
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(57 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(166 productos)
- LHRH(1 productos)
- Receptor de opioides(326 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(90 productos)
- Reductasa(50 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3371 productos de "Endocrinología / Hormonas"
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Epi-Cryptoacetalide
Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.Fórmula:C18H22O3Forma y color:SolidPeso molecular:286.371Fluorphine
CAS:Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41ODM-204
CAS:ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).Fórmula:C20H21F3N4Pureza:98%Forma y color:SolidPeso molecular:374.40MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Fórmula:C27H29ClN4O2Pureza:98%Forma y color:SolidPeso molecular:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57Keap1-IN-1
Keap1-IN-1 (Compound 27) is an inhibitor of Keap1, functioning by covalently modifying the Cys151 residue on the BTB domain of KEAP1, thereby disrupting the interaction between Keap and Nrf. It enhances the mRNA expression of the antioxidant response element (ARE) dependent gene NQO1, with an EC50 of 160 nM, and exhibits cytotoxicity in U2OS cells, with an EC50 of 527 nM.Fórmula:C17H21Cl2N2O5PS3Forma y color:SolidPeso molecular:531.434LY2623091
CAS:LY2623091, a mineralocorticoid receptor antagonist, is utilized in treating refractory hypertension. It demonstrates CYP3A4-dependent clearance and exhibits synergistic effects when combined with CYP3A4 inhibitors.Fórmula:C30H30FN5O3Peso molecular:527.59pTH (1-37) (human)
CAS:pTH (1-37) human fragment boosts cAMP, alkaline phosphatase, growth, and BMD, potential for osteoporosis research.Fórmula:C195H316N58O54S2Peso molecular:4401.08Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Fórmula:C20H23N3OForma y color:SolidPeso molecular:321.42BIBS 39
CAS:BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.Fórmula:C32H36N4O3Pureza:99.28%Forma y color:SolidPeso molecular:524.65β-Lipotropin (61-69)
CAS:β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Fórmula:C45H66N10O15SPeso molecular:1019.13PL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Fórmula:C31H38F3N5O7Peso molecular:649.66(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat)
CAS:'(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat), a peptide, functions as a ligand for parathyroid hormone (PTH) receptors [1].'Fórmula:C194H303N59O53Peso molecular:4309.85GPR88 agonist 2
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].Forma y color:Odour SolidGalloylalbiflorin
CAS:Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.Fórmula:C30H32O15Forma y color:SolidPeso molecular:632.57PROTAC ERα Degrader-10
CAS:PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.Fórmula:C45H49N5O4Peso molecular:723.9[Sar1, Ile8]-Angiotensin II acetate
'[Sar1, Ile8]-Angiotensin II acetate triggers oxidases and prompts superoxide in muscles; has varied vascular impacts.Fórmula:C48H77N13O12Pureza:99.36%Forma y color:SolidPeso molecular:1028.2Ref: TM-T7575L1
2mg35,00€5mg48,00€10mg64,00€25mg126,00€50mg202,00€100mg304,00€200mg439,00€1mL*10mM (DMSO)96,00€Kalata B7
CAS:Kalata B7, a cyclotide isolated from Oldenlandia affinis DC (Rubiaceae), possesses membrane-permeating capabilities and acts as a partial agonist of oxytocin- and vasopressin V1a-receptors [1] [2].Fórmula:C128H196N36O40S6Peso molecular:3071.53Acetalin-3
CAS:Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Fórmula:C42H61N11O8S2Peso molecular:912.13TD-802
CAS:TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.Fórmula:C52H61ClN10O6Forma y color:SolidPeso molecular:957.56

