G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ACTH 1-14 acetate(25696-21-3 free base)
ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.
Formula:
C79H113N21O22S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1740.96
Ref: TM-TP1238L
| 1mg | 50.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 380.00 € | ||
| 100mg | 540.00 € | ||
| 200mg | 713.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SKF 38393 hydrochloride
CAS:62717-42-4
SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.
Formula:
C16H17NO2·HCl
Purity:
98.70% - 99.1%
Color and Shape:
Solid
Molecular weight:
291.77
Ref: TM-T6988
| 1ml | 85.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 77.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
E7046
CAS:1369489-71-3
E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting …
Formula:
C22H18F5N3O4
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
483.4
Ref: TM-TQ0025
| 5mg | 52.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 209.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GW9508
CAS:885101-89-3
GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in …
Formula:
C22H21NO3
Purity:
97.89% - 99.19%
Color and Shape:
Solid
Molecular weight:
347.41
Ref: TM-T1781
| 1ml | 34.00 € | ||
| 10mg | 34.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 136.00 € | ||
| 200mg | 195.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
K 41498 aceate
K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for …
Purity:
96.40%
Molecular weight:
N/A
Ref: TM-TP2009L
| 1mg | 308.00 € | ||
| 5mg | 1,054.00 € | ||
| 10mg | 1,417.00 € | ||
| 25mg | 2,108.00 € | ||
| 50mg | 2,843.00 € | ||
| 100mg | 3,833.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
APD668
CAS:832714-46-2
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for …
Formula:
C21H24FN5O5S
Purity:
99.45% - 99.97%
Color and Shape:
Solid
Molecular weight:
477.51
Ref: TM-T2088
| 1mg | 49.00 € | ||
| 1ml | 115.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 453.00 € | ||
| 100mg | 639.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Adenosine receptor antagonist 4
CAS:133240-06-9
Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
Formula:
C10H13N3
Purity:
98.59% - 99.58%
Color and Shape:
Off-White Powder
Molecular weight:
175.23
Ref: TM-T21620
| 1ml | 47.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 133.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[D-Phe12]-Bombesin acetate](https://static.cymitquimica.com/products/TM/thumb/TP2239L.jpg)
[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
Formula:
C76H116N22O20S
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
1689.94
Ref: TM-TP2239L
| 1mg | 157.00 € | ||
| 5mg | 343.00 € | ||
| 10mg | 513.00 € | ||
| 25mg | 923.00 € | ||
| 50mg | 1,380.00 € | ||
| 100mg | 2,074.00 € | ||
| 200mg | 3,111.00 € | ||
| 500mg | 4,714.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bepotastine Besilate
CAS:190786-44-8
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
Formula:
C21H25ClN2O3·C6H6O3S
Purity:
99.83% - 99.90%
Color and Shape:
Brown Viscous Liquid
Molecular weight:
547.06
Ref: TM-T6405
| 1ml | 35.00 € | ||
| 100mg | 46.00 € | ||
| 500mg | 88.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
N-Oleoyl glycine
CAS:2601-90-3
N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of …
Formula:
C20H37NO3
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
339.51
Ref: TM-T13803
| 1ml | 77.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 318.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Human growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release …
Purity:
99.26%
Molecular weight:
N/A
Ref: TM-TP1155L
| 1mg | 185.00 € | ||
| 5mg | 460.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,747.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 …
Formula:
C169H276N52O55S2
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
3980.45
Ref: TM-TP1232L
| 1mg | 276.00 € | ||
| 5mg | 677.00 € | ||
| 10mg | 917.00 € | ||
| 25mg | 1,412.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,572.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Piperoxan hydrochloride
CAS:135-87-5
Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.
Formula:
C14H20ClNO2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
269.77
Ref: TM-T4526
| 1ml | 56.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 204.00 € | ||
| 200mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tolvaptan
CAS:150683-30-0
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that …
Formula:
C26H25ClN2O3
Purity:
97% - 99.78%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T2326
| 1mg | 38.00 € | ||
| 1ml | 126.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 357.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Myristyl nicotinate
CAS:273203-62-6
Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid …
Formula:
C20H33NO2
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
319.48
Ref: TM-T19438
| 1ml | 34.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 44.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID](https://static.cymitquimica.com/products/TM/thumb/T8913.jpg)
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:260555-42-8
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.
Formula:
C13H13NO5
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
263.25
Ref: TM-T8913
| 1ml | 44.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 164.00 € | ||
| 200mg | 238.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Urantide acetate(669089-53-6 free base)
Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in …
Formula:
C53H70N10O14S2
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
1135.31
Ref: TM-TP2106L
| 1mg | 112.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 757.00 € | ||
| 100mg | 1,056.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Naratriptan hydrochloride
CAS:143388-64-1
Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation …
Formula:
C17H25N3O2S·HCl
Purity:
99.17% - 99.89%
Color and Shape:
Beige Solid
Molecular weight:
371.93
Ref: TM-T6602
| 1ml | 53.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 131.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | 459.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - …
Purity:
95.44% - 96.09%
Molecular weight:
N/A
Ref: TM-TP1199L
| 1mg | 234.00 € | ||
| 5mg | 553.00 € | ||
| 10mg | 746.00 € | ||
| 25mg | 1,103.00 € | ||
| 50mg | 1,486.00 € | ||
| 100mg | 2,009.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
(S)-Amisulpride
CAS:71675-92-8
(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.
Formula:
C17H27N3O4S
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
369.48
Ref: TM-T26375
| 1mg | 49.00 € | ||
| 1ml | 121.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 326.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 898.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
