G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ESI-05
CAS:5184-64-5
ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and …
Formula:
C16H18O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
274.38
Ref: TM-T15247
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 270.00 € | ||
| 100mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
hGPR91 antagonist 1
CAS:1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Formula:
C31H23F4N3O
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
529.53
Ref: TM-T11560
| 1mg | 95.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 298.00 € | ||
| 25mg | 507.00 € | ||
| 50mg | 692.00 € | ||
| 100mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 224.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Bendazol
CAS:621-72-7
Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.
Formula:
C14H12N2
Purity:
98.7% - 99.81%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
208.26
Ref: TM-T1322
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Diphenhydramine hydrochloride
CAS:147-24-0
DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.
Formula:
C17H22ClNO
Purity:
99.84%
Color and Shape:
Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)
Molecular weight:
291.82
Ref: TM-T0330
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Diphenylpyraline hydrochloride
CAS:132-18-3
Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
Formula:
C19H23NO·HCl
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
317.85
Ref: TM-T0059
| 500mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Isoxsuprine hydrochloride
CAS:579-56-6
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular …
Formula:
C18H24ClNO3
Purity:
99.38%
Color and Shape:
Crystals From Water Solid
Molecular weight:
337.84
Ref: TM-T0324
| 200mg | 35.00 € | ||
| 500mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Granisetron hydrochloride
CAS:107007-99-8
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used …
Formula:
C18H25ClN4O
Purity:
99.88% - 99.93%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
348.87
Ref: TM-T1042
| 10mg | 38.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 127.00 € | ||
| 200mg | 178.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Acetophenazine dimaleate
CAS:5714-00-1
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the …
Formula:
C31H37N3O10S
Purity:
99.39% - 99.48%
Color and Shape:
Solid
Molecular weight:
643.71
Ref: TM-T10232
| 2mg | 42.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 183.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Fenoterol
CAS:13392-18-2
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and …
Formula:
C17H21NO4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
303.35
Ref: TM-T8358
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 230.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Indacaterol maleate
CAS:753498-25-8
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
Formula:
C28H32N2O7
Purity:
99.03% - 99.67%
Color and Shape:
Solid
Molecular weight:
508.56
Ref: TM-T1239
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 145.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Nicergoline
CAS:27848-84-6
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with …
Formula:
C24H26BrN3O3
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
484.39
Ref: TM-T1132
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 145.00 € | ||
| 500mg | 234.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Adrenalone hydrochloride
CAS:62-13-5
Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
Formula:
C9H11NO3·HCl
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
217.65
Ref: TM-T0948
| 1g | 145.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 50.00 € | ||
| 500mg | 97.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Ticagrelor
CAS:274693-27-5
Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.
Formula:
C23H28F2N6O4S
Purity:
98.08% - 99.77%
Color and Shape:
Solid
Molecular weight:
522.57
Ref: TM-T0179
| 1g | 364.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 66.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 154.00 € | ||
| 500mg | 245.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
JNJ-39758979
CAS:1046447-90-8
JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).
Formula:
C11H19N5
Purity:
98.3% - 99.62%
Color and Shape:
Solid
Molecular weight:
221.3
Ref: TM-T11723L
| 1mg | 74.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 905.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Aripiprazole
CAS:129722-12-9
Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
Formula:
C23H27Cl2N3O2
Purity:
99.43% - 99.62%
Color and Shape:
Colourless Flake Crystalline Solid
Molecular weight:
448.39
Ref: TM-T1566
| 1g | 133.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 84.00 € | ||
| 500mg | 101.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Aniracetam
CAS:72432-10-1
Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and …
Formula:
C12H13NO3
Purity:
99.89%
Color and Shape:
White Crystalline Or Crystalline Powde
Molecular weight:
219.24
Ref: TM-T0333
| 1g | 52.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Chlorprothixene hydrochloride
CAS:6469-93-8
Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
Formula:
C18H18ClNS·HCl
Purity:
99.16%
Color and Shape:
White Powder
Molecular weight:
352.32
Ref: TM-T0074L
| 100mg | 37.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Domperidone
CAS:57808-66-9
Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Formula:
C22H24ClN5O2
Purity:
98% - 99.82%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T0082
| 50mg | 46.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 89.00 € | ||
| 500mg | 145.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
2-Bromo-6-methoxynaphthalene
CAS:5111-65-9
2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.
Formula:
C11H9BrO
Purity:
98.51%
Color and Shape:
White To Off-White Powder
Molecular weight:
237.09
Ref: TM-T0663
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Levocetirizine
CAS:130018-77-8
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a …
Formula:
C21H25ClN2O3
Purity:
98% - 99.9%
Color and Shape:
White Powder
Molecular weight:
388.89
Ref: TM-T1469
| 5mg | 38.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 258.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
