G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ketanserin tartrate
CAS:83846-83-7
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study …
Formula:
C26H28FN3O9
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
545.51
Ref: TM-T1066L
| 25mg | 37.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 68.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Degarelix
CAS:214766-78-6
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
Formula:
C82H103ClN18O16
Color and Shape:
Solid
Molecular weight:
1632.26
Ref: TM-T10988
| 50mg | 793.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Virodhamine
CAS:287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of …
Formula:
C22H37NO2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
347.53
Ref: TM-T64371
| 2mg | 52.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
GLP-1R modulator C16
CAS:875005-43-9
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
Formula:
C21H26ClFN2O3
Purity:
99.6% - 99.6%
Color and Shape:
Solid
Molecular weight:
408.89
Ref: TM-T40997
| 1mg | 98.00 € | ||
| 2mg | 140.00 € | ||
| 5mg | 222.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Agomelatine (L(+)-Tartaric acid)
CAS:824393-18-2
Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, …
Formula:
C19H23NO8
Color and Shape:
Solid
Molecular weight:
393.39
Ref: TM-T10267
| 2mg | 40.00 € | ||
| 5mg | 57.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Taranabant racemate
CAS:701977-00-6
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
Formula:
C27H25ClF3N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.95
Ref: TM-T13081
| 2mg | 50.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
CB1/2 agonist 3
CAS:2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 …
Formula:
C25H41NO2
Color and Shape:
Solid
Molecular weight:
387.6
Ref: TM-T61736
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 447.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Clothiapine
CAS:2058-52-8
Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
Formula:
C18H18ClN3S
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
343.87
Ref: TM-T23900
| 1mg | 96.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
GLP-1R modulator L7-028
CAS:2648317-95-5
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
Formula:
C24H28N2O3
Purity:
98.76% - 98.76%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T40279
| 1mg | 64.00 € | ||
| 5mg | 136.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Tegaserod
CAS:145158-71-0
Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the …
Formula:
C16H23N5O
Purity:
99.89%
Color and Shape:
Liquid
Molecular weight:
301.39
Ref: TM-T60680
| 2mg | 37.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
ML224
CAS:1338824-21-7
ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' …
Formula:
C31H31N3O5
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
525.59
Ref: TM-T16106
| 1mg | 57.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 139.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
UCSF924
CAS:1434515-70-4
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 …
Formula:
C20H22N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
322.4
Ref: TM-T13245
| 2mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 205.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
GAT211
CAS:102704-40-5
GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study …
Formula:
C22H18N2O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
342.39
Ref: TM-T27405
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 322.00 € | ||
| 500mg | 776.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Motixafortide
CAS:664334-36-5
Motixafortide (BKT140 4-fluorobenzoyl) is an antagonist of CXCR4 (IC50: 1 nM).
Formula:
C97H144FN33O19S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2159.52
Ref: TM-T14665
| 25mg | 695.00 € | ||
| 50mg | 1,121.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Nebentan potassium
CAS:342005-82-7
Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is …
Formula:
C24H20KN5O5S
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
529.61
Ref: TM-T36008
| 1mg | 91.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 306.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,174.00 € | ||
| 500mg | 2,357.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
(Rac)-Rotigotine hydrochloride
CAS:102120-99-0
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, …
Formula:
C19H26ClNOS
Color and Shape:
Solid
Molecular weight:
351.93
Ref: TM-T12676
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
WAY-100635 maleate
CAS:634908-75-1
WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).
Formula:
C25H34N4O2·xC4H4O4
Purity:
100%
Color and Shape:
White Solid
Molecular weight:
538.645
Ref: TM-T3453
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 223.00 € | ||
| 100mg | 329.00 € | ||
| 500mg | 789.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
Kynurenic acid
CAS:492-27-3
Kynurenic acid (Quinurenic acid) is an NMDA, glutamate, α7 nicotinic acetylcholine receptor triple antagonist and …
Formula:
C10H7NO3
Purity:
99.69%
Color and Shape:
Liquid
Molecular weight:
189.17
Ref: TM-T65135
| 50mg | 36.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
TP-16
CAS:2332972-26-4
TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs …
Formula:
C24H22FNO4S
Purity:
98.83% - 99.33%
Color and Shape:
Solid
Molecular weight:
439.5
Ref: TM-T62525
| 1mg | 432.00 € | ||
| 5mg | 1,013.00 € | ||
| 25mg | 2,016.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
ACT-462206
CAS:1361321-96-1
ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used …
Formula:
C20H24N2O4S
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
388.48
Ref: TM-T26559
| 1mg | 44.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 697.00 € | ||
| 500mg | 1,393.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 27 Nov 2024
