G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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TUG-770
CAS:1402601-82-4
TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 …
Formula:
C19H14FNO2
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
307.32
Ref: TM-TQ0241
| 1mg | 64.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 650.00 € | ||
| 100mg | 933.00 € | ||
| 500mg | 1,872.00 € | ||
| 1mL*10mM (DMSO) | 201.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Fenoprofen
CAS:29679-58-1
Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, …
Formula:
C15H14O3
Color and Shape:
Solid
Molecular weight:
242.27
Ref: TM-T0184L
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 66.00 € | ||
| 100mg | 94.00 € | ||
| 500mg | 196.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
CB1/2 agonist 3
CAS:2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 …
Formula:
C25H41NO2
Color and Shape:
Liquid
Molecular weight:
387.6
Ref: TM-T61736
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 447.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
ML 145
CAS:1164500-72-4
ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)
Formula:
C24H22N2O5S2
Color and Shape:
Solid
Molecular weight:
482.57
Ref: TM-T12074
| 2mg | 88.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 342.00 € | ||
| 50mg | 509.00 € | ||
| 100mg | 731.00 € | ||
| 200mg | 1,049.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Fedovapagon
CAS:347887-36-9
Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder …
Formula:
C27H34N4O3
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
462.58
Ref: TM-T15273
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
(R)-Mirtazapine
CAS:61364-37-2
(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.
Formula:
C17H19N3
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 481.00 € | ||
| 100mg | 685.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Octreotide
CAS:83150-76-9
Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.
Formula:
C49H66N10O10S2
Purity:
99.64%
Color and Shape:
White Powder
Molecular weight:
1019.24
Ref: TM-T2584
| 1mg | 50.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 284.00 € | ||
| 50mg | 425.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
CGP 20712 A
CAS:105737-62-0
CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that …
Formula:
C24H29F3N4O8S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
590.57
Ref: TM-T10778
| 1mg | 95.00 € | ||
| 5mg | 271.00 € | ||
| 10mg | 401.00 € | ||
| 25mg | 654.00 € | ||
| 50mg | 907.00 € | ||
| 100mg | 1,199.00 € | ||
| 200mg | 1,649.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
BAN ORL 24 dihydrochloride
CAS:1401463-54-4
BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that …
Formula:
C27H37Cl2N3O2
Purity:
95.03%
Color and Shape:
Solid
Molecular weight:
506.51
Ref: TM-T10457
| 2mg | 78.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
cis-(Z)-Flupentixol dihydrochloride
CAS:51529-01-2
cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.
Formula:
C23H27Cl2F3N2OS
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
507.44
Ref: TM-T2564
| 5mg | 64.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 268.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
ML224
CAS:1338824-21-7
ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' …
Formula:
C31H31N3O5
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
525.59
Ref: TM-T16106
| 1mg | 57.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 139.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
GLP-1R modulator L7-028
CAS:2648317-95-5
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
Formula:
C24H28N2O3
Purity:
98.76% - 98.76%
Color and Shape:
Liquid
Molecular weight:
392.49
Ref: TM-T40279
| 1mg | 64.00 € | ||
| 5mg | 136.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
GLP-1R modulator C16
CAS:875005-43-9
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
Formula:
C21H26ClFN2O3
Purity:
99.6% - 99.6%
Color and Shape:
Liquid
Molecular weight:
408.89
Ref: TM-T40997
| 1mg | 98.00 € | ||
| 2mg | 140.00 € | ||
| 5mg | 222.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
WIN 51,708
CAS:144177-30-0
WIN 51,708 is an antagonist of neurokinin-1 receptor.
Formula:
C29H33N3O
Purity:
99%
Color and Shape:
Solid
Molecular weight:
439.59
Ref: TM-T29157
| 1mg | 274.00 € | ||
| 2mg | 408.00 € | ||
| 5mg | 675.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
GRK6-IN-2
CAS:2677786-27-3
GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 …
Formula:
C21H21FN6
Purity:
98.94%
Color and Shape:
Liquid
Molecular weight:
376.43
Ref: TM-T61556
| 2mg | 61.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 694.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
L-798106
CAS:244101-02-8
L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and …
Formula:
C27H22BrNO4S
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
536.44
Ref: TM-T15689
| 1mg | 50.00 € | ||
| 5mg | 106.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 334.00 € | ||
| 50mg | 536.00 € | ||
| 100mg | 858.00 € | ||
| 200mg | 1,133.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
GLP-1R modulator C5
CAS:421578-93-0
GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane …
Formula:
C24H21NO3
Purity:
99.59%
Color and Shape:
Liquid
Molecular weight:
371.43
Ref: TM-T61483
| 1mg | 42.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
SLIGRL-NH2
CAS:171436-38-7
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.
Formula:
C29H56N10O7
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
656.82
Ref: TM-TP1046
| 1mg | 95.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Virodhamine
CAS:287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of …
Formula:
C22H37NO2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
347.53
Ref: TM-T64371
| 2mg | 52.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Citalopram
CAS:59729-33-8
Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be …
Formula:
C20H21FN2O
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
324.39
Ref: TM-T20828
| 25mg | 35.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 147.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
