
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(164 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(34 productos)
- Receptor de vasopresina(48 productos)
Mostrar 6 subcategorías más
Se han encontrado 3419 productos de "Endocrinología / Hormonas"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Frakefamide TFA
Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.Fórmula:C32H35F4N5O7Forma y color:SolidPeso molecular:677.6415,26-Dihydroxylanosta-7,9(11),24-trien-3-one
CAS:15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is a natural product that can be used as a reference standard. The CAS number of 15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is 420781-85-7.Fórmula:C30H46O3Forma y color:SolidPeso molecular:454.7ICI 174,864
CAS:Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.Fórmula:C38H53N5O7Pureza:98%Forma y color:White SolidPeso molecular:691.87Hemorphin-7
CAS:Hemorphin-7, an atypical opioid peptide from hemoglobin, may enhance memory, promote cell growth, and is a potential breast cancer biomarker.Fórmula:C49H64N12O11Pureza:98%Forma y color:SolidPeso molecular:997.11BAY 1003803
CAS:BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.Fórmula:C21H18ClF5N2O4Forma y color:SolidPeso molecular:492.83PROTAC ERα Degrader-2
CAS:PROTAC ERα Degrader-2 is composed of a cIAP1 ligand binding group, a linker, and an estrogen receptor α (ERα) binding group, serving as an ERα degrader.Fórmula:C42H61N5O8Pureza:98%Forma y color:SolidPeso molecular:763.96Neuropeptide EI, rat
CAS:Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Fórmula:C63H98N16O23Pureza:98%Forma y color:SolidPeso molecular:1447.55WAY267464 HCl
CAS:WAY267464: nonpeptide OT agonist, anxiolytic, modulates selectivity, improves CNS entry and oral uptake.Fórmula:C32H37Cl2N7O4Pureza:98%Forma y color:SolidPeso molecular:654.59Dexamethasone phosphate
CAS:Dexamethasone phosphate is a synthetic adrenal corticosteroid. It also has potent anti-inflammatory properties.Fórmula:C22H30FO8PForma y color:SolidPeso molecular:472.44Vasopressin Dimer (parallel) (TFA)
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, andFórmula:C94H131F3N30O26S4Pureza:98%Forma y color:SolidPeso molecular:2282.49Dynorphin A (1-10)
CAS:Dynorphin A (1-10) is an opioid peptide, binds κ-opioid receptor, blocks NMDA current, IC50: 42.0 μM.Fórmula:C57H91N19O12Pureza:98%Forma y color:SolidPeso molecular:1234.45Angiotensin II 5-valine
CAS:ngiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors.Fórmula:C49H69N13O12Pureza:98%Forma y color:SolidPeso molecular:N/AERRγ agonist-2
CAS:ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a K d value of 6.5 μM.Fórmula:C27H21N5O2Forma y color:SolidPeso molecular:447.49OP-3633
CAS:OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.Fórmula:C30H39NO2Pureza:98%Forma y color:SolidPeso molecular:445.64Zankiren
CAS:Zankiren is a renin inhibitor. Zankiren can reduce blood pressure, plasma renin activity, and angiotension II.Fórmula:C35H55N5O6S2Forma y color:SolidPeso molecular:705.9711-Ketodihydrotestosterone
CAS:11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).Fórmula:C19H28O3Forma y color:SolidPeso molecular:304.42Koreanoside E
CAS:Koreanoside E is a useful organic compound for research related to life sciences. The catalog number is T125538 and the CAS number is 1804014-67-2.Fórmula:C27H30O11Forma y color:SolidPeso molecular:530.526Prednicarbate
CAS:Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.Fórmula:C27H36O8Pureza:99.88%Forma y color:SolidPeso molecular:488.57PROTAC ER Degrader-14
CAS:PROTAC ER Degrader-14 (compound 86) is a PROTAC-type estrogen receptor/ERR degrader. It comprises an E3 ubiquitin ligase ligand (blue part) (S)-Deoxy-thalidomide, a PROTAC linker (black part) N-Boc-piperazine, and a target protein ligand (red part) ER ligand-6. The combination of the E3 ligase and linker forms tert-Butyl (S)-4-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)piperazine-1-carboxylate.Fórmula:C44H46FN5O5Forma y color:SolidPeso molecular:743.865SNIPER(ER)-87
CAS:SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (Fórmula:C59H73N5O10SPureza:98%Forma y color:SolidPeso molecular:1044.32

