G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Sumanirole maleate
CAS:179386-44-8
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 …
Formula:
C15H17N3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
319.31
Ref: TM-TQ0140
| 2mg | 89.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Furprofen
CAS:66318-17-0
Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain …
Formula:
C14H12O4
Purity:
98.56% - 99.32%
Color and Shape:
Solid
Molecular weight:
244.24
Ref: TM-T11340
| 1mg | 50.00 € | ||
| 1ml | 106.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 293.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 743.00 € | ||
| 500mg | 1,526.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-543 Citrate
CAS:1415562-83-2
PF-543 Citrate is an inhibitor of sphingosine-competitive SPHK1(IC50 of 2 nM ).
Formula:
C33H39NO11S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
657.73
Ref: TM-T12436
| 2mg | 51.00 € | ||
| 5mg | 83.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
3-Hydroxy agomelatine
CAS:166526-99-4
3-Hydroxy agomelatine is an Agomelatine metabolite and a 5-HT2C receptor antagonist (IC50: 3.2 μM; Ki: …
Formula:
C15H17NO3
Color and Shape:
Solid
Molecular weight:
259.3
Ref: TM-T10114
| 1mg | 62.00 € | ||
| 5mg | 161.00 € | ||
| 10mg | 215.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 529.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Nebentan potassium
CAS:342005-82-7
Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is …
Formula:
C24H20KN5O5S
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
529.61
Ref: TM-T36008
| 1mg | 91.00 € | ||
| 1ml | 225.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 306.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,174.00 € | ||
| 500mg | 2,357.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Canagliflozin hemihydrate
CAS:928672-86-0
Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion …
Formula:
C48H52F2O11S2
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
907.05
Ref: TM-T1782L
| 1ml | 51.00 € | ||
| 25mg | 53.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Scopine hydrochloride
CAS:85700-55-6
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.
Formula:
C8H13NO2·HCl
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
191.66
Ref: TM-T6663
| 2mg | 35.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Alfuzosin
CAS:81403-80-7
Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and …
Formula:
C19H27N5O4
Purity:
99.64%
Color and Shape:
White Crystaline Powder
Molecular weight:
389.45
Ref: TM-T22232
| 1ml | 35.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 184.00 € | ||
| 500mg | 463.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ozanimod hydrochloride
CAS:1618636-37-5
Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS …
Formula:
C23H25ClN4O3
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
440.92
Ref: TM-T62552
| 1mg | 66.00 € | ||
| 1ml | 151.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | 409.00 € | ||
| 50mg | 641.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(R)-Mirtazapine
CAS:61364-37-2
(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.
Formula:
C17H19N3
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 481.00 € | ||
| 100mg | 685.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MRGPRX4 modulator-2
CAS:2492595-24-9
MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value …
Formula:
C15H9ClF4O3
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
348.68
Ref: TM-T61183
| 1mg | 61.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 199.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CGP 20712 A
CAS:105737-62-0
CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that …
Formula:
C24H29F3N4O8S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
590.57
Ref: TM-T10778
| 1mg | 146.00 € | ||
| 5mg | 353.00 € | ||
| 10mg | 520.00 € | ||
| 25mg | 824.00 € | ||
| 50mg | 1,110.00 € | ||
| 100mg | 1,489.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T39647
| 1mg | 68.00 € | ||
| 1ml | 160.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 492.00 € | ||
| 100mg | 727.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Atosiban
CAS:90779-69-4
Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions …
Formula:
C43H67N11O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
994.19
Ref: TM-T4996
| 5mg | 67.00 € | ||
| 10mg | 90.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 295.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:27964-99-4
Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant …
Formula:
(C6H14N2O2)x·xHBr
Color and Shape:
Solid
Molecular weight:
227.102
Ref: TM-T40363
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 212.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Dehydroaripiprazole
CAS:129722-25-4
Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.
Formula:
C23H25Cl2N3O2
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
446.37
Ref: TM-T10989
| 1mg | 37.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 342.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,078.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
L-368,899 hydrochloride
CAS:160312-62-9
L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may …
Formula:
C26H43ClN4O5S2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
591.23
Ref: TM-T11794
| 1ml | 211.00 € | ||
| 2mg | 111.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 460.00 € | ||
| 50mg | 720.00 € | ||
| 100mg | 1,010.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
ML224
CAS:1338824-21-7
ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' …
Formula:
C31H31N3O5
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
525.59
Ref: TM-T16106
| 1mg | 57.00 € | ||
| 1ml | 139.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 364.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Trazpiroben
CAS:1352993-39-5
Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.
Formula:
C31H39N3O4
Purity:
98.85% - 99.41%
Color and Shape:
Solid
Molecular weight:
517.66
Ref: TM-T38754
| 1mg | 277.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 933.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,872.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GLP-1R modulator L7-028
CAS:2648317-95-5
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
Formula:
C24H28N2O3
Purity:
98.76% - 98.76%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T40279
| 1mg | 64.00 € | ||
| 5mg | 136.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
