
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(271 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(98 productos)
- Lípido(58 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8626 productos de "Metabolismo"
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CALP3 acetate(261969-05-5 free base)
<p>CALP3 acetate blocks Ca2+ channels, mimics elevated [Ca2+]i, activates EF hands, and regulates CaM, channels, and pumps.</p>Fórmula:C46H72N10O11Pureza:96.49%Forma y color:SolidPeso molecular:941.12Lanthanum(III) chloride heptahydrate
CAS:<p>Lanthanum(III) chloride blocks divalent cation channels, useful for biochemical research.</p>Fórmula:Cl3H14LaO7Pureza:98%Forma y color:White Solid PowderPeso molecular:371.37YTX-465
CAS:<p>YTX-465 is an inhibitor of both stearoyl-CoA desaturase(IC50s = 39 nM) and Ole1 (IC50s = 30.4 μM).</p>Fórmula:C25H26N6O3Pureza:99.96%Forma y color:SolidPeso molecular:458.51AR7
CAS:<p>AR7 is a retinoic acid receptor α (RARα) antagonist.</p>Fórmula:C15H12ClNOPureza:98.12% - 99.86%Forma y color:SolidPeso molecular:257.71WWL229
CAS:<p>WWL229 selectively inhibits Ces3 without affecting Ces1f, ABHD6, or other serine hydrolases, mimicking WWL113 in adipocytes.</p>Fórmula:C16H22N2O5Pureza:98.14%Forma y color:SolidPeso molecular:322.36CAY10698
CAS:<p>CAY10698 is a 12-lipoxygenase inhibitor (12-LO; IC50 of 5.1 μM).</p>Fórmula:C17H17N3O4S2Pureza:98.97%Forma y color:SolidPeso molecular:391.46Udenafil
CAS:<p>Udenafil is an inhibitor of PDE5 .</p>Fórmula:C25H36N6O4SPureza:99.90%Forma y color:Off-White SolidPeso molecular:516.66Vonafexor
CAS:<p>Vonafexor (EYP001) is a farnesoid X receptor (FXR, NR1H4) agonist, with anti-HBV effects</p>Fórmula:C19H15Cl3N2O5SPureza:98.74%Forma y color:SolidPeso molecular:489.76IACS-13909
CAS:<p>IACS-13909 (BBP-398), a specific and potent allosteric inhibitor of SHP2, that suppresses signaling through the MAPK pathway.</p>Fórmula:C17H18Cl2N6Pureza:98.8%Forma y color:SolidPeso molecular:377.27U-73122
CAS:<p>U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.</p>Fórmula:C29H40N2O3Pureza:97.50%Forma y color:Solid Off-WhitePeso molecular:464.64Dimesna
CAS:<p>Dimesna (BNP-7787) is a synthetic derivative of dithio-ethane sulfonate with uroprotective properties.</p>Fórmula:C4H8Na2O6S4Pureza:99.90%Forma y color:SolidPeso molecular:326.34GSK 650394
CAS:<p>GSK 650394 is an inhibitor of serum- and glucocorticoid-regulated kinases (SGK). GSK 650394 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C25H22N2O2Pureza:97.46% - >99.99%Forma y color:SolidPeso molecular:382.45Benzamidine hydrochloride
CAS:<p>Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.</p>Fórmula:C7H9ClN2Pureza:99.25% - 99.97%Forma y color:White To Off-White PowderPeso molecular:156.61CID 2011756
CAS:<p>CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.</p>Fórmula:C22H21ClN2O3Pureza:98.15% - ≥95%Forma y color:SolidPeso molecular:396.87PSB-1491
CAS:PSB-1491 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 0.386 nM, >25000-fold selective versus MAO-A.Fórmula:C15H11Cl2N3OPureza:98.41% - 99.68%Forma y color:SolidPeso molecular:320.17Sulindac sulfone
CAS:<p>Sulindac sulfone is a metabolite of the nonsteroidal anti-inflammatory drug sulindac. Sulindac sulfone is an inhibitor of aldose reductase (IC50 =367 nM).</p>Fórmula:C20H17FO4SPureza:98.2% - 98.83%Forma y color:SolidPeso molecular:372.41ICI 63197
CAS:ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.Fórmula:C9H13N5OPureza:99.70%Forma y color:White SolidPeso molecular:207.23ML-030
CAS:<p>ML-030 is a potent PDE4 inhibitor, selective for subtypes (A1, B1, B2, C1, D2) with IC50 ranging from 6.7 to 452 nM.</p>Fórmula:C20H20N4O4SPureza:97.93%Forma y color:SolidPeso molecular:412.46Minaprine dihydrochloride
CAS:<p>Minaprine dihydrochloride: reversible MAO-A inhibitor, mild on acetylcholinesterase, used for depression.</p>Fórmula:C17H24Cl2N4OPureza:99.43% - 99.99%Forma y color:SolidPeso molecular:371.3W 36017
CAS:<p>W36017 is an impurity of lidocaine with a PKA of 7.4 for blocking neurologic activity.</p>Fórmula:C12H18N2OPureza:99.09%Forma y color:SolidPeso molecular:206.28(E)-3PO
CAS:<p>(E)-3PO is a PFKFB3 (6-phosphofructo-2-kinase/fructose-2, 6-bisphosphatase) inhibitor.</p>Fórmula:C13H10N2OPureza:98.8% - 98.92%Forma y color:SolidPeso molecular:210.23Mitapivat sulfate hydrate
CAS:<p>Mitapivat sulfate hydrate (AG 348 sulfate hydrate) is a pyruvate kinase (PK) allosteric activator, used to study pyruvate kinase deficiency.</p>Fórmula:C24H26N4O3S1H2SO43H2OPureza:99.22%Forma y color:SolidPeso molecular:526.6KML29
CAS:<p>KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.</p>Fórmula:C24H21F6NO7Pureza:98.65%Forma y color:SolidPeso molecular:549.42Proguanil hydrochloride
CAS:<p>Proguanil hydrochloride, a biguanide, metabolizes into cycloguanil, an anti-malaria agent that inhibits plasmodium's DNA and protein synthesis.</p>Fórmula:C11H17Cl2N5Pureza:98.34% - 98.39%Forma y color:SolidPeso molecular:290.19GN44028
CAS:<p>GN44028 is a HIF-1 inhibitor with an IC50 of 14 nM, stopping HIF-1α activity but not mRNA or protein levels, or dimerization.</p>Fórmula:C18H15N3O2Pureza:99.52%Forma y color:SolidPeso molecular:305.33CTPI-2
CAS:<p>CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.</p>Fórmula:C13H9ClN2O6SPureza:97.23%Forma y color:SolidPeso molecular:356.74Tiplaxtinin
CAS:<p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>Fórmula:C24H16F3NO4Pureza:99.16% - 99.93%Forma y color:SolidPeso molecular:439.38CH-223191
CAS:<p>CH-223191, a specific aryl hydrocarbon receptor (AhR) antagonist, inhibited TCDD-induced luciferase activity with an IC50 of 0.03 μM. High-Quality, Low-Cost!</p>Fórmula:C19H19N5OPureza:99.01% - 99.71%Forma y color:SolidPeso molecular:333.39GSK256066 Trifluoroacetate
CAS:GSK 256066 Trifluoroacetate: selective PDE4 inhibitor, IC50: 3.2 pM for PDE4B, treats COPD.Fórmula:C29H27F3N4O7SForma y color:SolidPeso molecular:632.61Celgosivir hydrochloride
CAS:<p>Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).</p>Fórmula:C12H22ClNO5Forma y color:SolidPeso molecular:295.76Umbralisib hydrochloride
CAS:<p>Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.</p>Fórmula:C31H25ClF3N5O3Pureza:98%Forma y color:SolidPeso molecular:608.01Inulin
CAS:<p>Inulin(Inulin and sodium chloride), a starch found in the tubers and roots of many plants.</p>Fórmula:C6nH10nO5nPureza:99% - ≥95%Forma y color:White PowderPeso molecular:490.411FPH1
CAS:FPH1 (BRD-6125) (BRD-6125) can promote the expansion of iPS-derived hepatocytes.Fórmula:C16H15ClF2N2O3SPureza:99.80%Forma y color:SolidPeso molecular:388.82Dimethylfraxetin
CAS:<p>Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki:0.0097 μM)</p>Fórmula:C12H12O5Pureza:99.96% - ≥95%Forma y color:SolidPeso molecular:236.221-Ethynylpyrene
CAS:<p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>Fórmula:C18H10Pureza:98.48%Forma y color:SolidPeso molecular:226.27FOY 251
CAS:<p>FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.</p>Fórmula:C17H19N3O7SPureza:97.11% - 99.33%Forma y color:SolidPeso molecular:409.41HNHA
CAS:<p>HNHA is an inhibitor of HDAC.</p>Fórmula:C17H21NO2SPureza:98.04%Forma y color:SolidPeso molecular:303.42CP-640186 hydrochloride
CAS:<p>CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat</p>Fórmula:C30H36ClN3O3Pureza:98.86%Forma y color:SolidPeso molecular:522.08Cecropin P1, porcine acetate
<p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>Fórmula:C149H257N45O45Pureza:95.4% - 98%Forma y color:SolidPeso molecular:3398.91Glycerol 3-phosphate biscyclohexylammonium salt
CAS:<p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>Fórmula:C15H35N2O6PPureza:99.94%Forma y color:SolidPeso molecular:370.42Linrodostat mesylate
CAS:<p>Linrodostat (BMS-986205) is an oral IDO1 inhibitor that boosts immune response and has anti-cancer properties.</p>Fórmula:C25H28ClFN2O4SPureza:98%Forma y color:SolidPeso molecular:507.02ZSET1446
CAS:<p>ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.</p>Fórmula:C15H12N2OPureza:99.32%Forma y color:SolidPeso molecular:236.27Olesoxime
CAS:<p>Olesoxime (TRO 19622) (TRO19622), A Mitochondrial-Targeted Neuroprotective Compound,is an experimental neuroprotective drug.</p>Fórmula:C27H45NOPureza:99.86%Forma y color:SolidPeso molecular:399.65Elafibranor
CAS:<p>Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) with</p>Fórmula:C22H24O4SPureza:98.42% - 98.78%Forma y color:SolidPeso molecular:384.49MK-8617
CAS:<p>MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).</p>Fórmula:C24H21N5O4Pureza:99.38% - >99.99%Forma y color:SolidPeso molecular:443.45Pirozadil
CAS:Pirozadil shows hypolipidemic activity.Fórmula:C27H29NO10Pureza:97.54% - 98.31%Forma y color:SolidPeso molecular:527.52SR9238
CAS:<p>SR9238 is a synthetic agonist of liver X receptor inverse (IC50s: 214 nM and 43 nM for LXRα and LXRβ, respectively).</p>Fórmula:C31H33NO7S2Pureza:99.19% - 99.95%Forma y color:SolidPeso molecular:595.73FG-2216
CAS:<p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>Fórmula:C12H9ClN2O4Pureza:97.1% - >99.99%Forma y color:SolidPeso molecular:280.66G6PDi-1
CAS:<p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>Fórmula:C14H12N4OSPureza:98.69%Forma y color:SolidPeso molecular:284.34GW0742
CAS:<p>GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).</p>Fórmula:C21H17F4NO3S2Pureza:99.75% - 99.85%Forma y color:SolidPeso molecular:471.49kb NB 142-70
CAS:<p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>Fórmula:C11H9NO2S2Pureza:98.15% - ≥95%Forma y color:SolidPeso molecular:251.32Mitapivat
CAS:<p>Mitapivat (PKR-IN-1), also known as PKM2 activator 1020 is a PKM2 activator (pyruvate kinase activator) for the treatment of pyruvate kinase deficiency.</p>Fórmula:C24H26N4O3SPureza:99.47% - 99.83%Forma y color:SolidPeso molecular:450.553-METHOXY-DL-TYROSINE
CAS:<p>3-Methoxy-DL-Tyrosine: natural, non-essential amino, precursor to dopamine, may aid in treating Parkinson's, depression, obesity.</p>Fórmula:C10H13NO4Pureza:99.90%Forma y color:SolidPeso molecular:211.21(E)-2-Decenoic acid
CAS:<p>(E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.</p>Fórmula:C10H18O2Pureza:98%Forma y color:SolidPeso molecular:170.25Perfluorooctanoic acid
CAS:<p>Perfluorooctanoic acid (PFOA) (PFOA) is a persistent and widespread industry-made chemical.</p>Fórmula:C8HF15O2Pureza:99.70%Forma y color:White To Off-White Powder OthersolidPeso molecular:414.07BVT 2733
CAS:<p>BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1.</p>Fórmula:C17H21ClN4O3S2Pureza:98% - 99.64%Forma y color:SolidPeso molecular:428.96LB-60-OF61 hydrochloride
CAS:<p>LB-60-OF61 hydrochloride is a potent NAMPT enzyme inhibitor with cytotoxic effects, targeting MYC-overexpressing cell lines.</p>Fórmula:C29H31ClN6O2Forma y color:SolidPeso molecular:531.064-Chlorophenylurea
CAS:<p>4-Chlorophenylurea (NSC-12971) is a novel orally bioavailable inhibitor of factor Xa.</p>Fórmula:C7H7ClN2OPureza:98.87%Forma y color:White Granular / PrillPeso molecular:170.6BW-A 78U
CAS:<p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>Fórmula:C13H12FN5Pureza:99.45%Forma y color:SolidPeso molecular:257.27Glutamyl-glutamic acid
CAS:<p>Glutamyl-glutamic acid (Glu-glu) is an Interpeptide Bridge in the Murein of Some Micrococci and Arthrobacter sp..</p>Fórmula:C10H16N2O7Pureza:≥98%Forma y color:SolidPeso molecular:276.24Belzutifan
CAS:<p>"Belzutifan (MK-6482) is an oral HIF-2α inhibitor for ccRCC, with enhanced potency (IC50: 9 nM)."</p>Fórmula:C17H12F3NO4SPureza:99.34% - 99.88%Forma y color:SolidPeso molecular:383.34p-Fluoro-L-phenylalanine
CAS:<p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>Fórmula:C9H10FNO2Pureza:99.63%Forma y color:White To Off-White PowderPeso molecular:183.18PRL-3 Inhibitor I
CAS:<p>PRL-3 Inhibitor I (BR-1) is a phosphatase of regenerating liver 3 (PRL-3) inhibitor which blocks the migration and invasion of metastatic cancer cells.</p>Fórmula:C17H11Br2NO2S2Pureza:98.11%Forma y color:SolidPeso molecular:485.21LW6
CAS:<p>LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.</p>Fórmula:C26H29NO5Pureza:98.1% - 98.22%Forma y color:SolidPeso molecular:435.51JNJ-42041935
CAS:<p>JNJ-42041935 (HIF-PHD Inhibitor II) is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes.</p>Fórmula:C12H6ClF3N4O3Pureza:99.58% - ≥95%Forma y color:SolidPeso molecular:346.65Enterostatin, human, mouse, rat acetate
<p>Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.</p>Fórmula:C23H40N8O8Pureza:99.91%Forma y color:SolidPeso molecular:556.61Dansylglycine
CAS:<p>Dansylglycine is a fluorescent probe for specific determination of halogenating activity of myeloperoxidase and eosinophil peroxidase[1].</p>Fórmula:C14H16N2O4SPureza:99.1%Forma y color:SolidPeso molecular:308.35Fluorometholone Acetate
CAS:<p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>Fórmula:C24H31FO5Pureza:99.76%Forma y color:SolidPeso molecular:418.50NDI-091143
CAS:<p>NDI-091143 is a potent and high-affinity human ATP-citrate lyase (ACLY) inhibitor with an IC50 of 2.1 nM (ADP-Glo assay),indirectly disrupting citrate binding</p>Fórmula:C20H14ClF2NO5SPureza:97.03% - ≥95%Forma y color:SolidPeso molecular:453.84CAY10650
CAS:<p>CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).</p>Fórmula:C28H25NO6Pureza:97.33%Forma y color:SolidPeso molecular:471.5AUDA
CAS:<p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>Fórmula:C23H40N2O3Pureza:99.50%Forma y color:SolidPeso molecular:392.58Ethyl potassium malonate
CAS:<p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>Fórmula:C5H7KO4Pureza:99.71%Forma y color:White Crystals Or PowderPeso molecular:170.213-Methylglutaric acid
CAS:<p>Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.</p>Fórmula:C6H10O4Pureza:98.64%Forma y color:SolidPeso molecular:146.14GSK2981278
CAS:<p>GSK2981278 (ROR gama modulator 1) is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).</p>Fórmula:C25H35NO5SPureza:99.31% - 99.67%Forma y color:SolidPeso molecular:461.61STF-31
CAS:<p>STF-31 is an inhibitor of glucose transporter 1 (GLUT1) with IC50 of 1 μM.</p>Fórmula:C23H25N3O3SPureza:99.55% - >99.99%Forma y color:SolidPeso molecular:423.53LXR-623
CAS:<p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>Fórmula:C21H12ClF5N2Pureza:97.91% - 99.24%Forma y color:SolidPeso molecular:422.78U-104
CAS:<p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>Fórmula:C13H12FN3O3SPureza:98.76% - 99.88%Forma y color:SolidPeso molecular:309.32Eliglustat
CAS:<p>Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.</p>Fórmula:C23H36N2O4Pureza:99% - 99.70%Forma y color:SolidPeso molecular:404.54Cilofexor
CAS:<p>Cilofexor inhibits binding of a synthetic peptide, Cilofexor is a farnesoid X receptor (FXR) agonist.</p>Fórmula:C28H22Cl3N3O5Pureza:99.86% - ≥95%Forma y color:SolidPeso molecular:586.85SR0987
CAS:<p>SR0987 is a RORγt agonist,</p>Fórmula:C16H10ClF6NO2Pureza:99.43%Forma y color:SolidPeso molecular:397.7Zinc Phytate
CAS:<p>Zinc Phytate, present in food, plays a crucial role in human nutrient absorption.</p>Fórmula:C6H6O24P6Zn6Pureza:98%Forma y color:SolidPeso molecular:1040AA38-3
CAS:<p>AA38-3 (1-Piperidinecarboxylic acid, 4-nitrophenyl ester) inhibites three SHs (ABHD6, ABHD11, and FAAH)</p>Fórmula:C12H14N2O4Pureza:99.56%Forma y color:SolidPeso molecular:250.25DMOG
CAS:<p>DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.</p>Fórmula:C6H9NO5Pureza:80.23% - 99.98%Forma y color:SolidPeso molecular:175.14Lazabemide hydrochloride
CAS:<p>Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki:7.9nM).</p>Fórmula:C8H11Cl2N3OPureza:98.65%Forma y color:SolidPeso molecular:236.098SW033291
CAS:<p>SW033291 is a small-molecule inhibitor of 15-PGDH (Ki=0.1 nM) that increases prostaglandin PGE2 levels in bone marrow and other tissues.</p>Fórmula:C21H20N2OS3Pureza:97.26% - 99.02%Forma y color:SolidPeso molecular:412.59CDC25B-IN-2
CAS:<p>BIA is an inhibitor of the interaction between TMBIM6 and mTORC2, which ultimately blocks AKT activation and cancer progression.</p>Fórmula:C15H12N2O3Pureza:99.12%Forma y color:SolidPeso molecular:268.27Lofemizole
CAS:<p>Lofemizole is an antagonist of CYP1A2.</p>Fórmula:C10H9ClN2Pureza:97.11%Forma y color:SolidPeso molecular:192.64Ensifentrine
CAS:<p>Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3(IC50: 0.4 nM) is 3,440 times higher than that for PDE4(IC50: 1479 nM), that</p>Fórmula:C26H31N5O4Pureza:99.76% - 99.94%Forma y color:SolidPeso molecular:477.56L-Leucyl-L-Leucine methyl ester hydrochloride
CAS:<p>L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.</p>Fórmula:C13H27ClN2O3Pureza:98.41% - 99.63%Forma y color:SolidPeso molecular:294.81TM5275 sodium
CAS:<p>TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).</p>Fórmula:C28H27ClN3NaO5Pureza:98.8% - 99.74%Forma y color:SolidPeso molecular:543.98AG-120 (racemic)
CAS:<p>AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.</p>Fórmula:C28H22ClF3N6O3Pureza:99.56%Forma y color:SolidPeso molecular:582.963-Amino-2-oxazolidinone
CAS:<p>3-Amino-2-oxazolidinone (AOZ) is the metabolite of Furazolidone. It is always be detected as a indicator of furazolidone residues in vivo.</p>Fórmula:C3H6N2O2Pureza:97.82%Forma y color:SolidPeso molecular:102.09Piclamilast
CAS:<p>Piclamilast (RP 73401) is a PDE4 inhibitor.</p>Fórmula:C18H18Cl2N2O3Pureza:98.28% - 99.57%Forma y color:SolidPeso molecular:381.25RPI-1
CAS:<p>RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.</p>Fórmula:C17H15NO4Pureza:98.91% - ≥95%Forma y color:SolidPeso molecular:297.31Ibudilast
CAS:Ibudilast (MN-166)(KC-404;AV-411;MN-166) is a relatively nonselective phosphodiesterase inhibitor. It is approved for use as an anti-inflammatory in Japan.Fórmula:C14H18N2OPureza:99.83% - >99.99%Forma y color:White SolidPeso molecular:230.31M1001
CAS:<p>M1001 is a HIF-2α agonist.</p>Fórmula:C17H17N3O2SPureza:98.83%Forma y color:SolidPeso molecular:327.4Fomepizole hydrochloride
CAS:<p>Fomepizole hydrochloride inhibits CYP2E1 and alcohol dehydrogenase, blocking toxic metabolites, and treats methanol/ethylene glycol poisoning.</p>Fórmula:C4H7ClN2Forma y color:SolidPeso molecular:118.56(R)-GNE-140
CAS:<p>(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.</p>Fórmula:C25H23ClN2O3S2Pureza:98.25% - 98.91%Forma y color:SolidPeso molecular:499.04Calcitriol
CAS:<p>Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM).</p>Fórmula:C27H44O3Pureza:98.81% - 99.64%Forma y color:Colorless Crystalline Solid SolidPeso molecular:416.64TMS
CAS:<p>TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).</p>Fórmula:C18H20O4Pureza:99.17% - 99.73%Forma y color:SolidPeso molecular:300.35Balipodect
CAS:<p>Balipodect (TAK063) is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is >15000-fold over other PDEs.</p>Fórmula:C23H17FN6O2Pureza:98% - 99.79%Forma y color:SolidPeso molecular:428.42N-Oxalylglycine
CAS:<p>N-Oxalylglycine (Oxalylglycine) is a cell permeable inhibitor of α-ketoglutarate-dependent enzymes.</p>Fórmula:C4H5NO5Pureza:99.23%Forma y color:Colourless SolidPeso molecular:147.09BVT-14225
CAS:BVT-14225 is a selective 11β-Hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor (IC50=52 nM).Fórmula:C16H20ClN3O3S2Pureza:97.78%Forma y color:SolidPeso molecular:401.93NL-1
CAS:<p>NL-1 is a mitoNEET inhibitor with antileukemic effect.</p>Fórmula:C18H25NO3SPureza:98.64%Forma y color:SolidPeso molecular:335.46Lotamilast
CAS:<p>Lotamilast (RVT-501) is a phosphodiesterase 4 (PDE-4) inhibitor (IC50: 2.8 nM) potentially for the treatment of atopic dermatitis.</p>Fórmula:C26H24N4O5Pureza:97.03% - 99.29%Forma y color:SolidPeso molecular:472.49Calcineurin Autoinhibitory Peptide acetate
<p>Calcineurin Autoinhibitory Peptide acetate is a selectivecalcineurin phosphatase inhibitor(IC50 ~ 10 μM).</p>Fórmula:C252H417N78O82S4Pureza:97.24%Forma y color:SolidPeso molecular:5979.742,2'-Methylenebis(6-tert-butyl-4-methylphenol)
CAS:<p>2,2′-Methylenbis(4-methyl-6-tert-butylphenol) ist ein Antioxidans aus der Gruppe der Bisphenole.</p>Fórmula:C23H32O2Pureza:99.74%Forma y color:White Solid PowderPeso molecular:340.506-Phosphogluconic acid
CAS:<p>6-Phosphogluconic acid competitively inhibits PGI with Ki: 0.048 mM for glucose 6-P, 0.042 mM for fructose 6-P.</p>Fórmula:C6H13O10PPureza:98%Forma y color:SolidPeso molecular:276.14KY-226
CAS:<p>KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,)</p>Fórmula:C27H31NO3S2Pureza:99.4%Forma y color:SolidPeso molecular:481.67Biocytin
CAS:<p>Biocytin, a D-biotin and L-lysine conjugate, maps brain connections via a secondary amide bond.</p>Fórmula:C16H28N4O4SPureza:97.23%Forma y color:White SolidPeso molecular:372.48Haloxyfop
CAS:<p>(±)-Haloxyfop (Haloxyfop Acid) is a herbicide.</p>Fórmula:C15H11ClF3NO4Pureza:99.94% - >99.99%Forma y color:SolidPeso molecular:361.7ML-095 hydrochloride
CAS:ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.Fórmula:C13H15ClN2O3Pureza:99.37%Forma y color:SolidPeso molecular:282.72TEPP-46
CAS:<p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C17H16N4O2S2Pureza:98.21% - 98.77%Forma y color:SolidPeso molecular:372.46A939572
CAS:<p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of <4 nM for mSCD1 and 37 nM for hSCD1.</p>Fórmula:C20H22ClN3O3Pureza:99.96% - ≥95%Forma y color:SolidPeso molecular:387.86Fabomotizole hydrochloride
CAS:<p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>Fórmula:C15H22ClN3O2SPureza:99.54% - >99.99%Forma y color:SolidPeso molecular:343.871-Ethynylnaphthalene
CAS:<p>1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 IB1</p>Fórmula:C12H8Pureza:99.05%Forma y color:Yellow To Brown LiquidPeso molecular:152.19Isavuconazole
CAS:<p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>Fórmula:C22H17F2N5OSPureza:99.74% - >99.99%Forma y color:SolidPeso molecular:437.47Vardenafil hydrochloride trihydrate
CAS:<p>Vardenafil hydrochloride trihydrate (BAY38-9456) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>Fórmula:C23H32N6O4S·HCl·3H2OPureza:99.77%Forma y color:SolidPeso molecular:579.11Bay K 8644
CAS:<p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>Fórmula:C16H15F3N2O4Pureza:99.41%Forma y color:Yellow PowderPeso molecular:356.3Levamlodipine besylate
CAS:<p>Levamlodipine besylate, or S-amlodipine (CAS 103129-82-4), is the active enantiomer of amlodipine, used to treat hypertension and angina.</p>Fórmula:C26H31ClN2O8SPureza:99.78% - 99.79%Forma y color:SolidPeso molecular:567.05Tryptophan, N-indol-3-ylacetyl- (6CI)
CAS:<p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>Fórmula:C21H19N3O3Pureza:99.55%Forma y color:SolidPeso molecular:361.4Efonidipine
CAS:Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Fórmula:C34H38N3O7PPureza:98.35% - 99.47%Forma y color:SolidPeso molecular:631.66Lactisole
CAS:<p>Lactisole (na-PMP) is an inhibitor of the glucose-sensing receptor</p>Fórmula:C10H11NaO4Pureza:99.9%Forma y color:White To Pale Cream Crystalline SolidPeso molecular:218.182-Deoxy-2-sulfoamino-D-glucose sodium
CAS:<p>2-Deoxy-2-sulfoamino-D-glucose sodium (GlcN-2S) is possible to effect reaction at arthritis.</p>Fórmula:C6H12NNaO8SPureza:99.76%Forma y color:SolidPeso molecular:281.22Ziritaxestat
CAS:<p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>Fórmula:C30H33FN8O2SPureza:97% - 99.85%Forma y color:SolidPeso molecular:588.7N-Valyltryptophan
CAS:<p>N-Valyltryptophan (Val-trp) is an incomplete breakdown product of protein catabolism or protein digestion.</p>Fórmula:C16H21N3O3Pureza:97.52%Forma y color:SolidPeso molecular:303.361-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine
CAS:<p>1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.</p>Fórmula:C46H84NO8PPureza:98%Forma y color:SolidPeso molecular:810.13Dichlorphenamide
CAS:<p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>Fórmula:C6H6Cl2N2O4S2Pureza:96.87% - 97.25%Forma y color:Needles From Dimethylsulfoxide + Water SolidPeso molecular:305.16CP-91149
CAS:<p>CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence of</p>Fórmula:C21H22ClN3O3Pureza:99.66% - 99.81%Forma y color:SolidPeso molecular:399.87S29434
CAS:<p>S29434 (NMDPEF) is a potent, competitiveinhibitor of quinone reductase 2 (QR2;IC50:5-16nM).</p>Fórmula:C21H18N4O3Pureza:99.92%Forma y color:SolidPeso molecular:374.39JNJ-1661010
CAS:<p>JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.</p>Fórmula:C19H19N5OSPureza:99.79% - 99.97%Forma y color:SolidPeso molecular:365.45Cyclosporine
CAS:<p>Cyclosporine is a calcineurin phosphatase pathway inhibitor, used as an immunosuppressant drug to prevent rejection in organ transplantation.</p>Fórmula:C62H111N11O12Pureza:99.68%Forma y color:White PowderPeso molecular:1202.61n-acetylciprofloxacin
CAS:<p>n-acetylciprofloxacin (3-Quinolinecarboxylic acid, 7-(4-acetyl-1-piperazinyl)-1-cyclopropyl-6-fluoro-1) is inhibitor of H37Rv.</p>Fórmula:C19H20FN3O4Pureza:99.83%Forma y color:SolidPeso molecular:373.38Fmoc-Phe(4-CN)-OH
CAS:<p>Fmoc-Phe(4-CN)-OH is an N-Fmoc protected phenylalanine derivative and potentially useful synthetic intermediate</p>Fórmula:C25H20N2O4Pureza:99.45%Forma y color:White PowderPeso molecular:412.44BMS-309403
CAS:BMS309403 is a potent and selective inhibitor of adipocyte fatty acid binding protein aFABP.Cost-effective and quality-assured.Fórmula:C31H26N2O3Pureza:99.52% - 99.76%Forma y color:SolidPeso molecular:474.55FT113
CAS:<p>FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity</p>Fórmula:C22H20FN3O4Pureza:97.05%Forma y color:SolidPeso molecular:409.41Doxercalciferol
CAS:<p>Doxercalciferol, a synthetic vitamin D2, curbs parathyroid activity for treating secondary hyperparathyroidism and bone disorders.</p>Fórmula:C28H44O2Pureza:99.03% - 99.69%Forma y color:White Crystalline PowderPeso molecular:412.65SEA0400
CAS:<p>SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.</p>Fórmula:C21H19F2NO3Pureza:98.88% - 99.55%Forma y color:SolidPeso molecular:371.38NCT-501 hydrochloride
CAS:<p>NCT-501 hydrochloride: potent, selective ALDH1A1 inhibitor based on theophylline; IC50 of 40 nM; highly discriminant against other ALDHs.</p>Fórmula:C21H33ClN6O3Forma y color:SolidPeso molecular:452.98Methyl 13-cis-4-Oxoretinoate
CAS:<p>Methyl 13-cis-4-Oxoretinoate (13-cis-4-Oxo-retinoic acid Methyl Ester) is a retinoic acid metabolite in neuroblastoma.</p>Fórmula:C21H28O3Pureza:96.6% - 99.08%Forma y color:SolidPeso molecular:328.45VAS2870
CAS:VAS2870 is an inhibitor of NADPH oxidase (NOX).Fórmula:C18H12N6OSPureza:99.74%Forma y color:SolidPeso molecular:360.39PF-8380 hydrochloride
CAS:<p>PF-8380 hydrochloride is a powerful inhibitor of autotaxin, exhibiting an IC(50) of 2.8 nM in isolated enzyme assays and 101 nM in human whole blood.</p>Fórmula:C22H22Cl3N3O5Forma y color:SolidPeso molecular:514.79Darexaban
CAS:<p>Darexaban (YM-150) selectively inhibits Factor Xa, reducing clotting and risk of heart/stroke events.</p>Fórmula:C27H30N4O4Pureza:98.33%Forma y color:SolidPeso molecular:474.55Panaxadiol
CAS:<p>Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng.</p>Fórmula:C30H52O3Pureza:98% - 99.9%Forma y color:SolidPeso molecular:460.73N-Biotinyl-6-aminohexanoic acid
CAS:<p>N-Biotinyl-6-aminohexanoic acid (N-(+)-Biotinyl-6-aminohexanoic acid) can be used to perform N-terminal biotinylation.</p>Fórmula:C16H27N3O4SPureza:98.61%Forma y color:SolidPeso molecular:357.47Ponalrestat
CAS:<p>Ponalrestat is an aldose reductase inhibitor.</p>Fórmula:C17H12BrFN2O3Pureza:97.34% - 99.86%Forma y color:SolidPeso molecular:391.193-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one
CAS:<p>DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 nM, respectively)</p>Fórmula:C18H13NOPureza:99.37%Forma y color:SolidPeso molecular:259.316α-Hydroxyprednisolone
<p>16α-Hydroxyprednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonide</p>Fórmula:C21H28O6Pureza:99.75%Forma y color:White SolidPeso molecular:376.44RS-25344
CAS:<p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>Fórmula:C19H13N5O4Pureza:98.98%Forma y color:SolidPeso molecular:375.34ML355
CAS:<p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>Fórmula:C21H19N3O4S2Pureza:98.02% - 98.2%Forma y color:SolidPeso molecular:441.52ZINC13466751
CAS:<p>ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).</p>Fórmula:C20H21N5O2Pureza:99.8%Forma y color:SolidPeso molecular:363.41IOX2
CAS:<p>IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.</p>Fórmula:C19H16N2O5Pureza:98% - 99.59%Forma y color:SolidPeso molecular:352.34Pranidipine
CAS:<p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>Fórmula:C25H24N2O6Pureza:99.95%Forma y color:Yellow SolidPeso molecular:448.47ML-298
CAS:<p>ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).</p>Fórmula:C22H23F3N4O2Pureza:99.35%Forma y color:SolidPeso molecular:432.44Icerguastat
CAS:Icerguastat (IFB-088) is a selective inhibitor of holophosphatase. Icerguastat selectively inhibited a regulatory subunit of protein phosphatase 1 in vivo.Fórmula:C8H9ClN4Pureza:97.95%Forma y color:SolidPeso molecular:196.64Fomepizole
CAS:<p>Fomepizole (4-Methylpyrazole), a competitive inhibitor of alcohol dehydrogenase, is used as an antidote in methanol or ethylene glycol poisoning.</p>Fórmula:C4H6N2Pureza:98.1% - 99.94%Forma y color:Yellow <13°C Solid >13°C LiquidPeso molecular:82.1Z-HA155
CAS:<p>Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.</p>Fórmula:C24H19BFNO5SPureza:99.18%Forma y color:SolidPeso molecular:463.29Antimalarial agent 14
CAS:<p>Antimalarial agent 14 (NSC-102533) is a bioactive chemical.</p>Fórmula:C16H10O3Pureza:99.68%Forma y color:SolidPeso molecular:250.25N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
CAS:<p>Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.</p>Fórmula:C23H28N6Pureza:98.35%Forma y color:SolidPeso molecular:388.511-Naphthyl phosphate potassium salt
CAS:<p>1-Naphthyl phosphate potassium salt inhibits non-specific phosphatase.</p>Fórmula:C10H7K2O4PPureza:99%Forma y color:SolidPeso molecular:300.33MLCK inhibitor peptide 18 acetate
<p>MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.</p>Fórmula:C62H109N23O13Pureza:99.57%Forma y color:SolidPeso molecular:1384.67Tazarotene
CAS:<p>Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.</p>Fórmula:C21H21NO2SPureza:97.01% - 99.14%Forma y color:White SolidPeso molecular:351.46Inosine
CAS:<p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>Fórmula:C10H12N4O5Pureza:99.51% - 99.89%Forma y color:SolidPeso molecular:268.23Alkaline Phosphatase
CAS:<p>Alkaline phosphatase is a membrane-bound glycoprotein that catalyzes the hydrolysis of phosphate monoesters under alkaline conditions. High-Quality, Low-Cost!</p>Pureza:≥98%Forma y color:SolidPeso molecular:N/AYM-750
CAS:<p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>Fórmula:C31H36N2OPureza:99.96%Forma y color:SolidPeso molecular:452.63Bepridil hydrochloride
CAS:<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Fórmula:C24H35ClN2OPureza:99.45% - 99.68%Forma y color:SolidPeso molecular:403ND-646
CAS:<p>ND-646 is an orally bioavailable and allosteric inhibitor of the ACC enzymes ACC1 and ACC2(IC50s of 3.5 nM and 4.1 nM for recombinant hACC1 and hACC2,</p>Fórmula:C28H32N4O7SPureza:98.64%Forma y color:SolidPeso molecular:568.64GEBR-7b
CAS:<p>GEBR-7b (3-(Cyclopentyloxy)-4-methoxybenzaldehyde) is a phosphodiesterase-4 (PDE4) inhibitor.</p>Fórmula:C13H16O3Pureza:99.533%Forma y color:SolidPeso molecular:220.26Tetrahydropapaverine hydrochloride
CAS:<p>Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.</p>Fórmula:C20H26ClNO4Pureza:99.08%Forma y color:White Crystal PowderPeso molecular:379.878Tropifexor
CAS:<p>Tropifexor (LJN452) is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM.</p>Fórmula:C29H25F4N3O5SPureza:99.3% - 99.85%Forma y color:SolidPeso molecular:603.58CVT-2738
CAS:<p>CVT-2738 (RS-94287) is a metabolite of Ranolazine. Ranolazine is a partial fatty acid oxidation (pFOX) inhibitor and anti-anginal drug.</p>Fórmula:C14H21N3OPureza:99.84%Forma y color:SolidPeso molecular:247.34BAY-218
CAS:<p>Bindarit (AF2838) is an aryl hydrocarbon receptor (AHR) antagonist.Cost-effective and quality-assured.</p>Fórmula:C20H17ClFN3O3Pureza:99.46% - 99.85%Forma y color:SolidPeso molecular:401.82Fmoc-N-Me-Leu-OH
CAS:Fmoc-N-Me-Leu-OH is available for the peptide-coupling reaction.Fórmula:C22H25NO4Pureza:99.51%Forma y color:White PowderPeso molecular:367.44SR33805
CAS:<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Fórmula:C32H40N2O5SPureza:99.15%Forma y color:SolidPeso molecular:564.74Angiotensin I (human, mouse, rat)
CAS:<p>Angiotensin I (human, mouse, rat) is the precursor to the vasoconstrictor peptide angiotensin II, cleaved by the angiotensin-converting enzyme (ACE).</p>Fórmula:C62H89N17O14Pureza:>99.99%Forma y color:SolidPeso molecular:1296.484-Methylumbelliferyl-β-D-Glucopyranoside
CAS:<p>4-Methylumbelliferyl-β-D-Glucopyranoside (4-MU-GLU) is used in the GCase activity assay based on the catalytic hydrolysis of 4-methylumbelliferyl β-D-</p>Fórmula:C16H18O8Pureza:99.89%Forma y color:White PowderPeso molecular:338.31BMS-823778 hydrochloride
CAS:<p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>Fórmula:C18H19Cl2N3OForma y color:SolidPeso molecular:364.274-Nonylphenylboronic acid
CAS:<p>4-Nonylphenylboronic acid is a inhibitor of FAAH.</p>Fórmula:C15H25BO2Pureza:97.63%Forma y color:SolidPeso molecular:248.171,2-Didecanoyl-sn-glycero-3-phosphocholi
CAS:<p>1,2-Didecanoyl PC: synthetic phospholipid aiding peptide drug and insulin absorption.</p>Fórmula:C28H56NO8PPureza:98%Forma y color:SolidPeso molecular:565.72Turofexorate Isopropyl
CAS:<p>Turofexorate Isopropyl (XL335) is a potent, selective, and orally bioavailable FXR agonist with EC50 of 4 nM</p>Fórmula:C25H24F2N2O3Pureza:98.55% - 99.73%Forma y color:SolidPeso molecular:438.47Idoxuridine hydrate
CAS:<p>Idoxuridine (5-IUdR) blocks DNA polymerase, treating herpes eye infections, with an IC50 of 4.3 μM against feline herpes.</p>Fórmula:C9H13IN2O6Forma y color:SolidPeso molecular:372.115Tebufenpyrad
CAS:<p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>Fórmula:C18H24ClN3OPureza:98.63% - 99.16%Forma y color:SolidPeso molecular:333.86Atglistatin
CAS:<p>Atglistatin: ATGL inhibitor, IC50 ~0.7 μM, inhibits lipolysis, non-toxic up to 50 μM.</p>Fórmula:C17H21N3OPureza:97.2% - 99.01%Forma y color:SolidPeso molecular:283.37SR9011 hydrochloride
CAS:<p>SR9011 hydrochloride is a REV-ERBα/β agonist, exhibiting an IC50 value of 790 nM for REV-ERBα and 560 nM for REV-ERBβ.</p>Fórmula:C23H32Cl2N4O3SForma y color:SolidPeso molecular:515.49Tauro-Obeticholic acid
CAS:<p>Tauro-Obeticholic acid is an active Obeticholic acid metabolite. Obeticholic acid is an orally bioavailable agonist of farnesoid-X receptor (FXR).</p>Fórmula:C28H49NO6SPureza:99.74% - 99.82%Forma y color:SolidPeso molecular:527.767-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS:<p>7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).</p>Fórmula:C15H16N4Pureza:99.22%Forma y color:SolidPeso molecular:252.31Kresoxim-Methyl
CAS:<p>Kresoxim-methyl is a strobilurin fungicide,inhibits conidial germination of V. inaequalis isolates from apple orchards .</p>Fórmula:C18H19NO4Pureza:99.24%Forma y color:SolidPeso molecular:313.35TM5007
CAS:<p>TM5007 is a poent inhibitor of plasminogen activator inhibitor-1 (PAI-1; IC50 of 29 uM).</p>Fórmula:C24H20N2O6S4Pureza:96.91%Forma y color:SolidPeso molecular:560.69Gcase activator 1
CAS:<p>Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator.</p>Fórmula:C20H30N4O2Pureza:99.25% - 99.31%Forma y color:SolidPeso molecular:358.48Tempol
CAS:<p>Tempol (Tanol) is a superoxide scavenger. It has anti-inflammatory, neuroprotective and analgesic effects.</p>Fórmula:C9H18NO2Pureza:97% - 99.74%Forma y color:4-Hydroxy-Tempo Appears As Orange Flakes Solid FlakesPeso molecular:172.25Monobenzyl phthalate
CAS:<p>Monobenzyl phthalate (Phthalic Acid Monobenzyl Ester) is Phthalate metabolite.</p>Fórmula:C15H12O4Pureza:99.11% - 99.38%Forma y color:SolidPeso molecular:256.256-Aminonicotinamide
CAS:<p>6-Aminonicotinamide (6-AN) is a well-established inhibitor of the NADP+-dependent enzyme.</p>Fórmula:C6H7N3OPureza:98.99% - 99.4%Forma y color:Physical Description White Crystalline Solid (Ntp 1992)Peso molecular:137.142-Ketoglutaric acid
CAS:<p>2-Ketoglutaric acid is a reversible inhibitor of tyrosinase (IC50=15 mM). 2-Ketoglutaric acid is an intermediate of the Krebs cycle. High-Quality, Low-Cost!</p>Fórmula:C5H6O5Pureza:99.28%Forma y color:SolidPeso molecular:146.1Orthanilamide
CAS:Orthanilamide (Orthanilamide) is a molecule containing the sulfonamide functional group attached to an aniline.Fórmula:C6H8N2O2SPureza:99.72% - 99.96%Forma y color:White To Pale Cream Crystalline Powder Or CrystalsPeso molecular:172.2Homo Sildenafil
CAS:<p>Homo Sildenafil is an analog of Sildenafil, It acts as a phosphodiesterase inhibitor.</p>Fórmula:C23H32N6O4SPureza:99.88%Forma y color:White SolidPeso molecular:488.6Dorzolamide hydrochloride
CAS:<p>Dorzolamide hydrochloride (MK507 hydrochloride) is the hydrochloride salt form of dorzolamide, an inhibitor of carbonic anhydrase, a zinc-containing enzyme that</p>Fórmula:C10H17ClN2O4S3Pureza:99.48% - 99.67%Forma y color:White Off-White Crystalline PowderPeso molecular:360.9HET0016
CAS:<p>HET0016: potent, selective 20-HETE synthase/CYP450 inhibitor; IC50s: 17.7-20.6 nM; inhibits angiogenesis, tumor growth.</p>Fórmula:C12H18N2OPureza:98.84%Forma y color:SolidPeso molecular:206.28TPPU
CAS:<p>TPPU is a potent inhibitor of both human and mouse sEH (IC50 of 3.7 and 2.8 nM, respectively)</p>Fórmula:C16H20F3N3O3Pureza:97.82%Forma y color:SolidPeso molecular:359.34SR9243
CAS:<p>SR9243, an LXR inverse agonist, can induce LXR-corepressor interaction; shows anticancer activity and selectively targets the lipogenesis and Warburg effect.</p>Fórmula:C31H32BrNO4S2Pureza:98% - 99.03%Forma y color:SolidPeso molecular:626.62N-desmethylmirtazapine
CAS:N-desmethylmirtazapine: mirtazapine metabolite; used for anxiety, sleep, nausea, appetite.Fórmula:C16H17N3Pureza:99.84%Forma y color:SolidPeso molecular:251.33
