G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Sumatriptan succinate
CAS:103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment …
Formula:
C18H27N3O6S
Purity:
97.53% - 99.51%
Color and Shape:
White Powder
Molecular weight:
413.49
Ref: TM-T0203
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 74.00 € | ||
| 500mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Spiperone
CAS:749-02-0
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
Formula:
C23H26FN3O2
Purity:
99.34% - 99.89%
Color and Shape:
Solid
Molecular weight:
395.47
Ref: TM-T0280
| 5mg | 47.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
L-DOPA
CAS:59-92-7
L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is …
Formula:
C9H11NO4
Purity:
99.16% - 99.99%
Color and Shape:
Colorless To White Crystals Or Crystalline Powder; Needles From Water Solid
Molecular weight:
197.19
Ref: TM-T0848
| 200mg | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Mizolastine
CAS:108612-45-9
Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever …
Formula:
C24H25FN6O
Purity:
98% - 99.77%
Color and Shape:
Solid
Molecular weight:
432.49
Ref: TM-T0118
| 10mg | 42.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 177.00 € | ||
| 500mg | 298.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Meptazinol hydrochloride
CAS:59263-76-2
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic …
Formula:
C15H23NO·HCl
Purity:
99.83%
Color and Shape:
White Solid
Molecular weight:
269.81
Ref: TM-T0201
| 5mg | 48.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 168.00 € | ||
| 200mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Buflomedil hydrochloride
CAS:35543-24-9
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of …
Formula:
C17H26ClNO4
Purity:
99.67% - 99.7%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
343.85
Ref: TM-T0317
| 1g | 86.00 € | ||
| 5g | 180.00 € | ||
| 100mg | 42.00 € | ||
| 500mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Quetiapine hemifumarate
CAS:111974-72-2
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, …
Formula:
C46H54N6O8S2
Purity:
100% - 97.63%
Color and Shape:
White Crystalline Solid
Molecular weight:
883.09
Ref: TM-T6241
| 1g | 52.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Rupatadine Fumarate
CAS:182349-12-8
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 …
Formula:
C26H26ClN3·C4H4O4
Purity:
99.64%
Color and Shape:
White Or Almost-White Powder
Molecular weight:
532.03
Ref: TM-T6242
| 1g | 183.00 € | ||
| 25mg | 38.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 70.00 € | ||
| 500mg | 127.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
NE 52-QQ57
CAS:1401728-56-0
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …
Formula:
C24H28N6O
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T11461
| 1mg | 73.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 394.00 € | ||
| 50mg | 587.00 € | ||
| 100mg | 835.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Linaclotide
CAS:851199-59-2
Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.
Formula:
C59H79N15O21S6
Purity:
97.93% - 98.71%
Color and Shape:
Solid
Molecular weight:
1526.74
Ref: TM-T11852
| 1mg | 66.00 € | ||
| 2mg | 93.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 490.00 € | ||
| 100mg | 700.00 € | ||
| 1mL*10mM (DMSO) | 269.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Tizanidine hydrochloride
CAS:64461-82-1
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Formula:
C9H9Cl2N5S
Purity:
99.87%
Color and Shape:
Solid White
Molecular weight:
290.17
Ref: TM-T0290
| 10mg | 51.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 105.00 € | ||
| 200mg | 133.00 € | ||
| 500mg | 212.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
p-MPPI hydrochloride
CAS:220643-77-6
p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.
Formula:
C25H28ClIN4O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
578.87
Ref: TM-T16421
| 10mg | 93.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 371.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Pizotifen Malate
CAS:5189-11-7
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based …
Formula:
C19H21NS·C4H6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
429.53
Ref: TM-T0225
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Moxisylyte hydrochloride
CAS:964-52-3
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Formula:
C16H26ClNO3
Purity:
99.93% - ≥95%
Color and Shape:
Solid
Molecular weight:
315.84
Ref: TM-T0394
| 50mg | 43.00 € | ||
| 100mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Deoxycholic acid
CAS:83-44-3
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.
Formula:
C24H40O4
Purity:
99.35%
Color and Shape:
Crystals From Alc Solid
Molecular weight:
392.57
Ref: TM-T2965
| 100mg | 58.00 € | ||
| 500mg | 79.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Metaraminol tartrate
CAS:33402-03-8
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.
Formula:
C13H19NO8
Purity:
99.53%
Color and Shape:
White Powder
Molecular weight:
317.29
Ref: TM-T0279
| 50mg | 46.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 87.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Fluoxetine
CAS:54910-89-3
Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.
Formula:
C17H18F3NO
Purity:
99.07% - 99.28%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T0450
| 10mg | 35.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 81.00 € | ||
| 200mg | 120.00 € | ||
| 500mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Alvimopan
CAS:156053-89-3
Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
Formula:
C25H32N2O4
Purity:
99.78% - 99.97%
Color and Shape:
Solid
Molecular weight:
424.53
Ref: TM-T1242
| 1mg | 49.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 560.00 € | ||
| 500mg | 1,216.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
BTRX-335140
CAS:2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic …
Formula:
C25H32FN5O2
Purity:
98% - 98.45%
Color and Shape:
Solid
Molecular weight:
453.55
Ref: TM-T14835
| 1mg | 105.00 € | ||
| 2mg | 155.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 406.00 € | ||
| 25mg | 840.00 € | ||
| 50mg | 1,378.00 € | ||
| 100mg | 1,882.00 € | ||
| 200mg | 2,632.00 € | ||
| 1mL*10mM (DMSO) | 283.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Quetiapine
CAS:111974-69-7
Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine …
Formula:
C21H25N3O2S
Purity:
100% - 99.14%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
383.51
Ref: TM-T0162
| 10mg | 55.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
