G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Histamine
CAS:51-45-6
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE.
Formula:
C5H9N3
Purity:
100% - 96.63%
Color and Shape:
Needles From Chloroform Solid
Molecular weight:
111.15
Ref: TM-T0965
| 50mg | 47.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 78.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Pemirolast potassium
CAS:100299-08-9
Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.
Formula:
C10H7KN6O
Purity:
98.91% - 99.63%
Color and Shape:
Crystals From Dimethylformamide Crystalline Solid
Molecular weight:
266.31
Ref: TM-T1425
| 5mg | 35.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 162.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ifenprodil
CAS:23210-56-2
Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, …
Formula:
C21H27NO2
Purity:
99.78%
Color and Shape:
White Crystalline Powder
Molecular weight:
325.44
Ref: TM-T1186L
| 1mg | 106.00 € | ||
| 1ml | 217.00 € | ||
| 5mg | 208.00 € | ||
| 10mg | 312.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 897.00 € | ||
| 200mg | 1,235.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Trazodone hydrochloride
CAS:25332-39-2
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive …
Formula:
C19H23Cl2N5O
Purity:
99.50% - 99.52%
Color and Shape:
Solid
Molecular weight:
408.33
Ref: TM-T1619
| 1ml | 36.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 57.00 € | ||
| 500mg | 83.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Bromopride
CAS:4093-35-0
Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the …
Formula:
C14H22BrN3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
344.25
Ref: TM-T1175
| 1mg | 39.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 390.00 € | ||
| 100mg | 554.00 € | ||
| 200mg | 773.00 € | ||
| 500mg | 1,180.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Agomelatine
CAS:138112-76-2
Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
Formula:
C15H17NO2
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
243.3
Ref: TM-T1445
| 1ml | 69.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 732.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Prucalopride
CAS:179474-81-8
Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these …
Formula:
C18H26ClN3O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
367.87
Ref: TM-T2542
| 1ml | 36.00 € | ||
| 10mg | 45.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
2-(1-Piperazinyl)pyrimidine
CAS:20980-22-7
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Formula:
C8H12N4
Purity:
98.86%
Color and Shape:
Liquid - Crystal - Lump
Molecular weight:
164.21
Ref: TM-T1696
| 1g | 38.00 € | ||
| 1ml | 49.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Alosetron hydrochloride
CAS:122852-69-1
Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin …
Formula:
C17H19ClN4O
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
330.81
Ref: TM-T2525
| 10mg | 36.00 € | ||
| 25mg | 76.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 256.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Adrenalone hydrochloride
CAS:62-13-5
Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
Formula:
C9H11NO3·HCl
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
217.65
Ref: TM-T0948
| 50mg | 54.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 100.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Moxisylyte hydrochloride
CAS:964-52-3
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Formula:
C16H26ClNO3
Purity:
98% - 99.97%
Color and Shape:
Solid
Molecular weight:
315.84
Ref: TM-T0394
| 1ml | 52.00 € | ||
| 50mg | 42.00 € | ||
| 100mg | 54.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Loperamide hydrochloride
CAS:34552-83-5
Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
Formula:
C29H34Cl2N2O2
Purity:
100% - 99.78%
Color and Shape:
Crystals Practically Insoluble In Water
Molecular weight:
513.498
Ref: TM-T0209
| 1ml | 55.00 € | ||
| 100mg | 59.00 € | ||
| 500mg | 88.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Indacaterol maleate
CAS:753498-25-8
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
Formula:
C28H32N2O7
Purity:
99.03% - 99.67%
Color and Shape:
Solid
Molecular weight:
508.56
Ref: TM-T1239
| 1ml | 55.00 € | ||
| 10mg | 36.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 100.00 € | ||
| 200mg | 149.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Olodaterol
CAS:868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding …
Formula:
C21H26N2O5
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T3457
| 1mg | 69.00 € | ||
| 2mg | 111.00 € | ||
| 5mg | 193.00 € | ||
| 10mg | 289.00 € | ||
| 25mg | 579.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Alprenolol
CAS:13655-52-2
Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of …
Formula:
C15H23NO2
Purity:
99.73% - 99.78%
Color and Shape:
Solid
Molecular weight:
249.35
Ref: TM-T4560
| 50mg | 52.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fenoterol
CAS:13392-18-2
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and …
Formula:
C17H21NO4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
303.35
Ref: TM-T8358
| 1ml | 71.00 € | ||
| 2mg | 38.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 4 Oct 2024
Bisoprolol hemifumarate
CAS:104344-23-2
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 …
Formula:
C20H33NO6
Purity:
99% - 99.95%
Color and Shape:
White To Offf-White Powder
Molecular weight:
383.49
Ref: TM-T0143
| 1ml | 56.00 € | ||
| 50mg | 51.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Metoprolol tartrate
CAS:56392-17-7
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
Formula:
C15H25NO3C4H6O6
Purity:
99.72% - 99.93%
Color and Shape:
White To Off-White / Powder
Molecular weight:
684.81
Ref: TM-T0487
| 1ml | 67.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 71.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Alvimopan
CAS:156053-89-3
Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
Formula:
C25H32N2O4
Purity:
99.78% - 99.97%
Color and Shape:
Solid
Molecular weight:
424.53
Ref: TM-T1242
| 1mg | 49.00 € | ||
| 1ml | 88.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 552.00 € | ||
| 500mg | 1,189.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Phentolamine mesylate
CAS:65-28-1
Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.
Formula:
C17H19N3O·CH4O3S
Purity:
99.77% - 99.9%
Color and Shape:
By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
Molecular weight:
377.46
Ref: TM-T1275
| 1ml | 55.00 € | ||
| 100mg | 60.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 152.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
