
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5593 produits trouvés pour "Apoptose"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
PF-573228
CAS :<p>PF-573228 is an ATP-competitive FAK inhibitor. In a cell-free assay, the IC50 of FAK is 4 nM.</p>Formule :C22H20F3N5O3SDegré de pureté :96.58% - 99.51%Couleur et forme :SolidMasse moléculaire :491.49PF-3758309 dihydrochloride
<p>PF-3758309 dihydrochloride is a potent PAK4 inhibitor (Kd = 2.7 nM, Ki = 18.7 nM), oral, ATP-competitive; blocks cell growth, induces apoptosis.</p>Formule :C25H32Cl2N8OSCouleur et forme :SolidMasse moléculaire :563.55Voreloxin hydrochloride
CAS :<p>Voreloxin hydrochloride (SNS-595 hydrochloride) is a potent inhibitor of Topoisomerase II with broad-spectrum anti-tumor activity.</p>Formule :C18H20ClN5O4SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :437.9Pioglitazone potassium
CAS :<p>Pioglitazone potassium is an oral PPARγ agonist with EC50 of 0.93 μM (human) and 0.99 μM (mouse), used in diabetes research.</p>Formule :C19H19KN2O3SCouleur et forme :SolidMasse moléculaire :394.53Atezolizumab
CAS :<p>Atezolizumab is an antibody inhibitor, a humanized monoclonal antibody, IgG1, which targets PD-L1. Atezolizumab has antitumor effect. Cost-effective and quality-assured.</p>Degré de pureté :95.10% - 99.3% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145 kDaBufotalin
CAS :<p>1. Bufotalin (Bufotaline)e is a kind of poisonous secretions of toads.</p>Formule :C26H36O6Degré de pureté :99.45% - 99.91%Couleur et forme :White To Off-White SolidMasse moléculaire :444.56Osthole
CAS :<p>Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.</p>Formule :C15H16O3Degré de pureté :99.93% - 99.96%Couleur et forme :Fine White PowderMasse moléculaire :244.29Alantolactone
CAS :<p>Alantolactone is a selective inhibitor of STAT3 that induces cancer-associated apoptosis and has antitumor activity.Cost-effective and quality-assured.</p>Formule :C15H20O2Degré de pureté :99.02% - 99.66%Couleur et forme :Crystalline PowderMasse moléculaire :232.32Bomedemstat
CAS :<p>Bomedemstat (IMG-7289),Irreversible LSD1 inhibitor. Active in MPN models. Antineoplastic effects. Used in AML and myelofibrosis research.</p>Formule :C28H34FN7O2Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :519.61Nodinitib-1
CAS :<p>Nodinitib-1 (CID-1088438) is a potent and selective NOD1 inhibitor with an IC50 of 0.56 μM.</p>Formule :C14H13N3O2SDegré de pureté :99.97% - >99.99%Couleur et forme :SolidMasse moléculaire :287.34Isoliensinine
CAS :<p>Isoliensinine (Isoliensinin) is a natural product, a bisbenzylisoquinoline alkaloid. Isoliensinine has antitumor and antioxidant effects. Cost effective and quality assured.</p>Formule :C37H42N2O6Degré de pureté :98.53% - 99.79%Couleur et forme :SolidMasse moléculaire :610.74A-1331852
CAS :<p>A-1331852 is a potent and selectiveBCL-XL inhibitor and may be useful in the treatment of cancer, immune and autoimmune diseases.</p>Formule :C38H38N6O3SDegré de pureté :98.15% - >99.99%Couleur et forme :SolidMasse moléculaire :658.81Guggulsterone
CAS :<p>Guggulsterone (Guggulsterone E&Z) E&Z is a 3-hydroxy steroid. It has a role as an androgen.</p>Formule :C21H28O2Degré de pureté :99.4% - 99.8%Couleur et forme :Light Yellow PowderMasse moléculaire :312.45BV6
CAS :<p>BV6 is an antagonist of c-IAP1 and XIAP, members of the inhibitors of apoptosis (IAP) family.</p>Formule :C70H96N10O8Degré de pureté :97.46% - 99.82%Couleur et forme :SolidMasse moléculaire :1205.57Calcimycin
CAS :<p>Calcimycin (A-23187) is a polyether antibiotic that transports Ca²⁺, uncouples phosphorylation, and inhibits ATPase in mitochondria.</p>Formule :C29H37N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :523.62Licochalcone D
CAS :<p>Licochalcone D may treat melanoma and heart injury, halt cell spread, and reduce inflammation and allergies.</p>Formule :C21H22O5Degré de pureté :99.03% - 99.9%Couleur et forme :SolidMasse moléculaire :354.4GSK1324726A
CAS :<p>GSK1324726A (I-BET726) is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM).</p>Formule :C25H23ClN2O3Degré de pureté :98.34% - 99.85%Couleur et forme :SolidMasse moléculaire :434.91TCS-PIM-1-4a
CAS :<p>SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).</p>Formule :C11H6F3NO2SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :273.23Dihydrorotenone
CAS :<p>Dihydrorotenone is a potent mitochondrial inhibitor and probably induces Parkinsonian syndrome.</p>Formule :C23H24O6Degré de pureté :98.98% - 99.58%Couleur et forme :SolidMasse moléculaire :396.43Methyl protodioscin
CAS :<p>Methyl protodioscin boosts HDL, lowers LDL and triglycerides, has anti-cancer effects, and promotes apoptosis via mitochondrial pathways.</p>Formule :C52H86O22Degré de pureté :99.308% - 99.73%Couleur et forme :SolidMasse moléculaire :1063.23Flurbiprofen Axetil
CAS :<p>Flurbiprofen Axetil (Lipfen) is an anti-inflammatory used as an analgesic.</p>Formule :C19H19FO4Degré de pureté :97.58% - 98%Couleur et forme :SolidMasse moléculaire :330.35NSC 73150
CAS :<p>6-Methyl-1H-pyrimidin-4-one (NSC 73150) shows antitumor effects, impeding growth in breast, lung, liver cancer, and inducing apoptosis.</p>Formule :C12H12N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :244.254E1rcat
CAS :<p>4E1RCat is a dual inhibitor of eIF4E:eIF4 g and eIF4E:4E-BP1 interaction. And it inhibits the binding of eIF4 g to eIF4E with IC50 of 3.2 μM.</p>Formule :C28H18N2O6Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :478.45pimpinellin
CAS :<p>Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity.</p>Formule :C13H10O5Degré de pureté :99.85% - ≥95%Couleur et forme :SolidMasse moléculaire :246.22DAPT
CAS :<p>DAPT (LY-374973) is a γ-secretase inhibitor that inhibits total Aβ and Aβ42 (IC50=115/200 nM) and is orally active.</p>Formule :C23H26F2N2O4Degré de pureté :98.06% - 99.81%Couleur et forme :White SolidMasse moléculaire :432.46Bay 11-7085
CAS :<p>Bay 11-7085 can irreversibly inhibit the IκBα phosphorylation induced by TNFα (IC50: 10 μM).</p>Formule :C13H15NO2SDegré de pureté :99.76% - 99.94%Couleur et forme :White SolidMasse moléculaire :249.33UNC1215
CAS :<p>UNC1215, a potent MBT antagonist, targets L3MBTL3 with high selectivity (IC50: 40 nM, Kd: 120 nM, 50x versus MBT family).</p>Formule :C32H43N5O2Degré de pureté :98% - 99.04%Couleur et forme :SolidMasse moléculaire :529.72AES-350
CAS :<p>AES-350, an HDAC6 inhibitor (IC50: 0.0244 μM), also targets HDAC-3, -8, -11, induces AML cell apoptosis, and aids AML research.</p>Formule :C18H20N2O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :312.36N-Formyl-Met-Leu-Phe
CAS :<p>N-Formyl-Met-Leu-Phe (N-Formyl-MLF) (fMLF) is a synthetic peptide that acts as an agonist at formyl peptide receptors (FPR; Ki = 0.8 pM).</p>Formule :C21H31N3O5SDegré de pureté :98.69% - ≥95%Couleur et forme :SolidMasse moléculaire :437.55Rotundic acid
CAS :<p>Rotundic acid fights various cancers: HepG2, A375, NCI-H446, MCF-7, and HT-29.</p>Formule :C30H48O5Degré de pureté :96.91% - 99.97%Couleur et forme :SolidMasse moléculaire :488.7Polyporenic acid C
CAS :<p>Polyporenic acid C shows inhibitory activity against human collagenase.</p>Formule :C31H46O4Degré de pureté :96.84% - 99.71%Couleur et forme :SolidMasse moléculaire :482.69RITA
CAS :<p>RITA (NSC-652287) forms DNA-DNA/protein cross-links without DNA breaks; disrupts p53/Mdm2 like nutlin-3.</p>Formule :C14H12O3S2Degré de pureté :98.49% - 99.55%Couleur et forme :SolidMasse moléculaire :292.37Danshensu
CAS :<p>Danshensu (Dan shen suan A) is an active ingredient of Salvia miltiorrhiza with wide cardiovascular benefit.</p>Formule :C9H10O5Degré de pureté :98.4% - 99.74%Couleur et forme :SolidMasse moléculaire :198.17Ketorolac
CAS :<p>Ketorolac (Acuvail) is an NSAID that blocks prostaglandin synthesis, related to heterocyclic acetic acids.</p>Formule :C15H13NO3Degré de pureté :99.68%Couleur et forme :White Crystalline Or White PowderMasse moléculaire :255.27ML162
CAS :<p>ML162 is a covalent glutathione peroxidase 4 (GPX4) inhibitor that induces ferroptosis. ML162 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C23H22Cl2N2O3SDegré de pureté :98.42% - 99.55%Couleur et forme :SolidMasse moléculaire :477.4Poziotinib
CAS :<p>Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).</p>Formule :C23H21Cl2FN4O3Degré de pureté :98.69% - 99.78%Couleur et forme :SolidMasse moléculaire :491.34BG45
CAS :<p>BG45 is an HDAC I type inhibitor with IC50 of 289 nM, 2.0 μM, 2.2 μM and >20 μM for HDAC3/1/2/6 in cell-free assays, respectively.</p>Formule :C11H10N4ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :214.22Thapsigargin
CAS :<p>Thapsigargin is a natural product, an inhibitor of sarcoplasmic/endoplasmic reticulum Ca2+ ATPase (SERCA) and an endoplasmic reticulum stress inducer.</p>Formule :C34H50O12Degré de pureté :99.07% - 99.3%Couleur et forme :Colourless FilmMasse moléculaire :650.75RAF265
CAS :<p>RAF265 (CHIR-265) inhibits C-Raf/B-Raf/V600E (IC50: 3-60 nM), blocks VEGFR2 (EC50: 30 nM), in Phase 2 trials.</p>Formule :C24H16F6N6ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :518.41Epieriocalyxin A
CAS :<p>Epieriocalyxin A can suppress Caco-2 colon cancer cell growth. It could be a potential drug for colon cancer therapy in the future.</p>Formule :C20H24O5Degré de pureté :97.00%Couleur et forme :SolidMasse moléculaire :344.4Helichrysetin
CAS :<p>Helichrysetin shows mild anti-HIV-1 activity and potential as an anticancer agent with cytotoxic effects on A549, MCF-7, Ca Ski, HT-29 cells.</p>Formule :C16H14O5Degré de pureté :96.32% - ≥95%Couleur et forme :SolidMasse moléculaire :286.28Flavokawain B
CAS :<p>Flavokawain B inhibits NO and PGE2, causes oxidative stress, and induces apoptosis, with potential for treating prostate cancer.</p>Formule :C17H16O4Degré de pureté :99.97% - >99.99%Couleur et forme :SolidMasse moléculaire :284.31Quinidine sulfate dihydrate
CAS :<p>Quinidine sulfate dihydrate (Pitayine Sodium) is a potent and selective cytochrome P450db inhibitor</p>Formule :C40H54N4O10SDegré de pureté :99.85%Couleur et forme :White To Light Yellow Crystal PowdeMasse moléculaire :782.9Paederosidic acid
CAS :<p>Paederosidic acid shows anti-tumor, anticonvulsant, and sedative properties, may treat epilepsy by modulating brain GABA and glutamate levels.</p>Formule :C18H24O12SDegré de pureté :98% - 99.56%Couleur et forme :SolidMasse moléculaire :464.44OsMundacetone
CAS :<p>OsMundacetone (4-(3,4-Dihydroxyphenyl)-3-buten-2-one) is a natual product isolated from Rhizoma osmundae.</p>Formule :C10H10O3Degré de pureté :99.59% - ≥95%Couleur et forme :SolidMasse moléculaire :178.18DL-Buthionine-(S,R)-sulfoximine
CAS :<p>DL-Buthionine-(S,R)-sulfoximine (Butionine sulfoximine) is an inhibitor of γ-glutamylcysteine synthetase for the treatment of solid tumors.</p>Formule :C8H18N2O3SDegré de pureté :98% - 99.64%Couleur et forme :White Fine PowderMasse moléculaire :222.31Orantinib
CAS :<p>Orantinib (NSC 702827) , a excellent effective against PDGFR autophosphorylation with Ki of 8 nM, also highly inhibits Flk-1 and FGFR1 trans-phosphorylation.</p>Formule :C18H18N2O3Degré de pureté :98.92% - 99.52%Couleur et forme :SolidMasse moléculaire :310.35Ginkgetin
CAS :<p>Ginkgetin: antiviral, antifungal, anti-inflammatory; COX-2 reducer; STAT3 inhibitor; pro-apoptotic in cancer; neuroprotective in Parkinson's.</p>Formule :C32H22O10Degré de pureté :98.63% - 99.94%Couleur et forme :SolidMasse moléculaire :566.51Valproic Acid
CAS :<p>Valproic Acid (2-Propylpentanoic Acid) is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels.</p>Formule :C8H16O2Degré de pureté :97.78% - 99%Couleur et forme :Colourless To Pale Yellow Liquid ViscousMasse moléculaire :144.21PRLX-93936
CAS :<p>PRLX-93936 is a selective Ras pathway protein inhibitor that modulates RAS/JNK pathway-associated protein phosphorylation, anticancer activity.</p>Formule :C21H24N4O2Couleur et forme :SolidMasse moléculaire :364.44PNU-74654
CAS :<p>PNU 74654 blocks β-catenin/Tcf4, disrupting Wnt signaling (Kd = 450 nM).</p>Formule :C19H16N2O3Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :320.34DD1
CAS :<p>DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.</p>Formule :C16H14N2O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :282.29SRS11-92
CAS :<p>SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1</p>Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.47Vanillyl Alcohol
CAS :<p>Vanillyl Alcohol (3-Methoxy-4-hydroxybenzyl alcohol) possesses anti-angiogenic, anticonvulsive, anti-inflammatory, anti-oxidant and anti-nociceptive activities.</p>Formule :C8H10O3Degré de pureté :97.02% - 98.42%Couleur et forme :Crystalline White To Off-White PowderMasse moléculaire :154.16Pyrogallol
CAS :<p>Pyrogallol (Piral) is a white crystalline powder and a powerful reducing agent prepared by heating gallic acid.</p>Formule :C6H6O3Degré de pureté :99.88%Couleur et forme :SoildMasse moléculaire :126.11NVP 231
CAS :<p>NVP-231 is a potent, specific and reversible CerK inhibitor(IC50=12±2 nM) that competitively inhibits ceramide binding to CerK.</p>Formule :C25H25N3O2SDegré de pureté :99.16% - ≥95%Couleur et forme :SolidMasse moléculaire :431.55Taurolidine
CAS :<p>Taurolidine is a synthetic taurine analog with antimicrobial and anti-neoplastic actions. It displays broad bactericidal and fungicidal activity.</p>Formule :C7H16N4O4S2Degré de pureté :99.79% - 99.81%Couleur et forme :SolidMasse moléculaire :284.36DC260126
CAS :<p>DC260126 is a small-molecule antagonist of FFA1 (GPR40)</p>Formule :C16H18FNO2SDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :307.38CCCP
CAS :<p>CCCP blocks STING activation, TBK1, IRF3 signaling, and IFN-β production by disrupting MMP.</p>Formule :C9H5ClN4Degré de pureté :97.15% - 99.64%Couleur et forme :Yellow To Orange PowderMasse moléculaire :204.62NSC 15364
CAS :<p>NSC 15364 (1,3-Bis(4-aminophenyl)urea) can be used for screening of ALR inhibitors by detection of hydrogen peroxide production Measured in Biochemical System.</p>Formule :C13H14N4ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :242.28W-7 hydrochloride
CAS :<p>W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride</p>Formule :C16H22Cl2N2O2SDegré de pureté :99.63%Couleur et forme :White Crystalline SolidMasse moléculaire :377.32Clobenpropit dihydrobromide
CAS :<p>Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)</p>Formule :C14H19Br2ClN4SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :470.7SCR130
CAS :<p>SCR130 (1,7,9-Triazaspiro[4.5]dec-1-ene-6,10-dione, 2,4-bis(4-chlorophenyl)-8-thioxo-) 是基于 SCR7 的 DNA 非同源末端连接抑制剂,可诱导细胞凋亡并,具有抗癌活性。 它特异性依赖连接酶 IV,抑制 DNA 的末端连接。</p>Formule :C19H13Cl2N3O2SDegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :418.3iCRT3
CAS :<p>iCRT3 is a Wnt and β-catenin-responsive transcription inhibitor.</p>Formule :C23H26N2O2SDegré de pureté :98.32% - 98.47%Couleur et forme :SolidMasse moléculaire :394.53Alvespimycin hydrochloride
CAS :<p>Alvespimycin hydrochloride (BMS 826476) is a potent HSP90 inhibitor with IC50 of 62 nM. Phase 2.</p>Formule :C32H48N4O8·HClDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :653.21Pembrolizumab
CAS :<p>Pembrolizumab (MK-3475) is a humanized monoclonal antibody.Cost-effective and quality-assured.</p>Degré de pureté :95% - 99.70%Couleur et forme :LiquidMasse moléculaire :149 kDaIITZ-01
CAS :<p>IITZ-01 is potent autophagy inhibitor with single-agent anticancer activity ( IC50 of 2.62 μM for PI3Kγ.)</p>Formule :C26H23FN8ODegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :482.513-Nitropropanoic acid
CAS :<p>3-Nitropropanoic acid (Bovinocidin) is an irreversible inhibitor of succinate dehydrogenase.</p>Formule :C3H5NO4Degré de pureté :98.35% - 99.94%Couleur et forme :Crystals From Chloroform Physical Description Golden Crystals (From Chloroform) (Ntp 1992)Masse moléculaire :119.08TM5441
CAS :<p>TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines with IC50 values ranging from 13.9 to 51.1 μM.Cost-effective and quality-assured.Cost-effective and quality-assured.</p>Formule :C21H17ClN2O6Degré de pureté :97.62% - 99.09%Couleur et forme :SolidMasse moléculaire :428.82Solamargine
CAS :<p>Solamargine, a steroidal alkaloid from Solanum nigrum, inhibits cancer cell growth and induces apoptosis.</p>Formule :C45H73NO15Degré de pureté :99.17% - 99.96%Couleur et forme :SolidMasse moléculaire :868.06Angiotensin II human
CAS :<p>Angiotensin II acts on AT1/AT2 receptors, 30% similar seven-transmembrane glycoproteins, converted from Ang I by ACE.</p>Formule :C50H71N13O12Degré de pureté :95% - >99.99%Couleur et forme :SolidMasse moléculaire :1046.18PD168393
CAS :<p>PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, FGFR, PDGFR, and insulin.</p>Formule :C17H13BrN4ODegré de pureté :99.13% - 99.83%Couleur et forme :SolidMasse moléculaire :369.22Mancozeb
CAS :<p>Mancozeb is a fungicide of ethylene-bis-dithiocarbamate.</p>Formule :C8H12MnN4S8ZnDegré de pureté :98%Couleur et forme :Grayish-Yellow PowderMasse moléculaire :541.08Sophocarpine
CAS :<p>Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.</p>Formule :C15H22N2ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :246.35CDPPB
CAS :<p>CDPPB is a modulator of mGluR5 positive allosteric(with an EC50 of 27 nM in Chinese hamster ovary cells expressing human mGluR5).</p>Formule :C23H16N4ODegré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :364.4Iproniazid
CAS :<p>Iproniazid is an irreversible monoamine oxidase inhibitor. It is used as an antidepressive agent.</p>Formule :C9H13N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.22CCPA
CAS :<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Formule :C15H20ClN5O4Degré de pureté :99.1%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8NUN82647
CAS :<p>NUN82647 (CU-242) is an Inhibitor of cell cycle at G2 phase, and apoptosis inducer.</p>Formule :C15H13N3O2SDegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :299.35Z-VAD(OMe)-FMK
CAS :<p>View and buy Z-VAD(OMe)-FMK from TargetMol.Z-VAD(OMe)-FMK is a cell-permeable and irreversible pan-caspase inhibitor.Cited in 10 publications.</p>Formule :C22H30FN3O7Degré de pureté :95.92% - 99.71%Couleur et forme :SolidMasse moléculaire :467.49Pevonedistat
CAS :<p>Pevonedistat (MLN4924) is a potent and selective NEDD8 activating enzyme (NAE) inhibitor (IC50=4.7 nM).</p>Formule :C21H25N5O4SDegré de pureté :95% - 99.92%Couleur et forme :SolidMasse moléculaire :443.521R,3S-RSL 3
CAS :<p>1R,3S-RSL 3 is a harmala alkaloid.</p>Formule :C23H21ClN2O5Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :440.88Amcasertib
CAS :<p>Amcasertib (BBI503) is an orally administered investigational agent designed to inhibit cancer stem cell pathways via targeting stemness kinases.</p>Formule :C31H33N5O2SDegré de pureté :97.56% - >99.99%Couleur et forme :SolidMasse moléculaire :539.69Isosorbide Mononitrate
CAS :<p>Isosorbide Mononitrate (Corangin) is a Nitrate Vasodilator, dilating the blood vessels so as to reduce the blood pressure.</p>Formule :C6H9NO6Degré de pureté :98.16%Couleur et forme :Isosorbide-5-Mononitrate Is A Crystalline Solid It Is Very Flammable And May Be Toxic By IngestionMasse moléculaire :191.14Romidepsin
CAS :<p>Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.</p>Formule :C24H36N4O6S2Degré de pureté :99.4% - 99.94%Couleur et forme :SolidMasse moléculaire :540.7Fluazinam
CAS :<p>Fluazinam: a pyridinamine fungicide, broad-spectrum, strongly inhibits S. sclerotiorum mycelial growth.</p>Formule :C13H4Cl2F6N4O4Degré de pureté :98% - 99.7%Couleur et forme :Light Yellow CrystalsMasse moléculaire :465.09Saquinavir
CAS :<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formule :C38H50N6O5Degré de pureté :99.50% - >99.99%Couleur et forme :SolidMasse moléculaire :670.84Tenilsetam
CAS :<p>Tenilsetam: an endonuclease, nootropic, AGE inhibitor potential for Alzheimer's.</p>Formule :C8H10N2OSDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :182.244-IBP
CAS :<p>4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .</p>Formule :C19H21IN2ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :420.29Lubiprostone
CAS :<p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>Formule :C20H32F2O5Degré de pureté :97.31% - 98.54%Couleur et forme :White Odorless Crystals Or Crystalline PowderMasse moléculaire :390.46RH01687
CAS :<p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>Formule :C12H9ClN6O2SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :336.76Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86Sodium benzoate
CAS :<p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>Formule :C7H5NaO2Degré de pureté :99.72%Couleur et forme :White Solid CrystallineMasse moléculaire :144.10HX 531
CAS :<p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>Formule :C29H29N3O4Degré de pureté :98.59% - 99.86%Couleur et forme :SolidMasse moléculaire :483.56Ceftiofur
CAS :<p>Ceftiofur is a semisynthetic antibiotic, with activity against various gram-positive/negative, anaerobic and aerobic bacteria encountered by domestic animals.</p>Formule :C19H17N5O7S3Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :523.56NSC 3852
CAS :<p>NSC 3852 is a potent inhibitor of histone deacetylase.</p>Formule :C9H6N2O2Degré de pureté :99.64%Couleur et forme :Slightly Yellow To Yellow-Green PowderMasse moléculaire :174.16ILK-IN-2
CAS :<p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>Formule :C30H30F3N5ODegré de pureté :99.30%Couleur et forme :SolidMasse moléculaire :533.59BMS202 hydrochloride (1675203-84-5(free base))
CAS :<p>BMS202 hydrochloride (1675203-84-5) is a potent PD-1/PD-L1 inhibitor (IC50: 18 nM) that promotes PD-L1 dimerization, blocking PD1 binding.</p>Formule :C25H30ClN3O3Degré de pureté :98.29% - 99.47%Couleur et forme :SolidMasse moléculaire :455.97NS-3-008 hydrochloride
CAS :<p>NS-3-008 hydrochloride (NS-3-008 HCl) is a transcriptional G0/G1 switch 2 (G0s2) inhibitor( IC50 of 2.25 μM).</p>Formule :C14H24ClN3Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :269.81PD184161
CAS :<p>PD184161 is a novel, orally-active MEK inhibitor. PD184161 inhibited MEK activity (IC50 = 10-100 nM) in a time- and concentration-dependent manner[1].</p>Formule :C17H13BrClF2IN2O2Degré de pureté :99.40%Couleur et forme :SolidMasse moléculaire :557.56Rhapontin
CAS :<p>Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.</p>Formule :C21H24O9Degré de pureté :99% - 99.91%Couleur et forme :Light YellowMasse moléculaire :420.41Perillyl alcohol
CAS :<p>Perillyl Alcohol, a monoterpene with antitumor properties, inhibits protein activation blocking cancer cell growth.</p>Formule :C10H16ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :152.23Z-DEVD-FMK
CAS :<p>Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,</p>Formule :C30H41FN4O12Degré de pureté :96.19% - 99.69%Couleur et forme :SolidMasse moléculaire :668.66ZM 336372
CAS :<p>ZM 336372 is a potent and selective c-Raf inhibitor.</p>Formule :C23H23N3O3Degré de pureté :97.24% - 97.51%Couleur et forme :SolidMasse moléculaire :389.45Notoginsenoside R1
CAS :<p>Notoginsenoside R1 (Sanchinoside R1) has been shown to exhibit antioxidant, antiapoptotic, anti-inflammatory, and immune-stimulatory properties.</p>Formule :C47H80O18Degré de pureté :99.57% - >99.99%Couleur et forme :SolidMasse moléculaire :933.13Geranylgeraniol
CAS :<p>Geranylgeraniol (FT0626663) is an isoprenoid found in fruits, vegetables, and grains, including rice.</p>Formule :C20H34ODegré de pureté :99.17% - ≥98%Couleur et forme :SolidMasse moléculaire :290.48Buparlisib
CAS :<p>Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM for p110α, p110β, and p110δ).</p>Formule :C18H21F3N6O2Degré de pureté :95.32% - 98.45%Couleur et forme :SolidMasse moléculaire :410.39SSE15206
CAS :<p>SSE15206 is a microtubule polymerization inhibitor that overcomes multidrug resistance.</p>Formule :C19H21N3O3SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :371.45Ac-DEVD-CHO acetate
<p>Caspase-3 Inhibitor I (N-acetyl-asp-glu-val-asp-al) is a specific inhibitor of Caspase-3.</p>Formule :C22H34N4O13Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :562.52Rigosertib sodium
CAS :<p>Rigosertib sodium (ON-01910), a non-ATP-competitive inhibitor of PLK1(IC50=9 nM), exhibits 30-fold higher specificity activity over Plk2 and no effect on Plk3.</p>Formule :C21H24NNaO8SDegré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :473.47Iberdomide
CAS :<p>Iberdomide (CC-220) is a modulator of cereblon( IC50 value of 60 nM in a competitive TR-FRET assay).</p>Formule :C25H27N3O5Degré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :449.5Tubastatin A Hydrochloride
CAS :<p>Tubastatin A Hydrochloride (TSA HCl) is an effective and specific HDAC6 inhibitor (IC50: 15 nM).</p>Formule :C20H21N3O2·HClDegré de pureté :97.24% - 99.15%Couleur et forme :SolidMasse moléculaire :371.86Ganoderenic acid D
CAS :<p>Ganoderenic acid D, extracted from Ganoderma lucidum, triggers apoptosis and halts cancer cell growth.</p>Formule :C30H40O7Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :512.63Necrostatin-1
CAS :<p>Necrostatin-1 (Nec-1) is a necrotic apoptosis inhibitor and RIP1 inhibitor with specificity.</p>Formule :C13H13N3OSDegré de pureté :99.25% - >99.99%Couleur et forme :SolidMasse moléculaire :259.33SNS-032
CAS :<p>SNS-032 (BMS-387032) is a selective inhibitor of CDK2 and is 10- and 20-fold selective over CDK1/CDK4. SNS-032 is sensitive to CDK7/9, and no effect on CDK6.</p>Formule :C17H24N4O2S2Degré de pureté :98.27% - 99.91%Couleur et forme :SolidMasse moléculaire :380.53SecinH3
CAS :<p>SecinH3 is selective cytohesin inhibitor.</p>Formule :C24H20N4O4SDegré de pureté :97.49% - 99.37%Couleur et forme :SolidMasse moléculaire :460.51NVP-CGM097
CAS :<p>NVP-CGM097 (CGM097) is an effective and specific MDM2 inhibitor (IC50: 1.7 nM for hMDM2).</p>Formule :C38H47ClN4O4Degré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :659.26Amifostine thiol dihydrochloride
CAS :<p>Amifostine (WR 1065) activates p53 via JNK and shields tissues from cancer drug toxicity.</p>Formule :C5H16Cl2N2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :207.165Cobimetinib
CAS :<p>Cobimetinib (GDC-0973) is a MEK1 inhibitor with selective and oral activity. Cobimetinib exhibits antitumor activity. Cost-effective and quality-assured.</p>Formule :C21H21F3IN3O2Degré de pureté :98% - 99.61%Couleur et forme :SolidMasse moléculaire :531.31TAK-243
CAS :<p>TAK-243 (MLN7243) is a selective inhibitor of the ubiquitin-activating enzyme UAE (IC50=1 nM).</p>Formule :C19H20F3N5O5S2Degré de pureté :98.09% - 98.93%Couleur et forme :SolidMasse moléculaire :519.52GSK2256098
CAS :<p>GSK2256098 (GTPL7939) is a small molecule FAK kinase inhibitor.</p>Formule :C20H23ClN6O2Degré de pureté :99.46% - 99.74%Couleur et forme :SolidMasse moléculaire :414.89Penicillic acid
CAS :<p>Penicillic acid, a mycotoxin from Aspergillus/Penicillium, blocks Fas ligand apoptosis and is cytotoxic to rat lung macrophages.</p>Formule :C8H10O4Degré de pureté :98%Couleur et forme :Needles From Petroleum Ether Slight Yellow PowderMasse moléculaire :170.16Thonningianin A
CAS :<p>Thonningianin A: an anti-cancer compound with antioxidant effects, GST inhibitor, and radical scavenger.</p>Formule :C42H34O21Degré de pureté :98.37% - 99.94%Couleur et forme :SolidMasse moléculaire :874.71CDDO-Im
CAS :<p>CDDO-Im (TP-235) is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).</p>Formule :C34H43N3O3Degré de pureté :98.3% - 99.61%Couleur et forme :SolidMasse moléculaire :541.72KEA1-97
CAS :<p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>Formule :C15H9Cl2FN4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :335.16Vistusertib
CAS :<p>Vistusertib (AZD2014) is an orally bioavailable inhibitor of the mammalian target of rapamycin (mTOR) with potential antineoplastic activity.</p>Formule :C25H30N6O3Degré de pureté :97.08% - 99.06%Couleur et forme :SolidMasse moléculaire :462.54NADPH tetrasodium salt
CAS :<p>NADPH tetrasodium salt is the reduced form of the electron acceptor nicotinamide adenine dinucleotide phosphate, which acts as an electron donor in a variety of</p>Formule :C21H26N7Na4O17P3Degré de pureté :97.15% - >99.99%Couleur et forme :SolidMasse moléculaire :833.35Vandetanib
CAS :<p>Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 and EGFR.</p>Formule :C22H24BrFN4O2Degré de pureté :99.7% - >99.99%Couleur et forme :White SolidMasse moléculaire :475.35CP-31398 dihydrochloride
CAS :<p>CP-31398 dihydrochloride is a p53 stabilizer which stabilizes the active conformation of p53 and promotes p53 activity in cancer cell lines.</p>Formule :C22H28Cl2N4ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :435.4ABT-737
CAS :<p>ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.</p>Formule :C42H45ClN6O5S2Degré de pureté :98.15% - >99.99%Couleur et forme :SolidMasse moléculaire :813.43C25-140
CAS :<p>C25-140 is a small-molecule inhibitor of TRAF6-Ubc13.</p>Formule :C26H31N7ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :457.57Ziyuglycoside II
CAS :<p>1.</p>Formule :C35H56O8Degré de pureté :99.52% - ≥95%Couleur et forme :SolidMasse moléculaire :604.81Tubastatin A
CAS :<p>Tubastatin A: Selective HDAC6 inhibitor, IC50 of 15 nM, 1000x less effective on other isozymes except HDAC8.</p>Formule :C20H21N3O2Degré de pureté :97.22% - 99.51%Couleur et forme :SolidMasse moléculaire :335.4Isosilybin A
CAS :<p>Isosilybin A is a partial PPARγ agonist, it significantly induced ABCA1 protein expression, it inhibited both monophenolase (IC50=1.7-7.6μM) and diphenolase (</p>Formule :C25H22O10Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :482.44Linalool
CAS :<p>Linalool, in essential oils, offers antinociceptive, antimicrobial, and anti-inflammatory effects, protects the liver, and boosts plant defense.</p>Formule :C10H18ODegré de pureté :98.22%Couleur et forme :Colorless Liquid Drypowder Liquid Othersolid LiquidMasse moléculaire :154.25Nutlin-3b
CAS :<p>Nutlin-3b, a less potent (+)-enantiomer of Nutlin-3, inhibits p53/MDM2 at IC50: 13.6 μM, 150x weaker than Nutlin-3a.</p>Formule :C30H30Cl2N4O4Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :581.49SRS16-86
CAS :<p>SRS16-86 is a novel third-generation ferrostatin, is an inhibitor of ferroptosis.</p>Formule :C26H32N4O2Degré de pureté :97.73%Couleur et forme :SolidMasse moléculaire :432.562,5-dimethyl Celecoxib
CAS :<p>2,5-dimethyl Celecoxib, a derivative targeting mPGES-1, inhibits PGE2 synthesis in inflammation.</p>Formule :C18H16F3N3O2SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :395.4PhiKan 083
CAS :<p>PhiKan 083 is a carbazole derivative</p>Formule :C16H18N2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :238.33Hirsutine
CAS :<p>Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive and</p>Formule :C22H28N2O3Degré de pureté :99.36% - 99.98%Couleur et forme :SolidMasse moléculaire :368.47(Rac)-Antineoplaston A10
CAS :<p>Antineoplaston A10 is the first identified human antineoplaston, naturally occurring with anti-proliferative properties.</p>Formule :C13H14N2O3Degré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :246.26A-1210477
CAS :<p>A-1210477 is an effective and specific MCL-1 and Bcl-2 inhibitor (Ki/IC50: 0.454/26.2 nM).</p>Formule :C46H55N7O7SDegré de pureté :99.17% - 99.37%Couleur et forme :SolidMasse moléculaire :850.04PF-3758309 hydrochloride
CAS :<p>PF-3758309 hydrochloride (PF-03758309 hydrochloride) , is a PAK4 inhibitor, is also a n orally bioavailable small-molecule inhibitor of p21-activated kinase 4 (</p>Formule :C25H31ClN8OSDegré de pureté :98.83% - >99.99%Couleur et forme :SolidMasse moléculaire :527.08PP121
CAS :<p>PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.</p>Formule :C17H17N7Degré de pureté :98.45% - 99.67%Couleur et forme :SolidMasse moléculaire :319.36Garcinol
CAS :<p>Garcinol: inhibits HATs/PCAF (IC50=7/5 μM), anti-inflammatory, anti-cancer, anti-cholinesterase (AChE IC50=0.66 μM, BChE IC50=7.39 μM).</p>Formule :C38H50O6Degré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :602.8Cucurbitacin B
CAS :<p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>Formule :C32H46O8Degré de pureté :97.1% - 99.33%Couleur et forme :SolidMasse moléculaire :558.7Kinsenoside
CAS :<p>Kinsenoside ((+)-Kinsenoside) shows significant antihepatotoxic, and anti-inflammatory activities.</p>Formule :C10H16O8Degré de pureté :99.2% - >99.99%Couleur et forme :SolidMasse moléculaire :264.23FX1
CAS :<p>FX1 is an effective and selective BCL6 inhibitor (IC50: 35 μM).</p>Formule :C14H9ClN2O4S2Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :368.82ZM-447439
CAS :<p>ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.</p>Formule :C29H31N5O4Degré de pureté :99.11% - 99.59%Couleur et forme :Pale Yellow SolidMasse moléculaire :513.59Rottlerin
CAS :<p>Rottlerin (NSC-56346), a Mallotus Philippinensis extract, inhibits PKC (3-100 μM IC50); triggers apoptosis by activating caspase 3.</p>Formule :C30H28O8Degré de pureté :97.41% - 99.44%Couleur et forme :Orange To Brown PowderMasse moléculaire :516.54ASK1-IN-2
CAS :<p>ASK1-IN-2: oral ASK1 inhibitor, IC50 32.8 nM, potential ulcerative colitis treatment.</p>Formule :C19H17FN6ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :364.38GSK-923295
CAS :<p>GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).</p>Formule :C32H38ClN5O4Degré de pureté :96.22% - 98.02%Couleur et forme :SolidMasse moléculaire :592.13PHA-767491 hydrochloride
CAS :<p>PHA-767491 (CAY-10572) is a potent Cdc7/CDK9 inhibitor (IC50: 10/34 nM), selective against GSK3-β, CDK1/2, CDK5, MK2, CHK2, PLK1.</p>Formule :C12H12ClN3ODegré de pureté :99.56% - 99.92%Couleur et forme :SolidMasse moléculaire :249.69α-Thujone
CAS :<p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>Formule :C10H16ODegré de pureté :97.02% - 98.41%Couleur et forme :Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Masse moléculaire :152.23CP-724714
CAS :<p>CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against EGFR, Abl, InsR, PDGFR, IRG-1R, Src, VEGFR2</p>Formule :C27H27N5O3Degré de pureté :97.1% - 98.82%Couleur et forme :SolidMasse moléculaire :469.54ASP3026
CAS :<p>ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies,and Positive for Anaplastic Lymphoma Kinase.</p>Formule :C29H40N8O3SDegré de pureté :98.78% - 99.81%Couleur et forme :SolidMasse moléculaire :580.74CCT 137690
CAS :<p>CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).</p>Formule :C26H31BrN8ODegré de pureté :98.51% - 99.89%Couleur et forme :SolidMasse moléculaire :551.48COTI-2
CAS :<p>COTI-2, an orally available thiosemicarbazone, is an activator of mutant forms of the p53 protein with potential antineoplastic activity.</p>Formule :C19H22N6SDegré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :366.48C-DIM12
CAS :<p>C-DIM12 boosts Nurr1 gene expression, heightens Nurr1 protein in neurons, and improves survival against 6-OHDA.</p>Formule :C23H17ClN2Degré de pureté :97.72% - ≥95%Couleur et forme :SolidMasse moléculaire :356.85L-685458
CAS :<p>L-685458 (L-685,458) is a specific and potent inhibitor of A beta PP gamma-secretase activity with Ki of 17 nM.</p>Formule :C39H52N4O6Degré de pureté :99.62% - 99.80%Couleur et forme :SolidMasse moléculaire :672.85Momelotinib
CAS :<p>Momelotinib (LM-1149), an oral JAK1/2 inhibitor with IC50s 11/18 nM, blocks ATP binding, disrupting JAK-STAT pathway and reducing tumor growth.</p>Formule :C23H22N6O2Degré de pureté :97.47% - 99.56%Couleur et forme :SolidMasse moléculaire :414.46BC-1258
CAS :<p>BC-1258 is a unique small molecule F-box/LRR-repeat protein 2 (FBXL2) activator.</p>Formule :C22H22N4S2Degré de pureté :97.48% - 99.64%Couleur et forme :SolidMasse moléculaire :406.57Dubermatinib
CAS :<p>Dubermatinib (TP0903) is a potent and selective Axl kinase inhibitor.</p>Formule :C24H30ClN7O2SDegré de pureté :98.65% - 99.58%Couleur et forme :SolidMasse moléculaire :516.06R406
CAS :<p>R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.</p>Formule :C22H23FN6O5·C6H6O3SDegré de pureté :97.67% - 98.82%Couleur et forme :SolidMasse moléculaire :628.63Mito-LND
CAS :<p>Mito-LND (Mito-Loidamine) is an orally active and mitochondria-targeted inhibitor of oxidative phosphorylation.</p>Formule :C43H45BrCl2N3OPDegré de pureté :97.25% - 98.34%Couleur et forme :SolidMasse moléculaire :801.62AZD-3463
CAS :<p>AZD-3463 (ALK/IGF1R inhibitor) , an orally bioavailable ALK inhibitor (Ki: 0.75 nM), can inhibit IGF1R with equivalent potency.</p>Formule :C24H25ClN6ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :448.95Etalocib
CAS :<p>Etalocib (LY293111) is a potent diaryl ether inhibitor blocking LTB4 receptor and 5'-lipoxygenase, with antineoplastic properties.</p>Formule :C33H33FO6Degré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :544.6Tiplaxtinin
CAS :<p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>Formule :C24H16F3NO4Degré de pureté :99.16% - 99.93%Couleur et forme :SolidMasse moléculaire :439.38Toyocamycin
CAS :<p>Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (</p>Formule :C12H13N5O4Degré de pureté :98.1% - 98.17%Couleur et forme :SolidMasse moléculaire :291.26Adalimumab
CAS :<p>Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.</p>Degré de pureté :95% - 99.50%Couleur et forme :LiquidMasse moléculaire :145.4 kDaIcaritin
CAS :<p>Icaritin (Anhydroicaritin) has hormone regulation activity and cardiovascular function improvement activity.</p>Formule :C21H20O6Degré de pureté :97.69% - 99.76%Couleur et forme :SolidMasse moléculaire :368.38Se-Methylselenocysteine
CAS :<p>Se-Methylselenocysteine (Se-MSC) is a potent chemopreventive agent in many test systems and has been shown to inhibit tumor promotion and induce apoptosis.</p>Formule :C4H9NO2SeDegré de pureté :99.49% - 99.87%Couleur et forme :White To Slightly Yellow PowderMasse moléculaire :182.08Divalproex Sodium
CAS :<p>Divalproex Sodium (Valproate semisodium) binds to and inhibits gamma-aminobutyric acid (GABA) transaminase and its anticonvulsant activity may be exerted by</p>Formule :C8H16O2·C8H15O2·NaDegré de pureté :99.87%Couleur et forme :A White Powder With A Characteristic OdorMasse moléculaire :310.41PCI-34051
CAS :<p>PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM).</p>Formule :C17H16N2O3Degré de pureté :97.219% - 98.29%Couleur et forme :SolidMasse moléculaire :296.32MI-136
CAS :<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Formule :C23H21F3N6SDegré de pureté :98.63% - 99.12%Couleur et forme :SolidMasse moléculaire :470.51HS-173
CAS :<p>HS-173 is an effective PI3Kα inhibitor (IC50: 0.8 nM).</p>Formule :C21H18N4O4SDegré de pureté :99.33% - 99.64%Couleur et forme :SolidMasse moléculaire :422.46RHPS4
CAS :<p>RHPS4 (RHPS 4 methosulfate) is a potent inhibitor of Telomerase at submicromolar.</p>Formule :C22H17F2N2·CH3O4SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :458.48Leachianone A
CAS :<p>Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced cytotoxicity.</p>Formule :C26H30O6Degré de pureté :98.53% - 99.79%Couleur et forme :SolidMasse moléculaire :438.51Citric acid
CAS :<p>Citric acid (Citro) is a weak organic tricarboxylic acid found in citrus fruits, a food additive and a natural preservative. High-Quality, Low-Cost!</p>Formule :C6H8O7Degré de pureté :98.88%Couleur et forme :White Solid CrystallineMasse moléculaire :192.12Ursonic Acid
CAS :<p>Ursonic Acid (TOS-BB-0966) belongs to the family of Ursane Triterpenes whose structure is based on the pentacyclic ursane skeleton.</p>Formule :C30H46O3Degré de pureté :98.90% - >99.99%Couleur et forme :SolidMasse moléculaire :454.68Polydatin
CAS :<p>Polydatin, a resveratrol glycoside from Polygonum cuspidatum, inhibits platelet aggregation, alters lipid ratios, and modulates cell functions.</p>Formule :C20H22O8Degré de pureté :97.2% - 98.94%Couleur et forme :White Fine PowderMasse moléculaire :390.38Piperlongumine
CAS :<p>Piperlongumine (Piplartine) is a natural alkaloid from Piper longum L.</p>Formule :C17H19NO5Degré de pureté :97.03% - 99.90%Couleur et forme :SolidMasse moléculaire :317.34ODQ
CAS :<p>ODQ is an effective and selective soluble guanylyl cyclase (sGC) inhibitor.</p>Formule :C9H5N3O2Degré de pureté :98.98%Couleur et forme :Off-White To Light Yellow PowderMasse moléculaire :187.15Cycleanine
CAS :<p>Cycleanine has potent antibacterial, antifungal, antiplasmodial, and cytotoxic activities.</p>Formule :C38H42N2O6Degré de pureté :98.04% - 99.57%Couleur et forme :SolidMasse moléculaire :622.75PS47
CAS :<p>PS-47(PS 47) is an inactive E-isomer of PS48. PS48 is an activator of PDK1.</p>Formule :C17H15ClO2Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :286.75D4476
CAS :<p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>Formule :C23H18N4O3Degré de pureté :99.7% - 99.96%Couleur et forme :SolidMasse moléculaire :398.41Capsazepine
CAS :<p>Capsazepine, a TRPV1 antagonist (IC50: 562 nM), blocks capsaicin-induced heat pain.</p>Formule :C19H21ClN2O2SDegré de pureté :98% - 99.78%Couleur et forme :White To Off-White PowderMasse moléculaire :376.9SC144
CAS :<p>SC144 is an orally active small-molecule gp130 inhibitor.</p>Formule :C16H11FN6ODegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :322.3Dapivirine
CAS :<p>Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>Formule :C20H19N5Degré de pureté :98% - 99.77%Couleur et forme :SolidMasse moléculaire :329.4Bafetinib
CAS :<p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>Formule :C30H31F3N8ODegré de pureté :94.16% - 99.68%Couleur et forme :SolidMasse moléculaire :576.62PHT-427
CAS :<p>PHT-427 (CS-0223) is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity binding for the PH domains of Akt and PDPK1).</p>Formule :C20H31N3O2S2Degré de pureté :97.54% - >99.99%Couleur et forme :SolidMasse moléculaire :409.61Benzyl isothiocyanate
CAS :<p>BITC, found in cruciferous veggies, exhibits anticancer, antimicrobial, and immunomodulatory effects.</p>Formule :C8H7NSDegré de pureté :99.25% - 99.83%Couleur et forme :Clear Yellow LiquidMasse moléculaire :149.21T0901317
CAS :<p>T0901317 is a potent and selective agonist for both LXR and FXR, with EC50 of ~50 nM and 5 μM, respectively; it inhibits nuclear factor/κB (NF/κB).</p>Formule :C17H12F9NO3SDegré de pureté :98% - 99.64%Couleur et forme :SolidMasse moléculaire :481.33Onvansertib
CAS :<p>Onvansertib (NMS-1286937) is a PLK1 inhibitor with high selectivity and oral activity. Onvansertib has antitumor activity. Cost-effective and quality-assured.</p>Formule :C24H27F3N8O3Degré de pureté :98.3% - 99.88%Couleur et forme :SolidMasse moléculaire :532.52SBI-0640756
CAS :<p>SBI-0640756 (SBI-756) (SBI-756) is a first-in-class inhibitor that targets eIF4G1 and disrupts the eIF4F complex.</p>Formule :C23H14ClFN2O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :404.82Piperazine Erastin
CAS :<p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>Formule :C35H41ClN6O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :645.19PluriSIn 1
CAS :<p>PluriSIn 1 (NSC 14613) blocks SCD1, key in oleic acid creation, showing lipid metabolism's role in hPSCs.</p>Formule :C12H11N3ODegré de pureté :99.19% - 99.63%Couleur et forme :SolidMasse moléculaire :213.24BTSA1
CAS :<p>BTSA1: High-affinity BAX activator inducing conformational changes for apoptosis.</p>Formule :C21H14N6OS2Degré de pureté :99.60% - 99.71%Couleur et forme :SolidMasse moléculaire :430.51Cambinol
CAS :<p>Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.</p>Formule :C21H16N2O2SDegré de pureté :98.02% - 99.83%Couleur et forme :SolidMasse moléculaire :360.43LYN-1604 dihydrochloride
CAS :<p>LYN-1604 is a novel ULK1 activator.It inducing cell death involved in ATF3, RAD21, and caspase3, accompanied by autophagy and apoptosis.</p>Formule :C33H45Cl4N3O2Degré de pureté :98.95% - 99.92%Couleur et forme :SolidMasse moléculaire :657.54Azadirachtin
CAS :<p>Azadirachtin has antifungal activity, used as an insecticide.</p>Formule :C35H44O16Degré de pureté :98.11% - 99.713%Couleur et forme :SolidMasse moléculaire :720.71

