
GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.020 productos)
- Receptor de adenosina(249 productos)
- Receptor adrenérgico(3.022 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(60 productos)
- CXCR(157 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(216 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(442 productos)
- Receptor de endotelina(83 productos)
- Receptor GNRH(83 productos)
- GPCR19(33 productos)
- GRK(32 productos)
- GTPasa(23 productos)
- Receptor de glucagón(195 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(322 productos)
- PAFR(13 productos)
- PKA(51 productos)
- Receptor S1P(17 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
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Se han encontrado 5938 productos de "GPCR / proteína G"
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Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Fórmula:C23H29ClFN3O4Pureza:99.77%Forma y color:White To Slightly Biege Powder SolidPeso molecular:465.95DPTN dihydrochloride
CAS:DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Fórmula:C22H20Cl2N4OSPureza:99.95%Forma y color:SoildPeso molecular:459.39LCKLSL hydrochloride
LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.Fórmula:C30H58ClN7O8SPureza:98.02% - 99.31%Forma y color:SolidPeso molecular:712.34Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Fórmula:C16H21N3·HClPureza:99.54% - 99.81%Forma y color:White SolidPeso molecular:291.82Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Forma y color:SolidPeso molecular:1347.5Gevotroline
CAS:Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.Fórmula:C19H20FN3Pureza:99.45%Forma y color:SolidPeso molecular:309.38Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Fórmula:C163H273N49O44Pureza:96.87%Forma y color:SolidPeso molecular:3623.21ESI-05
CAS:ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.Fórmula:C16H18O2SPureza:97.22%Forma y color:SolidPeso molecular:274.38Dexpramipexole dihydrochloride
CAS:Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamineFórmula:C10H19Cl2N3SPureza:99.75% - 99.88%Forma y color:SolidPeso molecular:284.25Anamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Fórmula:C31H42N6O3Pureza:99.35% - 99.94%Forma y color:SolidPeso molecular:546.7PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Fórmula:C31H30FN5O4Pureza:97.19% - 99.56%Forma y color:SolidPeso molecular:555.6Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Pureza:SDS-PAGE:95% SEC-HPLC:98.90%Forma y color:LiquidPeso molecular:146.43 kDaDesipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Fórmula:C18H23ClN2Pureza:99.58% - 99.94%Forma y color:White To Off-White PowderPeso molecular:302.842Sergliflozin A
CAS:Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.Fórmula:C20H24O7Pureza:99.71%Forma y color:SolidPeso molecular:376.4Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Fórmula:C24H28N2O3Pureza:99.60% - 99.97%Forma y color:White Crystalline PowderPeso molecular:392.49Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Fórmula:C19H23NO·HClPureza:98.72%Forma y color:SolidPeso molecular:317.85Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Fórmula:C17H20N4SPureza:99.86% - ≥95%Forma y color:Yellowish Crystalline PowderPeso molecular:312.43Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Fórmula:C18H30ClN3O5Pureza:99.53% - 99.61%Forma y color:White SolidPeso molecular:403.91Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:99.87% - 99.93%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFórmula:C32H40ClNO4Pureza:>99.99%Forma y color:White Crystalline PowderPeso molecular:538.12Fenspiride hydrochloride
CAS:Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Forma y color:SolidPeso molecular:296.79Citalopram hydrobromide
CAS:Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFórmula:C20H22BrFN2OPureza:99.81%Forma y color:White Crystalline PowderPeso molecular:405.304Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Forma y color:SolidPeso molecular:643.71Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Fórmula:C19H21N·HClPureza:98.54% - 99.98%Forma y color:SolidPeso molecular:299.84Filorexant
CAS:Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).Fórmula:C24H25FN4O2Pureza:98.88%Forma y color:SolidPeso molecular:420.48Indusatumab
CAS:<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Pureza:> 95% - > 95%Forma y color:LiquidPeso molecular:145.18 kDaJNJ-18038683
CAS:JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Fórmula:C26H28ClN3O7Pureza:97.29%Forma y color:SolidPeso molecular:529.97Erenumab
CAS:Erenumab: human antibody blocking CGRP receptors to prevent migraines.Pureza:99.43% (SEC-HPLC) - > 95%Forma y color:LiquidPeso molecular:146.2 kDaFluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Forma y color:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.58%Forma y color:SoildPeso molecular:784.58Urapidil hydrochloride
CAS:Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Fórmula:C20H29N5O3·HClPureza:99.58%Forma y color:White Or Off-White Crystalline PowderPeso molecular:423.94Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Fórmula:C18H25ClN4OPureza:99.88% - 99.93%Forma y color:White To Off-White Crystalline SolidPeso molecular:348.87NF-56-EJ40 hydrochloride
CAS:NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.Fórmula:C27H31Cl2N3O3Pureza:99.33%Forma y color:SoildPeso molecular:516.46Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Fórmula:C17H18F3NOPureza:99.07% - 99.28%Forma y color:SolidPeso molecular:309.33Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Fórmula:C17H21ClN2SPureza:99.90%Forma y color:SolidPeso molecular:320.88Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Fórmula:C23H30FN3Pureza:99.85%Forma y color:SolidPeso molecular:367.5Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Forma y color:SolidPeso molecular:408.33Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Fórmula:C14H15Cl2NSPureza:99.85% - >99.99%Forma y color:White PowderPeso molecular:300.25PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Fórmula:C25H37Cl2N3O2Pureza:99.68%Forma y color:SolidPeso molecular:482.49Palonosetron hydrochloride
CAS:Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Forma y color:White SolidPeso molecular:332.87Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Fórmula:C26H27N5O2Pureza:99.61%Forma y color:Light Yellow SolidPeso molecular:441.52Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Fórmula:C9H11NO3·HClPureza:99.94%Forma y color:SolidPeso molecular:217.65Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Pureza:97.76%Forma y color:SoildAcebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Fórmula:C18H29ClN2O4Pureza:99.92% - >99.99%Forma y color:White Or Slightly Off-White Crystalline Powder SolidPeso molecular:372.89Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Fórmula:C28H32ClN3O8SPureza:99.78%Forma y color:Off-White PowderPeso molecular:606.09Rimonabant hydrochloride
CAS:Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。Fórmula:C22H22Cl4N4OPureza:98.24% - 99.5%Forma y color:Off-White To White Crystalline PowderPeso molecular:500.25Ondansetron hydrochloride dihydrate
CAS:Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Fórmula:C18H19N3O·HCl·2H2OPureza:99.92%Forma y color:White Crystal PowderPeso molecular:365.86Indacaterol maleate
CAS:Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.Fórmula:C28H32N2O7Pureza:99.03% - 99.67%Forma y color:SolidPeso molecular:508.56Dopexamine hydrochloride
CAS:Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.Fórmula:C22H34Cl2N2O2Pureza:98.55%Forma y color:SolidPeso molecular:429.422-Bromo-6-methoxynaphthalene
CAS:2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Fórmula:C11H9BrOPureza:98.51%Forma y color:White To Off-White PowderPeso molecular:237.09CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Fórmula:C15H18Cl2N4OPureza:99.5%Forma y color:SolidPeso molecular:341.24Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Fórmula:C18H18ClNS·HClPureza:99.76%Forma y color:White PowderPeso molecular:352.32Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Fórmula:C26H35NO7Pureza:98.53% - 99.43%Forma y color:CoaPeso molecular:473.57Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Fórmula:C19H31ClF3NO3Pureza:99.55%Forma y color:SolidPeso molecular:413.9Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Fórmula:C19H21NSPureza:99.93%Forma y color:SolidPeso molecular:295.44Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Forma y color:White Or Almost White Crystalline PowderPeso molecular:463.79CYM 50769
CAS:CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).Fórmula:C24H17ClN2O3Pureza:98% - 99.08%Forma y color:SolidPeso molecular:416.86Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Forma y color:White Crystalline PowderPeso molecular:313.86Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Forma y color:SolidPeso molecular:307.39ML-180
CAS:ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .Fórmula:C20H25ClN4O2Pureza:99.74%Forma y color:SolidPeso molecular:388.89hGPR91 antagonist 1
CAS:hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).Fórmula:C31H23F4N3OPureza:98.89%Forma y color:SolidPeso molecular:529.53Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Fórmula:C19H27N5O4·HClPureza:99.78%Forma y color:White To Off-White SolidPeso molecular:425.91KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Fórmula:C26H40N4O8Pureza:98.46%Forma y color:SolidPeso molecular:536.62Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Forma y color:SolidPeso molecular:449.4Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:98.55%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Forma y color:Colorless To Pink SolidPeso molecular:495.53Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Forma y color:White Or Kind Of White PowderPeso molecular:287.36Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Forma y color:White To Off-White Crystalline PowderPeso molecular:383.51Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Fórmula:C19H26ClNO2Pureza:99.35%Forma y color:SolidPeso molecular:335.87Noradrenaline bitartrate
CAS:Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.Fórmula:C12H19NO10Pureza:99.53% - >99.99%Forma y color:SolidPeso molecular:337.28Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H11ClFNO2Pureza:99.98%Forma y color:SoildPeso molecular:231.65Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Fórmula:C18H26ClN3O3Pureza:>99.99%Forma y color:SolidPeso molecular:367.87Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Forma y color:White Crystalline PowderPeso molecular:341.43Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Fórmula:C25H37NO4Pureza:99.2% - 99.9%Forma y color:SolidPeso molecular:415.57Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Forma y color:PowderPeso molecular:522.55Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFórmula:C17H19N3·HClPureza:98% - 99.53%Forma y color:White Or Almost White Crystalline PowderPeso molecular:301.82Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Fórmula:C13H16N4Pureza:98.34% - 99.73%Forma y color:SolidPeso molecular:228.29Senktide acetate
Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.Fórmula:C42H59N7O13SPureza:98.26%Forma y color:SolidPeso molecular:902.02Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Forma y color:Colourless Flake Crystalline SolidPeso molecular:448.39Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Forma y color:SolidPeso molecular:461.81(3aR,9aR)-Fluparoxan
CAS:<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H10FNO2Pureza:97.82%Forma y color:SoildPeso molecular:195.19Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Fórmula:C17H22Cl2N4Pureza:99.79%Forma y color:SolidPeso molecular:353.29AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Fórmula:C17H14O5Pureza:97.59%Forma y color:SolidPeso molecular:298.29Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFórmula:C10H13NO4Pureza:98.95% - 99.86%Forma y color:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Forma y color:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:99.08%Forma y color:SolidPeso molecular:631.59Olinciguat
CAS:Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.Fórmula:C21H16F5N7O3Pureza:99.33% - 99.71%Forma y color:SolidPeso molecular:509.39Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Fórmula:C9H15ClNO5PPureza:99.84%Forma y color:SolidPeso molecular:283.65MP-A08
CAS:MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.Fórmula:C27H25N3O4S2Pureza:97.44%Forma y color:SolidPeso molecular:519.64Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Fórmula:C16H26ClNO3Pureza:99.94% - ≥95%Forma y color:SolidPeso molecular:315.84YNT-185
CAS:YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,Fórmula:C33H37N5O5SPureza:99.67%Forma y color:SolidPeso molecular:615.74Phenothiazine
CAS:Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.Fórmula:C12H9NSPureza:99.95%Forma y color:Yellow Solid PelletsPeso molecular:199.27NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Fórmula:C20H24ClN3OPureza:99.56%Forma y color:SolidPeso molecular:357.88Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Forma y color:SolidPeso molecular:266.55Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Forma y color:SolidPeso molecular:395.43Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Forma y color:SolidPeso molecular:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Fórmula:C21H24ClNOPureza:99.77% - >99.99%Forma y color:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Forma y color:SolidPeso molecular:384.9Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Fórmula:C31H38N2OPureza:97.49%Forma y color:SolidPeso molecular:454.65

