
Benzimidazole and Imidazole Derivatives
Benzimidazole is a compound consisting of a benzene ring fused to an imidazole ring, a five-membered structure containing two nitrogen atoms. Benzimidazole derivatives, such as albendazole, are known for their antiparasitic and antifungal activity, used in the treatment of parasitic infections and certain parasitic diseases in animals and humans. Imidazole, on the other hand, is a five-membered structure with two nitrogen atoms found in various biologically active compounds. Imidazole derivatives, such as metronidazole, have antimicrobial and antiparasitic properties. These compounds are also used in the pharmaceutical industry for treating bacterial infections, parasitic diseases, and some fungal infections, as well as in organic chemistry as catalysts.
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Found 10373 products of "Benzimidazole and Imidazole Derivatives"
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Itraconazole-d5 (major)
CAS:Controlled Product<p>Applications An isotopically labelled, orally active antimycotic structurally related to Ketoconazole.A representative lot was 88% d5, 12% d4 with no d0. It is a COVID19-related research product.<br>References Espinel-Ingroff, A., et al.: Antimicrob. Agents Chemother., 26, 5 (1984), Heykants, J., et al.: Mycoses, 32, Suppl 1, 67 (1989), Sugar, A.M., et al.: Curr. Clin. Top. Infect. Dis., 13, 74 (1993),<br></p>Formula:C352H5H33Cl2N8O4Color and Shape:NeatMolecular weight:710.661,3-dibenzyl-1H-benzo[d]imidazol-3-ium chloride
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:334.85000610351562-(3-Aminophenyl)-1H-benzo[d]imidazol-6-amine
CAS:Purity:97.0%Color and Shape:SolidMolecular weight:224.26699829101562rac Desethyl Oxybutynin-d5 Hydrochloride
CAS:Controlled Product<p>Applications A labelled metabolite of the drug Oxybutynin (D289475). Used in the treatment of incontinence.<br>References Hughes, K., et al.: Xenobiotica, 22, 859 (1992), Oki, T., et al.: Biol. Pharm. Bull., 24, 491 (2001), Fetscher, C., et al.: Br. J. Pharmacol., 136, 64 (2002), Zobrist, R., et al.: Pharm. Res., 20, 103 (2003)<br></p>Formula:C20H22D5NO3·HClColor and Shape:White To Off-WhiteMolecular weight:334.47 + (36.46)5-amino-1-propyl-1H-imidazole-4-carboxamide
CAS:Formula:C7H12N4OPurity:95.0%Color and Shape:SolidMolecular weight:168.2Bis(4-cyanophenyl)methanol
CAS:Controlled Product<p>Stability Light Sensitive<br>Applications A metabolite of Letrozole.<br>References Koyama, E., et al.: Ther. Drug Monit., 15, 224 (1993), Pfister, C., et al.: J. Pharm. Sci., 83, 520 (1994), Vander H.Y., et al.: J. Pharm. Biomed. Anal., 24, 723 (2001), Cohen, M., et al.: Clin. Cancer Res., 8, 665 (2002),<br></p>Formula:C15H10N2OColor and Shape:NeatMolecular weight:234.25N-(tert-Butyl)-2-((4,5-diphenyloxazol-2-yl)thio)propanamide
CAS:Purity:97.0%Molecular weight:380.510009765625Albendazole Sulfoxide
CAS:<p>Impurity Albendazole EP Impurity B<br>Applications Albendazole Sulfoxide (Albendazole EP Impurity B) is a metabolite of Albendazole, an anthelmintic.<br>References Dominguez, L., et al.: Farmaco, 50, 697 (1995), De Laurentis, N., et al.: Pharm. Pharmacol Lett., 6, 2: 51 (1996)<br></p>Formula:C12H15N3O3SColor and Shape:White To BrownMolecular weight:281.332-Chlorobenzophenone
CAS:<p>Impurity Clotrimazole EP Impurity E<br>Applications 2-Chlorobenzophenone (Clotrimazole EP Impurity E) is a metabolite of Clofedanol (C586920). Chlorobenzophenone is also used as a catalyst in the photocrosslinking of polyethylenes.<br>References Qu, B. et al.: J. Appl. Polym. Sci., 48, 701 (1993); Eckhardt, G. et al.: J. Clin. Chem. Clin. Biochem., 15, 687 (1977);<br></p>Formula:C13H9ClOColor and Shape:NeatMolecular weight:216.66Lansoprazole Sulfide
CAS:Controlled Product<p>Impurity Lansoprazole EP Impurity C; USP Impurity B<br>Applications Lansoprazole Sulfide (Lansoprazole EP Impurity C; USP Impurity B) is a metabolite of Lansoprazole, as gastric pump inhibitor.<br>References Oie, et al.: J. Pharm. Sci., 68, 1203 (1979), Naesdal, J., et al.: Clin. Pharmacol. Ther., 40, 344 (1986), Dube, L., et al.: Biopharm. Drug Dispos., 10, 55 (1989), Barradell, L., et al.: Drugs, 44, 225 (1992),<br></p>Formula:C16H14F3N3OSColor and Shape:WhiteMolecular weight:353.36rel-(1R,3S,5S)-8-Methyl-8-azabicyclo[3,2,1]oct-6-en-yl-2-hydroxy-2,2-dithiophen-2-yl acetate
CAS:Controlled Product<p>Impurity Tiotropium EP impurity D<br>Applications (1R,3S,5S)-8-Methyl-8-azabicyclo[3,2,1]oct-6-en-yl-2-hydroxy-2,2-dithiophen-2-ylacetate is an impurity in the synthesis of Tiotropium Bromide (T444850), a muscarinic receptor antagonist. Bronchodilator.<br>References Haddad, E.-B., et al.: Mol. Pharmacol., 45, 899 (1994); Donohue, J. F., et al.: Chest, 122, 47 (2002); Profita, M., et al.: Allergy, 60, 1361 (2005); Dusser, D., et al.: Eur. Respir. J., 27, 547 (2006);<br></p>Formula:C18H19NO3S2Color and Shape:NeatMolecular weight:361.48Nocodazole
CAS:<p>M05733 - Nocodazole</p>Formula:C14H11N3O3SPurity:98%Color and Shape:Solid, Beige powderMolecular weight:301.32000732421875rac 5-Hydroxymethyl Tolterodine-d14
CAS:Controlled ProductFormula:C22H17D14NO2Purity:90%Color and Shape:NeatMolecular weight:355.572-(4-Bromo-phenyl)-1-methyl-1H-benzoimidazole
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:287.1600036621094Secnidazole-d3
CAS:Controlled Product<p>Applications Labelled Secnidazole (S225000). Analog of Metronidazole. Antiamebic. Antiprotozoal (Trichomonas).<br>References Cosar, C., et al.: Arzneim.-Forsch., 16, 23 (1966), Videau, D., et al.: Br. J. Vener. Dis., 54, 77 (1978), Symonds, J., et al.: J. Antimicrob. Chemother., 5, 484 (1979),<br></p>Formula:C7H8D3N3O3Color and Shape:White To Off-WhiteMolecular weight:188.2N-Nitroso Varenicline
CAS:Controlled Product<p>Applications N-Nitroso Varenicline is a derivative of Varenicline (V215635(M)), which is a useful medication for smoking cessation.<br>References Hart, E., et al.: Behavioural Brain Research, 397, 112887 (2021)<br></p>Formula:C13H12N4OColor and Shape:NeatMolecular weight:240.2613,4-Diaminoanisole
CAS:<p>Applications 3,4-Diaminoanisole (cas# 102-51-2) is a compound useful in organic synthesis.<br></p>Formula:C7H10N2OColor and Shape:NeatMolecular weight:138.174-Methylpentanal (up to 75% hydrated form)
CAS:Controlled Product<p>Applications An intermediate used in the synthesis of Pregabalin (P704800) and related compounds.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Posadas, I., et al.: Br. J. Pharmacol., 142, 331 (2004),<br></p>Formula:C6H12OColor and Shape:Colourless LiquidMolecular weight:100.163,5-Didesamino-3,5-dioxo Lamotrigine
CAS:Controlled Product<p>Impurity Lamotrigine EP Impurity D<br>Applications 3,5-Didesamino-3,5-dioxo Lamotrigine (Lamotrigine EP Impurity D) is an impurity of the anticonvulsant Lamotrigine (L173250).<br>References Hlavac, J. et al.: ARKIVOC, 1, 22 (2003);<br></p>Formula:C9H5Cl2N3O2Color and Shape:NeatMolecular weight:258.064-(4-Cyanobenzyl)-1,2,4-triazole
CAS:Controlled Product<p>Applications 4-(4-Cyanobenzyl)-1,2,4-triazole is an intermediate in the synthesis of Letrozole (L330100), an oral, non-steroidal, aromatase inhibitor generally used to treat breast cancer as a result of hormone response after surgery.<br>References Bhatnagar, A.S., et al: J. Steroid Biochem. Mol. Biol., 37, 1021 (1990), Pfister, C.U., et al.: J. Pharm. Sci., 83, 520 (1994), Lipton, A., et al.: Cancer, 75, 2132 (1995),<br></p>Formula:C10H8N4Color and Shape:NeatMolecular weight:184.20Carbamazepine-d2 (Major)
CAS:Controlled Product<p>Applications Labelled Carbamazepine (C175840). Used in treatment of pain associated with trigeminal neuralgia. Anticonvulsant.<br>References Stenger, E.G., et al.: Med. Exp., 11, 191 (1964), Pynnonen, S., et al.: Ther. Drug Monit., 1, 409 (1979), Sidebottom, A., et al.: J. Clin. Pharm. Ther., 20, 31 (1995)<br></p>Formula:C15H10D2N2OColor and Shape:NeatMolecular weight:238.28Efinaconazole-N-oxide
CAS:Controlled Product<p>Applications Efinaconazole-N-oxide is a degradation product and potentially a metabolite of the anti-fungal drug Efinaconazole (E435070).<br>References Sugiura, K., et. al.: Antimicrob. Agents CH., 58, 3837 (2014);<br></p>Formula:C18H22F2N4O2Color and Shape:NeatMolecular weight:364.392-(1H-benzimidazol-2-ylthio)-1-cyclopropylethanone
CAS:Purity:95.0%Molecular weight:232.30000305175785-(3-BROMOPHENYL)-1H-TETRAZOLE
CAS:Formula:C7H5BrN4Purity:98%Color and Shape:SolidMolecular weight:225.049Albendazole-d7
CAS:Controlled Product<p>Applications Labelled Albendazole (A511610). An anthelmintic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Zhao, Y., et al.: Org. Biomol. Chem., 6, 4509 (2008), Sanderson, H., et al.: Toxicol. Lett., 187, 84 (2009),<br></p>Formula:C12H8D7N3O2SColor and Shape:NeatMolecular weight:272.37α,α,2,6-Tetrachloro-toluene
CAS:Controlled Product<p>Impurity Isoconazole Impurity 9<br>Applications α,α,2,6-Tetrachloro-toluene (Isoconazole Impurity 9) is an impurity of Isoconazole (I798250), an antibacterial and antifungal agent used to treat vaginitis.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Asikoglu, M. et al.: J. Pharm. Pharmacol. 47, 717 (1995); Marrero-Ponce, Y. et al.: Bioorg. Med. Chem. 13, 2881 (2005)<br></p>Formula:C7H4Cl4Color and Shape:Light YellowMolecular weight:229.922-(PYRIDIN-2-YLMETHYL)-1H-BENZO[D]IMIDAZOLE-6-CARBOXYLIC ACID
Purity:90.0%Molecular weight:253.26100158691406N-Methyl Omeprazole (Mixture of isomers with the methylated nitrogens of imidazole)
CAS:Controlled Product<p>Applications Omeprazole (O635000) impurity.<br>References Allenmark, S., et al.: Anal. Biochem., 136, 293 (1984), Besancon, M., et al.: J. Biol. Chem., 272, 22438 (1997),<br></p>Formula:C18H21N3O3SColor and Shape:Off White SolidMolecular weight:359.44(1R)-(-)-10-Camphorsulfonic Acid
CAS:Controlled Product<p>Impurity Voriconazole EP Impurity E (1R)-Isomer<br>Stability Hygroscopic<br>Applications (1R)-(-)-10-Camphorsulfonic Acid (Voriconazole EP Impurity E (1R)-Isomer) is a chiral derivative of Camphor. Used in the preparation of a chiral recognition polymer that is used in the chiral separation of amino acids. A catalyst in direct animation of α-branched aldehydes (including important biological molecules such as α-Me phenylglycine) with near perfect enantioselectivity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Guo, H. et al.: Polym. Preprints Am. Chem. Soc., 40, 506 (1999); Liu, C. et al.: Org. Lett., 13, 2638 (2011);<br></p>Formula:C10H16O4SColor and Shape:WhiteMolecular weight:232.30Hydroxy Voriconazole
Controlled Product<p>Applications A hydroxylated derivative of Voriconazole (V760000), a systemic antifungal and ergosterol biosynthesis inhibitor.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sanati, H., et al.: Antimicrob. Ag. Chemother., 41, 2492 (1997).<br></p>Formula:C16H14F3N5O2Color and Shape:NeatMolecular weight:365.31Luliconazole
CAS:Controlled Product<p>Stability Light Sensitive<br>Applications Luliconazole is an azole antifungal drug.<br>References Uhida, K., et al.: J. Infect. Chemother., 10, 216 (2004); Niwano, ., et al.: Antimicro. Agents Chemother., 42, 967 (1998),<br></p>Formula:C14H9Cl2N3S2Color and Shape:Off-White To Light YellowMolecular weight:354.28Modafinil Carboxylate Methyl Ester
CAS:Controlled Product<p>Impurity Modafinil EP Impurity C<br>Applications Modafinil Carboxylate Methyl Ester (Modafinil EP Impurity C) is a Modafinil derivative.<br>References Lehr, H., et al.: J. Med. Chem., 6, 136 (1963), Saikawa, I., et al.: Chem. Pharm. Bull., 33, 5534 (1985),<br></p>Formula:C16H16O3SColor and Shape:NeatMolecular weight:288.365-Chloro-6-(2,3-dichlorophenoxy)-1,3-dihydro-2H-benzimidazol-2-one
CAS:<p>Applications 5-Chloro-6-(2,3-dichlorophenoxy)-1,3-dihydro-2H-benzimidazol-2-one is a metabolite of Triclabendazole (T774175), the only anthelmintic drug, which is active against immature, mature and adult stages of fluke.<br>References Whelan, M., et al.: J. Chromato., 1275, 41 (2013); Barrera, S., et al.; Antimicrob. Agent. Chemother., 56, 3535 (2012);<br></p>Formula:C13H7Cl3N2O2Color and Shape:Off-White To BrownMolecular weight:329.57N-Nitroso Methyl Aniline Derivative
CAS:Formula:C14H11ClN2O2Color and Shape:WhiteMolecular weight:274.7023Omeprazole Sulfide Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Omeprazole Sulfide Hydrochloride is a metabolite of Omeprazole (O635000), which binds covalently to proton pump. It inhibits gastric secretion. Used as an anttiulcerative.<br>References Muller, P., et al.: Arzneimittel-Forsch., 33, 1685 (1983); Wallmark, B., et al.: Biochim. Biophys. Acta., 778, 549 (1984); Morii, M., et al.: J. Biol. chem., 268, 21553 (1993); Ritter, M., et al.: Br. J. Pharmacol., 124, 627 (1998)<br></p>Formula:C17H19N3O2S·HClColor and Shape:NeatMolecular weight:329.42 + 36.46Carbimazole
CAS:<p>Applications Carbimazole, a prodrug of Methimazole (M260300), is used in the treatment of hyperthyroidism.<br>References Marchant, B., et al.: J. Clin. Endocrinol. Metab., 45, 1187 (1977), Johnsson, E., et al.: Lancet, 350, 1520 (1997),<br></p>Formula:C7H10N2O2SColor and Shape:NeatMolecular weight:186.23Lamotrigine
CAS:Controlled Product<p>Applications An anticonvulsant. Inhibits glutamate release, possible through inhibition of Sodium, Potassium and Calcium currents. Used in treatment of bipolar depression.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Miller, A.A., et al.: Epilepsia, 27, 483 (1986), Grunze, et al.: Neuropsychobiology, 38, 131 (1998), Calabrese, J.R., et al.: J. Clin. Psychiatry, 60, 79 (1999),<br></p>Formula:C9H7Cl2N5Color and Shape:NeatMolecular weight:256.09Climbazole-d4
CAS:Controlled ProductFormula:C15D4H13ClN2O2Color and Shape:Off White SolidMolecular weight:296.792-Butyl-3-[2'-(1H-tetrazol-5-yl)biphenyl-4-ylmethyl]1,3-diaza-spiro[4.4]non-1-en-4-one
CAS:Purity:97.0%Color and Shape:Solid, White - Almost white powderMolecular weight:428.5400085449219Tiotropium Bromide
CAS:Formula:C19H22NO4S2·BrColor and Shape:White To Off-WhiteMolecular weight:472.42N-methyl-1-(1-phenyl-1H-tetrazol-5-yl)cyclohexanamine
CAS:Purity:95.0%Molecular weight:257.34100341796875Lamotrigine 3,3-Dimer
CAS:Controlled Product<p>Applications Lamotrigine 3,3-Dimer is a dimer impurity of the anticonvulsant Lamotrigine (L173250).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Formula:C19H14Cl4N10Color and Shape:NeatMolecular weight:524.19Ref: 10-F987646
1gTo inquire5gTo inquire5mg80.00€10mg102.00€25mg211.00€50mg362.00€100mgTo inquire250mgTo inquire5-Hydroxy Omeprazole-d3 Sodium Salt
CAS:Controlled ProductFormula:C17H15D3N3NaO4SColor and Shape:White To Light YellowMolecular weight:386.425-[(2-methyl-1H-benzimidazol-1-yl)methyl]-2-furoic acid
CAS:Purity:95.0%Molecular weight:256.2609863281252-(4-Chlorobenzyl)-1H-benzimidazole
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:242.71000671386721H-Benzo[d]imidazole-5-carbohydrazide
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:176.17900085449225,6-DIMETHYL-2-(PYRIDIN-3-YL)-1H-BENZO[D]IMIDAZOLE
CAS:Purity:95.0%Molecular weight:223.27900695800784-(1H-Benzimidazol-2-yl)-1,2,5-oxadiazol-3-amine
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:201.18899536132812(E)-2-(4-(1H-Imidazol-4-yl)styryl)-1H-indene-1,3(2H)-dione
CAS:Purity:95.0%Molecular weight:314.343994140625(-)-Donepezil
CAS:Controlled Product<p>Applications (-)-Donepezil is an isomer of Donepezil (D531750), a nootropic, acting as an inhibitor of acetylcholinesterase.<br>References Ohnishi, A., et al.: J. Clin. Pharmacol., 33, 1086 (1993), Galli, A., et al.: Eur. J. Pharmacol., 270, 189 (1994)<br></p>Formula:C24H29NO3Color and Shape:NeatMolecular weight:379.49Itraconazole N,N-Dioxide
Controlled Product<p>Stability Hygroscopic<br>Applications Itraconazole N,N-Dioxide is a derivative of Itraconazole (I937500). Itraconazole is an orally active antimycotic structurally related to Ketoconazole. Antifungal. It is a COVID19-related research product.<br>References Espinel-Ingroff, A., et al.: Antimicrob. Agents Chemother., 26, 5 (1984), Heykants, J., et al.: Mycoses, 32, Suppl 1, 67 (1989), Sugar, A.M.,et al.: Curr. Clin. Top. Infect. Dis., 13, 74 (1993),<br></p>Formula:C35H38Cl2N8O6Color and Shape:NeatMolecular weight:737.632-Amino-5(6)-benzoylbenzimidazole
CAS:<p>Impurity Mebendazole EP Impurity A<br>Applications The minor urinary metabolite of Mebendazole (M200500) in man. Mebendazole impurity.<br>References Leban, J., et al.: Bioorg. Med. Chem. Lett., 17, 5858 (2007),<br></p>Formula:C14H11N3OColor and Shape:NeatMolecular weight:237.266-Bromo-5-(2-fluoro-4-nitrophenoxy)-1-methyl-1H-indazole
CAS:Purity:95.0%Molecular weight:366.14599609375Metronidazole-d4
CAS:Controlled Product<p>Applications Metronidazole-d4 is a labelled analog of Metronidazole (M338880). Used as an antibacterial in the treatment of rosacea. Antiprotozoal (trichomonas). A potential human carcinogen.<br>References Carballo, M., et al.: J. App. Toxicol., 29, 248 (2009), Leitsch, D., et al.: Mol. Microbiol., 72, 518 (2009), Sanderson, H., et al.: Toxicol. Lett., 187, 84 (2009),<br></p>Formula:C62H4H5N3O3Color and Shape:Light YellowMolecular weight:175.18Lansoprazole-d4
CAS:Controlled ProductFormula:C162H4H10F3N3O2SColor and Shape:NeatMolecular weight:373.39Midazolam
CAS:Controlled Product<p>Applications Anesthetic; anticonvulsant; sedative; hypnotic. Positive allosteric modulator of the GABAA receptor. Neuroprotective & Neuroresearch products.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Dundee, J. W., et al.: Drugs, 28, 519 (1984), Lahat, E., et al.: Br. Med. J., 321, 83 (2000)<br></p>Formula:C18H13ClFN3Color and Shape:White To Off-WhiteMolecular weight:325.77(S)-Pregabalin-13C3
CAS:Controlled Product<p>Applications (S)-Pregabalin-13C3, is the labeled analogue of (S)-Pregabalin (P704790), a S-Enantiomer of Pregabalin. A GABA analogue used as an anticonvulsant. Anxiolytic analgesic used to treat peripheral neuropathic pain and fibromyalgia.<br>References Taylor, C.P., at al.: Epilepsy Res., 14, 11 (1993), Field, M.J., et al.: Pain, 80, 391 (1999)<br></p>Formula:C513C3H17NO2Color and Shape:Off-WhiteMolecular weight:162.2(R)-Lansoprazole
CAS:<p>Stability Hygroscopic<br>Applications The R-enantiomer of Lansoprazole; a gastric proton pump inhibitor. An antiulcerative.<br>References Figgitt, D., et al.: Drugs, 60, 925 (2000), Katsuki, H., et al.: Eur. J. Clin. Pharmacol., 57, 709 (2001), Barradell, L.B., et al.: Drugs, 44, 225 (1992), Kim, K., et al.: Clin. Pharmacol. Ther., 72, 90 (2002), Niioka, T., et al.: Ther. Drug Monit., 28, 321 (2006),<br></p>Formula:C16H14F3N3O2SColor and Shape:Off White To Dark BrownMolecular weight:369.36N-Desmethyl,-N-nitroso-promethazine
CAS:Controlled ProductFormula:C16H17N3OSColor and Shape:NeatMolecular weight:299.393-Methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinemethanol
CAS:Controlled ProductFormula:C9H10F3NO2Color and Shape:Light Beige To Light BrownMolecular weight:221.071-(4-Chloro-2-(2-fluorobenzoyl)phenyl)-2-methyl-1H-imidazole-5-carboxylic Acid
CAS:Controlled Product<p>Applications 1-(4-Chloro-2-(2-fluorobenzoyl)phenyl)-2-methyl-1H-imidazole-5-carboxylic Acid is a metalobilite of Midazolam(M343000) which is a anesthetic; anticonvulsant; sedative; hypnotic. Positive allosteric modulator of the GABAA receptor. Neuroprotective & Neuroresearch products.<br>References Dundee, J. W., et al.: Drugs, 28, 519 (1984), Lahat, E., et al.: Br. Med. J., 321, 83 (2000),<br></p>Formula:C18H12ClFN2O3Color and Shape:NeatMolecular weight:358.75Carbamazepine 10,11-Epoxide-d2 (Major)
CAS:Controlled Product<p>Applications A labelled metabolite of Carbamazepine (C175840).<br>References Bellucci, G., et al.: J. Med. Chem., 30, 768 (1987), Johannessen, S., et al.: Ther. Drug. Monit., 27, 710 (2005), Bialer, M., et al.: Expert Opin. Invest. Drugs, 15, 637 (2006), Williams, J., et al.: J. Clin. Pharmacol., 46, 258 (2006),<br></p>Formula:C15H10D2N2O2Color and Shape:NeatMolecular weight:254.28Rufinamide-15N,d2
CAS:Controlled Product<p>Applications Labelled Rufinamide (R701552). Antiepileptic triazole derivative which decreases firing by neurons at sodium channels. Anticonvulsant.<br>References Cheung, W.K., et al.: Pharm. Res., 12, 1878 (1995), Cardot, J.-M., et al.: Biopharm. Drug Dispos., 19, 259 (1998), Palhagen, S., et al.: Epilepsy Res., 43, 115 (2001),<br></p>Formula:C10H6D2F2N315NOColor and Shape:White SolidMolecular weight:241.2Oxazepam
CAS:Controlled Product<p>Applications Anxiolytic; muscle relaxant (skeletal); anticonvulsant; ligand for the GABAA receptor benzodiazepine modulatory site. Controlled substance (depressant).<br>References Goldenthal, E.I., et al.: Toxicol. Appl. Pharmacol., 18, 185 (1971), Sisenwine, et al.: Arzneim. Forsch., 22, 682 (1972), Shearer, C.M., et al.: Anal. Profiles Drug Subs., 3, 441 (1974), Greenblatt, D.J., et al.: Clin. Pharmacokinet., 6, 89 (1981),<br></p>Formula:C15H11ClN2O2Color and Shape:White To Off-WhiteMolecular weight:286.71cis-2-(2,4-Dichlorophenyl)-2-(1H-1,2,4-triazol-1-ylmethyl)-1,3-dioxolane-4-methanol
CAS:Controlled ProductFormula:C13H13Cl2N3O3Color and Shape:NeatMolecular weight:330.174-Isobutyl-2-pyrrolidinone (pregabalin lactam impurity)
CAS:<p>Impurity Pregabalin USP Related Compound C<br>Applications Pregabalin (P704800) intermediate. Pregabalin USP Related Compound C<br>References Taylor, C.P., at al.: Epilepsy Res., 14, 11 (1993), Field, M.J., et al.: Pain, 80, 391 (1999)<br></p>Formula:C8H15NOColor and Shape:Light YellowMolecular weight:141.21Voriconazole-d3
CAS:Controlled Product<p>Applications Labelled Vorizonazole (V760000), used as an antifungal (systemic). An Ergosterol Biosynthesis inhibitor.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sanati, H., et al.: Antimicrob. Ag. Chemother., 41, 2492 (1997),<br></p>Formula:C162H3H11F3N5OColor and Shape:White To BeigeMolecular weight:352.33Iminostilbene
CAS:Controlled Product<p>Impurity Carbamazepine EP Impurity D<br>Applications A metabolite of Carbamazepine (CBZ) (C175840).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Lertratanangkoon, K., et al.: Drug Metab. Dispos., 10, 1 (1982), Deleu, D., et al.: Eur. J. Clin. Pharmacol., 57, 243 (2001),<br></p>Formula:C14H11NColor and Shape:Yellow To Dark OrangeMolecular weight:193.24Omeprazole Sulfone N-Oxide
CAS:<p>Impurity Omeprazole EP Impurity I<br>Applications Omeprazole Sulfone N-Oxide (Omeprazole EP Impurity I) is a metabolite of Omeprazole. Impurity I.<br>References Stevens, C.M., et al.: J. Biol. Chem., 75, 182 (1950), Okamoto, S., et al.: Biochem. Biophys. Res. Commun., 101, 440 (1981)<br></p>Formula:C17H19N3O5SColor and Shape:NeatMolecular weight:377.414'-Ethoxyacetophenone
CAS:<p>Applications 4'-Ethoxyacetophenone, is an acetophenone derivative that can be used as an antibacterial agent. It is a reagent for plymerization. It can also be used as a flavoring agent in fabricating cigarettes with flavored filter tips.<br>References Sivakumar, P., et al.: Chem. Bio. Drug Design, 72, 303 (2008); Mathis, D. E., Beitraege zur Tabakforschung Int., 12, 1 (1983);<br></p>Formula:C10H12O2Color and Shape:White To Off-WhiteMolecular weight:164.20para-Clotrimazole Isomer
CAS:Controlled Product<p>Impurity Clotrimazole EP Impurity B<br>Applications para-Clotrimazole Isomer (Clotrimazole EP Impurity B) is a positional isomer of the antifungal agent (C587400). It showed agonistic activity on the pregnane X receptor and regulated the levels of apoA1 and HDL-cholesterol in rodents.<br>References Buechel, K.H. et al.: Drugs Made Ger., 15, 79 (1972); Bachmann, K. et al.: Pharmacol. Res., 50, 237 (2004);<br></p>Formula:C22H17ClN2Color and Shape:NeatMolecular weight:344.84


