G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Quetiapine
CAS:111974-69-7
Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine …
Formula:
C21H25N3O2S
Purity:
100% - 99.14%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
383.51
Ref: TM-T0162
| 10mg | 59.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 118.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Fluoxetine
CAS:54910-89-3
Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.
Formula:
C17H18F3NO
Purity:
99.07% - 99.28%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T0450
| 10mg | 40.00 € | ||
| 25mg | 53.00 € | ||
| 50mg | 67.00 € | ||
| 100mg | 85.00 € | ||
| 200mg | 124.00 € | ||
| 500mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Metaraminol tartrate
CAS:33402-03-8
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.
Formula:
C13H19NO8
Purity:
99.53%
Color and Shape:
White Powder
Molecular weight:
317.29
Ref: TM-T0279
| 50mg | 50.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 90.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Pizotifen Malate
CAS:5189-11-7
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based …
Formula:
C19H21NS·C4H6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
429.53
Ref: TM-T0225
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Buflomedil hydrochloride
CAS:35543-24-9
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of …
Formula:
C17H26ClNO4
Purity:
99.67% - 99.7%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
343.85
Ref: TM-T0317
| 1g | 84.00 € | ||
| 5g | 175.00 € | ||
| 100mg | 41.00 € | ||
| 500mg | 58.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Spiperone
CAS:749-02-0
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
Formula:
C23H26FN3O2
Purity:
99.34% - 99.89%
Color and Shape:
Solid
Molecular weight:
395.47
Ref: TM-T0280
| 5mg | 46.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Sumatriptan succinate
CAS:103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment …
Formula:
C18H27N3O6S
Purity:
97.53% - 99.51%
Color and Shape:
White Powder
Molecular weight:
413.49
Ref: TM-T0203
| 50mg | 41.00 € | ||
| 100mg | 55.00 € | ||
| 500mg | 147.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Betaxolol hydrochloride
CAS:63659-19-8
Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.
Formula:
C18H30ClNO3
Purity:
98.64% - 99.56%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T0226
| 25mg | 37.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 82.00 € | ||
| 200mg | 92.00 € | ||
| 500mg | 154.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Eletriptan hydrobromide
CAS:177834-92-3
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D …
Formula:
C22H27BrN2O2S
Purity:
100% - 97.8%
Color and Shape:
Tan Solid
Molecular weight:
463.43
Ref: TM-T0216
| 5mg | 36.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 325.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
CE3F4
CAS:143703-25-7
CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of …
Formula:
C11H10Br2FNO
Purity:
97% - 97.15%
Color and Shape:
Solid
Molecular weight:
351.01
Ref: TM-T12616L
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 273.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Sertraline hydrochloride
CAS:79559-97-0
Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the …
Formula:
C17H18Cl3N
Purity:
99.12% - 99.86%
Color and Shape:
Solid Powder
Molecular weight:
342.691
Ref: TM-T0482
| 5mg | 51.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 298.00 € | ||
| 500mg | 507.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
(R)-Terazosin
CAS:109351-34-0
R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 …
Formula:
C19H25N5O4
Purity:
98.87% - 98.96%
Color and Shape:
Solid
Molecular weight:
387.43
Ref: TM-T12643
| 1mg | 46.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 484.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Bromperidol
CAS:10457-90-6
Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
Formula:
C21H23BrFNO2
Purity:
99.89%
Color and Shape:
Tan Solid
Molecular weight:
420.32
Ref: TM-T14830
| 10mg | 43.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Itopride hydrochloride
CAS:122892-31-3
Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
Formula:
C20H27ClN2O4
Purity:
99.76%
Color and Shape:
White Or Pale Brownish Crystal
Molecular weight:
394.9
Ref: TM-T1552
| 50mg | 41.00 € | ||
| 100mg | 54.00 € | ||
| 500mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Chlorpheniramine maleate
CAS:113-92-8
Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, …
Formula:
C20H23ClN2O4
Purity:
99.67%
Color and Shape:
Odorless White Crystalline Solid Or White Powder With A Bitter Taste
Molecular weight:
390.87
Ref: TM-T1553
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
BP 897 hydrochloride
CAS:314776-92-6
BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low …
Formula:
C26H32ClN3O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T14767
| 1mg | 36.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
ONC206
CAS:1638178-87-6
ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the …
Formula:
C23H22F2N4O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T16392
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Pranlukast
CAS:103177-37-3
Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.
Formula:
C27H23N5O4
Purity:
99.85%
Color and Shape:
Off-White Solid
Molecular weight:
481.5
Ref: TM-T0694
| 25mg | 54.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 124.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
Prasugrel
CAS:150322-43-3
Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent …
Formula:
C20H20FNO3S
Purity:
98.62% - 99.76%
Color and Shape:
White Solid
Molecular weight:
373.44
Ref: TM-T0230
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 76.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 190.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 26 Nov 2024
