G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Pemirolast potassium
CAS:100299-08-9
Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.
Formula:
C10H7KN6O
Purity:
98.91% - 99.63%
Color and Shape:
Crystals From Dimethylformamide Crystalline Solid
Molecular weight:
266.31
Ref: TM-T1425
| 5mg | 35.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 162.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Ziprasidone hydrochloride
CAS:122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows …
Formula:
C21H22CL2N4OS
Purity:
98.37% - 99.34%
Color and Shape:
Solid
Molecular weight:
449.4
Ref: TM-T0031L
| 5mg | 44.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 163.00 € | ||
| 500mg | 388.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Promazine hydrochloride
CAS:53-60-1
Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
Formula:
C17H21ClN2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
320.88
Ref: TM-T0766
| 1g | 49.00 € | ||
| 5g | 94.00 € | ||
| 10g | 139.00 € | ||
| 500mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Ursodeoxycholic acid
CAS:128-13-2
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
Formula:
C24H40O4
Purity:
99.74% - ≥95%
Color and Shape:
White - Almost White Solid Powder
Molecular weight:
392.57
Ref: TM-T0700
| 1g | 54.00 € | ||
| 5g | 111.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 66.00 € | ||
| 500mg | 53.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Metipranolol
CAS:22664-55-7
Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic …
Formula:
C17H27NO4
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
309.4
Ref: TM-T8899
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 473.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Atenolol
CAS:29122-68-7
Atenolol (Tenormin) is a selective β1 receptor antagonist.
Formula:
C14H22N2O3
Purity:
99.07%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
266.3361
Ref: TM-T0007
| 1ml | 54.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Alverine citrate
CAS:5560-59-8
Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
Formula:
C26H35NO7
Purity:
100% - 99.83%
Color and Shape:
Coa
Molecular weight:
473.57
Ref: TM-T0428
| 1g | 80.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
MRS-1706
CAS:264622-53-9
MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.
Formula:
C27H29N5O5
Purity:
97.95%
Color and Shape:
Solid
Molecular weight:
503.55
Ref: TM-T16136
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 678.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
N6-Cyclohexyladenosine
CAS:36396-99-3
N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.
Formula:
C16H23N5O4
Purity:
99.84% - 99.98%
Color and Shape:
Solid
Molecular weight:
349.38
Ref: TM-T12160
| 10mg | 34.00 € | ||
| 25mg | 60.00 € | ||
| 50mg | 101.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Pizotifen
CAS:15574-96-6
Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available …
Formula:
C19H21NS
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
295.44
Ref: TM-T1442
| 1g | 104.00 € | ||
| 100mg | 35.00 € | ||
| 500mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist.
Formula:
C10H13ClN4O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
256.69
Ref: TM-T15432
| 1mg | 72.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 633.00 € | ||
| 100mg | 900.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Alfuzosin hydrochloride
CAS:81403-68-1
Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign …
Formula:
C19H27N5O4·HCl
Purity:
99.61%
Color and Shape:
White To Off-White Solid
Molecular weight:
425.91
Ref: TM-T0091
| 10mg | 44.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 151.00 € | ||
| 200mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
JNJ-18038683
CAS:851376-05-1
JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for …
Formula:
C26H28ClN3O7
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
529.97
Ref: TM-T11720
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 373.00 € | ||
| 200mg | 530.00 € | ||
| 1mL*10mM (DMSO) | 54.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Solabegron
CAS:252920-94-8
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese …
Formula:
C23H23ClN2O3
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T12970
| 1mg | 57.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 459.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 825.00 € | ||
| 200mg | 1,090.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
PF429242 dihydrochloride
CAS:2248666-66-0
PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Formula:
C25H37Cl2N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
482.49
Ref: TM-T12437
| 1mg | 43.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Mebhydrolin napadisylate
CAS:6153-33-9
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, …
Formula:
C19H20N2C10H8O6S2
Purity:
99.35% - 99.77%
Color and Shape:
White Or Almost White Crystalline
Molecular weight:
420.52
Ref: TM-T0113
| 1g | 62.00 € | ||
| 5g | 131.00 € | ||
| 10g | 182.00 € | ||
| 500mg | 45.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Urapidil hydrochloride
CAS:64887-14-5
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Formula:
C20H29N5O3·HCl
Purity:
99.93%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
423.94
Ref: TM-T0088
| 1g | 132.00 € | ||
| 100mg | 45.00 € | ||
| 200mg | 60.00 € | ||
| 500mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Naftopidil
CAS:57149-07-2
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as …
Formula:
C24H28N2O3
Purity:
99.4% - 99.97%
Color and Shape:
White Crystalline Powder
Molecular weight:
392.49
Ref: TM-T0696
| 1g | 68.00 € | ||
| 500mg | 46.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
LY2940094
CAS:1307245-86-8
LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
Formula:
C22H23ClF2N4O2S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
480.96
Ref: TM-T15799
| 1mg | 80.00 € | ||
| 2mg | 105.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 270.00 € | ||
| 25mg | 533.00 € | ||
| 50mg | 764.00 € | ||
| 100mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
