Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(33 productos)
- Receptor de vasopresina(48 productos)
Mostrar 6 subcategorías más
Se han encontrado 3420 productos de "Endocrinología / Hormonas"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
KNT-127
CAS:KNT-127 is an agonist of δ-Opioid receptor.Fórmula:C24H24N2O2Pureza:98%Forma y color:SolidPeso molecular:372.46AP5
CAS:AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.Fórmula:C28H28FNO4Pureza:98%Forma y color:SolidPeso molecular:461.52Naltrindole 5′-isothiocyanate
CAS:Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.Fórmula:C27H25N3O3SForma y color:SolidPeso molecular:471.571Urotensin-II receptor antagonist-1
CAS:Urotensin-II receptor antagonist-1 (compound 1) is a human Urotensin II receptor antagonist with low oral bioavailability (F=0-3% in rats) and a Ki of 16 nM in HEK293 cells expressing human recombinant UT receptors. It inhibits cytochrome P450 enzymes (IC50=0.75 μM for CYP2D6; 1.4 μM for CYP3A4), suppresses κ opioid receptors (EC50=3.2 μM), and targets cardiac sodium channels (Ki=2.5 μM).Fórmula:C25H31Cl2N3OForma y color:SolidPeso molecular:460.439THR-β agonist 4
CAS:THR-β agonist 4 is a potent agonist of THR-β.Fórmula:C16H11Cl2F2N5O6SForma y color:SolidPeso molecular:510.26Androgen receptor antagonist 11
CAS:Androgen receptor antagonist 11 (compound N29) is a selective, orally available antagonist.Fórmula:C20H19F3N4O3SForma y color:SolidPeso molecular:452.45U 80215
CAS:U 80215 is an enzyme-competitive inhibitor.Fórmula:C42H60N8O6SForma y color:SolidPeso molecular:805.04Saprisartan potassium
CAS:Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.Fórmula:C25H21BrF3KN4O4SForma y color:SolidPeso molecular:649.52Novokinin
CAS:Angiotensin AT2 receptor agonistFórmula:C39H61N11O7Pureza:98%Forma y color:SolidPeso molecular:795.9721-Deacetoxy deflazacort
CAS:21-Deacetoxy deflazacort is a dehydrogenated derivative of Deflazacort, which is a glucocorticoid. As an inactive precursor, Deflazacort rapidly converts into the active metabolite, 21-Desacetyldeflazacort. This compound serves as both an anti-inflammatory and immunosuppressive agent.Fórmula:C23H29NO4Forma y color:SolidPeso molecular:383.485′-Guanidinonaltrindole
CAS:5′-Guanidinonaltrindole (GNTI) is a selective antagonist of the kappa opioid receptor.Fórmula:C27H29N5O3Forma y color:SolidPeso molecular:471.551L162389
CAS:L162389 is an angiotensin II receptor antagonist with a balanced affinity for AT1 and AT2 receptor and stimulates the conversion of phosphatidylinositol.Fórmula:C31H38N4O4SPureza:99.11% - 99.57%Forma y color:SolidPeso molecular:562.72BMS-248360
CAS:BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.Fórmula:C36H45N5O5SPureza:98%Forma y color:SolidPeso molecular:659.84GDC-0927 Racemate
CAS:GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.Fórmula:C28H28FNO4Pureza:98%Forma y color:SolidPeso molecular:461.52Erα-IN-1
Erα-IN-1 (compound 3c) is an inhibitor of the estrogen receptor α (ERα), effectively blocking ERα activity in MCF7/ERE-LUC cells.Fórmula:C16H11FN2Forma y color:SolidPeso molecular:250.27BNTX
CAS:BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.Fórmula:C27H27NO4Forma y color:SolidPeso molecular:429.508OSU-ERb-12
CAS:OSU-ERb-12 is an ERβ agonist that suppresses ovarian cancer cell proliferation both in vitro and in vivo, and decreases the expression of Snail [1] [2].Fórmula:C15H30B10O2Forma y color:SolidPeso molecular:350.51GW856464
CAS:GW856464 is an antagonist of MCHR1. It is utilized in research related to cardiovascular diseases and obesity.Fórmula:C23H20ClN3O3SForma y color:SolidPeso molecular:453.94BU72
CAS:BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.Fórmula:C28H32N2O2Forma y color:SolidPeso molecular:428.57GSK866
CAS:GSK866 is a selective glucocorticoid receptor agonist (SEGRA).Fórmula:C23H21Cl2F4N5O3Forma y color:SolidPeso molecular:562.34
