Ciclo celular / Checkpoint
Los inhibidores del ciclo celular/puntos de control son compuestos que interrumpen la progresión normal del ciclo celular, particularmente en puntos de control regulatorios clave. Estos inhibidores son cruciales para estudiar la división celular, comprender la proliferación de células cancerosas y desarrollar terapias anticancerígenas. Al dirigirse a fases específicas del ciclo celular, estos inhibidores pueden inducir la detención del ciclo celular, lo que lleva a apoptosis o senescencia en células de división rápida. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad del ciclo celular/puntos de control para apoyar su investigación en biología del cáncer, biología celular y desarrollo de fármacos.
Subcategorías de "Ciclo celular / Checkpoint"
- Aurora quinasa(114 productos)
- CDK(546 productos)
- Detención del ciclo celular(5 productos)
- Chk(48 productos)
- DYRK(47 productos)
- Dynamin(27 productos)
- Ferroptosis(227 productos)
- HSP(180 productos)
- Integrin(269 productos)
- Kinesina(87 productos)
- LIM quinasa(20 productos)
- Asociado a microtúbulos(274 productos)
- PKC(126 productos)
- PLK(25 productos)
- ROCK(62 productos)
- Rho(6 productos)
- Wee1(14 productos)
- c-Myc(76 productos)
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Se han encontrado 3904 productos de "Ciclo celular / Checkpoint"
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Meturedepa
CAS:Meturedepa is an antineoplastic agent.Fórmula:C11H22N3O3PPureza:98%Forma y color:SolidPeso molecular:275.28DHODH-IN-13
CAS:DHODH-IN-13 is an inhibitor of DHODH with IC50 of 4.3 μM for rat liver. DHODH-IN-13 can be used in studies about rheumatoid arthritis.Fórmula:C10H6F3N3O3Pureza:99.66%Forma y color:SolidPeso molecular:273.17hDHODH-IN-5
CAS:hDHODH-IN-5 is an inhibitor of human dihydroorotate dehydrogenase (hDHODH, IC50 = 0.91 μM).Fórmula:C21H21F3N2O2Pureza:99.55%Forma y color:SolidPeso molecular:390.4Ref: TM-T11029
1mg80,00€5mg158,00€10mg221,00€25mg356,00€50mg530,00€100mg755,00€1mL*10mM (DMSO)172,00€CCT068127
CAS:CCT068127 is a potent CDK2 and CDK9 inhibitor.Fórmula:C19H27N7OForma y color:SolidPeso molecular:369.46BzDANP
CAS:BzDANP is a modulator of pre-miR-29a maturation by Dicer.Fórmula:C18H24N6Forma y color:SolidPeso molecular:324.42L 703014
CAS:L 703014 is an antagonist of the fibrinogen receptor.Fórmula:C24H34N4O4Pureza:98%Forma y color:SolidPeso molecular:442.55SEC inhibitor KL-2
CAS:KL-2: potent SEC inhibitor, selectively disrupts AFF4-CCNT1, dose-dependent, Ki: 1.50 μM.Fórmula:C17H13ClFNO3Pureza:99.86%Forma y color:SolidPeso molecular:333.74L-Fd4A
CAS:L-Fd4A (compound 36) is an adenine derivative with anti-HIV (EC50=1.5μM) and anti-HBV (EC50=1.7μM) effects, low cytotoxicity.Fórmula:C10H10FN5O2Forma y color:SolidPeso molecular:251.22AM-TS23
CAS:AM-TS23 is used as a DNA polymerase lambda and beta inhibitor.Fórmula:C17H12N2O3S3Pureza:98%Forma y color:SolidPeso molecular:388.48Nucleoside-Analog-1
CAS:Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.Fórmula:C9H9N5O5Pureza:98%Forma y color:SolidPeso molecular:267.2ML366
CAS:ML366 is a Vibrio cholerae Quorum Sensing inhibitor Acting via the LuxO response regulator.Fórmula:C17H19N3O4Pureza:98%Forma y color:SolidPeso molecular:329.35HBX28258
CAS:HBX28258, a human USP7 inhibitor, binds covalently and selectively deactivates USP7 in colon cancer and kidney cells.Fórmula:C26H30ClN3OPureza:98%Forma y color:SolidPeso molecular:435.99XL-188
CAS:XL-188: Potent, selective USP7 inhibitor, IC50 = 193 nM (domain), 90 nM (full). Boosts p53, p21; degrades HDM2. Unique among DUB inhibitors.Fórmula:C32H42N6O4Forma y color:SolidPeso molecular:574.71JNJ-9676
CAS:JNJ-9676 is an orally active inhibitor of the coronavirus membrane protein, thereby blocking viral assembly and release.coronavirus and SARS-CoV.Fórmula:C28H21F2N5O2Pureza:99.83%Forma y color:SoildPeso molecular:497.5Ref: TM-T205924
1mg137,00€5mg330,00€10mg532,00€25mg1.108,00€50mg1.738,00€100mg2.592,00€1mL*10mM (DMSO)354,00€OXA-06 Dihydrochloride
CAS:OXA-06 Dihydrochloride is a PANC-1 cell migration and MYPT1 phosphorylation inhibitor.Fórmula:C21H18FN3Pureza:98%Forma y color:SolidPeso molecular:331.39Levofloxacin sodium
CAS:Levofloxacin sodium: synthetic antibacterial, stops DNA replication by inhibiting bacterial DNA gyrase.Fórmula:C18H20FN3NaO4Pureza:98%Forma y color:SolidPeso molecular:384.363LY 207702
CAS:LY 207702, a difluorinated purine nucleoside, exhibits antitumor activity in preclinical models.Fórmula:C10H12F2N6O3Pureza:98%Forma y color:SolidPeso molecular:302.24CDK4/6-IN-12
CAS:CDK4/6-IN-12 inhibits CDK4/6 with IC50s of 592.3 nM & 3090 nM, useful in cancer research.Fórmula:C12H10N6Forma y color:SolidPeso molecular:238.25Codon readthrough inducer 1
CAS:Codon readthrough inducer 1 contains pyrimidine bases and shows good readthrough activity.Fórmula:C15H11N3O5Pureza:98%Forma y color:SolidPeso molecular:313.26MS0017509
CAS:MS0017509 is a DNA damage repair inhibitor.Fórmula:C11H10N4Pureza:98%Forma y color:SolidPeso molecular:198.222'-Fluorothymidine
CAS:2'-Fluorothymidine is a selective substrate for TK2, related to thymidine and methyluridine.Fórmula:C10H13FN2O5Pureza:99.98%Forma y color:SolidPeso molecular:260.22Ref: TM-T19101
1mg50,00€5mg105,00€10mg161,00€25mg276,00€50mg416,00€100mg625,00€200mg837,00€1mL*10mM (DMSO)101,00€Kira8 Hydrochloride
CAS:Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Fórmula:C31H30Cl2N6O3SPureza:98%Forma y color:SolidPeso molecular:637.58SC-203885
CAS:SC-203885 is a checkpoint kinase 2 inhibitor.Fórmula:C15H13N5O2Pureza:98%Forma y color:SolidPeso molecular:295.3hDHODH-IN-4
CAS:hDHODH-IN-4, a potent DHODH inhibitor, has a pIC50 of 7.8 and blocks measles virus replication with a pMIC50 of 8.8.Fórmula:C21H24N4O2Pureza:99.87%Forma y color:SolidPeso molecular:364.44Tetrahydrouridine
CAS:Tetrahydrouridine (NSC-112907; THU) is a multidrug resistance modulator.Fórmula:C9H16N2O6Pureza:98%Forma y color:SolidPeso molecular:248.23BMH-23
CAS:BMH-23 is an RNA polymerase I inhibitor that acts by causing nucleolar stress and showing potent anticancer activity across many tumor types.Fórmula:C15H15N3Pureza:98%Forma y color:SolidPeso molecular:237.3AnnH31
CAS:AnnH31 is a potent Dyrk1A inhibitor with an IC50 value of 81 nM.AnnH31 inhibits MAO-A with an IC50 of 3.2 μM.AnnH31 can be used as a probe to confirm theFórmula:C15H13N3OPureza:99.99%Forma y color:SolidPeso molecular:251.28Phelorphan
CAS:Phelorphan is an inhibitor of enkephalinase.Fórmula:C20H22N2O4SPureza:98%Forma y color:SolidPeso molecular:386.46CDK8-IN-10
CAS:CDK8-IN-10 is a selective and potent inhibitor of cell cycle protein-dependent kinase (CDK8) (IC50: 8.25 nM) that can be used to study cancer.Fórmula:C25H15ClF3N5O3Forma y color:SolidPeso molecular:525.87A 65282
CAS:A 65282: antibacterial isothiazoloquinolone, inhibits P4-unknotting, causes DNA breaks via topoisomerase II.Fórmula:C17H16F2N4O2SPureza:98%Forma y color:SolidPeso molecular:378.4RP-106
CAS:RP-106 is an ATP-competitive inhibitor of CDK5/p25, CDK1/cyclin B, and GSK-3.Fórmula:C17H19N3OPureza:98%Forma y color:SolidPeso molecular:281.35CFM-1
CAS:CFM-1 is an antagonist of the anaphase-promoting complex (APC)-2. It also is a cell cycle and apoptosis regulatory protein (CARP)-1 interaction antagonist.Fórmula:C12H7BrN2O2S2Pureza:98%Forma y color:SolidPeso molecular:355.23PD 130883
CAS:PD 130883 is a potent lipophilic quinazoline antifolate.Fórmula:C18H15N5O3Pureza:98%Forma y color:SolidPeso molecular:349.34Apricitabine
CAS:Apricitabine (SPD754) is a highly selective and orally active HIV-1 reverse transcriptase inhibitor (Ki=0.08 μM), the (-) enantiomer of 2′-deoxy-3′-oxy-4′-Fórmula:C8H11N3O3SPureza:99.45%Forma y color:SolidPeso molecular:229.26Ref: TM-T14313
1mg283,00€5mg507,00€10mg628,00€25mg962,00€50mg1.601,00€100mg2.682,00€1mL*10mM (DMSO)592,00€RUC-1
CAS:RUC-1 is an αIIbβ3-selective ADP-induced platelet aggregation inhibitor.Fórmula:C11H15N5OSPureza:98%Forma y color:SolidPeso molecular:265.33Homocarbonyltopsentin
CAS:Homocarbonyltopsentin: Small molecule, binds TSL2 pentaloops, enhances SMN2 E7 splicing, EC50 16 μM.Fórmula:C21H14N4O3Pureza:98%Forma y color:SolidPeso molecular:370.36Guanoctine hydrochloride
CAS:Guanoctine hydrochloride has antihypertensive activity.Fórmula:C9H22ClN3Forma y color:SolidPeso molecular:207.74ROCK-IN-D2
CAS:ROCK-IN-D2 is an effective and selective inhibitor of ROCK.Fórmula:C22H28N6OPureza:98%Forma y color:SolidPeso molecular:392.5RHI002-Me
CAS:RHI002-Me is a methylated derivative of RHI002, a selective inhibitor of human RNaseH2.Fórmula:C18H19N3O2S2Pureza:98%Forma y color:SolidPeso molecular:373.49MFH290
CAS:MFH290 is a selective CDK12/13 inhibitor, covalently bonding with CDK12 Cys-1039, blocks Pol II CTD phosphorylation, and enhances olaparib's efficacy.Fórmula:C26H31N5O3S2Forma y color:SolidPeso molecular:525.69A 65281
CAS:A 65281: antibacterial isothiazoloquinolone, inhibits P4-unknotting, induces DNA breakage via topoisomerase II.Fórmula:C17H16F2N4O2SPureza:98%Forma y color:SolidPeso molecular:378.4Balamapimod
CAS:Balamapimod is a reversible inhibitor of Ras/Raf/MEK. It also has a potential anti-tumor activity.Fórmula:C30H32ClN7OSPureza:98%Forma y color:SolidPeso molecular:574.14CDK9-IN-15
CAS:CDK9-IN-15: potent CDK9 inhibitor, blocks P-TEFb phosphorylation, inhibits transcription, reduces mRNA, induces tumor cell apoptosis.Fórmula:C16H11N3OSPureza:99.32%Forma y color:SolidPeso molecular:293.34Ref: TM-T60619
5mg46,00€10mg71,00€25mg126,00€50mg180,00€100mg260,00€200mg364,00€1mL*10mM (DMSO)44,00€Capzimin
CAS:Capzimin is a selective inhibitor of proteasome isopeptidase Rpn11.Fórmula:C30H24N6O2S4Pureza:98.31% - 99.32%Forma y color:SolidPeso molecular:628.81Ref: TM-T10672
1mg48,00€2mgA consultar5mg95,00€10mg150,00€25mg300,00€50mg515,00€1mL*10mM (DMSO)131,00€(E/Z)-BIO-acetoxime
CAS:(E/Z)-BIO-acetoxime: potent GSK-3 α/β inhibitor; IC50: GSK-3α/β 10nM, CDK5/p25 2.4μM, CDK2/A 4.3μM, CDK1/B 63μM.Fórmula:C18H12BrN3O3Forma y color:SolidPeso molecular:398.21Zaurategrast ethyl ester
CAS:Zaurategrast ethyl ester, an α4β1/α4β7 integrin antagonist prodrug of CT7758, treats inflammatory/autoimmune conditions.Fórmula:C28H29BrN4O3Pureza:98%Forma y color:SolidPeso molecular:549.46CTP Synthetase-IN-1
CAS:CTP Synthetase-IN-1 is a cytidine 5'-triphosphate synthetase (CTPS) inhibitor with antitumor activity for the study of arthritis and rheumatoid arthritis.Fórmula:C20H19F3N6O3S2Pureza:98.11% - 99.18%Forma y color:SolidPeso molecular:512.53Ref: TM-T72505
1mg65,00€5mg141,00€10mg230,00€25mg477,00€50mg803,00€100mg1.378,00€1mL*10mM (DMSO)158,00€BRD9185
CAS:BRD9185 is an inhibitor of Dihydroorotate dehydrogenase (DHODH) with an EC50 of 16 nM against multidrug-resistant blood-stage parasites in vitro.Fórmula:C23H21F6N3O2Pureza:98%Forma y color:SolidPeso molecular:485.42Scaff10-8
CAS:Scaff10-8 blocks AKAP-Lbc-RhoA, aiding aquaporin-2 movement in kidney cells.Fórmula:C22H18O6Pureza:98%Forma y color:SolidPeso molecular:378.37DHODH-IN-1
CAS:DHODH-IN-1 is a potent dihydroorotate dehydrogenase (DHODH) inhibitor with IC50 of 25 nM. DHODH-IN-1 is an inhibitor of the pyrimidine biosynthetic pathway.Fórmula:C21H20F3N3O2Pureza:99.76%Forma y color:SolidPeso molecular:403.4Aurora A/PKC-IN-1
CAS:Aurora A/PKC-IN-1 inhibits AurA (IC50: 6.9 nM), PKCα (IC50: 16.9 nM), and hinders breast cancer cell growth and spread.Fórmula:C16H14N6OSe2Forma y color:SolidPeso molecular:464.24D-Xylofuranose, 1,2,3,5-tetraacetate
CAS:1,2,3,5-Tetra-O-acetyl-D-xylofuranose is a starting material for the synthesis of nucleosides.Fórmula:C13H18O9Forma y color:SolidPeso molecular:318.28NSC666715
CAS:NSC666715 is the strand-displacement activity of DNA polymerase inhibitor.Fórmula:C15H13Cl2N5O2S2Pureza:98%Forma y color:SolidPeso molecular:430.33FD-IN-1
CAS:FD-IN-1 is an orally active Factor D (FD) inhibitor (IC50=12 nM), inhibits Factor XIa and Tryptase β2 with IC50 values of 7.7 and 6.5 μM, respectively.Fórmula:C23H23NO4Pureza:98.85%Forma y color:SolidPeso molecular:377.43XU1
CAS:XU1（Benzo[c][1,8]naphthyridin-6(5h)-One） is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation orFórmula:C12H8N2OPureza:97.81% - 99.59%Forma y color:SolidPeso molecular:196.2Zaurategrast ethyl ester sulfate
CAS:Zaurategrast ethyl ester sulfate is a α4β1/α4β7 integrin antagonist, and used for the treatment of inflammatory and autoimmune disorders.Fórmula:C56H60Br2N8O10SPureza:98%Forma y color:SolidPeso molecular:1197.01NSC 693868
CAS:CDKs and GSK-3 inhibitorFórmula:C9H7N5Pureza:98%Forma y color:SolidPeso molecular:185.19KIF18A-IN-4
CAS:KIF18A-IN-4: Non-competitive KIF18A inhibitor, IC50 6.16 μM, targets mitotic kinesins/kinases, anti-tumor.Fórmula:C22H27N3O3SForma y color:SolidPeso molecular:413.53Y-9738
CAS:Y-9738 is an agent of hypolipidemic.Fórmula:C15H16ClNO4Pureza:98%Forma y color:SolidPeso molecular:309.74TDRL-551
CAS:TDRL-551 is a novel and potent replication protein A (RPA) inhibitor (IC50=18 µM) with potential anticancer activity.TDRL-551 inhibits RPA-DNA interaction andFórmula:C25H23ClIN3O4Pureza:98.09%Forma y color:SolidPeso molecular:591.83Ref: TM-T28935
1mg73,00€5mg160,00€10mg250,00€25mg505,00€50mg803,00€100mg1.288,00€1mL*10mM (DMSO)202,00€Lysine-methotrexate
CAS:Lysine-methotrexate is an anticancer drug. It is an inhibitor of dihydrofolate reductase.Fórmula:C21H27N9O3Pureza:98%Forma y color:SolidPeso molecular:453.5Piposulfan
CAS:Piposulfan, a water-insoluble alkylating agent, is used as an antineoplastic and anti-tumor agent.Fórmula:C12H22N2O8S2Forma y color:SolidPeso molecular:386.44Flurocitabine
CAS:Flurocitabine is a therapeutic agent with antineoplastic activity.Fórmula:C9H10FN3O4Pureza:98%Forma y color:SolidPeso molecular:243.19LCAHA
CAS:LCAHA is a USP2a inhibitor. LCAHA inhibits growth of cyclin D1-dependent cells.Fórmula:C24H41NO3Forma y color:SolidPeso molecular:391.59DHFR-IN-5
CAS:DHFR-IN-5: potent, oral DHFR inhibitor, Ki 0.54 nM against mutant P. falciparum, anti-malarial.Fórmula:C18H24N4O4Forma y color:SolidPeso molecular:360.41Valomaciclovir
CAS:Valomaciclovir is a DNA polymerase inhibitor potentially for treatment of acute herpes zoster and EB virus infection.Fórmula:C15H24N6O4Forma y color:SolidPeso molecular:352.39HBV-IN-22
CAS:HBV-IN-22 (Compound LC5f) is an HBV DNA replication inhibitor that acts on both wild-type HBV (IC50: 0.71 μM) and drug-resistant HBV (IC50: 0.84 μM).Fórmula:C26H29N3O2S2Forma y color:SolidPeso molecular:479.66ROCK2-IN-5
ROCK2-IN-5, a compound blending fasudil, caffeic, and ferulic acids, shows promise for ALS research involving SOD1 mutations.Fórmula:C23H25N3O5SForma y color:SolidPeso molecular:455.53ATB107
CAS:ATB107 is a potent and novel inhibitor of indole-3-glycerol phosphate synthase (IGPS, KD: 3 μM).Fórmula:C21H28N8Pureza:98%Forma y color:SolidPeso molecular:392.5KIRA-7
CAS:KIRA-7: imidazopyrazine, anti-fibrotic, inhibits IRE1α RNase (IC50: 110 nM) allosterically.Fórmula:C27H23FN6OForma y color:SolidPeso molecular:466.51Mycro2
CAS:Mycro2 is an inhibitor of the protein-protein interactions between the bHLHZip proteins c-Myc and Max.Fórmula:C17H11F3N4OS2Forma y color:SolidPeso molecular:408.42Nitracrine dihydrochloride
CAS:Nitracrine dihydrochloride is an acridine antineoplastic agent used in mammary and ovarian tumors. It inhibits RNA synthesis.Fórmula:C18H22Cl2N4O2Forma y color:SolidPeso molecular:397.3DHFR-IN-2
CAS:DHFR-IN-2 (4e) is a potent MtDHFR uncompetitive inhibitor with a 7 μM IC50, promising for TB research.Fórmula:C14H13NO2Forma y color:SolidPeso molecular:227.26Metralindole
CAS:Metralindole is a reversible inhibitor of monoamine oxidase A (RIMA).Fórmula:C15H17N3OForma y color:SolidPeso molecular:255.32RET-IN-19
CAS:RET-IN-19, a potent RET inhibitor, anticancer: IC50 6.8 nM (RET-wt), 13.51 nM (RET V804M); for NSCLC research.Fórmula:C28H28N6O4SForma y color:SolidPeso molecular:544.62(R)-Filanesib
CAS:(R)-Filanesib is the R-enantiomer of ARRY-520. (R)-Filanesib is a synthetic kinesin spindle protein (KSP) inhibitor (IC50: 6 nM).Fórmula:C20H22F2N4O2SForma y color:SolidPeso molecular:420.48CDK4/6-IN-8
CAS:CDK4/6-IN-8 (Compound 7p) is a selective inhibitor of CDK4 (IC50=5.01 nM) and CDK6 (IC50=3.97 nM).Fórmula:C18H18N6O5Forma y color:SolidPeso molecular:398.37IMB-10
CAS:IMB-10 is an alphaMbeta2 integrin modulator, inhibiting leukocyte migration and recruitment in vitro and in vivo.Fórmula:C19H15NOS2Forma y color:SolidPeso molecular:337.46Remdesivir maleate
CAS:Remdesivir (GS-5734) is a broad-spectrum antiviral prodrug effective against SARS-CoV-2 and Ebola, used for research, not human treatment.Fórmula:C31H39N6O12PForma y color:SolidPeso molecular:718.656Tenofovir exalidex
CAS:Tenofovir exalidex (CMX 157) is a lipid-conjugated acyclic nucleotide analog of Tenofovir, demonstrating efficacy against wild-type and antiretroviral-resistantFórmula:C28H52N5O5PPureza:99.83%Forma y color:SolidPeso molecular:569.72BPIC
CAS:BPIC is an agent of anti-tumor that acts by inhibiting inflammation and scavenging free radicals.Fórmula:C27H20N2O5Forma y color:SolidPeso molecular:452.46CLK1-IN-2
CLK1-IN-2: Metabolically stable, Clk1-selective inhibitor; IC50=1.7nM; useful in tumor, Duchenne MD, HIV-1, influenza research.Fórmula:C16H12Cl2N2O2SForma y color:SolidPeso molecular:367.25MK-0668 Mesylate
CAS:MK-0668 Mesylate is the mesylate form of MK-0668 that is a very potent and orally active very late antigen-4 antagonist.Fórmula:C32H34Cl2N6O9S2Forma y color:SolidPeso molecular:781.68αvβ1 integrin-IN-1 TFA (1689540-62-2 free base)
αvβ1 integrin-IN-1 TFA is an effective and selective αvβ1 integrin inhibitor (IC50: 0.63 nM).Fórmula:C28H35F3N6O8SPureza:98%Forma y color:SolidPeso molecular:672.67TDRL-X80
CAS:TDRL-X80 inhibits XPA DNA binding; effective on single, double, and cisplatin-damaged DNA; IC50: 18-29 μM (FP), 21-39 μM (ELISA).Fórmula:C23H15ClN2O6Forma y color:SolidPeso molecular:450.83BPKDi
CAS:BPKDi is a potent and selective inhibitor of PKD (protein kinase D).Fórmula:C21H28N6OPureza:98%Forma y color:SolidPeso molecular:380.49SLM6
CAS:SLM6, an inhibitor of cyclin-dependent kinase-9 (CDK9), exhibits potent anti-multiple myeloma activity.Fórmula:C12H17N7O4Forma y color:SolidPeso molecular:323.31POLA1 inhibitor 1
CAS:POLA1 inhibitor 1: oral, antitumor, effective on various cancers and Adaroten-resistant cells.Fórmula:C26H27NO4Forma y color:SolidPeso molecular:417.5Aloisine A
CAS:Aloisine A, a CDK/GSK-3 inhibitor with IC50: Cdk1/B-150nM, Cdk2/A-120nM, Cdk2/E-400nM, Cdk5/25-200nM, Cdk5/35-160nM, GSK-3α-500nM, GSK-3β-650nM, JNK-3-10μM.Fórmula:C16H17N3OPureza:98%Forma y color:SolidPeso molecular:267.33CDK9/10/GSK3β-IN-1
CAS:CDK9/10/GSK3β-IN-1 is a kinase inhibitor (Flavopiridol analogue) that effectively inhibits HsGSK3β, HsCDK9/CyclinT, HsCDK5/p25 and HsCDK2/CyclinA with IC50Fórmula:C29H24ClN3O4SForma y color:SolidPeso molecular:546.04Alsterpaullone, 2-Cyanoethyl
CAS:Alsterpaullone, 2-Cyanoethyl is a selective dual inhibitor of Cdk1/cyclin B and GSK-3β.Fórmula:C19H14N4O3Forma y color:SolidPeso molecular:346.34CK0106023
CAS:CK0106023, a KSP inhibitor, shows strong antitumor effects in mice, outperforming paclitaxel, and induces monopolar spindles.Fórmula:C30H32BrClN4O2Forma y color:SolidPeso molecular:595.96TP1287
CAS:TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.Fórmula:C21H21ClNO8PForma y color:SolidPeso molecular:481.82Teloxantrone HCl
CAS:Teloxantrone, a DNA topoisomerase II inhibitor, is used potentially for the treatment of solid tumors.Fórmula:C21H28ClN5O5Forma y color:SolidPeso molecular:465.94Nexinhib20
CAS:Nexinhib20 is an inhibitor of exosome synthesis and transport with anti-inflammatory activity, inhibits RAB27A and neutral sphingomyelinase 2 (nSMase2) nsMase2.Fórmula:C15H16N4O3Pureza:99.89%Forma y color:SolidPeso molecular:300.31Braco-19 trihydrochloride
CAS:BRACO19 3HCl inhibits telomerase, blocking its capping function, and prevents HAdV viral replication.Fórmula:C35H46Cl3N7O2Pureza:98.74%Forma y color:SolidPeso molecular:703.14Aminopterin sodium
CAS:Aminopterin sodium is an immunosuppressive anticancer drug, blocking folate synthesis by inhibiting dihydrofolate reductase.Fórmula:C19H20N8NaO5Forma y color:SolidPeso molecular:463.41SMAPP1
CAS:SMAPP1 is an activator of protein phosphatase 1 (PP1). SMAPP1 induces PP1 activity in vitro and activates latent HIV-1 provirus in cultured and primary T cells.Fórmula:C27H25N5O5S2Pureza:98%Forma y color:SolidPeso molecular:563.65Yoshi-864
CAS:Yoshi-864, an alkyl sulfonate, alkylates DNA to hinder replication; potential anti-cancer agent.Fórmula:C8H20ClNO6S2Forma y color:SolidPeso molecular:325.83Synucleozid
CAS:Synucleozid is a potent the SNCA mRNA inhibitor that encodes α-synuclein protein (IC50=1.5 μM), has the potential for the investigation of Parkinson’s disease.Fórmula:C22H20N6Pureza:98%Forma y color:SolidPeso molecular:368.43
