Enzyme Modulators
Enzyme modulators are compounds that can enhance or inhibit the activity of enzymes, thereby regulating the rate of biochemical reactions. These modulators play a critical role in controlling metabolic pathways, cell signaling, and various physiological processes. Enzyme modulators are widely used in research and drug development to study enzyme functions and to develop therapeutic agents. At CymitQuimica, we offer a comprehensive range of high-quality enzyme modulators to support your research in enzyme regulation and drug discovery.
Subcategories of "Enzyme Modulators"
Found 693 products of "Enzyme Modulators"
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Mirodenafil dihydrochloride
CAS:<p>Mirodenafil dihydrochloride is a potent phosphodiesterase-5 (PDE5) inhibitor, which is a synthetic compound with a primarily chemical origin. Its mode of action involves the inhibition of the enzyme PDE5, which predominantly resides in the smooth muscle cells lining blood vessels. By inhibiting PDE5, Mirodenafil dihydrochloride effectively increases the levels of cyclic guanosine monophosphate (cGMP), leading to the relaxation of smooth muscle tissues and vasodilation.</p>Formula:C26H39Cl2N5O5SPurity:Min. 97 Area-%Color and Shape:White PowderMolecular weight:604.59 g/molMefenamic acid
CAS:<p>COX1 inhibitor; blocker of Ca2+-activated non-selective cation channels</p>Formula:C15H15NO2Purity:Min. 99 Area-%Color and Shape:White PowderMolecular weight:241.29 g/molMetformin HCl - Bio-X ™
CAS:<p>Metformin is a widely used anti-hyperglycemic (anti-diabetic) agent for the treatment of type 2 diabetes mellitus. This is due to it decreasing blood glucose by decreasing hepatic glucose product by activation of the AMP-activated protein kinase AMPK. Studies have also demonstrated Metformin to have anti-cancer activity, attributed to several mechanisms such as inhibition of mammalian target of rapamycin (mTOR), cancer stem cells and inflammation.</p>Formula:C4H11N5•HClPurity:Min. 95%Color and Shape:PowderMolecular weight:165.62 g/molLenvatinib mesylate - Bio-X ™
CAS:<p>Lenvatinib is an anti-cancer drug that is a multi-kinase inhibitor for VEGFR1, VEGFR2 and VEGFR. It has been shown to be effective against several cancers such as thyroid cancer and is currently in clinical trials for the treatment of leukaemia and prostate cancer. Furthermore, Lenvatinib also inhibits the activity of other protein kinases, including those involved in inflammatory responses.</p>Formula:C22H23ClN4O7SPurity:Min. 95%Color and Shape:PowderMolecular weight:522.96 g/molPexidartinib
CAS:<p>Inhibitor of CSF1R receptor</p>Formula:C20H15ClF3N5Purity:Min. 95%Color and Shape:PowderMolecular weight:417.81 g/molTH 5487
CAS:<p>Specific inhibitor of 8-oxoguanine glycosylase OGG1 with IC50 in submicromolar range. The compound inhibits binding of OGG1 to its substrate 8-oxoguanine, a guanine analog generated in the presence of reactive oxygen species (ROS). It was shown that TH5487 decreases inflammation level by inhibiting the base excision DNA repair in mice and altering the OGG1 chromatin dynamics. The compound also has implications in cancer biology since OGG1 inhibitors sensitise tumours to chemotherapy.</p>Formula:C19BrH18IN4O2Purity:Min. 95%Color and Shape:SolidMolecular weight:541.18 g/molPitavastatin lactone
CAS:<p>Inhibitor of HMG-CoA reductase</p>Formula:C25H22FNO3Purity:Min. 95%Color and Shape:PowderMolecular weight:403.45 g/mol(R)-Lansoprazole
CAS:<p>Gastric proton pump inhibitor</p>Formula:C16H14F3N3O2SPurity:Min. 95%Color and Shape:PowderMolecular weight:369.36 g/molN-ω-Propyl-L-arginine
CAS:<p>Neuronal selective nitric oxide synthase inhibitor</p>Formula:C9H20N4O2Purity:Min. 95%Color and Shape:White PowderMolecular weight:216.28 g/molZoledronic acid, disodium salt, tetrahydrate
CAS:<p>Farnesyl pyrophosphate synthase inhibitor; hepatic de novo lipogenesis inhibitor</p>Formula:C5H8N2Na2O7P2·4H2OPurity:Min. 98 Area-%Color and Shape:PowderMolecular weight:388.11 g/molUNC 3230
CAS:<p>Inhibitor of PIP5K1C</p>Formula:C17H20N4O2SPurity:Min. 95%Color and Shape:SolidMolecular weight:344.43 g/molIrinotecan hydrochloride trihydrate - Bio-X ™
CAS:<p>Irinotecan hydrochloride trihydrate is a topoisomerase I inhibitor that is used as chemotherapy drug for colorectal cancer. By inhibiting topoisomerase I, Irinotecan hydrochloride trihydrate prevents the replication of DNA in cells, and stops the cancer cells from growing and dividing. When used for chemotherapy, Irinotecan hydrochloride trihydrate is usually part of combination therapy with other chemotherapy drugs, such as 5-fluorouracil (5-FU) and leucovorin for other cancers.</p>Formula:C33H38N4O6•HCl•(H2O)3Purity:Min. 95%Color and Shape:PowderMolecular weight:677.18 g/molLenvatinib base - Bio-X ™
CAS:<p>Lenvatinib is a tyrosine kinase inhibitor that is used to treat cancers such as solid tumours. This drug inhibits the activity of VEGR receptors. It also inhibits other receptors such as fibroblast growth factor.</p>Formula:C21H19ClN4O4Purity:Min. 95%Color and Shape:PowderMolecular weight:426.85 g/molTandutinib
CAS:<p>Tyrosine kinase inhibitor; antineoplastic activity; pro-apoptotic</p>Formula:C31H42N6O4Purity:Min. 95%Color and Shape:PowderMolecular weight:562.7 g/molVorinostat - Bio-X ™
CAS:<p>Vorinostat is a histone deacetylase inhibitor which interferes with gene transcription regulatory mechanisms. It is used to treat cutaneous manifestations in patients with progressive, persistent, or recurrent cutaneous T- cell lymphoma (CTCL) following prior systemic therapies. This drug inhibits the enzymatic activity of histone deacetylases HDAC1, HDAC2 and HDAC3 (Class I) and HDAC6 (Class II).</p>Formula:C14H20N2O3Purity:Min. 99 Area-%Color and Shape:PowderMolecular weight:264.32 g/molDarapladib
CAS:<p>Inhibitor of lipoprotein-associated phospholipase A2</p>Formula:C36H38F4N4O2SPurity:Min. 98 Area-%Color and Shape:PowderMolecular weight:666.77 g/molQuizartinib
CAS:<p>Inhibitor of FLT3 receptor tyrosine kinases; anti-neoplastic</p>Formula:C29H32N6O4SPurity:Min. 95%Color and Shape:White PowderMolecular weight:560.67 g/molAzaserine
CAS:<p>Glutamine analogue and antagonist of glutamine-dependent amidotransferases, with antibiotic and antifungal properties. Inhibits purine biosynthesis, FGAM synthetase and glucosamine-6-phosphate isomerase that contributes to its antineoplastic property. Azaserine can also act as a carcinogen, by inducing DNA carboxymethylation. Protects endothelial cells from inflammation under hyperglycemic conditions, via antioxidant mechanisms, independent of hexosamine biosynthetic pathway.</p>Formula:C5H7N3O4Purity:Min. 98 Area-%Color and Shape:Slightly Yellow PowderMolecular weight:173.13 g/mol(Z)-PugNAc
CAS:<p>Inhibitor of O-GlcNAcase and N-acetylhexosaminidases</p>Formula:C15H19N3O7Purity:Min. 97 Area-%Color and Shape:White PowderMolecular weight:353.33 g/molAZ 960
CAS:<p>ATP competitive JAK2 inhibitor</p>Formula:C18H16F2N6Purity:Min. 95%Color and Shape:PowderMolecular weight:354.36 g/mol
