Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
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Subcategories of "Inhibitors"
Angiogenesis
Apoptosis
Cell Cycle/Checkpoint
Chromatin/Epigenetics
Cytoskeletal Signaling
DNA Damage/DNA Repair
Endocrinology/Hormones
Enzyme
GPCR/G-Protein
Immunology and Inflammation
Influenza Virus
JAK/STAT signaling
MAPK Signaling
Membrane Transporter/Ion Channel
Metabolism
Microbiology/Virology
Neuroscience
Other Inhibitors
Oxidation-Reduction
PI3K/Akt/mTOR Signaling
Proteases/Proteasome
Stem Cell and Derivatives
Tyrosine Kinase/Adaptors
Ubiquitination
Show 16 more subcategories
Products of "Inhibitors"
DYRK1-IN-1
CAS:2814486-79-6
DYRK1-IN-1: Selective DYRK1A inhibitor with IC50 of 220 nM, good permeability, CNS penetrant for research, …
Formula:
C12H12N6
Color and Shape:
Liquid
Molecular weight:
240.26
Ref: TM-T60334
| 100mg | 1,371.00 € | ||
| 200mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
KAG-308
CAS:1215192-68-9
KAG-308: selective EP4 agonist; Ki: 2.57 nM, EC50: 17 nM; suppresses colitis, promotes mucosal healing, …
Formula:
C24H30F2N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
460.52
Ref: TM-T15642
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Mar 2025
SIK1 activator 1
CAS:2769850-83-9
SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.
Formula:
C23H32O6
Color and Shape:
Liquid
Molecular weight:
404.5
Ref: TM-T61992
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Mar 2025
Anti-Aβ agent 1A
Anti-Aβ agent 1A is a potent anti-amyloid-β agent.
Formula:
C35H49NO4
Color and Shape:
Liquid
Molecular weight:
547.77
Ref: TM-T63873
| 25mg | 1,418.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
L5-DA
L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with …
Formula:
C32H34N6O2
Color and Shape:
Liquid
Molecular weight:
534.65
Ref: TM-T63765
| 25mg | 1,418.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
GSK3368715
CAS:1629013-22-4
GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases …
Formula:
C20H38N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
366.54
Ref: TM-T11500
| 25mg | 2,523.00 € | ||
| 50mg | 3,348.00 € | ||
| 100mg | 4,583.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
COX-2/NO-IN-1
COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.
Formula:
C15H15NO3
Color and Shape:
Liquid
Molecular weight:
257.28
Ref: TM-T60403
| 25mg | 1,418.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
AVE-1330A sodium
CAS:396731-20-7
AVE-1330A sodium is a beta-Lactamase inhibitor.
Formula:
C7H10N3NaO6S
Color and Shape:
Liquid
Molecular weight:
287.23
Ref: TM-T69299
| 25mg | 2,396.00 € | ||
| 50mg | 3,152.00 € | ||
| 100mg | 4,289.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
COX-2/PI3K-IN-2
COX-2/PI3K-IN-2 (5f): anti-inflammatory & anti-cancer, selectively inhibits COX-2 (Ki=3.02nM), potently blocks PI3K (IC50=2.78nM).
Formula:
C16H17N5O2
Color and Shape:
Liquid
Molecular weight:
311.34
Ref: TM-T60769
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € | ||
| 100mg | 2,364.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
GLP-1R agonist 8
CAS:2736446-82-3
GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 < 2 nM).
Formula:
C33H32N4O5
Color and Shape:
Liquid
Molecular weight:
564.63
Ref: TM-T63999
| 25mg | 2,023.00 € | ||
| 50mg | 2,633.00 € | ||
| 100mg | 3,328.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
BMS-748730
CAS:910297-57-3
BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.
Formula:
C22H26ClN7O3S
Color and Shape:
Solid
Molecular weight:
504.01
Ref: TM-T30540
| 1mg | 963.00 € | ||
| 5mg | 1,908.00 € | ||
| 10mg | 2,595.00 € | ||
| 25mg | 3,842.00 € | ||
| 50mg | 5,218.00 € | ||
| 100mg | 7,041.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
BMS 310705
CAS:280578-49-6
BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.
Formula:
C27H42N2O6S
Color and Shape:
Liquid
Molecular weight:
522.7
Ref: TM-T73084
| 25mg | 4,074.00 € | ||
| 50mg | 5,389.00 € | ||
| 100mg | 7,645.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
T-3861174
CAS:2209057-94-1
T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with …
Formula:
C26H25FN6O2
Color and Shape:
Liquid
Molecular weight:
472.51
Ref: TM-T69800
| 25mg | 2,117.00 € | ||
| 50mg | 2,779.00 € | ||
| 100mg | 3,730.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
Pociredir
CAS:2490674-02-5
Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.
Formula:
C22H18FN5O2
Color and Shape:
Liquid
Molecular weight:
403.41
Ref: TM-T61975
| 25mg | 1,996.00 € | ||
| 50mg | 2,597.00 € | ||
| 100mg | 3,282.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
Massarilactone H
CAS:1393110-39-8
Massarilactone H, a polyketide, is a neuraminidase inhibitor, with an IC 50 of 8.18 µM …
Formula:
C11H12O5
Color and Shape:
Liquid
Molecular weight:
224.21
Ref: TM-T72732
| 25mg | 2,396.00 € | ||
| 50mg | 3,152.00 € | ||
| 100mg | 4,289.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
Emapticap pegol
CAS:1390630-22-4
Emapticap pegol inhibits pro-inflammatory CCL2, is a 40-nt Spiegelmer aptamer for humans (NOX-E36) and mice …
Color and Shape:
Liquid
Ref: TM-T64256
| 25mg | 1,418.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
L-365260 hemihydrate
L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.
Formula:
C24H24N4O3
Color and Shape:
Liquid
Molecular weight:
407.47
Ref: TM-T62039
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Mar 2025
H 218-54
CAS:117760-71-1
H 218-54 is a renin inhibitor.
Formula:
C37H56N2O5S
Color and Shape:
Liquid
Molecular weight:
640.92
Ref: TM-T71318
| 25mg | 2,396.00 € | ||
| 50mg | 3,152.00 € | ||
| 100mg | 4,289.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
TH-6
TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, …
Formula:
C22H24FN3O5
Color and Shape:
Liquid
Molecular weight:
429.44
Ref: TM-T62366
| 25mg | 1,119.00 € | ||
| 50mg | 1,455.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
MAO A/HDAC-IN-1
MAO A/HDAC-IN-1 is an effective monoamine oxidase A (MAO A) and HDAC dual inhibitor, which …
Formula:
C21H24ClN3O3
Color and Shape:
Liquid
Molecular weight:
401.89
Ref: TM-T61958
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € | ||
| 100mg | 2,364.00 € |
Estimated delivery in United States, on Tuesday 18 Mar 2025
