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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"

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  • ML418

    CAS:
    <p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>
    Fórmula:C19H24ClN3O3
    Pureza:99.3%
    Forma y color:Solid
    Peso molecular:377.87
  • IK1 inhibitor PA-6

    CAS:
    <p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>
    Fórmula:C31H32N4O2
    Pureza:98.9%
    Forma y color:Solid
    Peso molecular:492.61
  • Glibenclamide

    CAS:
    <p>Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.</p>
    Fórmula:C23H28ClN3O5S
    Pureza:99.05% - 99.75%
    Forma y color:Solid
    Peso molecular:494.00
  • NaV1.7 inhibitor-1

    CAS:
    <p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>
    Fórmula:C23H30FNO4S
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:435.55
  • Fluxametamide

    CAS:
    <p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>
    Fórmula:C20H16Cl2F3N3O3
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:474.26
  • Bemegride

    CAS:
    <p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>
    Fórmula:C8H13NO2
    Pureza:99.89%
    Forma y color:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)
    Peso molecular:155.19
  • VU0134992 hydrochloride

    CAS:
    <p>VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).</p>
    Fórmula:C20H32BrClN2O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:447.84
  • Pramocaine hydrochloride

    CAS:
    <p>Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.</p>
    Fórmula:C17H27NO3·HCl
    Pureza:99.15% - 99.61%
    Forma y color:Crystals White Or Off White Crystalline Powder
    Peso molecular:329.86
  • Omeprazole sulfide

    CAS:
    <p>Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.</p>
    Fórmula:C17H19N3O2S
    Pureza:98.83%
    Forma y color:White To Slightly Collored Solid Solid Crystalline
    Peso molecular:329.42
  • Phenformin hydrochloride

    CAS:
    <p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>
    Fórmula:C10H16ClN5
    Pureza:97.11% - 99.80%
    Forma y color:Lactic Acidosis
    Peso molecular:241.72
  • Bupivacaine hydrochloride

    CAS:
    <p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>
    Fórmula:C18H28N2O·HCl
    Pureza:99.9% - >99.99%
    Forma y color:Solid
    Peso molecular:324.89
  • γ-Aminobutyric acid

    CAS:
    <p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>
    Fórmula:C4H9NO2
    Pureza:99.95%
    Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid Powder
    Peso molecular:103.12
  • Dooku1

    CAS:
    <p>Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.</p>
    Fórmula:C13H9Cl2N3OS
    Pureza:98.87% - 99.74%
    Forma y color:Solid
    Peso molecular:326.2
  • Prilocaine hydrochloride

    CAS:
    <p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>
    Fórmula:C13H21ClN2O
    Pureza:99.97%
    Forma y color:Needles White Or Off White Crystalline Powder
    Peso molecular:256.77
  • Ciclopirox olamine

    CAS:
    <p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>
    Fórmula:C14H24N2O3
    Pureza:99.16% - >99.99%
    Forma y color:White To Yellow Solid Solid Particulate/Powder
    Peso molecular:268.35
  • Methocarbamol

    CAS:
    <p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>
    Fórmula:C11H15NO5
    Pureza:99.96%
    Forma y color:Crystals From Benzene Solid
    Peso molecular:241.24
  • Lotilaner

    CAS:
    <p>Lotilaner is a parasiticide.</p>
    Fórmula:C20H14Cl3F6N3O3S
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:596.76
  • Phenibut

    CAS:
    <p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>
    Fórmula:C10H13NO2
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:179.22
  • Suloctidil

    CAS:
    <p>Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.</p>
    Fórmula:C20H35NOS
    Pureza:99.75% - >99.99%
    Forma y color:Solid
    Peso molecular:337.56
  • Glipizide

    CAS:
    <p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>
    Fórmula:C21H27N5O4S
    Pureza:99.67% - 99.75%
    Forma y color:Solid
    Peso molecular:445.54