G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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p-MPPI hydrochloride
CAS:220643-77-6
p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.
Formula:
C25H28ClIN4O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
578.87
Ref: TM-T16421
| 10mg | 91.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 366.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CE3F4
CAS:143703-25-7
CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of …
Formula:
C11H10Br2FNO
Purity:
97% - 97.15%
Color and Shape:
Solid
Molecular weight:
351.01
Ref: TM-T12616L
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 273.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sulpiride
CAS:15676-16-1
Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as …
Formula:
C15H23N3O4S
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
341.43
Ref: TM-T1201
| 50mg | 43.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 69.00 € | ||
| 500mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tetrahydrozoline
CAS:84-22-0
Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the …
Formula:
C13H16N2
Purity:
97.85% - 99.77%
Color and Shape:
Solid
Molecular weight:
200.28
Ref: TM-T0397
| 10mg | 28.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 115.00 € | ||
| 500mg | 186.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Reparixin L-lysine salt
CAS:266359-93-7
Reparixin L-lysine salt (Repertaxin L-lysine salt) is an allosteric chemokine receptor 1/2 (CXCR1/2) activation inhibitor.
Formula:
C20H35N3O5S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
429.57
Ref: TM-T12705
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alverine citrate
CAS:5560-59-8
Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
Formula:
C26H35NO7
Purity:
100% - 99.83%
Color and Shape:
Coa
Molecular weight:
473.57
Ref: TM-T0428
| 1g | 80.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CYM50308
CAS:1345858-76-5
CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).
Formula:
C20H21F2N3O2S
Purity:
99.43% - 99.63%
Color and Shape:
Solid
Molecular weight:
405.46
Ref: TM-T15032
| 1mg | 61.00 € | ||
| 5mg | 139.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 321.00 € | ||
| 50mg | 450.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 831.00 € | ||
| 500mg | 1,197.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Eletriptan hydrobromide
CAS:177834-92-3
Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D …
Formula:
C22H27BrN2O2S
Purity:
100% - 97.8%
Color and Shape:
Tan Solid
Molecular weight:
463.43
Ref: TM-T0216
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 422.00 € | ||
| 200mg | 549.00 € | ||
| 500mg | 871.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Centanafadine hydrochloride
CAS:923981-14-0
Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA …
Formula:
C15H16ClN
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
245.75
Ref: TM-T10758L
| 1mg | 59.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 639.00 € | ||
| 100mg | 1,003.00 € | ||
| 200mg | 1,346.00 € | ||
| 500mg | 2,006.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Betaxolol hydrochloride
CAS:63659-19-8
Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.
Formula:
C18H30ClNO3
Purity:
98.64% - 99.56%
Color and Shape:
Solid
Molecular weight:
343.89
Ref: TM-T0226
| 25mg | 37.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 82.00 € | ||
| 200mg | 92.00 € | ||
| 500mg | 154.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alvimopan
CAS:156053-89-3
Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
Formula:
C25H32N2O4
Purity:
99.78% - 99.97%
Color and Shape:
Solid
Molecular weight:
424.53
Ref: TM-T1242
| 1mg | 49.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 552.00 € | ||
| 500mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Acetophenazine dimaleate
CAS:5714-00-1
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the …
Formula:
C31H37N3O10S
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
643.71
Ref: TM-T10232
| 2mg | 40.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sumatriptan succinate
CAS:103628-48-4
Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment …
Formula:
C18H27N3O6S
Purity:
97.53% - 99.51%
Color and Shape:
White Powder
Molecular weight:
413.49
Ref: TM-T0203
| 25mg | 53.00 € | ||
| 50mg | 65.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 119.00 € | ||
| 500mg | 244.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Spiperone
CAS:749-02-0
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
Formula:
C23H26FN3O2
Purity:
99.34% - 99.89%
Color and Shape:
Solid
Molecular weight:
395.47
Ref: TM-T0280
| 5mg | 46.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Citalopram hydrobromide
CAS:59729-32-7
Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal …
Formula:
C20H22BrFN2O
Purity:
99.35%
Color and Shape:
White Crystalline Powder
Molecular weight:
405.304
Ref: TM-T1483
| 10mg | 52.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 156.00 € | ||
| 500mg | 243.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mepyramine maleate
CAS:59-33-6
Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and …
Formula:
C21H27N3O5
Purity:
99.7% - 99.71%
Color and Shape:
White Crystalline Powder
Molecular weight:
401.47
Ref: TM-T1232
| 1g | 83.00 € | ||
| 500mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lofepramine
CAS:23047-25-8
Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.
Formula:
C26H27ClN2O
Purity:
98.38%
Color and Shape:
Crystals From Methanol Or Acetone Solid
Molecular weight:
418.96
Ref: TM-T15773
| 2mg | 48.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 396.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Antazoline hydrochloride
CAS:2508-72-7
Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and …
Formula:
C17H19N3·HCl
Purity:
98% - 99.76%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
301.82
Ref: TM-T0092
| 1g | 113.00 € | ||
| 100mg | 41.00 € | ||
| 500mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(+)-Dropropizine
CAS:99291-24-4
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved …
Formula:
C13H20N2O2
Purity:
99.92%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.31
Ref: TM-T0217L
| 1g | 49.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Olinciguat
CAS:1628732-62-6
Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.
Formula:
C21H16F5N7O3
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
509.39
Ref: TM-T16383
| 1mg | 176.00 € | ||
| 5mg | 446.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,375.00 € | ||
| 100mg | 1,821.00 € | ||
| 1mL*10mM (DMSO) | 499.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
