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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • CALP3 acetate(261969-05-5 free base)


    <p>CALP3 acetate blocks Ca2+ channels, mimics elevated [Ca2+]i, activates EF hands, and regulates CaM, channels, and pumps.</p>
    Fórmula:C46H72N10O11
    Pureza:96.49%
    Forma y color:Solid
    Peso molecular:941.12
  • Lanthanum(III) chloride heptahydrate

    CAS:
    <p>Lanthanum(III) chloride blocks divalent cation channels, useful for biochemical research.</p>
    Fórmula:Cl3H14LaO7
    Pureza:98%
    Forma y color:White Solid Powder
    Peso molecular:371.37
  • YTX-465

    CAS:
    <p>YTX-465 is an inhibitor of both stearoyl-CoA desaturase(IC50s = 39 nM) and Ole1 (IC50s = 30.4 μM).</p>
    Fórmula:C25H26N6O3
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:458.51
  • AR7

    CAS:
    <p>AR7 is a retinoic acid receptor α (RARα) antagonist.</p>
    Fórmula:C15H12ClNO
    Pureza:98.12% - 99.86%
    Forma y color:Solid
    Peso molecular:257.71
  • WWL229

    CAS:
    <p>WWL229 selectively inhibits Ces3 without affecting Ces1f, ABHD6, or other serine hydrolases, mimicking WWL113 in adipocytes.</p>
    Fórmula:C16H22N2O5
    Pureza:98.14%
    Forma y color:Solid
    Peso molecular:322.36
  • CAY10698

    CAS:
    <p>CAY10698 is a 12-lipoxygenase inhibitor (12-LO; IC50 of 5.1 μM).</p>
    Fórmula:C17H17N3O4S2
    Pureza:98.97%
    Forma y color:Solid
    Peso molecular:391.46
  • Udenafil

    CAS:
    <p>Udenafil is an inhibitor of PDE5 .</p>
    Fórmula:C25H36N6O4S
    Pureza:99.90%
    Forma y color:Off-White Solid
    Peso molecular:516.66
  • Vonafexor

    CAS:
    <p>Vonafexor (EYP001) is a farnesoid X receptor (FXR, NR1H4) agonist, with anti-HBV effects</p>
    Fórmula:C19H15Cl3N2O5S
    Pureza:98.74%
    Forma y color:Solid
    Peso molecular:489.76
  • IACS-13909

    CAS:
    <p>IACS-13909 (BBP-398), a specific and potent allosteric inhibitor of SHP2, that suppresses signaling through the MAPK pathway.</p>
    Fórmula:C17H18Cl2N6
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:377.27
  • U-73122

    CAS:
    <p>U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.</p>
    Fórmula:C29H40N2O3
    Pureza:97.50%
    Forma y color:Solid Off-White
    Peso molecular:464.64
  • Dimesna

    CAS:
    <p>Dimesna (BNP-7787) is a synthetic derivative of dithio-ethane sulfonate with uroprotective properties.</p>
    Fórmula:C4H8Na2O6S4
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:326.34
  • GSK 650394

    CAS:
    <p>GSK 650394 is an inhibitor of serum- and glucocorticoid-regulated kinases (SGK). GSK 650394 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C25H22N2O2
    Pureza:97.46% - >99.99%
    Forma y color:Solid
    Peso molecular:382.45
  • Benzamidine hydrochloride

    CAS:
    <p>Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.</p>
    Fórmula:C7H9ClN2
    Pureza:99.25% - 99.97%
    Forma y color:White To Off-White Powder
    Peso molecular:156.61
  • CID 2011756

    CAS:
    <p>CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.</p>
    Fórmula:C22H21ClN2O3
    Pureza:98.15% - ≥95%
    Forma y color:Solid
    Peso molecular:396.87
  • PSB-1491

    CAS:
    PSB-1491 is a selective and competitive monoamine oxidase B inhibitor with IC50 of 0.386 nM, >25000-fold selective versus MAO-A.
    Fórmula:C15H11Cl2N3O
    Pureza:98.41% - 99.68%
    Forma y color:Solid
    Peso molecular:320.17
  • Sulindac sulfone

    CAS:
    <p>Sulindac sulfone is a metabolite of the nonsteroidal anti-inflammatory drug sulindac. Sulindac sulfone is an inhibitor of aldose reductase (IC50 =367 nM).</p>
    Fórmula:C20H17FO4S
    Pureza:98.2% - 98.83%
    Forma y color:Solid
    Peso molecular:372.41
  • ICI 63197

    CAS:
    ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.
    Fórmula:C9H13N5O
    Pureza:99.70%
    Forma y color:White Solid
    Peso molecular:207.23
  • ML-030

    CAS:
    <p>ML-030 is a potent PDE4 inhibitor, selective for subtypes (A1, B1, B2, C1, D2) with IC50 ranging from 6.7 to 452 nM.</p>
    Fórmula:C20H20N4O4S
    Pureza:97.93%
    Forma y color:Solid
    Peso molecular:412.46
  • Minaprine dihydrochloride

    CAS:
    <p>Minaprine dihydrochloride: reversible MAO-A inhibitor, mild on acetylcholinesterase, used for depression.</p>
    Fórmula:C17H24Cl2N4O
    Pureza:99.43% - 99.99%
    Forma y color:Solid
    Peso molecular:371.3
  • W 36017

    CAS:
    <p>W36017 is an impurity of lidocaine with a PKA of 7.4 for blocking neurologic activity.</p>
    Fórmula:C12H18N2O
    Pureza:99.09%
    Forma y color:Solid
    Peso molecular:206.28
  • (E)-3PO

    CAS:
    <p>(E)-3PO is a PFKFB3 (6-phosphofructo-2-kinase/fructose-2, 6-bisphosphatase) inhibitor.</p>
    Fórmula:C13H10N2O
    Pureza:98.8% - 98.92%
    Forma y color:Solid
    Peso molecular:210.23
  • Mitapivat sulfate hydrate

    CAS:
    <p>Mitapivat sulfate hydrate (AG 348 sulfate hydrate) is a pyruvate kinase (PK) allosteric activator, used to study pyruvate kinase deficiency.</p>
    Fórmula:C24H26N4O3S1H2SO43H2O
    Pureza:99.22%
    Forma y color:Solid
    Peso molecular:526.6
  • KML29

    CAS:
    <p>KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.</p>
    Fórmula:C24H21F6NO7
    Pureza:98.65%
    Forma y color:Solid
    Peso molecular:549.42
  • Proguanil hydrochloride

    CAS:
    <p>Proguanil hydrochloride, a biguanide, metabolizes into cycloguanil, an anti-malaria agent that inhibits plasmodium's DNA and protein synthesis.</p>
    Fórmula:C11H17Cl2N5
    Pureza:98.34% - 98.39%
    Forma y color:Solid
    Peso molecular:290.19
  • GN44028

    CAS:
    <p>GN44028 is a HIF-1 inhibitor with an IC50 of 14 nM, stopping HIF-1α activity but not mRNA or protein levels, or dimerization.</p>
    Fórmula:C18H15N3O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:305.33
  • CTPI-2

    CAS:
    <p>CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.</p>
    Fórmula:C13H9ClN2O6S
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:356.74
  • Tiplaxtinin

    CAS:
    <p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>
    Fórmula:C24H16F3NO4
    Pureza:99.16% - 99.93%
    Forma y color:Solid
    Peso molecular:439.38
  • CH-223191

    CAS:
    <p>CH-223191, a specific aryl hydrocarbon receptor (AhR) antagonist, inhibited TCDD-induced luciferase activity with an IC50 of 0.03 μM. High-Quality, Low-Cost!</p>
    Fórmula:C19H19N5O
    Pureza:99.01% - 99.71%
    Forma y color:Solid
    Peso molecular:333.39
  • GSK256066 Trifluoroacetate

    CAS:
    GSK 256066 Trifluoroacetate: selective PDE4 inhibitor, IC50: 3.2 pM for PDE4B, treats COPD.
    Fórmula:C29H27F3N4O7S
    Forma y color:Solid
    Peso molecular:632.61
  • Celgosivir hydrochloride

    CAS:
    <p>Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).</p>
    Fórmula:C12H22ClNO5
    Forma y color:Solid
    Peso molecular:295.76
  • Umbralisib hydrochloride

    CAS:
    <p>Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.</p>
    Fórmula:C31H25ClF3N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:608.01
  • Inulin

    CAS:
    <p>Inulin(Inulin and sodium chloride), a starch found in the tubers and roots of many plants.</p>
    Fórmula:C6nH10nO5n
    Pureza:99% - ≥95%
    Forma y color:White Powder
    Peso molecular:490.411
  • FPH1

    CAS:
    FPH1 (BRD-6125) (BRD-6125) can promote the expansion of iPS-derived hepatocytes.
    Fórmula:C16H15ClF2N2O3S
    Pureza:99.80%
    Forma y color:Solid
    Peso molecular:388.82
  • Dimethylfraxetin

    CAS:
    <p>Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki:0.0097 μM)</p>
    Fórmula:C12H12O5
    Pureza:99.96% - ≥95%
    Forma y color:Solid
    Peso molecular:236.22
  • 1-Ethynylpyrene

    CAS:
    <p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>
    Fórmula:C18H10
    Pureza:98.48%
    Forma y color:Solid
    Peso molecular:226.27
  • FOY 251

    CAS:
    <p>FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.</p>
    Fórmula:C17H19N3O7S
    Pureza:97.11% - 99.33%
    Forma y color:Solid
    Peso molecular:409.41
  • HNHA

    CAS:
    <p>HNHA is an inhibitor of HDAC.</p>
    Fórmula:C17H21NO2S
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:303.42
  • CP-640186 hydrochloride

    CAS:
    <p>CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat</p>
    Fórmula:C30H36ClN3O3
    Pureza:98.86%
    Forma y color:Solid
    Peso molecular:522.08
  • Cecropin P1, porcine acetate


    <p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>
    Fórmula:C149H257N45O45
    Pureza:95.4% - 98%
    Forma y color:Solid
    Peso molecular:3398.91
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Fórmula:C15H35N2O6P
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:370.42
  • Linrodostat mesylate

    CAS:
    <p>Linrodostat (BMS-986205) is an oral IDO1 inhibitor that boosts immune response and has anti-cancer properties.</p>
    Fórmula:C25H28ClFN2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:507.02
  • ZSET1446

    CAS:
    <p>ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.</p>
    Fórmula:C15H12N2O
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:236.27
  • Olesoxime

    CAS:
    <p>Olesoxime (TRO 19622) (TRO19622), A Mitochondrial-Targeted Neuroprotective Compound,is an experimental neuroprotective drug.</p>
    Fórmula:C27H45NO
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:399.65
  • Elafibranor

    CAS:
    <p>Elafibranor (GFT505) is an agonist of the peroxisome proliferator-activated receptor-α (PPAR-α) and peroxisome proliferator-activated receptor-δ (PPAR-δ) with</p>
    Fórmula:C22H24O4S
    Pureza:98.42% - 98.78%
    Forma y color:Solid
    Peso molecular:384.49
  • MK-8617

    CAS:
    <p>MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).</p>
    Fórmula:C24H21N5O4
    Pureza:99.38% - >99.99%
    Forma y color:Solid
    Peso molecular:443.45
  • Pirozadil

    CAS:
    Pirozadil shows hypolipidemic activity.
    Fórmula:C27H29NO10
    Pureza:97.54% - 98.31%
    Forma y color:Solid
    Peso molecular:527.52
  • SR9238

    CAS:
    <p>SR9238 is a synthetic agonist of liver X receptor inverse (IC50s: 214 nM and 43 nM for LXRα and LXRβ, respectively).</p>
    Fórmula:C31H33NO7S2
    Pureza:99.19% - 99.95%
    Forma y color:Solid
    Peso molecular:595.73
  • FG-2216

    CAS:
    <p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>
    Fórmula:C12H9ClN2O4
    Pureza:97.1% - >99.99%
    Forma y color:Solid
    Peso molecular:280.66
  • G6PDi-1

    CAS:
    <p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>
    Fórmula:C14H12N4OS
    Pureza:98.69%
    Forma y color:Solid
    Peso molecular:284.34
  • GW0742

    CAS:
    <p>GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for human PPARδ/α/γ).</p>
    Fórmula:C21H17F4NO3S2
    Pureza:99.75% - 99.85%
    Forma y color:Solid
    Peso molecular:471.49
  • kb NB 142-70

    CAS:
    <p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>
    Fórmula:C11H9NO2S2
    Pureza:98.15% - ≥95%
    Forma y color:Solid
    Peso molecular:251.32
  • Mitapivat

    CAS:
    <p>Mitapivat (PKR-IN-1), also known as PKM2 activator 1020 is a PKM2 activator (pyruvate kinase activator) for the treatment of pyruvate kinase deficiency.</p>
    Fórmula:C24H26N4O3S
    Pureza:99.47% - 99.83%
    Forma y color:Solid
    Peso molecular:450.55
  • 3-METHOXY-DL-TYROSINE

    CAS:
    <p>3-Methoxy-DL-Tyrosine: natural, non-essential amino, precursor to dopamine, may aid in treating Parkinson's, depression, obesity.</p>
    Fórmula:C10H13NO4
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:211.21
  • (E)-2-Decenoic acid

    CAS:
    <p>(E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.</p>
    Fórmula:C10H18O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:170.25
  • Perfluorooctanoic acid

    CAS:
    <p>Perfluorooctanoic acid (PFOA) (PFOA) is a persistent and widespread industry-made chemical.</p>
    Fórmula:C8HF15O2
    Pureza:99.70%
    Forma y color:White To Off-White Powder Othersolid
    Peso molecular:414.07
  • BVT 2733

    CAS:
    <p>BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1.</p>
    Fórmula:C17H21ClN4O3S2
    Pureza:98% - 99.64%
    Forma y color:Solid
    Peso molecular:428.96
  • LB-60-OF61 hydrochloride

    CAS:
    <p>LB-60-OF61 hydrochloride is a potent NAMPT enzyme inhibitor with cytotoxic effects, targeting MYC-overexpressing cell lines.</p>
    Fórmula:C29H31ClN6O2
    Forma y color:Solid
    Peso molecular:531.06
  • 4-Chlorophenylurea

    CAS:
    <p>4-Chlorophenylurea (NSC-12971) is a novel orally bioavailable inhibitor of factor Xa.</p>
    Fórmula:C7H7ClN2O
    Pureza:98.87%
    Forma y color:White Granular / Prill
    Peso molecular:170.6
  • BW-A 78U

    CAS:
    <p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>
    Fórmula:C13H12FN5
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:257.27
  • Glutamyl-glutamic acid

    CAS:
    <p>Glutamyl-glutamic acid (Glu-glu) is an Interpeptide Bridge in the Murein of Some Micrococci and Arthrobacter sp..</p>
    Fórmula:C10H16N2O7
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:276.24
  • Belzutifan

    CAS:
    <p>"Belzutifan (MK-6482) is an oral HIF-2α inhibitor for ccRCC, with enhanced potency (IC50: 9 nM)."</p>
    Fórmula:C17H12F3NO4S
    Pureza:99.34% - 99.88%
    Forma y color:Solid
    Peso molecular:383.34
  • p-Fluoro-L-phenylalanine

    CAS:
    <p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>
    Fórmula:C9H10FNO2
    Pureza:99.63%
    Forma y color:White To Off-White Powder
    Peso molecular:183.18
  • PRL-3 Inhibitor I

    CAS:
    <p>PRL-3 Inhibitor I (BR-1) is a phosphatase of regenerating liver 3 (PRL-3) inhibitor which blocks the migration and invasion of metastatic cancer cells.</p>
    Fórmula:C17H11Br2NO2S2
    Pureza:98.11%
    Forma y color:Solid
    Peso molecular:485.21
  • LW6

    CAS:
    <p>LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.</p>
    Fórmula:C26H29NO5
    Pureza:98.1% - 98.22%
    Forma y color:Solid
    Peso molecular:435.51
  • JNJ-42041935

    CAS:
    <p>JNJ-42041935 (HIF-PHD Inhibitor II) is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes.</p>
    Fórmula:C12H6ClF3N4O3
    Pureza:99.58% - ≥95%
    Forma y color:Solid
    Peso molecular:346.65
  • Enterostatin, human, mouse, rat acetate


    <p>Enterostatin, human, mouse, rat acetate is a pentapeptide mainly formed in the intestine by the cleavage of secreted pancreatic procolipase.</p>
    Fórmula:C23H40N8O8
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:556.61
  • Dansylglycine

    CAS:
    <p>Dansylglycine is a fluorescent probe for specific determination of halogenating activity of myeloperoxidase and eosinophil peroxidase[1].</p>
    Fórmula:C14H16N2O4S
    Pureza:99.1%
    Forma y color:Solid
    Peso molecular:308.35
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Fórmula:C24H31FO5
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:418.50
  • NDI-091143

    CAS:
    <p>NDI-091143 is a potent and high-affinity human ATP-citrate lyase (ACLY) inhibitor with an IC50 of 2.1 nM (ADP-Glo assay),indirectly disrupting citrate binding</p>
    Fórmula:C20H14ClF2NO5S
    Pureza:97.03% - ≥95%
    Forma y color:Solid
    Peso molecular:453.84
  • CAY10650

    CAS:
    <p>CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).</p>
    Fórmula:C28H25NO6
    Pureza:97.33%
    Forma y color:Solid
    Peso molecular:471.5
  • AUDA

    CAS:
    <p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>
    Fórmula:C23H40N2O3
    Pureza:99.50%
    Forma y color:Solid
    Peso molecular:392.58
  • Ethyl potassium malonate

    CAS:
    <p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>
    Fórmula:C5H7KO4
    Pureza:99.71%
    Forma y color:White Crystals Or Powder
    Peso molecular:170.21
  • 3-Methylglutaric acid

    CAS:
    <p>Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.</p>
    Fórmula:C6H10O4
    Pureza:98.64%
    Forma y color:Solid
    Peso molecular:146.14
  • GSK2981278

    CAS:
    <p>GSK2981278 (ROR gama modulator 1) is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).</p>
    Fórmula:C25H35NO5S
    Pureza:99.31% - 99.67%
    Forma y color:Solid
    Peso molecular:461.61
  • STF-31

    CAS:
    <p>STF-31 is an inhibitor of glucose transporter 1 (GLUT1) with IC50 of 1 μM.</p>
    Fórmula:C23H25N3O3S
    Pureza:99.55% - >99.99%
    Forma y color:Solid
    Peso molecular:423.53
  • LXR-623

    CAS:
    <p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>
    Fórmula:C21H12ClF5N2
    Pureza:97.91% - 99.24%
    Forma y color:Solid
    Peso molecular:422.78
  • U-104

    CAS:
    <p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>
    Fórmula:C13H12FN3O3S
    Pureza:98.76% - 99.88%
    Forma y color:Solid
    Peso molecular:309.32
  • Eliglustat

    CAS:
    <p>Eliglustat (Genz 99067) is an oral inhibitor of glucosylceramide synthase which is used in the therapy of type 1 Gaucher disease.</p>
    Fórmula:C23H36N2O4
    Pureza:99% - 99.70%
    Forma y color:Solid
    Peso molecular:404.54
  • Cilofexor

    CAS:
    <p>Cilofexor inhibits binding of a synthetic peptide, Cilofexor is a farnesoid X receptor (FXR) agonist.</p>
    Fórmula:C28H22Cl3N3O5
    Pureza:99.86% - ≥95%
    Forma y color:Solid
    Peso molecular:586.85
  • SR0987

    CAS:
    <p>SR0987 is a RORγt agonist,</p>
    Fórmula:C16H10ClF6NO2
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:397.7
  • Zinc Phytate

    CAS:
    <p>Zinc Phytate, present in food, plays a crucial role in human nutrient absorption.</p>
    Fórmula:C6H6O24P6Zn6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1040
  • AA38-3

    CAS:
    <p>AA38-3 (1-Piperidinecarboxylic acid, 4-nitrophenyl ester) inhibites three SHs (ABHD6, ABHD11, and FAAH)</p>
    Fórmula:C12H14N2O4
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:250.25
  • DMOG

    CAS:
    <p>DMOG (Dimethyloxalylglycine), an antagonist of the α-ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.</p>
    Fórmula:C6H9NO5
    Pureza:80.23% - 99.98%
    Forma y color:Solid
    Peso molecular:175.14
  • Lazabemide hydrochloride

    CAS:
    <p>Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki:7.9nM).</p>
    Fórmula:C8H11Cl2N3O
    Pureza:98.65%
    Forma y color:Solid
    Peso molecular:236.098
  • SW033291

    CAS:
    <p>SW033291 is a small-molecule inhibitor of 15-PGDH (Ki=0.1 nM) that increases prostaglandin PGE2 levels in bone marrow and other tissues.</p>
    Fórmula:C21H20N2OS3
    Pureza:97.26% - 99.02%
    Forma y color:Solid
    Peso molecular:412.59
  • CDC25B-IN-2

    CAS:
    <p>BIA is an inhibitor of the interaction between TMBIM6 and mTORC2, which ultimately blocks AKT activation and cancer progression.</p>
    Fórmula:C15H12N2O3
    Pureza:99.12%
    Forma y color:Solid
    Peso molecular:268.27
  • Lofemizole

    CAS:
    <p>Lofemizole is an antagonist of CYP1A2.</p>
    Fórmula:C10H9ClN2
    Pureza:97.11%
    Forma y color:Solid
    Peso molecular:192.64
  • Ensifentrine

    CAS:
    <p>Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3(IC50: 0.4 nM) is 3,440 times higher than that for PDE4(IC50: 1479 nM), that</p>
    Fórmula:C26H31N5O4
    Pureza:99.76% - 99.94%
    Forma y color:Solid
    Peso molecular:477.56
  • L-Leucyl-L-Leucine methyl ester hydrochloride

    CAS:
    <p>L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.</p>
    Fórmula:C13H27ClN2O3
    Pureza:98.41% - 99.63%
    Forma y color:Solid
    Peso molecular:294.81
  • TM5275 sodium

    CAS:
    <p>TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).</p>
    Fórmula:C28H27ClN3NaO5
    Pureza:98.8% - 99.74%
    Forma y color:Solid
    Peso molecular:543.98
  • AG-120 (racemic)

    CAS:
    <p>AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.</p>
    Fórmula:C28H22ClF3N6O3
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:582.96
  • 3-Amino-2-oxazolidinone

    CAS:
    <p>3-Amino-2-oxazolidinone (AOZ) is the metabolite of Furazolidone. It is always be detected as a indicator of furazolidone residues in vivo.</p>
    Fórmula:C3H6N2O2
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:102.09
  • Piclamilast

    CAS:
    <p>Piclamilast (RP 73401) is a PDE4 inhibitor.</p>
    Fórmula:C18H18Cl2N2O3
    Pureza:98.28% - 99.57%
    Forma y color:Solid
    Peso molecular:381.25
  • RPI-1

    CAS:
    <p>RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.</p>
    Fórmula:C17H15NO4
    Pureza:98.91% - ≥95%
    Forma y color:Solid
    Peso molecular:297.31
  • Ibudilast

    CAS:
    Ibudilast (MN-166)(KC-404;AV-411;MN-166) is a relatively nonselective phosphodiesterase inhibitor. It is approved for use as an anti-inflammatory in Japan.
    Fórmula:C14H18N2O
    Pureza:99.83% - >99.99%
    Forma y color:White Solid
    Peso molecular:230.31
  • M1001

    CAS:
    <p>M1001 is a HIF-2α agonist.</p>
    Fórmula:C17H17N3O2S
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:327.4
  • Fomepizole hydrochloride

    CAS:
    <p>Fomepizole hydrochloride inhibits CYP2E1 and alcohol dehydrogenase, blocking toxic metabolites, and treats methanol/ethylene glycol poisoning.</p>
    Fórmula:C4H7ClN2
    Forma y color:Solid
    Peso molecular:118.56
  • (R)-GNE-140

    CAS:
    <p>(R)-GNE-140 (GNE-140) is an effective LDHA/LDHB inhibitor (IC50s: 3/5 nM) and is 18-fold more potent than S enantiomer.</p>
    Fórmula:C25H23ClN2O3S2
    Pureza:98.25% - 98.91%
    Forma y color:Solid
    Peso molecular:499.04
  • Calcitriol

    CAS:
    <p>Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM).</p>
    Fórmula:C27H44O3
    Pureza:98.81% - 99.64%
    Forma y color:Colorless Crystalline Solid Solid
    Peso molecular:416.64
  • TMS

    CAS:
    <p>TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).</p>
    Fórmula:C18H20O4
    Pureza:99.17% - 99.73%
    Forma y color:Solid
    Peso molecular:300.35
  • Balipodect

    CAS:
    <p>Balipodect (TAK063) is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is &gt;15000-fold over other PDEs.</p>
    Fórmula:C23H17FN6O2
    Pureza:98% - 99.79%
    Forma y color:Solid
    Peso molecular:428.42
  • N-Oxalylglycine

    CAS:
    <p>N-Oxalylglycine (Oxalylglycine) is a cell permeable inhibitor of α-ketoglutarate-dependent enzymes.</p>
    Fórmula:C4H5NO5
    Pureza:99.23%
    Forma y color:Colourless Solid
    Peso molecular:147.09
  • BVT-14225

    CAS:
    BVT-14225 is a selective 11β-Hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor (IC50=52 nM).
    Fórmula:C16H20ClN3O3S2
    Pureza:97.78%
    Forma y color:Solid
    Peso molecular:401.93
  • NL-1

    CAS:
    <p>NL-1 is a mitoNEET inhibitor with antileukemic effect.</p>
    Fórmula:C18H25NO3S
    Pureza:98.64%
    Forma y color:Solid
    Peso molecular:335.46
  • Lotamilast

    CAS:
    <p>Lotamilast (RVT-501) is a phosphodiesterase 4 (PDE-4) inhibitor (IC50: 2.8 nM) potentially for the treatment of atopic dermatitis.</p>
    Fórmula:C26H24N4O5
    Pureza:97.03% - 99.29%
    Forma y color:Solid
    Peso molecular:472.49
  • Calcineurin Autoinhibitory Peptide acetate


    <p>Calcineurin Autoinhibitory Peptide acetate is a selectivecalcineurin phosphatase inhibitor(IC50 ~ 10 μM).</p>
    Fórmula:C252H417N78O82S4
    Pureza:97.24%
    Forma y color:Solid
    Peso molecular:5979.74
  • 2,2'-Methylenebis(6-tert-butyl-4-methylphenol)

    CAS:
    <p>2,2′-Methylenbis(4-methyl-6-tert-butylphenol) ist ein Antioxidans aus der Gruppe der Bisphenole.</p>
    Fórmula:C23H32O2
    Pureza:99.74%
    Forma y color:White Solid Powder
    Peso molecular:340.50
  • 6-Phosphogluconic acid

    CAS:
    <p>6-Phosphogluconic acid competitively inhibits PGI with Ki: 0.048 mM for glucose 6-P, 0.042 mM for fructose 6-P.</p>
    Fórmula:C6H13O10P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:276.14
  • KY-226

    CAS:
    <p>KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,)</p>
    Fórmula:C27H31NO3S2
    Pureza:99.4%
    Forma y color:Solid
    Peso molecular:481.67
  • Biocytin

    CAS:
    <p>Biocytin, a D-biotin and L-lysine conjugate, maps brain connections via a secondary amide bond.</p>
    Fórmula:C16H28N4O4S
    Pureza:97.23%
    Forma y color:White Solid
    Peso molecular:372.48
  • Haloxyfop

    CAS:
    <p>(±)-Haloxyfop (Haloxyfop Acid) is a herbicide.</p>
    Fórmula:C15H11ClF3NO4
    Pureza:99.94% - >99.99%
    Forma y color:Solid
    Peso molecular:361.7
  • ML-095 hydrochloride

    CAS:
    ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.
    Fórmula:C13H15ClN2O3
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:282.72
  • TEPP-46

    CAS:
    <p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C17H16N4O2S2
    Pureza:98.21% - 98.77%
    Forma y color:Solid
    Peso molecular:372.46
  • A939572

    CAS:
    <p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of &lt;4 nM for mSCD1 and 37 nM for hSCD1.</p>
    Fórmula:C20H22ClN3O3
    Pureza:99.96% - ≥95%
    Forma y color:Solid
    Peso molecular:387.86
  • Fabomotizole hydrochloride

    CAS:
    <p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>
    Fórmula:C15H22ClN3O2S
    Pureza:99.54% - >99.99%
    Forma y color:Solid
    Peso molecular:343.87
  • 1-Ethynylnaphthalene

    CAS:
    <p>1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 IB1</p>
    Fórmula:C12H8
    Pureza:99.05%
    Forma y color:Yellow To Brown Liquid
    Peso molecular:152.19
  • Isavuconazole

    CAS:
    <p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>
    Fórmula:C22H17F2N5OS
    Pureza:99.74% - >99.99%
    Forma y color:Solid
    Peso molecular:437.47
  • Vardenafil hydrochloride trihydrate

    CAS:
    <p>Vardenafil hydrochloride trihydrate (BAY38-9456) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>
    Fórmula:C23H32N6O4S·HCl·3H2O
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:579.11
  • Bay K 8644

    CAS:
    <p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>
    Fórmula:C16H15F3N2O4
    Pureza:99.41%
    Forma y color:Yellow Powder
    Peso molecular:356.3
  • Levamlodipine besylate

    CAS:
    <p>Levamlodipine besylate, or S-amlodipine (CAS 103129-82-4), is the active enantiomer of amlodipine, used to treat hypertension and angina.</p>
    Fórmula:C26H31ClN2O8S
    Pureza:99.78% - 99.79%
    Forma y color:Solid
    Peso molecular:567.05
  • Tryptophan, N-indol-3-ylacetyl- (6CI)

    CAS:
    <p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>
    Fórmula:C21H19N3O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:361.4
  • Efonidipine

    CAS:
    Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.
    Fórmula:C34H38N3O7P
    Pureza:98.35% - 99.47%
    Forma y color:Solid
    Peso molecular:631.66
  • Lactisole

    CAS:
    <p>Lactisole (na-PMP) is an inhibitor of the glucose-sensing receptor</p>
    Fórmula:C10H11NaO4
    Pureza:99.9%
    Forma y color:White To Pale Cream Crystalline Solid
    Peso molecular:218.18
  • 2-Deoxy-2-sulfoamino-D-glucose sodium

    CAS:
    <p>2-Deoxy-2-sulfoamino-D-glucose sodium (GlcN-2S) is possible to effect reaction at arthritis.</p>
    Fórmula:C6H12NNaO8S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:281.22
  • Ziritaxestat

    CAS:
    <p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>
    Fórmula:C30H33FN8O2S
    Pureza:97% - 99.85%
    Forma y color:Solid
    Peso molecular:588.7
  • N-Valyltryptophan

    CAS:
    <p>N-Valyltryptophan (Val-trp) is an incomplete breakdown product of protein catabolism or protein digestion.</p>
    Fórmula:C16H21N3O3
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:303.36
  • 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine

    CAS:
    <p>1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.</p>
    Fórmula:C46H84NO8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:810.13
  • Dichlorphenamide

    CAS:
    <p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>
    Fórmula:C6H6Cl2N2O4S2
    Pureza:96.87% - 97.25%
    Forma y color:Needles From Dimethylsulfoxide + Water Solid
    Peso molecular:305.16
  • CP-91149

    CAS:
    <p>CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence of</p>
    Fórmula:C21H22ClN3O3
    Pureza:99.66% - 99.81%
    Forma y color:Solid
    Peso molecular:399.87
  • S29434

    CAS:
    <p>S29434 (NMDPEF) is a potent, competitiveinhibitor of quinone reductase 2 (QR2;IC50:5-16nM).</p>
    Fórmula:C21H18N4O3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:374.39
  • JNJ-1661010

    CAS:
    <p>JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows &gt;100-fold selectivity for FAAH-1 than FAAH-2.</p>
    Fórmula:C19H19N5OS
    Pureza:99.79% - 99.97%
    Forma y color:Solid
    Peso molecular:365.45
  • Cyclosporine

    CAS:
    <p>Cyclosporine is a calcineurin phosphatase pathway inhibitor, used as an immunosuppressant drug to prevent rejection in organ transplantation.</p>
    Fórmula:C62H111N11O12
    Pureza:99.68%
    Forma y color:White Powder
    Peso molecular:1202.61
  • n-acetylciprofloxacin

    CAS:
    <p>n-acetylciprofloxacin (3-Quinolinecarboxylic acid, 7-(4-acetyl-1-piperazinyl)-1-cyclopropyl-6-fluoro-1) is inhibitor of H37Rv.</p>
    Fórmula:C19H20FN3O4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:373.38
  • Fmoc-Phe(4-CN)-OH

    CAS:
    <p>Fmoc-Phe(4-CN)-OH is an N-Fmoc protected phenylalanine derivative and potentially useful synthetic intermediate</p>
    Fórmula:C25H20N2O4
    Pureza:99.45%
    Forma y color:White Powder
    Peso molecular:412.44
  • BMS-309403

    CAS:
    BMS309403 is a potent and selective inhibitor of adipocyte fatty acid binding protein aFABP.Cost-effective and quality-assured.
    Fórmula:C31H26N2O3
    Pureza:99.52% - 99.76%
    Forma y color:Solid
    Peso molecular:474.55
  • FT113

    CAS:
    <p>FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity</p>
    Fórmula:C22H20FN3O4
    Pureza:97.05%
    Forma y color:Solid
    Peso molecular:409.41
  • Doxercalciferol

    CAS:
    <p>Doxercalciferol, a synthetic vitamin D2, curbs parathyroid activity for treating secondary hyperparathyroidism and bone disorders.</p>
    Fórmula:C28H44O2
    Pureza:99.03% - 99.69%
    Forma y color:White Crystalline Powder
    Peso molecular:412.65
  • SEA0400

    CAS:
    <p>SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.</p>
    Fórmula:C21H19F2NO3
    Pureza:98.88% - 99.55%
    Forma y color:Solid
    Peso molecular:371.38
  • NCT-501 hydrochloride

    CAS:
    <p>NCT-501 hydrochloride: potent, selective ALDH1A1 inhibitor based on theophylline; IC50 of 40 nM; highly discriminant against other ALDHs.</p>
    Fórmula:C21H33ClN6O3
    Forma y color:Solid
    Peso molecular:452.98
  • Methyl 13-cis-4-Oxoretinoate

    CAS:
    <p>Methyl 13-cis-4-Oxoretinoate (13-cis-4-Oxo-retinoic acid Methyl Ester) is a retinoic acid metabolite in neuroblastoma.</p>
    Fórmula:C21H28O3
    Pureza:96.6% - 99.08%
    Forma y color:Solid
    Peso molecular:328.45
  • VAS2870

    CAS:
    VAS2870 is an inhibitor of NADPH oxidase (NOX).
    Fórmula:C18H12N6OS
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:360.39
  • PF-8380 hydrochloride

    CAS:
    <p>PF-8380 hydrochloride is a powerful inhibitor of autotaxin, exhibiting an IC(50) of 2.8 nM in isolated enzyme assays and 101 nM in human whole blood.</p>
    Fórmula:C22H22Cl3N3O5
    Forma y color:Solid
    Peso molecular:514.79
  • Darexaban

    CAS:
    <p>Darexaban (YM-150) selectively inhibits Factor Xa, reducing clotting and risk of heart/stroke events.</p>
    Fórmula:C27H30N4O4
    Pureza:98.33%
    Forma y color:Solid
    Peso molecular:474.55
  • Panaxadiol

    CAS:
    <p>Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng.</p>
    Fórmula:C30H52O3
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:460.73
  • N-Biotinyl-6-aminohexanoic acid

    CAS:
    <p>N-Biotinyl-6-aminohexanoic acid (N-(+)-Biotinyl-6-aminohexanoic acid) can be used to perform N-terminal biotinylation.</p>
    Fórmula:C16H27N3O4S
    Pureza:98.61%
    Forma y color:Solid
    Peso molecular:357.47
  • Ponalrestat

    CAS:
    <p>Ponalrestat is an aldose reductase inhibitor.</p>
    Fórmula:C17H12BrFN2O3
    Pureza:97.34% - 99.86%
    Forma y color:Solid
    Peso molecular:391.19
  • 3-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one

    CAS:
    <p>DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 nM, respectively)</p>
    Fórmula:C18H13NO
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:259.3
  • 16α-Hydroxyprednisolone


    <p>16α-Hydroxyprednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonide</p>
    Fórmula:C21H28O6
    Pureza:99.75%
    Forma y color:White Solid
    Peso molecular:376.44
  • RS-25344

    CAS:
    <p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>
    Fórmula:C19H13N5O4
    Pureza:98.98%
    Forma y color:Solid
    Peso molecular:375.34
  • ML355

    CAS:
    <p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>
    Fórmula:C21H19N3O4S2
    Pureza:98.02% - 98.2%
    Forma y color:Solid
    Peso molecular:441.52
  • ZINC13466751

    CAS:
    <p>ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).</p>
    Fórmula:C20H21N5O2
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:363.41
  • IOX2

    CAS:
    <p>IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.</p>
    Fórmula:C19H16N2O5
    Pureza:98% - 99.59%
    Forma y color:Solid
    Peso molecular:352.34
  • Pranidipine

    CAS:
    <p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>
    Fórmula:C25H24N2O6
    Pureza:99.95%
    Forma y color:Yellow Solid
    Peso molecular:448.47
  • ML-298

    CAS:
    <p>ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).</p>
    Fórmula:C22H23F3N4O2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:432.44
  • Icerguastat

    CAS:
    Icerguastat (IFB-088) is a selective inhibitor of holophosphatase. Icerguastat selectively inhibited a regulatory subunit of protein phosphatase 1 in vivo.
    Fórmula:C8H9ClN4
    Pureza:97.95%
    Forma y color:Solid
    Peso molecular:196.64
  • Fomepizole

    CAS:
    <p>Fomepizole (4-Methylpyrazole), a competitive inhibitor of alcohol dehydrogenase, is used as an antidote in methanol or ethylene glycol poisoning.</p>
    Fórmula:C4H6N2
    Pureza:98.1% - 99.94%
    Forma y color:Yellow <13°C Solid >13°C Liquid
    Peso molecular:82.1
  • Z-HA155

    CAS:
    <p>Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.</p>
    Fórmula:C24H19BFNO5S
    Pureza:99.18%
    Forma y color:Solid
    Peso molecular:463.29
  • Antimalarial agent 14

    CAS:
    <p>Antimalarial agent 14 (NSC-102533) is a bioactive chemical.</p>
    Fórmula:C16H10O3
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:250.25
  • N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine

    CAS:
    <p>Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.</p>
    Fórmula:C23H28N6
    Pureza:98.35%
    Forma y color:Solid
    Peso molecular:388.51
  • 1-Naphthyl phosphate potassium salt

    CAS:
    <p>1-Naphthyl phosphate potassium salt inhibits non-specific phosphatase.</p>
    Fórmula:C10H7K2O4P
    Pureza:99%
    Forma y color:Solid
    Peso molecular:300.33
  • MLCK inhibitor peptide 18 acetate


    <p>MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.</p>
    Fórmula:C62H109N23O13
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:1384.67
  • Tazarotene

    CAS:
    <p>Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.</p>
    Fórmula:C21H21NO2S
    Pureza:97.01% - 99.14%
    Forma y color:White Solid
    Peso molecular:351.46
  • Inosine

    CAS:
    <p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>
    Fórmula:C10H12N4O5
    Pureza:99.51% - 99.89%
    Forma y color:Solid
    Peso molecular:268.23
  • Alkaline Phosphatase

    CAS:
    <p>Alkaline phosphatase is a membrane-bound glycoprotein that catalyzes the hydrolysis of phosphate monoesters under alkaline conditions. High-Quality, Low-Cost!</p>
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:N/A
  • YM-750

    CAS:
    <p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>
    Fórmula:C31H36N2O
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:452.63
  • Bepridil hydrochloride

    CAS:
    <p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>
    Fórmula:C24H35ClN2O
    Pureza:99.45% - 99.68%
    Forma y color:Solid
    Peso molecular:403
  • ND-646

    CAS:
    <p>ND-646 is an orally bioavailable and allosteric inhibitor of the ACC enzymes ACC1 and ACC2(IC50s of 3.5 nM and 4.1 nM for recombinant hACC1 and hACC2,</p>
    Fórmula:C28H32N4O7S
    Pureza:98.64%
    Forma y color:Solid
    Peso molecular:568.64
  • GEBR-7b

    CAS:
    <p>GEBR-7b (3-(Cyclopentyloxy)-4-methoxybenzaldehyde) is a phosphodiesterase-4 (PDE4) inhibitor.</p>
    Fórmula:C13H16O3
    Pureza:99.533%
    Forma y color:Solid
    Peso molecular:220.26
  • Tetrahydropapaverine hydrochloride

    CAS:
    <p>Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.</p>
    Fórmula:C20H26ClNO4
    Pureza:99.08%
    Forma y color:White Crystal Powder
    Peso molecular:379.878
  • Tropifexor

    CAS:
    <p>Tropifexor (LJN452) is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM.</p>
    Fórmula:C29H25F4N3O5S
    Pureza:99.3% - 99.85%
    Forma y color:Solid
    Peso molecular:603.58
  • CVT-2738

    CAS:
    <p>CVT-2738 (RS-94287) is a metabolite of Ranolazine. Ranolazine is a partial fatty acid oxidation (pFOX) inhibitor and anti-anginal drug.</p>
    Fórmula:C14H21N3O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:247.34
  • BAY-218

    CAS:
    <p>Bindarit (AF2838) is an aryl hydrocarbon receptor (AHR) antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C20H17ClFN3O3
    Pureza:99.46% - 99.85%
    Forma y color:Solid
    Peso molecular:401.82
  • Fmoc-N-Me-Leu-OH

    CAS:
    Fmoc-N-Me-Leu-OH is available for the peptide-coupling reaction.
    Fórmula:C22H25NO4
    Pureza:99.51%
    Forma y color:White Powder
    Peso molecular:367.44
  • SR33805

    CAS:
    <p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>
    Fórmula:C32H40N2O5S
    Pureza:99.15%
    Forma y color:Solid
    Peso molecular:564.74
  • Angiotensin I (human, mouse, rat)

    CAS:
    <p>Angiotensin I (human, mouse, rat) is the precursor to the vasoconstrictor peptide angiotensin II, cleaved by the angiotensin-converting enzyme (ACE).</p>
    Fórmula:C62H89N17O14
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1296.48
  • 4-Methylumbelliferyl-β-D-Glucopyranoside

    CAS:
    <p>4-Methylumbelliferyl-β-D-Glucopyranoside (4-MU-GLU) is used in the GCase activity assay based on the catalytic hydrolysis of 4-methylumbelliferyl β-D-</p>
    Fórmula:C16H18O8
    Pureza:99.89%
    Forma y color:White Powder
    Peso molecular:338.31
  • BMS-823778 hydrochloride

    CAS:
    <p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>
    Fórmula:C18H19Cl2N3O
    Forma y color:Solid
    Peso molecular:364.27
  • 4-Nonylphenylboronic acid

    CAS:
    <p>4-Nonylphenylboronic acid is a inhibitor of FAAH.</p>
    Fórmula:C15H25BO2
    Pureza:97.63%
    Forma y color:Solid
    Peso molecular:248.17
  • 1,2-Didecanoyl-sn-glycero-3-phosphocholi

    CAS:
    <p>1,2-Didecanoyl PC: synthetic phospholipid aiding peptide drug and insulin absorption.</p>
    Fórmula:C28H56NO8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:565.72
  • Turofexorate Isopropyl

    CAS:
    <p>Turofexorate Isopropyl (XL335) is a potent, selective, and orally bioavailable FXR agonist with EC50 of 4 nM</p>
    Fórmula:C25H24F2N2O3
    Pureza:98.55% - 99.73%
    Forma y color:Solid
    Peso molecular:438.47
  • Idoxuridine hydrate

    CAS:
    <p>Idoxuridine (5-IUdR) blocks DNA polymerase, treating herpes eye infections, with an IC50 of 4.3 μM against feline herpes.</p>
    Fórmula:C9H13IN2O6
    Forma y color:Solid
    Peso molecular:372.115
  • Tebufenpyrad

    CAS:
    <p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>
    Fórmula:C18H24ClN3O
    Pureza:98.63% - 99.16%
    Forma y color:Solid
    Peso molecular:333.86
  • Atglistatin

    CAS:
    <p>Atglistatin: ATGL inhibitor, IC50 ~0.7 μM, inhibits lipolysis, non-toxic up to 50 μM.</p>
    Fórmula:C17H21N3O
    Pureza:97.2% - 99.01%
    Forma y color:Solid
    Peso molecular:283.37
  • SR9011 hydrochloride

    CAS:
    <p>SR9011 hydrochloride is a REV-ERBα/β agonist, exhibiting an IC50 value of 790 nM for REV-ERBα and 560 nM for REV-ERBβ.</p>
    Fórmula:C23H32Cl2N4O3S
    Forma y color:Solid
    Peso molecular:515.49
  • Tauro-Obeticholic acid

    CAS:
    <p>Tauro-Obeticholic acid is an active Obeticholic acid metabolite. Obeticholic acid is an orally bioavailable agonist of farnesoid-X receptor (FXR).</p>
    Fórmula:C28H49NO6S
    Pureza:99.74% - 99.82%
    Forma y color:Solid
    Peso molecular:527.76
  • 7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine

    CAS:
    <p>7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).</p>
    Fórmula:C15H16N4
    Pureza:99.22%
    Forma y color:Solid
    Peso molecular:252.31
  • Kresoxim-Methyl

    CAS:
    <p>Kresoxim-methyl is a strobilurin fungicide,inhibits conidial germination of V. inaequalis isolates from apple orchards .</p>
    Fórmula:C18H19NO4
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:313.35
  • TM5007

    CAS:
    <p>TM5007 is a poent inhibitor of plasminogen activator inhibitor-1 (PAI-1; IC50 of 29 uM).</p>
    Fórmula:C24H20N2O6S4
    Pureza:96.91%
    Forma y color:Solid
    Peso molecular:560.69
  • Gcase activator 1

    CAS:
    <p>Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator.</p>
    Fórmula:C20H30N4O2
    Pureza:99.25% - 99.31%
    Forma y color:Solid
    Peso molecular:358.48
  • Tempol

    CAS:
    <p>Tempol (Tanol) is a superoxide scavenger. It has anti-inflammatory, neuroprotective and analgesic effects.</p>
    Fórmula:C9H18NO2
    Pureza:97% - 99.74%
    Forma y color:4-Hydroxy-Tempo Appears As Orange Flakes Solid Flakes
    Peso molecular:172.25
  • Monobenzyl phthalate

    CAS:
    <p>Monobenzyl phthalate (Phthalic Acid Monobenzyl Ester) is Phthalate metabolite.</p>
    Fórmula:C15H12O4
    Pureza:99.11% - 99.38%
    Forma y color:Solid
    Peso molecular:256.25
  • 6-Aminonicotinamide

    CAS:
    <p>6-Aminonicotinamide (6-AN) is a well-established inhibitor of the NADP+-dependent enzyme.</p>
    Fórmula:C6H7N3O
    Pureza:98.99% - 99.4%
    Forma y color:Physical Description White Crystalline Solid (Ntp 1992)
    Peso molecular:137.14
  • 2-Ketoglutaric acid

    CAS:
    <p>2-Ketoglutaric acid is a reversible inhibitor of tyrosinase (IC50=15 mM). 2-Ketoglutaric acid is an intermediate of the Krebs cycle. High-Quality, Low-Cost!</p>
    Fórmula:C5H6O5
    Pureza:99.28%
    Forma y color:Solid
    Peso molecular:146.1
  • Orthanilamide

    CAS:
    Orthanilamide (Orthanilamide) is a molecule containing the sulfonamide functional group attached to an aniline.
    Fórmula:C6H8N2O2S
    Pureza:99.72% - 99.96%
    Forma y color:White To Pale Cream Crystalline Powder Or Crystals
    Peso molecular:172.2
  • Homo Sildenafil

    CAS:
    <p>Homo Sildenafil is an analog of Sildenafil, It acts as a phosphodiesterase inhibitor.</p>
    Fórmula:C23H32N6O4S
    Pureza:99.88%
    Forma y color:White Solid
    Peso molecular:488.6
  • Dorzolamide hydrochloride

    CAS:
    <p>Dorzolamide hydrochloride (MK507 hydrochloride) is the hydrochloride salt form of dorzolamide, an inhibitor of carbonic anhydrase, a zinc-containing enzyme that</p>
    Fórmula:C10H17ClN2O4S3
    Pureza:99.48% - 99.67%
    Forma y color:White Off-White Crystalline Powder
    Peso molecular:360.9
  • HET0016

    CAS:
    <p>HET0016: potent, selective 20-HETE synthase/CYP450 inhibitor; IC50s: 17.7-20.6 nM; inhibits angiogenesis, tumor growth.</p>
    Fórmula:C12H18N2O
    Pureza:98.84%
    Forma y color:Solid
    Peso molecular:206.28
  • TPPU

    CAS:
    <p>TPPU is a potent inhibitor of both human and mouse sEH (IC50 of 3.7 and 2.8 nM, respectively)</p>
    Fórmula:C16H20F3N3O3
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:359.34
  • SR9243

    CAS:
    <p>SR9243, an LXR inverse agonist, can induce LXR-corepressor interaction; shows anticancer activity and selectively targets the lipogenesis and Warburg effect.</p>
    Fórmula:C31H32BrNO4S2
    Pureza:98% - 99.03%
    Forma y color:Solid
    Peso molecular:626.62
  • N-desmethylmirtazapine

    CAS:
    N-desmethylmirtazapine: mirtazapine metabolite; used for anxiety, sleep, nausea, appetite.
    Fórmula:C16H17N3
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:251.33