00 € | ||
| 25mg | 38.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 125.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Meptazinol hydrochloride
CAS:59263-76-2
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic …
Formula:
C15H23NO·HCl
Purity:
99.83%
Color and Shape:
White Solid
Molecular weight:
269.81
Ref: TM-T0201
| 1ml | 55.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 166.00 € | ||
| 200mg | 222.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
L-DOPA
CAS:59-92-7
L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is …
Formula:
C9H11NO4
Purity:
99.16% - 99.99%
Color and Shape:
Colorless To White Crystals Or Crystalline Powder; Needles From Water Solid
Molecular weight:
197.19
Ref: TM-T0848
| 200mg | 54.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
AH 6809
CAS:33458-93-4
AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse …
Formula:
C17H14O5
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
298.29
Ref: TM-T14148
| 1ml | 71.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Protriptyline hydrochloride
CAS:1225-55-4
Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.
Formula:
C19H21N·HCl
Purity:
98.54% - 99.98%
Color and Shape:
Solid
Molecular weight:
299.84
Ref: TM-T0204
| 1ml | 36.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 153.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Azacyclonol
CAS:115-46-8
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
Formula:
C18H21NO
Purity:
99.61%
Color and Shape:
Solid Powder
Molecular weight:
267.37
Ref: TM-T0318
| 1g | 34.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
NTP42
CAS:2055599-51-2
NTP42 is an antagonist of thromboxane A2 (TXA2) receptor(IC50 of 3.278 nM)
Formula:
C25H23F2N3O5S
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
515.53
Ref: TM-T12268
| 1mg | 39.00 € | ||
| 1ml | 92.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 446.00 € | ||
| 200mg | 621.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Labetalol hydrochloride
CAS:32780-64-6
Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic …
Formula:
C19H25ClN2O3
Purity:
99.29% - 99.85%
Color and Shape:
Solid
Molecular weight:
364.87
Ref: TM-T0348
| 1ml | 63.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 112.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
NEO 376
CAS:496921-73-4
NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing …
Formula:
C20H24ClN3O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
357.88
Ref: TM-T12207
| 1mg | 72.00 € | ||
| 1ml | 150.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 208.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 504.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 909.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ticlopidine hydrochloride
CAS:53885-35-1
Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement …
Formula:
C14H15Cl2NS
Purity:
99.82% - 99.98%
Color and Shape:
White Powder
Molecular weight:
300.25
Ref: TM-T0362
| 1ml | 36.00 € | ||
| 200mg | 34.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fezagepras
CAS:1002101-19-0
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist …
Formula:
C13H18O2
Purity:
96.73% - 99.38%
Color and Shape:
Solid
Molecular weight:
206.28
Ref: TM-T12883
| 1mg | 52.00 € | ||
| 1ml | 92.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 4 Oct 2024
MP-A08
CAS:219832-49-2
MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 …
Formula:
C27H25N3O4S2
Purity:
98.04%
Color and Shape:
Solid
Molecular weight:
519.64
Ref: TM-T16128
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 313.00 € | ||
| 200mg | 436.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Amantadine hydrochloride
CAS:665-66-7
Amantadine hydrochloride (CI-719) is an antiviral that is used in the prophylactic or symptomatic treatment …
Formula:
C10H18ClN
Purity:
99.86%
Color and Shape:
Solid Crystalline
Molecular weight:
187.71
Ref: TM-T1406
| 1g | 39.00 € | ||
| 5g | 57.00 € | ||
| 1ml | 36.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Risperidone
CAS:106266-06-2
Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 …
Formula:
C23H27FN4O2
Purity:
100%
Color and Shape:
Crystalline Solid
Molecular weight:
410.48
Ref: TM-T0351
| 1ml | 53.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 203.00 € | ||
| 500mg | 338.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Docusate sodium
CAS:577-11-7
Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to …
Formula:
C20H37NaO7S
Purity:
99.77%
Color and Shape:
White Wax-Like Solid With Water (Uscg 1999)
Molecular weight:
444.56
Ref: TM-T0929
| 1ml | 55.00 € | ||
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 500mg | 120.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
