Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(56 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(166 productos)
- LHRH(1 productos)
- Receptor de opioides(326 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(90 productos)
- Reductasa(50 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(46 productos)
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Se han encontrado 3369 productos de "Endocrinología / Hormonas"
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Retosiban
CAS:Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).Fórmula:C27H34N4O5Pureza:98%Forma y color:SolidPeso molecular:494.58SNIPER(ER)-110
SNIPER(ER)-110 links cIAP1 and estrogen ligands. SNIPER(ER)-51 degrades ER protein; DC50 <3 nM at 4h, 7.7 nM at 48h.Fórmula:C66H83N5O11Pureza:98%Forma y color:SolidPeso molecular:1122.39PRO20
<p>PRO20 is a specific and competitive antagonist of the (pro)renin receptor (PRR). It inhibits the calcium influx induced by Proproin with an IC50 value of 81 nmol/L. By blocking the binding of Prorenin to PRR, PRO20 inhibits the activation of the renin-angiotensin system (RAS), reducing the production of angiotensin II (Ang II) and exerting antihypertensive effects. PRO20 holds promise for research in antihypertensive agents.</p>Forma y color:Odour Solid[Glu4]-Oxytocin
CAS:'[Glu4]-Oxytocin is a variant for studying 'oxytocin-like' molecule shapes in water.'Fórmula:C43H65N11O13S2Peso molecular:1008.18DPC-AJ1951 TFA
DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.Fórmula:C78H128F3N23O21Forma y color:SolidPeso molecular:1781.02DBPR116
CAS:DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.Fórmula:C19H18FNO3SForma y color:SolidPeso molecular:359.4215-keto Prostaglandin A1
CAS:PGA1, derived from PGE1 in semen, creates 15-keto PGA1 via dehydrogenase, inducing vasoconstriction at 6μM like angiotensin II.Fórmula:C20H30O4Forma y color:SolidPeso molecular:334.45PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like macrophages in mouse TNBC tumors.Fórmula:C17H21BrCl2N6SPureza:99.99%Forma y color:SoildPeso molecular:492.26(Glu2)-TRH
CAS:(Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.Fórmula:C15H22N4O6Forma y color:SolidPeso molecular:354.36TF-505
CAS:TF-505, a steroid 5α-reductase inhibitor, is used potentially for the treatment of benign prostatic hyperplasia.Fórmula:C33H37NO4Pureza:98%Forma y color:SolidPeso molecular:511.65Osteostatin
CAS:Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presentingFórmula:C27H41N9O8Forma y color:SolidPeso molecular:619.67Perindoprilat
CAS:Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.Fórmula:C17H28N2O5Pureza:99.21%Forma y color:SolidPeso molecular:340.41AT-121 hydrochloride
CAS:<p>AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.</p>Fórmula:C24H39ClN4O3SPureza:97.28% - >99.99%Forma y color:SolidPeso molecular:499.11Angiotensin II (5-8), human
CAS:Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin IIFórmula:C26H36N6O5Pureza:98%Forma y color:SolidPeso molecular:512.6Deacylcortivazol
CAS:Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.Fórmula:C30H36N2O4Forma y color:SolidPeso molecular:488.62PL-017
CAS:μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.Fórmula:C29H37N5O5Pureza:98%Forma y color:SolidPeso molecular:535.64Gridegalutamide
CAS:Gridegalutamide exhibits anti-androgen and anti-tumor activities.Fórmula:C41H45F3N8O5SForma y color:SolidPeso molecular:818.91Nurr1 agonist 6
Compound 13, a Nurr1 agonist, exhibits a dissociation constant (Kd) of 1.5 μM and an effective concentration for 50% response (EC50) of 3 μM [1].Forma y color:Odour SolidPROTAC ERRα Degrader-3
CAS:PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein.Fórmula:C47H50F6N6O7SForma y color:SolidPeso molecular:957.07α-(Thiomethyl)spironolactone
CAS:7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.Fórmula:C23H32O3SPureza:>99.99%Forma y color:SolidPeso molecular:388.56
