
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(164 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(34 productos)
- Receptor de vasopresina(48 productos)
Mostrar 6 subcategorías más
Se han encontrado 3419 productos de "Endocrinología / Hormonas"
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2-Ethylhexyl trans-4-methoxycinnamate
CAS:2-Ethylhexyl trans-4-methoxycinnamate is a sunscreen agent.Fórmula:C18H26O3Pureza:98.92%Forma y color:Pale Yellow LiquidPeso molecular:290.4Angiotensin amide
CAS:Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.Fórmula:C49H70N14O11Pureza:98%Forma y color:SolidPeso molecular:1031.174'-hydroxy Tamoxifen
CAS:It is a metabolite of tamoxifen and an estrogen receptor modulator.Fórmula:C26H29NO2Pureza:98%Forma y color:SolidPeso molecular:387.511α-Hydroxy-3-epi-vitamin D3
CAS:1α-Hydroxy-3-epi-vitamin D3, a natural metabolite derived from 1alpha,25-dihydroxyvitamin D3, effectively suppresses parathyroid hormone (PTH) secretion[1].Fórmula:C27H44O2Forma y color:SolidPeso molecular:400.647Ac-RYYRIK-NH2
CAS:NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.Fórmula:C44H70N14O9Pureza:98%Forma y color:SolidPeso molecular:939.12Antitumor agent-195
Antitumor agent-195 (compound 16c) is a dual-targeting agent that simultaneously targets STAT3 and NQO1. At a concentration of 1 μM, it significantly inhibits the phosphorylation of STAT3 at the Tyr705 site and effectively induces apoptosis in MDA-MB-231 and MDA-MB-468 breast cancer cells. As a substrate of NQO1, Antitumor agent-195 markedly increases ROS production, causing severe DNA damage in a dose-dependent manner. It also demonstrates strong antitumor properties in MDA-MB-231 xenograft models.Fórmula:C22H22N2O4Forma y color:SolidPeso molecular:378.42BigLEN(mouse)
CAS:GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.Fórmula:C78H130N24O22Pureza:98%Forma y color:SolidPeso molecular:1756.03(rel)-PROTAC ERRα Degrader-1
(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader.Fórmula:C54H49Cl2F6N7O8Pureza:98%Forma y color:SolidPeso molecular:1108.91PROTAC ER Degrader-4
CAS:PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).Fórmula:C53H67F3N6O8SPureza:98%Forma y color:SolidPeso molecular:1005.2DAMGO (TFA)
CAS:DAMGO is a selective peptide agonist of the µ-opioid receptor .Fórmula:C28H36F3N5O8Pureza:98%Forma y color:SolidPeso molecular:627.61OT-R antagonist 2
CAS:OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .Fórmula:C28H29N3O4Pureza:98%Forma y color:SolidPeso molecular:471.55BI 653048
CAS:BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.Fórmula:C23H25F4N3O4SPureza:98%Forma y color:SolidPeso molecular:515.523-epi-25-hydroxy Vitamin D3
CAS:3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.Fórmula:C27H44O2Forma y color:SolidPeso molecular:400.64GNE-274
CAS:GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.Fórmula:C29H31NO4Forma y color:SolidPeso molecular:457.57Cgp 38560
CAS:CGP 38560 is a potent renin inhibitor.Fórmula:C40H67N5O9S2Forma y color:SolidPeso molecular:826.12Nurr1 agonist 2
CAS:Nurr1 agonist 2 with EC50 of 0.07 μM, boosts TH & VMAT2 mRNA, binds Nurr1 LBD at Kd 0.14 μM, for parkinsonism study.Fórmula:C18H14O3SPureza:98.78%Forma y color:SoildPeso molecular:310.37Methylprednisolone Acetate
Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.Fórmula:C24H32O6Pureza:99.74%Forma y color:Off-White SolidPeso molecular:416.51Axelopran
CAS:Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.Fórmula:C26H39N3O4Forma y color:SolidPeso molecular:457.61Raloxifene 6-glucuronide
CAS:Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.Fórmula:C34H35NO10SPureza:98%Forma y color:SolidPeso molecular:649.71PTP1B/AKR1B1-IN-1
PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50sFórmula:C22H21NO4S2Pureza:98%Forma y color:SolidPeso molecular:427.54

