
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(230 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(164 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(126 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(34 productos)
- Receptor de vasopresina(48 productos)
Mostrar 6 subcategorías más
Se han encontrado 3420 productos de "Endocrinología / Hormonas"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cgp 29287
CAS:Cgp 29287 is a primate-specific renin inhibitor. It also has a prolonged duration of action.Fórmula:C72H110N20O15Forma y color:SolidPeso molecular:1495.77PROTAC ERα Degrader-10
CAS:PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.Fórmula:C45H49N5O4Peso molecular:723.9(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat)
CAS:'(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat), a peptide, functions as a ligand for parathyroid hormone (PTH) receptors [1].'Fórmula:C194H303N59O53Peso molecular:4309.85C-Type Natriuretic Peptide (1-53), human
CAS:CNP, from natriuretic family, first in pigs, now in other species, processes into CNP-22/CNP-53, similar to ANP/BNP, with varying potencies.Fórmula:C251H417N81O71S3Pureza:98%Forma y color:SolidPeso molecular:5801.77Ethamoxytriphetol
CAS:Ethamoxytriphetol is a non-steroidal estrogen antagonist.Fórmula:C27H33NO3Forma y color:SolidPeso molecular:419.56Nurr1 agonist 6
Compound 13, a Nurr1 agonist, exhibits a dissociation constant (Kd) of 1.5 μM and an effective concentration for 50% response (EC50) of 3 μM [1].Forma y color:Odour SolidPL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Fórmula:C31H38F3N5O7Peso molecular:649.66Bradykinin potentiator-5
CAS:Bradykinin potentiator-5 is a peptide inflammatory mediator, causes blood vessels to dilate (enlarge), and therefore causes blood pressure to fall.Fórmula:C30H41N7O7Pureza:98%Forma y color:SolidPeso molecular:611.69Aclerastide
CAS:Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.Fórmula:C42H64N12O11Forma y color:SolidPeso molecular:913.03Dehydroisoandrosterone 3-acetate
CAS:Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.Fórmula:C21H30O3Pureza:>99.99%Forma y color:SolidPeso molecular:330.46RLA-4842
RLA-4842: iron-based anti-androgen; inhibits mCRPC cell proliferation.Fórmula:C42H46F3N5O8SForma y color:SolidPeso molecular:837.94A7C-301
4A7C-301, a Nurr1 agonist, exhibits potent neuroprotective effects in vitro and markedly mitigates neuropathological abnormalities while enhancing motor andForma y color:Odour SolidDBPR116
CAS:DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.Fórmula:C19H18FNO3SForma y color:SolidPeso molecular:359.42α-Neoendorphin (1-8)
CAS:α-Neoendorphin (1-8) is a 8-amino acid peptide derived from the N-terminal of α-Neoendorphin.Fórmula:C49H70N12O11Pureza:98%Forma y color:SolidPeso molecular:1003.15ARCC-4
CAS:ARCC-4: A VHL-recruiting, low-nanomolar (DC50=5nM) AR degrader; outshines enzalutamide; degrades AR mutants resistant to therapy.Fórmula:C53H56F3N7O7S2Pureza:98%Forma y color:SolidPeso molecular:1024.18Parathyroid hormone (1-34) (rat)
CAS:Parathyroid hormone (PTH) receptor agonist. Increases serum PTH levels and bone mass in rats.Fórmula:C180H291N55O48S2Pureza:98%Forma y color:SolidPeso molecular:4057.74Biphalin TFA
CAS:Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.Fórmula:C46H56N10O10·xC2HF3O2Pureza:98%Forma y color:SolidPeso molecular:909.00 (free base)PROTAC ERα Degrader-8
CAS:PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].Fórmula:C47H51N5O4Forma y color:SolidPeso molecular:749.94Betamethasone acibutate
CAS:Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.Fórmula:C28H37FO7Pureza:98%Forma y color:SolidPeso molecular:504.59Remikiren
CAS:Remikiren is a highly specific renin inhibitor with oral activity for the treatment of hypertensio.Fórmula:C33H50N4O6SForma y color:SolidPeso molecular:630.84

