
Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65562 products of "Quinazoline and Quinoline Derivatives"
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Tafamidis
CAS:<p>Tafamidis stabilizes TTR, preventing amyloid buildup; binds with negative cooperativity (Kd1: 3 nM, Kd2: 278 nM); treats familial amyloid polyneuropathy.</p>Formula:C14H7Cl2NO3Purity:99.34% - 99.65%Color and Shape:SolidMolecular weight:308.12Terazosin
CAS:<p>Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.</p>Formula:C19H25N5O4Color and Shape:SolidMolecular weight:387.43Betahistine dihydrochloride
CAS:<p>Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.</p>Formula:C8H14Cl2N2Purity:99.34% - 99.88%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:209.12(S)-Afatinib
CAS:<p>(S)-Afatinib (BIBW2992) is an irreversible EGFR family inhibitor with IC50s of 0.5/0.4/10/14/1 nM for EGFRwt, L858R, L858R/T790M, HER2, and HER4, respectively.</p>Formula:C24H25ClFN5O3Purity:99.22% - >99.99%Color and Shape:Off-White SolidMolecular weight:485.94Elenbecestat free base
CAS:<p>Elenbecestat (E2609) is a BACE1 inhibitor that reduces Aβ peptide formation, potentially preventing amyloid plaques in the brain.</p>Formula:C19H15F6N5O2SColor and Shape:SolidMolecular weight:491.41Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54Bedaquiline
CAS:<p>Bedaquiline, an anti-TB drug, blocks mycobacterial ATP synthesis, effective against all Mycobacterium tuberculosis states.</p>Formula:C32H31BrN2O2Purity:98% - 99.8%Color and Shape:SolidMolecular weight:555.5Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Formula:C12H19Cl2NOPurity:99.24% - >99.99%Color and Shape:Appearance White Crystalline PowderMolecular weight:264.19Benidipine
CAS:<p>Benidipine: potent oral calcium blocker, boosts nitric oxide synthase, enhances coronary flow, protects heart cells post-ischemia.</p>Formula:C28H31N3O6Color and Shape:SolidMolecular weight:505.56Barnidipine
CAS:<p>Barnidipine (YM-09730-5(Free base)) is a calcium channel blocker.</p>Formula:C27H29N3O6Purity:99.98%Color and Shape:SolidMolecular weight:491.54Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Formula:C20H25NO2S2Purity:99.25%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55eCF506
CAS:<p>eCF506 is a potent and selective inhibitor of SRC (IC50 < 0.5 nM)</p>Formula:C26H38N8O3Purity:97.85% - 98.16%Color and Shape:SolidMolecular weight:510.631-Phenylpropane-1,2-dione
CAS:<p>1-Phenylpropane-1,2-dione (Acetyl benzoyl) is a eukaryotic metabolite produced in plant metabolic reactions.</p>Formula:C9H8O2Purity:97.12%Color and Shape:LiquidMolecular weight:148.16Morroniside
CAS:<p>Morroniside regulates liver inflammation, lipid metabolism, protects against diabetic kidney damage, and guards the brain from ischemic injury.</p>Formula:C17H26O11Purity:99.70% - 99.84%Color and Shape:SolidMolecular weight:406.38Pyr10
CAS:<p>Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.</p>Formula:C18H13F6N3O2SPurity:99.69% - 99.7%Color and Shape:SolidMolecular weight:449.37Paritaprevir
CAS:<p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。</p>Formula:C40H43N7O7SPurity:99.72%Color and Shape:SolidMolecular weight:765.88

