Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(230 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(164 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(126 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(34 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3420 productos de "Endocrinología / Hormonas"
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PROTAC ERα Degrader-7
CAS:PROTAC ERα Degrader-7 (Compound i-320) is a powerful PROTAC degrader targeting the estrogen receptor alpha (ERα), exhibiting a DC50 of 0.000006 µM. This compound consists of a cereblon-binding segment, LBM, connected to ERBM, an ERα-binding ligand that includes a benzofused partially saturated 6-membered carbocyclic or heterocyclic ring [1].Fórmula:C46H49F2N5O4Forma y color:SolidPeso molecular:773.91ER ligand-9
CAS:ER ligand-9 is a conjugate of an estrogen receptor (Estrogen Receptor/ERR) ligand and a linker, utilized in the synthesis of PROTACs ERD-1233.Fórmula:C31H33NO3Forma y color:SolidPeso molecular:467.599Melanin Concentrating Hormone, salmon TFA
MCH (salmon) TFA is a 19-amino-acid neuropeptide affecting appetite, energy, sleep, and heart health via GPCR SLC-1/GPR24 and MCHR2.Fórmula:C91H140F3N27O26S4Forma y color:SolidPeso molecular:2213.5SB 205607 dihydrobromide
CAS:non-peptide δ1 opioid receptor agonistFórmula:C23H24N2OPureza:98%Forma y color:SolidPeso molecular:344.45[Sar1, Ile8]-Angiotensin II acetate
'[Sar1, Ile8]-Angiotensin II acetate triggers oxidases and prompts superoxide in muscles; has varied vascular impacts.Fórmula:C48H77N13O12Pureza:99.36%Forma y color:SolidPeso molecular:1028.2Ref: TM-T7575L1
2mg34,00€5mg46,00€10mg60,00€1mL*10mM (DMSO)90,00€25mg119,00€50mg192,00€100mg289,00€200mg415,00€Galloylalbiflorin
CAS:Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.Fórmula:C30H32O15Forma y color:SolidPeso molecular:632.57Zavacorilant
CAS:Zavacorilant is capable of modulating glucocorticoid receptor (GR).Fórmula:C25H26FN7O3S2Forma y color:SolidPeso molecular:555.65[Glu4]-Oxytocin
CAS:'[Glu4]-Oxytocin is a variant for studying 'oxytocin-like' molecule shapes in water.'Fórmula:C43H65N11O13S2Peso molecular:1008.18PROTAC AR Degrader-4 TFA
PROTAC AR Degrader-4: IAP ligand, linker, AR binder; it's a SNIPER that degrades AR non-genetically.Fórmula:C45H68F3N3O11Forma y color:SolidPeso molecular:884.03Premarin
CAS:Premarin (Estrone 3-sulfate) is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.Fórmula:C18H22O5SPureza:99.74%Forma y color:SoildPeso molecular:350.43Ref: TM-T36857L
1mg175,00€5mg394,00€1mL*10mM (DMSO)413,00€10mg582,00€25mg888,00€50mg1.243,00€100mg1.674,00€KOR agonist 4
KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.Fórmula:C21H25N3Forma y color:SolidPeso molecular:319.44HINT1-IN-1
HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).Fórmula:C23H24N8O5Forma y color:SolidPeso molecular:492.49GPR88 agonist 2
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].Forma y color:Odour Solid15-keto Prostaglandin A1
CAS:PGA1, derived from PGE1 in semen, creates 15-keto PGA1 via dehydrogenase, inducing vasoconstriction at 6μM like angiotensin II.Fórmula:C20H30O4Forma y color:SolidPeso molecular:334.45Acetalin-3
CAS:Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Fórmula:C42H61N11O8S2Peso molecular:912.13PROTAC AR-V7 degrader-1
CAS:Potent, oral AR-V7 degrader (Compound 6); DC50: 0.32µM; targets AR-DBD via VHL E3; EC50: 0.88µM in 22Rv1 cells.Fórmula:C41H52N6O6S2Forma y color:SolidPeso molecular:789.02Benazeprilat
CAS:Benazeprilat(CGS 14831) is an orally active active metabolite of Benazepril.Benazeprilat has potent antihypertensive activity and can be used in combinationFórmula:C22H24N2O5Pureza:99.23%Forma y color:Crystalline SolidPeso molecular:396.44BI 653048 phosphate
CAS:BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).Fórmula:C23H28F4N3O8PSPureza:98%Forma y color:SolidPeso molecular:613.52Kalata B7
CAS:Kalata B7, a cyclotide isolated from Oldenlandia affinis DC (Rubiaceae), possesses membrane-permeating capabilities and acts as a partial agonist of oxytocin- and vasopressin V1a-receptors [1] [2].Fórmula:C128H196N36O40S6Peso molecular:3071.53Enclomiphene-d4
Enclomiphene-d4 is the deuterium-labeled analog of Enclomiphene. Enclomiphene functions as a potent and orally active estrogen receptor antagonist, exhibiting antiestrogenic properties.Forma y color:Odour Solid
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