G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GR79236
CAS:124555-18-6
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has …
Formula:
C15H21N5O5
Color and Shape:
Solid
Molecular weight:
351.36
Ref: TM-TQ0136
| 2mg | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GW-1100
CAS:306974-70-9
GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic …
Formula:
C27H25FN4O4S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
520.58
Ref: TM-T15448
| 1mg | 35.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Tamsulosin
CAS:106133-20-4
Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.
Formula:
C20H28N2O5S
Purity:
99.94%
Color and Shape:
White Crystals
Molecular weight:
408.51
Ref: TM-T0210L
| 10mg | 36.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 96.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Spiroxatrine
CAS:1054-88-2
Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the …
Formula:
C22H25N3O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T23382
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 569.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AF-710B
CAS:1235733-73-9
AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors …
Formula:
C20H27N3OS
Purity:
98.62% - 99.89%
Color and Shape:
Solid
Molecular weight:
357.51
Ref: TM-T23649
| 1mg | 311.00 € | ||
| 2mg | 462.00 € | ||
| 5mg | 737.00 € | ||
| 10mg | 1,044.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,039.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Alfuzosin
CAS:81403-80-7
Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and …
Formula:
C19H27N5O4
Purity:
99.64%
Color and Shape:
White Crystaline Powder
Molecular weight:
389.45
Ref: TM-T22232
| 10mg | 47.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 184.00 € | ||
| 500mg | 463.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sumanirole maleate
CAS:179386-44-8
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 …
Formula:
C15H17N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
319.31
Ref: TM-TQ0140
| 2mg | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MRS-3777 hemioxalate
CAS:1186195-57-2
MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its …
Formula:
C17H19N5OC2H2O4
Purity:
97.10%
Color and Shape:
Solid
Molecular weight:
354.39
Ref: TM-T12107
| 1mg | 77.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
445.51
Ref: TM-T39647
| 1mg | 68.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 160.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Kushenol A
CAS:99217-63-7
Kushenol A is a kind of Adenosine 3', 5'-cyclic monophosphate(cAMP)phosphodiesterase inhibitiors, it shows selective alpha-glucosidase …
Formula:
C25H28O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
408.49
Ref: TM-TN1841
| 5mg | 741.00 € | ||
| 1mL*10mM (DMSO) | 1,021.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Atosiban
CAS:90779-69-4
Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions …
Formula:
C43H67N11O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
994.19
Ref: TM-T4996
| 5mg | 67.00 € | ||
| 10mg | 90.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 295.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:27964-99-4
Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant …
Formula:
(C6H14N2O2)x·xHBr
Color and Shape:
Liquid
Molecular weight:
227.102
Ref: TM-T40363
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 212.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neurotensin(8-13)
CAS:60482-95-3
Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) …
Formula:
C38H64N12O8
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
816.99
Ref: TM-T7617
| 1mg | 171.00 € | ||
| 2mg | 277.00 € | ||
| 5mg | 410.00 € | ||
| 10mg | 793.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
L-798106
CAS:244101-02-8
L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and …
Formula:
C27H22BrNO4S
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
536.44
Ref: TM-T15689
| 1mg | 50.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 332.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 855.00 € | ||
| 200mg | 1,129.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Fedovapagon
CAS:347887-36-9
Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder …
Formula:
C27H34N4O3
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
462.58
Ref: TM-T15273
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GAT211
CAS:102704-40-5
GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study …
Formula:
C22H18N2O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
342.39
Ref: TM-T27405
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 322.00 € | ||
| 500mg | 776.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Setiptiline
CAS:57262-94-9
Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with …
Formula:
C19H19N
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
261.36
Ref: TM-T12900
| 5mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MRGPRX4 modulator-2
CAS:2492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value …
Formula:
C15H9ClF4O3
Purity:
99.24%
Color and Shape:
Liquid
Molecular weight:
348.68
Ref: TM-T61183
| 1mg | 61.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Virodhamine
CAS:287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of …
Formula:
C22H37NO2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
347.53
Ref: TM-T64371
| 2mg | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dihydromunduletone
CAS:674786-20-0
Dihydromunduletone (DHM) is an adhesion G protein-coupled receptor (aGPCR) antagonist inhibits GPR56 and GPR114/ADGRG5, which …
Formula:
C25H28O6
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
424.49
Ref: TM-T11044
| 1mg | 172.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
