Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65576 products of "Quinazoline and Quinoline Derivatives"
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N-Formyl Linagliptin
Controlled Product<p>Stability Hygroscopic<br>Applications N-Formyl Linagliptin is a derivative of Linagliptin (L465900), a novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.<br>References Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011); Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011);<br></p>Formula:C26H28N8O3Color and Shape:NeatMolecular weight:500.55Bupivacaine Hydrochloride Monohydrate
CAS:<p>Applications Sodium channel blocker, local anesthetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),<br></p>Formula:C18H28N2O·ClH·H2OColor and Shape:WhiteMolecular weight:324.89Rivastigmine-d4 Tartrate Salt
CAS:Controlled Product<p>Applications Rivastigmine-d4 Tartrate Salt, is the labeled analogue of Rivastigmine Tartrate Salt (R541000), a brain selective acetylcholinesterase inhibitor. Nootropic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Rosler, M., et al.: Brit. Med. J., 318, 633 (1999), Enz, A., et al.: Prog. Brain Res., 98, 431 (1993),<br></p>Formula:C18H24D4N2O8Color and Shape:NeatMolecular weight:404.45N-(2,3-Dichlorophenyl)piperazine Hydrochloride
CAS:Controlled ProductFormula:C10H12Cl2N2·ClHColor and Shape:WhiteMolecular weight:267.58Metaflumizone
CAS:<p>Applications Metaflumizone is a semicarbazone insecticide that works by blocking sodium channel in target insects resulting in paralyzation associated with blocking nerve activity. Metaflumizone is useful as a heartworm control treatment.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Zhang, Zhe,, et al.: J. Integrat. Agri. 11, 1145 (2012); Kuhn, D., et al.: Modern. Crop. Protect. Compound., 3, 1273 (2012);<br></p>Formula:C24H16F6N4O2Color and Shape:WhiteMolecular weight:506.40N-(2,6-Dimethylphenyl)-1-piperazineacetamide
CAS:Formula:C14H21N3OColor and Shape:NeatMolecular weight:247.34Prulifloxacin
CAS:<p>Applications Prulifloxacin is a synthetic chemotherapeutic antibiotic of the fluoroquinolone drug class. Prulifloxacin is a prodrug for active metabolite, Ulifloxacin. Antibacterial.<br>References Ozaki, M., et al.: Antimicrob. Agents Chemother., 35, 2496 (1991), Segawa, J., et al.: J. Med. Chem., 35, 4727 (1992), Nakashima, M., et al.: J. Clin. Pharmacol., 34, 930 (1994),<br></p>Formula:C21H20FN3O6SColor and Shape:NeatMolecular weight:461.46N-Boc-L-cis-4,5-Methanoprolineamide
CAS:Controlled Product<p>Applications N-Boc-L-cis-4,5-Methanoprolineamide is an intermediate used to prepare methanoprolinenitrile-contg. dipeptide mimetics as DPP-IV inhibitors and as antidiabetic agents.<br>References Magnin, D., et al.: J. Med. Chem., 47, 2587 (2004)<br></p>Formula:C11H18N2O3Color and Shape:NeatMolecular weight:226.272De-4-fluoro 5-Fluoro Chidamide
CAS:<p>Applications De-5-fluoro 4-Fluorochidamide is an analogue of Chidamide (CAS 743420-02-0), a hitsone deacetylase inhibitor (HDACI) that enhances gemcitabine (G305000) cytotoxicity in pancreatic cancer cells.<br>References Qiao, Z., et. al.: Biochem. Bioph. Res. Co., 434, 95 (2013)<br></p>Formula:C22H19FN4O2Color and Shape:Off White PowderMolecular weight:390.413-(1H-2-INDOLYL)-4-(4-METHOXYPHENYL)-1-METHYL-1H-2-QUINOLINONE
CAS:Purity:97.0%Molecular weight:380.4469909667969Ref: 10-F673022
1gTo inquire2gTo inquire5gTo inquire10gTo inquire100mgTo inquire250mgTo inquire500mgTo inquireN-Nitroso Paroxetine
CAS:Formula:C19H19FN2O4Color and Shape:White To Light YellowMolecular weight:358.3645-Chloro-N-cyclohexylpentanamide
CAS:<p>Stability Hygroscopic<br>Applications 5-Chloro-N-cyclohexylpentanamide (cas# 15865-18-6) is a compound useful in organic synthesis.<br></p>Formula:C11H20ClNOColor and Shape:NeatMolecular weight:217.736N-(4-Hydroxybenzyl)-3,4-dimethoxybenzamide
CAS:Controlled Product<p>Applications N-(4-Hydroxybenzyl)-3,4-dimethoxybenzamide is an intermediate in the synthesis of Itopride (I931500, HCl); a dopamine D2-receptor antagonist with anticholinesterase activity. Also gastroprokinetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Iwanaga, Y., et al; Jpn. J. Pharmacol., 56, 261 (1991); Mushiroda, T., et al.: Drug Metab. Dispos., 28, 1231 (2000); Khamar, B.M., et al.: PCT Int. Appl. WO 2007074386 A2 20070705. Jul 5, 2007<br></p>Formula:C16H17NO4Color and Shape:NeatMolecular weight:287.31cis-Hydroxy Praziquantel
CAS:<p>Applications The main cis-monohydroxylated metabolite of Praziquantel (P702095).<br>References Buehring, K., et al.: Eur. J. Drug Metab. Pharm., 3, 179 (1978), Moldeus, P., et al.: Methods Enzymol., 52, 60 (1978), Cioli, D., et al.: Pharmacol. Ther., 68, 35 (1995),<br></p>Formula:C19H24N2O3Color and Shape:NeatMolecular weight:328.407-Hydroxy-4-(3-pyridyl)coumarin
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:239.229995727539062-Bromo-4,5-dimethoxybenzyl Alcohol
CAS:Controlled Product<p>Applications 2-Bromo-4,5-dimethoxybenzyl Alcohol is an intermediate compound used for the synthetic preparation of pharmaceutical goods. 2-Bromo-4,5-dimethoxybenzyl Alcohol have been used in the synthesis of rotenoids.<br>References Feng, L.S., et al.: Euro. J. Med. Chem., 55, 125 (2012); Candito, D.A., et al.: J. Am. Chem. Soc., 134, 15572 (2012);<br></p>Formula:C9H11BrO3Color and Shape:Off WhiteMolecular weight:247.09rac,trans-Milnacipran Hydrochloride
CAS:Controlled Product<p>Applications rac,trans-Milnacipran Hydrochloride is an impurity of rac-Milnacipran Hydrochloride (M344600), an antidepressant and a selective norepinephrine and serotonin reuptake inhibitor.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Moret, C., et al.: Neuropharmacology, 24, 1211 (1985), Palmier, C., et al.: Eur. J. Clin. Pharmacol., 37, 235 (1989), Spencer, C.M., et al.: Drugs, 56, 405 (1998)<br></p>Formula:C15H23ClN2OColor and Shape:NeatMolecular weight:282.81N-Desmethyl Danofloxacin
CAS:<p>Applications A metabolite of Danofloxacin.<br>References Kiely, J.S., et al.: J. Med. Chem., 43, 656 (1991)<br></p>Formula:C18H18FN3O3Color and Shape:NeatMolecular weight:343.35exo-Granisetron
CAS:<p>Impurity Granisetron EP Impurity F<br>Applications Granisetron Impurity F. Granisetron EP Impurity F.<br>References Fozard, J. R., et al.: Br. J. Pharmacol., 61, 130 (1977), Bradley, P.B., et al.: Neuropharmacology, 25, 563 (1986),<br></p>Formula:C18H24N4OColor and Shape:NeatMolecular weight:312.41N-(4-Amino-6,7-dimethoxyquinazol-2-yl)-N-methylpropylenediamine Formamide Hydrochloride
CAS:Controlled Product<p>Impurity Alfuzosin Hydrochloride EP Impurity E<br>Applications Alfuzosin (A532000) impurity. Alfuzosin (A532000) is an α1-Adrenoceptor antagonist structurally similar to Prozosin. Antihypertensive. Used in treatment of benign prostatic hypertrophy. (Alfuzosin Hydrochloride EP Impurity E )<br>References Ramage, A.G., et al.: Eur. J. Pharmacol., 129, 307 (1986), Deering, A.H.,: Brit. J. Clin. Pharmacol., 25, 417 (1988), Priolo, L.D., et al.: Eur. J. Clin. Pharmacol., 35, 25 (1988),<br></p>Formula:C15H21N5O3·HClColor and Shape:White To Off-WhiteMolecular weight:319.37 + (36.46)N-(2-Hydroxyethyl)-P,P-bisaziridinyl Thiophosphamide
CAS:Controlled ProductFormula:C6H14N3OPSColor and Shape:NeatMolecular weight:207.23Desfluoro Ezetimibe
CAS:Controlled Product<p>Impurity Ezetimibe Desfluoroaniline Analog (USP)<br>Stability Hygroscopic<br>Applications An impurity of the cholesterol absorption inhibitor Ezetimibe (E975000). Ezetimibe Desfluoroaniline Analog (USP).<br>References Anon.: IP.com J., 7, 4 (2007);<br></p>Formula:C24H22FNO3Color and Shape:White To Off-WhiteMolecular weight:391.43(R,S)(S,R)-Benidipine Hydrochloride
CAS:Formula:C28H31N3O6·HClColor and Shape:NeatMolecular weight:542.023Lodenafil Carbonate
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Lodenafil carbonate is a new PDE-5 inhibitor used for oral therapy in erectile dysfunction.<br>References Rosen, R., et al.: Urology, 49, 822 (1997), Chew, K., et al.: J. Sex Med., 5, 928 (2008), Teixeira, C., et al.: Eur. J. Pharmacol., 591, 189 (2008),<br></p>Formula:C47H62N12O11S2Color and Shape:NeatMolecular weight:1035.20Chlorpromazine Sulfoxide
CAS:<p>Impurity Chlorpromazine EP Impurity A<br>Applications Chlorpromazine Sulfoxide is a derivative of Chlorpromazine Hydrochloride (C424750), which is a dopamine antagonist of the typical antipsychotic class of medications possessing additional antiadrenergic, antiserotonergic, anticholinergic and antihistaminergic properties used for schizophrenia treatment.<br>References Anden, N.-E., et al.: Eur. J. Pharmacol., 11, 303 (1970), Curzon, G., et al.: Trends Pharmacol. Sci., 11, 61 (1990), Yuhas, D., Svi. Smer. Mind, (March 2003),<br></p>Formula:C17H19ClN2OSColor and Shape:Light YellowMolecular weight:334.864-(4-Methylpiperidin-4-yl)morpholinedihydrochloride
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:257.20001220703125Pibrentasvir
CAS:Controlled Product<p>Applications Pibrentasvir (CAS# 1353900-92-1) is an antiviral used for hepatitis C virus NS3/4A protease inhibition.<br>References Ng, T. I.; et al.: Antimicrob. Agents Chemother., 62, 1 (2018).<br></p>Formula:C57H65F5N10O8Color and Shape:Off-White To Light YellowMolecular weight:1113.18(2R)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile
CAS:Controlled Product<p>Applications (2R)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile, can be used in the synthesis of 1-[[(3-Hydroxy-1-adamantyl)amino]acetyl]-2-cyano-(S)-pyrrolidine, and Vildagliptin (C363780), which are potent, selective, and orally bioavailable dipeptidyl peptidase IV Inhibitor with Antihyperglycemic properties, that might be used for the treatment of type 2 diabetes.<br>References Singh, S.K., et al.: Beil. J. Org. Chem., 4, 20 (2008); Villhauer, E. B., et al.: J. Med. Chem., 46, 2774 (2003);<br></p>Formula:C7H9ClN2OColor and Shape:NeatMolecular weight:172.61Saquinavir
CAS:Controlled Product<p>Applications Saquinavir (CAS# 127779-20-8) is a useful research chemical compound.<br></p>Formula:C38H50N6O5Color and Shape:White To Off-WhiteMolecular weight:670.84rac 8,14-Dihydroxy Efavirenz-d4
CAS:Controlled Product<p>Applications A labelled metabolite of Efavirenz (E425000) (secondary metabolism).<br>References Gorski, J., et al.: Biochem. Pharmacol., 47, 1643 (1994), Desta, Z., et al.: J. Pharmacol. Exp. Ther., 285, 428 (1998), Langmann, P., et al.: Eur. J. Med. Res., 7, 309 (2002), Chang, T., et al.: Drug Metab. Dispos., 31, 7 (2003),<br></p>Formula:C14H5D4ClF3NO4Color and Shape:NeatMolecular weight:351.70Ethyl Ethanesulfonate
CAS:Controlled Product<p>Applications Ethyl Ethanesulfonate is used as a reactant in stereoselective Friedel-Crafts alkylation reactions. Also used in the preparation of 1-alkyl-3-methylimidazolium alkanesulfonate ionic liquids.<br>References Stadler, D., Bach, T.: Chem. Asian J., 3, 272 (2008); Blesic, M., et al.: Phys. Chem. Chem. Phys., 11, 8939 (2009);<br></p>Formula:C4H10O3SColor and Shape:NeatMolecular weight:138.19(R)-4-Hydroxy Propranolol Hydrobromide
CAS:Controlled Product<p>Applications The main metabolite of (R)-Propranolol.<br>References Shwed, J., et al.: Xenobiotica, 22, 973 (1992), Fujita, K., et al.: Biol. Pharm. Bull., 22, 446 (1999), Walle, U., et al.: Drug Metab. Dispos., 30, 564 (2002),<br></p>Formula:C16H21NO3·HBrColor and Shape:NeatMolecular weight:356.25(1-(4-Methylphenyl)-3-(4-(methylthio)phenyl)-1H-pyrazol-4-yl)methanol
CAS:Molecular weight:310.42001342773443-Chloro-4-nitropyridine N-oxide
CAS:Formula:C5H3ClN2O3Purity:95%Color and Shape:SolidMolecular weight:174.54Nitisinone-13C6
CAS:<p>Applications Labelled Nitisinone. Nitisinone is a herbicidal triketone that inhibits 4-hydroxyphenylpyruvate dioxygenase (HPPD), an enzyme involved in plastoquinone biosynthesis in plants and in tyrosine catabolism in mammals. It is used in treatment of inherited tyrosinemia type I.<br>References Lindstedt, S., et al.: Lancet, 340, 813 (1992), Ellis, M.K., et al.: Toxicol. Appl. Pharmacol., 133, 12 (1995), Lock, E.A., et al.: J. Inherited Metab. Dis., 21, 498 (1998),<br></p>Formula:C813C6H10F3NO5Color and Shape:Light Beige To BrownMolecular weight:335.18(3S,3'S)-4,4'-(7-Chloropyrido[2,3-d]pyrimidine-2,4-diyl)bis(3-methylmorpholine)
CAS:Purity:95.0%Molecular weight:363.85000610351564-(2-Aminophenyl)-3-morpholinone
CAS:<p>Applications 4-(2-Aminophenyl)-3-morpholinone is a reagent used in the preparation of various Morpholine based pharmaceuticals.<br>References Mederski, W., et al.: Bioorg. Med. Chem. Lett., 14, 3763 (2004), Roehrig, S., et al.: J. Med. Chem., 48, 5900 (2005),<br></p>Formula:C10H12N2O2Color and Shape:Off White SolidMolecular weight:192.214(R)-(+)-O-Desmethyl Carvedilol
CAS:Controlled Product<p>Applications An optically active metabolite of Carvedilol (C184625), a nonselective ß-adrenergic blocker with α-1-blocking activity. [α]D= +18.7 (c= 0.1 methanol)<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., et al.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Clohs, L., et al.: J. Pharm. Biomed. Anal., 31, 407 (2003),<br></p>Formula:C23H24N2O4Color and Shape:NeatMolecular weight:392.45(E)-3-(3-(3,4-dimethoxyphenyl)-1-phenyl-1H-pyrazol-4-yl)acrylic acid
CAS:Purity:98%Molecular weight:350.3739929199219(±)-Sibutramine
CAS:Controlled Product<p>Applications (±)-Sibutramine is a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure.<br>References Hanotin, C., et al.: Int. J. Obesity, 22, 32 (1998)<br></p>Formula:C17H26ClNColor and Shape:Off White SolidMolecular weight:279.85Methocarbamol β-D-Glucuronide Sodium Salt(Mixture of Diastereromers)
CAS:Controlled Product<p>Applications A metabolite of Methocarbamol (M225950).<br>References Thompson, R.M., et al.: Xenobiotica, 5,145 (1975),<br></p>Formula:C17H22NNaO11Color and Shape:White To Off-WhiteMolecular weight:439.35Deferiprone-d3
CAS:Controlled Product<p>Applications A chelator that could replace disferrioxamine. It is orally and parenterally effective in the removal of iron in vivo from rabbits and mice and also from transferrin and ferritin in vitro.<br>References Kontoghiorghes, G.J.: Lancet I, 817 (1985), Kontoghiorghes, G.J., et al.: Br. J. Haematol., 62, 607 (1986), Kontoghiorghes, G.J., et al.: Biochem. Biophys. Acta, 869, 141 (1986), Kontoghiorghes, G.J., et al.: Arzneim.-Forsch., 37, 1099 (1987),<br></p>Formula:C7H6D3NO2Color and Shape:White To Off-WhiteMolecular weight:142.17(R)-3-Aminopiperidine Dihydrochloride
CAS:Controlled Product<p>Applications (R)-3-Aminopiperidine Dihydrochloride has been used as a reactant for the preparation of dipeptidyl peptidase IV inhibitors derived from Alogliptin.<br>References Xie, Hui., et. al.: Eur. J. Med. Chem., 68, 312 (2013)<br></p>Formula:C5H14Cl2N2Color and Shape:NeatMolecular weight:173.08Edoxaban Tosylate Monohydrate
CAS:<p>Applications Edoxaban is an anticoagulant drug which acts as a direct factor Xa inhibitor.<br>References Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010)<br></p>Formula:C31H38ClN7O7S2•xH2OColor and Shape:White To Off-WhiteMolecular weight:720.26Dutasteride
CAS:Controlled Product<p>Applications Dutasteride is a dual inhibitor of 5α-reductase isoenzymes type 1 and 2; structurally related to Finasteride (F342000). Dutasteride is used in the treatment of benign prostatic hyperplasia.<br>References Bakshi, R.K., et al.: J. Med. Chem., 38, 3189 (1995), Gisleskog, P.O., et al.: Brit. J. Clin. Pharmacol., 47, 53 (1999), Djavan, B., et al.: Expert Opin. Pharmacother., 6, 311 (2005),<br></p>Formula:C27H30F6N2O2Color and Shape:NeatMolecular weight:528.532-[(2-Aminophenyl)amino]-5-methyl-3-thiophenecarbonitrile(Olanzapine Impurity)
CAS:Controlled Product<p>Applications An impurity of Olanzapine (O253750).<br>References Rao, R. et al.: J. Sep. Sci., 31, 107 (2008); Leyva-Perez, A. et al.: Tetrahedron, 66, 8203 (2010);<br></p>Formula:C12H11N3SColor and Shape:NeatMolecular weight:229.30Cloperastine Fendizoate
CAS:<p>Stability Hygroscopic<br>Applications Cloperastine fendizoate is used in the treatment of chronic non-productive cough. Antitussive. it is the salt of Cloperastine (CAS:3703-76-2)<br>References Aliprandi, P. et al.: Clin. Drug Invest. 22, 209 (2002)<br></p>Formula:C20H24ClNO·C20H14O4Color and Shape:White To Off-WhiteMolecular weight:648.19Trityl Chloride
CAS:Controlled Product<p>Applications Trityl Chloride is an alkyl halide commonly used in organic synthesis to introduce the trityl protecting group. Trityl Chloride is used in the preparation of S-trityl-L-cysteine (STLC), a tight-binding inhibitor of Eg5 that prevents mitotic progression.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References DeBonis, S. et al.: J. Med. Chem., 51, 1115 (2008); Chadwick, D.J. et al.: J. Chem. Soc. Perk. Trans. Org. Bio-Org. Chem., 1, 102 (1983);<br></p>Formula:C19H15ClColor and Shape:NeatMolecular weight:278.7822-Hydroxy Mifepristone-d6
CAS:Controlled Product<p>Applications A labelled metabolite of Mifepristone.<br>References Heikinheimo, O., et al.: J. Steroid Biochem., 26, 279 (1987), Brogden, R., et al.: Drugs, 45, 384 (1993), Shi, Y., et al.: Contraception, 48, 133 (1993), Jang, G., et al.: Biochem. Pharmacol., 52, 753 (1996), Gainer, E., et al.: Steroids, 68, 1005 (2003),<br></p>Formula:C29H29D6NO3Color and Shape:NeatMolecular weight:451.63Thiourea
CAS:Controlled Product<p>Applications Thiourea is used in biochemistry to increase the solubility (and resolution) of membrane proteins in two-dimensional electrophoresis. Thiourea is also used to treat thyrotoxicosis, a hypermetabolic clinical syndrome that is induced by multiple causes (Graves’ disease, hyperthyroidism, etc.).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Jabbour, S.: Am. J. Clin. Dermatol., 4, 315 (2003); Himsworth, H.: Lancet, 242, 465 (1943); Rabilloud, T., et al.: Electrophoresis, 19, 758 (1998)<br></p>Formula:CH4N2SColor and Shape:WhiteMolecular weight:76.124-phenyl-3-(2-thienyl)-1,2,4-triazoline-5-thione 98%
CAS:Purity:98.0%Molecular weight:259.3500061035156Anastrozole Dimer Impurity
CAS:Controlled Product<p>Impurity Anastrozole EP Impurity B / Anastrozole USP Related Compound C<br>Stability Hygroscopic<br>Applications Anastrozole Dimer Impurity (Anastrozole EP Impurity B) is an impurity of Anastrozole (A637425) (impurity C).<br></p>Formula:C30H31N9Color and Shape:Light YellowMolecular weight:517.631-[5-(Hydroxymethyl)-2-furyl]-2-methyl-1,2,3,4-tetrahydroisochinolin-4,6-diol
CAS:Controlled Product<p>Applications 1-[5-(Hydroxymethyl)-2-furyl]-2-methyl-1,2,3,4-tetrahydroisochinolin-4,8-diol is a degradation product of phenylephrine during the synthesis of the anti-cold medicine.<br>References Dousa, M. et al.: J. Pharm. Biomed. Anal., 55, 949 (2011);<br></p>Formula:C15H17NO4Color and Shape:NeatMolecular weight:275.30ETHYL 2-(3-METHYL-4-OXO-3,4-DIHYDROPHTHALAZIN-1-YL)ACETATE
CAS:Purity:95.0%Molecular weight:246.26600646972656Methocarbamol-d5
CAS:Controlled ProductFormula:C112H5H10NO5Color and Shape:NeatMolecular weight:246.27Carvedilol b-D-Glucuronide (mixture of diasteromers)
CAS:Controlled Product<p>Applications A metabolite of Carvedilol (C184625).<br>References McGurk, K., et al.: Biochem. Pharmacol., 55, 1005 (1998), Tukey, R., et al.: Annu. Rev. Pharmacol. Toxicol., 40, 581 (2000), Bowalgaha, K., et al.: Br. J. Clin. Pharmacol., 52, 605 (2001), Richardson, T., et al.: Drug Metab. Dispos., 34, 351 (2006),<br></p>Formula:C30H34N2O10Color and Shape:NeatMolecular weight:582.60N-(5-chloropyridin-2-yl)-2-(4-cyanobenzamido)-5-methoxybenzamide
CAS:Purity:97%Molecular weight:406.8299865722656Nicarbazine
CAS:Controlled Product<p>Applications Nicarbazine, is a coccidiostat, which is an antiprotozoal agent that acts upon Coccidia parasites.<br>References Ksenija Sinigoj, G., et al.: Slovenski Kemijski Dnevi, (2012); Kyung-Woo, L., et al.: Han'guk Kagum Hakhoechi, 39, 17 (2012);<br></p>Formula:C13H10N4O5·C6H8N2OColor and Shape:NeatMolecular weight:426.38Phenformin Hydrochloride
CAS:<p>Applications It is an anti-diabetic drug from the biguanide class.<br>References Moody, J.E., Anal. Profiles Drug Subs., 4, 319 (1975),<br></p>Formula:C10H15N5·ClHColor and Shape:NeatMolecular weight:241.727-Hydroxy-N-des{[2-(2-hydroxy)ethoxy]ethyl} Quetiapine Dihydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A metabolite of Quetiapine.<br>References McConville, B., et al.: J. Clin. Psychiatry, 61, 252 (2000), Wong, Y., et al.: J. Clin. Psychopharmacol, 21, 89 (2001), Cooper, K., et al.: Eur. J. Clin. Pharmacol., 59, 51 (2003),<br></p>Formula:C17H17N3OS·2ClHColor and Shape:White To Off-WhiteMolecular weight:384.324-Amino-6-ethoxy-5-[[4-[(4R)-1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl]phenyl]azo]-α-[[4-[(4R)-1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl]phenyl]hydrazono]-2-pyrimidineacetonitrile
CAS:<p>Applications 4-Amino-6-ethoxy-5-[[4-[(4R)-1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl]phenyl]azo]-α-[[4-[(4R)-1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl]phenyl]hydrazono]-2-pyrimidineacetonitrile is a levosimendan dimer impurity, which is a bioactive enantiomer of racemate, Simendan. Positive inotropic agent with vasodilating activity. Cardiotonic.<br>References Sandell, E.-P., et al.: J. Cardiovasc. Pharmacol., 26, S57 (1995), Pagel, P.S., et al.: Cardiovasc. Drug Rev., 14, 286 (1996),<br></p>Formula:C30H30N12O3Color and Shape:NeatMolecular weight:606.64Dehydro Levetiracetam
CAS:<p>Impurity Levetiracetam EP Impurity B<br>Stability Light Sensitive<br>Applications Dehydro Levetiracetam (Levetiracetam EP Impurity B) is an impurity of Levetiracetam (L331500) which is an (S)-enantiomer of Etiracetam (E932970) and the ethyl analog of Piracetam (P500800). Used as an anticonvulsant.<br>References Gower, A. J., et al.: Eur. J. Pharmacol., 222, 193 (1992); Kasteleijn-Noist Trenite, D.G.A., et al.: Epilepsy Res., 25, 225 (1996); Patsalos, P.N., et al.: Pharmacol. Ther., 85, 77 (2000)<br></p>Formula:C8H12N2O2Color and Shape:WhiteMolecular weight:168.192,3-Dihydro-3,5-dihydroxy-6-methyl-4-pyrone
CAS:Controlled ProductFormula:C6H8O4Color and Shape:NeatMolecular weight:144.13Norketamine-d4
CAS:Controlled Product<p>Applications A labelled metabolite of Ketamine (K165300).<br>References Sullivan, H., et al.: J. Med. Chem., 16, 909 (1973), Moreton, J., et al.: J. Pharmacol. Exp. Ther., 203, 303 (1977), Lin, H., et al.: J. Food Drug Anal., 13, 107 (2005),<br></p>Formula:C12H10D4ClNOColor and Shape:NeatMolecular weight:227.72Ethyl 7-chloro-8-cyano-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylate
CAS:Purity:95+%Molecular weight:334.73001098632811,5-Dihydroxyempagliflozin
CAS:Controlled ProductFormula:C23H29ClO8Color and Shape:NeatMolecular weight:468.92Reserpine-d9
CAS:Controlled Product<p>Applications Labelled Reserpine (R144600). An indole alkaloid found in Rauwolfia serpentina. Inhibits vesicular uptake of catecholamines and serotonin. Reserpine is reasonably anticipated to be a human carcinogen. Antihypertensive.<br>References Muller, J.M., et al.: Experientia, 8, 338 (1952), Schirmer, R.E., et al.: Anal. Profiles Drug Subs., 4, 384 (1975), Diener, R.M., et al.: Toxicol. Pathol., 8, 1 (1980),<br></p>Formula:C332H9H31N2O9Color and Shape:NeatMolecular weight:617.733-Methyl-1-phenyl-1H-pyrazole-5-carboxylic acid
CAS:Formula:C11H10N2O2Purity:98%Color and Shape:SolidMolecular weight:202.213Cyanuric Acid (1 mg/10 mL in 84:16% ACN:H2O)
CAS:Controlled ProductFormula:C3H3N3O3Color and Shape:Single SolutionMolecular weight:129.07Brexpiprazole N-Oxide
CAS:Controlled Product<p>Stability Not Stable in DMSO<br>Applications Brexpiprazole N-Oxide is an impurity and potential metabolite of Brexpiprazole (B677385), a drug candidate useful in treatment and prevention of mental disorders including CNS disorders.<br>References Yamashita, H., et al.: PCT Int. Appl., WO 2006112464 A1 20061026 (2006);<br></p>Formula:C25H27N3O3SColor and Shape:NeatMolecular weight:449.57Asenapine N-Oxide
CAS:Controlled Product<p>Applications A metabolite of Asenapine (A788000).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Ven der Wildenberg, H.M., et al.: Arzneim.-Forsch., 40, 540 (1990),<br></p>Formula:C17H16ClNO2Color and Shape:NeatMolecular weight:301.77Etomidate
CAS:Controlled Product<p>Applications Etomidate is a hypnotic. Neuroprotective & Neuroresearch Products<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Goetz, E., et al.: Anaesthesist, 23, 331 (1974), Chang, Z. L., et al.: Anal. Profiles Drug Subs., 12, 191 (1983),<br></p>Formula:C14H16N2O2Color and Shape:Off-WhiteMolecular weight:244.29Desisopropyl Atrazine-d5
CAS:Controlled Product<p>Applications A labelled metabolite of Atrazine (ATR) (A794600).<br>References Compton, D., et al.: Eur. J. Pharmacol., 110, 157 (1985), Das, P., et al.: Toxicol. Sci., 59, 127 (2001), Das, P., et al.: Life Sci., 73, 3123 (2003), Coban, A., et al.: J. Neurochem., 100, 1177 (2007),<br></p>Formula:C52H5H3ClN5Color and Shape:Off-WhiteMolecular weight:178.63Meloxicam-d3
CAS:Controlled Product<p>Applications Labelled form of Meloxicam. Preferential cyclooxygenase (COX-2) inhibitor. Used as an anti-inflammatory.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hawkey, C., et al.: Br. J. Rheumatol., 35, Suppl. 1, 1 (1996), Fleischmann, R., et al.: Expert Opin. Pharmacother., 3, 1501 (2002),<br></p>Formula:C142H3H10N3O4S2Color and Shape:Light Yellow To YellowMolecular weight:354.42Desmethyl Sibutramine
CAS:Controlled Product<p>Applications Desmethyl Sibutramine is a metabolite of Sibutramine (S422500), a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure.<br>References Hanotin, C., et al.: Int. J. Obesity, 22, 32 (1998); Woolard, J., et al.: J. Pharmacol. Exp. Ther., 308, 1102 (2004); Geranton, S., et al.: Neuropharmacol., 46, 511 (2004)<br></p>Formula:C16H24ClNColor and Shape:Colourless To YellowMolecular weight:265.822-(5-Methylthiophen-2-yl)quinoline-4-carboxylic acid
CAS:Color and Shape:SolidMolecular weight:269.32000732421875Mizolastine
CAS:<p>Applications A highly selective histamine H1-receptor antagonist (with no anticholinergic, antiadrenergic, or antiserotonin activity) for use in the treatment of allergic disorders, especially rhinitis and urticaria.<br>References Simons, F.E.R.: Clin. Alp. Allergy, 29, 3 (1999); Brostoff, J. et al.: Allergy, 51, 251 (1996); Gensthaler, B.M.: Pharm. Zeit., 143, 228 (1998);<br></p>Formula:C24H25FN6OColor and Shape:NeatMolecular weight:432.49
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