Trasportatore di membrana/canale ionico
Gli inibitori dei trasportatori di membrana e dei canali ionici sono composti che bloccano la funzione delle proteine responsabili del trasporto di ioni, nutrienti e altre molecole attraverso le membrane cellulari. Questi inibitori sono cruciali per studiare la regolazione dell'omeostasi cellulare, la trasduzione del segnale e la neurotrasmissione. Gli inibitori dei trasportatori di membrana e dei canali ionici sono anche importanti per sviluppare trattamenti per disturbi come l'epilessia, le malattie cardiovascolari e le sindromi metaboliche. Presso CymitQuimica, offriamo una vasta selezione di inibitori di alta qualità dei trasportatori di membrana e dei canali ionici per supportare la tua ricerca in fisiologia, neuroscienze e farmacologia.
Sottocategorie di "Trasportatore di membrana/canale ionico"
- ABC(3 prodotti)
- ATPasi(101 prodotti)
- Recettore dell'adiponectina(5 prodotti)
- CFTR(65 prodotti)
- Ricettore CGRP(54 prodotti)
- Canale del calcio(541 prodotti)
- Canale del cloruro(53 prodotti)
- Ricettore GABA(365 prodotti)
- Trasportatore di monoammine(30 prodotti)
- Trasportatore di monocarbossilato(18 prodotti)
- NKCC(2 prodotti)
- NPC1L1(3 prodotti)
- Cotrasportatore Na-K-Cl(10 prodotti)
- OAT(32 prodotti)
- OCT(7 prodotti)
- P-gp(54 prodotti)
- Canale del potassio(280 prodotti)
- Pompa protonica(42 prodotti)
- SGLT(31 prodotti)
- Canale del sodio(209 prodotti)
- Canale TRP/TRPV(95 prodotti)
Mostrare 13 più sottocategorie
Trovati 2512 prodotti di "Trasportatore di membrana/canale ionico"
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GABAA receptor agent 1
CAS:<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formula:C13H8ClN3O2Purezza:99.31%Colore e forma:SolidPeso molecolare:273.675,5-Dimethyloxazolidine-2,4-dione
CAS:5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Formula:C5H7NO3Purezza:99.12%Colore e forma:Drypowder PelletslargecrystalsPeso molecolare:129.11Vinpocetine
CAS:Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).Formula:C22H26N2O2Purezza:99.85% - 99.98%Colore e forma:White Crystalline SolidPeso molecolare:350.45FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Formula:C13H11N3OPurezza:98.75%Colore e forma:SolidPeso molecolare:225.25NS5806
CAS:NS5806 activates K+ currents, slows KV4.2/4.3 decay with KChIP2, and boosts KV4.3/KChIP2 peaks (EC50=5.3μM).Formula:C16H8Br2F6N6OPurezza:97.95%Colore e forma:SolidPeso molecolare:574.07VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Formula:C20H32BrClN2O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:447.84Ref: TM-T13316
5mg37,00€10mg59,00€25mg104,00€50mg170,00€100mg283,00€200mg437,00€1mL*10mM (DMSO)42,00€Omeprazole
CAS:Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Formula:C17H19N3O3SPurezza:98.43% - 98.48%Colore e forma:White SolidPeso molecolare:345.42Piracetam
CAS:Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.Formula:C6H10N2O2Purezza:97.16%Colore e forma:Crystals From Isopropanol SolidPeso molecolare:142.16Zamicastat
CAS:Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).Formula:C21H21F2N3OSPurezza:99.58%Colore e forma:SolidPeso molecolare:401.47Ref: TM-T13383
1mg96,00€5mg205,00€10mg309,00€25mg557,00€50mg838,00€100mg1.216,00€1mL*10mM (DMSO)221,00€Flufenamic acid
CAS:<p>Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.</p>Formula:C14H10F3NO2Purezza:98.68%Colore e forma:White To Light Yellow Crystalline PowderPeso molecolare:281.23Halothane
CAS:Halothane (Anestan) 可以减弱内皮依赖性舒张作用。Formula:C2HBrClF3Purezza:99.80% - >99.99%Colore e forma:Colorless Volatile Liquid Density 1 875 G / Cm3 Boiling Point 122 4°F (50 2°C) NoncombustiblePeso molecolare:197.384-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Formula:C5H6N2Purezza:91.61%Colore e forma:SolidPeso molecolare:94.11Suloctidil
CAS:Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.Formula:C20H35NOSPurezza:99.75% - >99.99%Colore e forma:SolidPeso molecolare:337.56Riparin III
CAS:Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.Formula:C16H17NO4Purezza:95.13%Colore e forma:SolidPeso molecolare:287.31Celivarone
CAS:<p>Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.</p>Formula:C34H47NO4Purezza:99.53%Colore e forma:SolidPeso molecolare:533.74ATP synthase inhibitor 1
CAS:ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.Formula:C17H18ClN3O3S2Purezza:99.83%Colore e forma:SolidPeso molecolare:411.93RUVBL1/2 ATPase-IN-1
CAS:RUVBL1/2 ATPase-IN-1 inhibits RUVBL1/2 ATPase (IC50: 6.0/7.7 μM); useful in cancer research.Formula:C28H28F3N5OPurezza:99.92%Colore e forma:SolidPeso molecolare:507.55Norverapamil hydrochloride
CAS:Norverapamil HCl, a Verapamil metabolite, blocks L-type calcium channels and inhibits P-gp function.Formula:C26H37ClN2O4Purezza:99.47%Colore e forma:SolidPeso molecolare:477.04Ref: TM-T16339
1mg37,00€5mg111,00€10mg187,00€25mg315,00€50mg472,00€100mg635,00€200mg888,00€1mL*10mM (DMSO)116,00€PF-04885614
CAS:PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.Formula:C13H14F3N3OPurezza:98.02%Colore e forma:SolidPeso molecolare:285.27Ref: TM-T12421
2mg42,00€5mg64,00€10mg92,00€25mg170,00€50mg316,00€100mg447,00€200mg628,00€1mL*10mM (DMSO)64,00€Afoxolaner
CAS:Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.Formula:C26H17ClF9N3O3Purezza:99.1% - 99.38%Colore e forma:SolidPeso molecolare:625.87Gliclazide
CAS:Gliclazide (SE1702), an oral antihyperglycemic agent, belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating beta-cells of theFormula:C15H21N3O3SPurezza:99.58%Colore e forma:SolidPeso molecolare:323.41(Z)-Capsaicin
CAS:<p>(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer of</p>Formula:C18H27NO3Purezza:97.33% - 98.91%Colore e forma:SolidPeso molecolare:305.41Nicorandil
CAS:Nicorandil (SG-75)(Ikorel) acts by relaxing the smooth muscle of the blood vessels, especially those of the venous system.Formula:C8H9N3O4Purezza:98.14% - >99.99%Colore e forma:White Or Off-White PowderPeso molecolare:211.17Alinidine
CAS:Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.Formula:C12H13Cl2N3Purezza:98.91% - >99.99%Colore e forma:SolidPeso molecolare:270.16IA-Alkyne
CAS:IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.Formula:C8H12INOPurezza:99.76%Colore e forma:SolidPeso molecolare:265.09Ref: TM-T15543
1mg59,00€5mg126,00€10mg187,00€25mg264,00€50mg329,00€100mg455,00€1mL*10mM (DMSO)120,00€Hydrochlorothiazide
CAS:Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。Formula:C7H8ClN3O4S2Purezza:99.43% - 99.50%Colore e forma:Crystals Physical Description Crystals Or White Powder (Ntp 1992)Peso molecolare:297.74VU6036720
<p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>Formula:C20H22ClFN4O2SPurezza:98.1%Colore e forma:SoildPeso molecolare:436.93Oxiracetam
CAS:<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formula:C6H10N2O3Purezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:158.16Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Formula:C6H11NO2Purezza:99.90%Colore e forma:SolidPeso molecolare:129.16Cromolyn sodium
CAS:Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.Formula:C23H14Na2O11Purezza:99.4% - 99.95%Colore e forma:Colorless Crystals From Ethanol + Ether White Crystalline PowderPeso molecolare:512.33FFN 511
CAS:Fluorescent false neurotransmitter (FFN)Formula:C17H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:284.35Clomethiazole
CAS:Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.Formula:C6H8ClNSPurezza:99.06%Colore e forma:SolidPeso molecolare:161.65Clorsulon
CAS:Clorsulon (L631529) is utilized for the treatment of Fasciola hepatica infections in calves and sheep.Formula:C8H8Cl3N3O4S2Purezza:99.66% - 99.87%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:380.66NS3623
CAS:NS3623 is an activator of human ether-a-go-go-related gene potassium channels.Formula:C15H10BrF3N6OPurezza:97.06%Colore e forma:SolidPeso molecolare:427.18Mebeverine hydrochloride
CAS:Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gutFormula:C25H35NO5Purezza:99.81% - 99.81%Colore e forma:SolidPeso molecolare:429.55Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formula:C8H14N2O4SPurezza:98.38% - 99.83%Colore e forma:SolidPeso molecolare:234.27Ropivacaine hydrochloride
CAS:Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activityFormula:C17H26N2O·HClPurezza:99.85% - 99.95%Colore e forma:SolidPeso molecolare:310.86Endovion
CAS:Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.Formula:C16H9BrF6N6OPurezza:98.51%Colore e forma:SolidPeso molecolare:495.18Gabapentin
CAS:Gabapentin (Neurontin) is an Anti-epileptic Agent.Formula:C9H17NO2Purezza:99.55% - 99.91%Colore e forma:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidPeso molecolare:171.24NS8593 hydrochloride
CAS:NS8593 hydrochloride (NS8593 HCl) is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels) .Formula:C17H18ClN3Purezza:99.77%Colore e forma:SolidPeso molecolare:299.8Ref: TM-T12256
1mg46,00€2mg59,00€5mg93,00€10mg159,00€25mg350,00€50mg525,00€100mg757,00€1mL*10mM (DMSO)96,00€QX-314 chloride
CAS:QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.Formula:C16H27ClN2OPurezza:99.73%Colore e forma:SolidPeso molecolare:298.85Ropivacaine
CAS:Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.Formula:C17H26N2OPurezza:97.75% - >99.99%Colore e forma:SolidPeso molecolare:274.40Linopirdine
CAS:Linopirdine (DuP 996) is a TRPV1 agonist.Formula:C26H21N3OPurezza:99.45% - 99.78%Colore e forma:SolidPeso molecolare:391.46Ref: TM-T15758
1mg43,00€2mg56,00€5mg88,00€10mg126,00€25mg227,00€50mg393,00€100mg560,00€200mg810,00€500mg1.206,00€1mL*10mM (DMSO)87,00€AR-C155858
CAS:AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).Formula:C21H27N5O5SPurezza:98.96% - 99.42%Colore e forma:SolidPeso molecolare:461.53Ref: TM-T14316
1mg96,00€5mg283,00€10mg492,00€25mg800,00€50mg1.103,00€100mg1.491,00€1mL*10mM (DMSO)296,00€Oxybutynin chloride
CAS:Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.Formula:C22H32ClNO3Purezza:99.27% - >99.99%Colore e forma:White PowderPeso molecolare:393.96Meticrane
CAS:Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.Formula:C10H13NO4S2Purezza:99.16%Colore e forma:SolidPeso molecolare:275.34Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formula:C12H21NO8SPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:339.36VU591
CAS:VU591 is a selective extra-renal potassium channel inhibitor with an IC₅₀ of 0.24 μM.Formula:C16H12N6O5Purezza:99.29% - 99.53%Colore e forma:SolidPeso molecolare:368.3Ref: TM-T13320L
5mg50,00€10mg80,00€25mg140,00€50mg244,00€100mg364,00€500mg780,00€1mL*10mM (DMSO)51,00€Gut restricted-7
CAS:Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.Formula:C25H40FNaO6SPurezza:98.81% - 99.27%Colore e forma:SolidPeso molecolare:510.64Tuvatexib
CAS:<p>Tuvatexib is a small molecule VDAC/HK2 dual modulator.</p>Formula:C21H23NO3Purezza:97.29% - 99.80%Colore e forma:SolidPeso molecolare:337.41E 0747 FA
E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.Formula:C22H30ClN3O6Purezza:98.54%Colore e forma:SolidPeso molecolare:467.94Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Formula:C25H14BrF11N2O2Purezza:99.82%Colore e forma:SolidPeso molecolare:663.29Ref: TM-T10618
1mg52,00€2mg74,00€5mg111,00€10mg180,00€25mg358,00€50mg588,00€100mg835,00€1mL*10mM (DMSO)131,00€Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Formula:C21H17ClF3N3O3Purezza:99.86%Colore e forma:SolidPeso molecolare:451.83Ref: TM-T15207
1mg62,00€5mg116,00€10mg170,00€25mg283,00€50mg424,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)128,00€Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Formula:C66H92F3N19O24Purezza:99.89%Colore e forma:SolidPeso molecolare:1592.55BMS-191095
CAS:BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.Formula:C22H21ClN4O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:408.88Ref: TM-T10566
1mg96,00€5mg202,00€10mg305,00€25mg550,00€50mg747,00€100mg1.008,00€1mL*10mM (DMSO)224,00€Omeprazole sulfide
CAS:Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.Formula:C17H19N3O2SPurezza:98.83%Colore e forma:White To Slightly Collored Solid Solid CrystallinePeso molecolare:329.42DSP-2230
CAS:<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Formula:C20H20F3N5O2Purezza:97.14%Colore e forma:SolidPeso molecolare:419.4Hydroxyhexamide
CAS:Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.Formula:C15H22N2O4SPurezza:98.91%Colore e forma:SolidPeso molecolare:326.41Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purezza:98% - >99.99%Colore e forma:1992)Peso molecolare:213.66Vigabatrin
CAS:Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-Formula:C6H11NO2Purezza:99.47% - 99.88%Colore e forma:SolidPeso molecolare:129.16Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Formula:C10H14O3Purezza:99.49%Colore e forma:SolidPeso molecolare:182.22Linoleoyl glycine
CAS:<p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>Formula:C20H35NO3Purezza:98.96%Colore e forma:SolidPeso molecolare:337.5MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFormula:C11H6BrN3O3Purezza:98.459%Colore e forma:SolidPeso molecolare:308.09Ref: TM-T12110
1mg96,00€5mg202,00€10mg329,00€25mg655,00€50mg1.103,00€100mg1.483,00€1mL*10mM (DMSO)224,00€BMS-195270
CAS:BMS-195270 is a bio-active chemical.Formula:C15H9ClF3N3O2Purezza:98.7%Colore e forma:SolidPeso molecolare:355.7Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Formula:C24H26ClNO4Purezza:99.78%Colore e forma:White SolidPeso molecolare:427.92Tocainide
CAS:Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.Formula:C11H16N2OPurezza:99.84%Colore e forma:SolidPeso molecolare:192.26Vocacapsaicin hydrochloride
CAS:<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Formula:C26H42ClN3O4Purezza:99.66% - 99.80%Colore e forma:SolidPeso molecolare:496.08TRPV4 agonist-1 free base
CAS:TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).Formula:C25H22F2N4O2Purezza:99.79%Colore e forma:SolidPeso molecolare:448.46NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formula:C20H24ClN3OPurezza:99.56%Colore e forma:SolidPeso molecolare:357.88Ref: TM-T12207
1mg74,00€5mg140,00€10mg215,00€25mg373,00€50mg522,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)156,00€Elexacaftor
CAS:Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.Formula:C26H34F3N7O4SPurezza:98.87% - 99.87%Colore e forma:SolidPeso molecolare:597.65Ref: TM-T14935
1mg87,00€2mg137,00€5mg243,00€10mg393,00€25mg772,00€50mg1.074,00€100mg1.444,00€1mL*10mM (DMSO)320,00€Phenazopyridine hydrochloride
CAS:Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.Formula:C11H12ClN5Purezza:99.27%Colore e forma:Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionPeso molecolare:249.7GFB-8438
CAS:GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).Formula:C16H14ClF3N4O2Purezza:99.58%Colore e forma:SolidPeso molecolare:386.76Ref: TM-T11394
2mg35,00€5mg52,00€10mg81,00€25mg117,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)58,00€MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formula:C25H25N3O2Purezza:99.77% - 99.8%Colore e forma:SolidPeso molecolare:399.48Sulfacarbamide
CAS:Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.Formula:C7H9N3O3SPurezza:95.6% - 99.72%Colore e forma:SolidPeso molecolare:215.23Econazole
CAS:Econazole ((±)-Econazol) is an imidazole derivative that is commonly used as a topical antifungal agent.Formula:C18H15Cl3N2OPurezza:98.11% - 99.97%Colore e forma:SolidPeso molecolare:381.68Ornidazole (Levo-)
CAS:<p>Ornidazole (Levo-) (Levornidazole) is the levo-isomer of Ornidazole.</p>Formula:C7H10ClN3O3Purezza:99.8%Colore e forma:SolidPeso molecolare:219.63Doxapram hydrochloride hydrate
CAS:Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.Formula:C24H33ClN2O3C24H30N2O2·ClH·H2OPurezza:99.64% - >99.99%Colore e forma:SolidPeso molecolare:432.99Oxybutynin
CAS:Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.Formula:C22H31NO3Purezza:97.81% - 99.57%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:357.49Verapamil hydrochloride
CAS:Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.Formula:C27H39ClN2O4Purezza:98.7% - 99.98%Colore e forma:White To Off-White PowderPeso molecolare:491.06Etifoxine hydrochloride
CAS:Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.Formula:C17H18Cl2N2OPurezza:99.36%Colore e forma:SolidPeso molecolare:337.24CRAC intermediate 2
CAS:CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.Formula:C11H7F6N3Purezza:99.69%Colore e forma:SolidPeso molecolare:295.18VU591 hydrochloride
CAS:VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.Formula:C16H13ClN6O5Purezza:98.93% - 99.22%Colore e forma:SolidPeso molecolare:404.76Ref: TM-T13320
1mg35,00€5mg74,00€10mg111,00€25mg226,00€50mg386,00€100mg540,00€200mg735,00€1mL*10mM (DMSO)84,00€Tolazamide
CAS:Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C14H21N3O3SPurezza:98% - >99.99%Colore e forma:SolidPeso molecolare:311.40Ref: TM-T1333
2mg35,00€5mg52,00€10mg70,00€25mg97,00€50mg125,00€100mg160,00€200mg230,00€1mL*10mM (DMSO)62,00€Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormula:C56H81NO15Purezza:98.68%Colore e forma:SolidPeso molecolare:1008.256L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formula:C3H6N2O2Purezza:99.75% - 99.99%Colore e forma:Crystals White PowderPeso molecolare:102.09Acetohexamide
CAS:Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.Formula:C15H20N2O4SPurezza:99.19% - 99.85%Colore e forma:Crystals From 90% Aq EthanolPeso molecolare:324.40LAU159
CAS:LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Formula:C17H12ClN3O2Purezza:98.7% - 99.38%Colore e forma:SolidPeso molecolare:325.75Ref: TM-T11822
1mg116,00€2mg169,00€5mg230,00€10mg418,00€25mg690,00€50mg938,00€100mg1.311,00€500mg2.632,00€Azosemide
CAS:Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).Formula:C12H11ClN6O2S2Purezza:99.84%Colore e forma:SolidPeso molecolare:370.84Permethrin
CAS:Permethrin (NRDC-143) is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.Formula:C21H20Cl2O3Purezza:99.37% - 99.54%Colore e forma:Colorless Crystals To A Viscous Liquid; Color White To Pale Yellow Permethrin Is A Pale Brown Liquid Relatively Water Insoluble Used As An InsecticidePeso molecolare:391.29URAT1 inhibitor 7
CAS:URAT1 inhibitor 7, a uric acid transporter protein URAT1 inhibitor.URAT1 inhibitor 7 inhibits CYP2C9 and can be used in the study of hyperuricemia and gout.Formula:C19H10ClFN4O3SPurezza:97.14%Colore e forma:SoildPeso molecolare:428.82Dyclonine hydrochloride
CAS:Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .Formula:C18H27NO2·HClPurezza:99.35%Colore e forma:White Crystalline SolidPeso molecolare:325.87ICA-27243
CAS:<p>ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.</p>Formula:C12H7ClF2N2OPurezza:99.54%Colore e forma:SolidPeso molecolare:268.65DCEBIO
CAS:<p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>Formula:C9H8Cl2N2OPurezza:99.89%Colore e forma:SolidPeso molecolare:231.08Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Formula:C11H12ClNO3SPurezza:99.88% - >99.99%Colore e forma:Crystals SolidPeso molecolare:273.74NS19504
CAS:NS19504 is an activator of Ca2+-activated K+ channel with EC50 of 11.0 µM.Formula:C10H9BrN2SPurezza:99.87%Colore e forma:SolidPeso molecolare:269.16Ref: TM-T12255
5mg49,00€10mg88,00€25mg170,00€50mg296,00€100mg444,00€500mg938,00€1mL*10mM (DMSO)55,00€Lansoprazole
CAS:Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISONFormula:C16H14F3N3O2SPurezza:99.18% - 99.84%Colore e forma:White Crystalline PowderPeso molecolare:369.36BIIB 722 Mesylate
CAS:<p>BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.</p>Formula:C19H23F3N6O5SPurezza:99.57%Colore e forma:SoildPeso molecolare:504.483Eact
CAS:<p>Eact is a potent TMEM16A activator that also triggers TRPV1, causing itch, pain, and heat sensitivity.</p>Formula:C22H24N2O5SPurezza:98.14%Colore e forma:SolidPeso molecolare:428.5TPC2-A1-P
CAS:TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).Formula:C20H21BrF3NO3Purezza:98.49%Colore e forma:SolidPeso molecolare:460.29Ref: TM-T36806
1mg97,00€5mg236,00€10mg394,00€25mg750,00€50mg1.216,00€100mg1.853,00€1mL*10mM (DMSO)240,00€Chlorpropamide
CAS:<p>Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary</p>Formula:C10H13ClN2O3SPurezza:98.90%Colore e forma:Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Peso molecolare:276.74Nav1.8-IN-4
CAS:Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.Formula:C20H14F4N2O3Purezza:99.83%Colore e forma:SoildPeso molecolare:406.33Ref: TM-T77693
1mg59,00€2mg85,00€5mg125,00€10mg188,00€25mg376,00€50mg612,00€100mg938,00€500mg1.882,00€Omeprazole metabolite Omeprazole sulfone
CAS:Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.Formula:C17H19N3O4SPurezza:99.87%Colore e forma:SolidPeso molecolare:361.42Ref: TM-T12309
1mg49,00€2mg65,00€5mg97,00€10mg154,00€25mg298,00€50mg445,00€100mg642,00€500mg1.320,00€1mL*10mM (DMSO)106,00€Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formula:C6H10N4Purezza:99.67% - 99.90%Colore e forma:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Peso molecolare:138.17Nikethamide
CAS:Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormula:C10H14N2OPurezza:99.42%Colore e forma:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Peso molecolare:178.23NaV1.7 inhibitor-1
CAS:NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Formula:C23H30FNO4SPurezza:99.89%Colore e forma:SolidPeso molecolare:435.55Ref: TM-T12181
1mg104,00€5mg255,00€10mg406,00€25mg700,00€50mg938,00€100mg1.378,00€1mL*10mM (DMSO)280,00€ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Formula:C19H24ClN3O3Purezza:99.3%Colore e forma:SolidPeso molecolare:377.87Ref: TM-T16110
1mg39,00€5mg84,00€10mg117,00€25mg188,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)93,00€DCPIB
CAS:<p>DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM</p>Formula:C22H28Cl2O4Purezza:99.79% - 99.87%Colore e forma:SolidPeso molecolare:427.36Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purezza:99.72% - 99.98%Colore e forma:Less Crystals Colourless CrystalsPeso molecolare:303.29Isoguvacine hydrochloride
CAS:<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Formula:C6H10ClNO2Purezza:99.59%Colore e forma:SolidPeso molecolare:163.6NS1652
CAS:<p>NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.</p>Formula:C15H11F3N2O3Purezza:99.62%Colore e forma:SolidPeso molecolare:324.25Ethaverine hydrochloride
CAS:Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Formula:C24H30ClNO4Purezza:99.66% - 99.90%Colore e forma:SolidPeso molecolare:431.96Ref: TM-T0369
2mg47,00€5mg66,00€10mg107,00€25mg177,00€50mg264,00€100mg378,00€200mg558,00€1mL*10mM (DMSO)89,00€CIQ
CAS:CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.Formula:C26H26ClNO5Purezza:99.5%Colore e forma:SolidPeso molecolare:467.94BI-749327
CAS:BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).Formula:C23H21F3N4O2Purezza:99.68% - 99.84%Colore e forma:SolidPeso molecolare:442.43Ref: TM-T10537
1mg133,00€2mg177,00€5mg274,00€10mg432,00€25mg630,00€50mg825,00€100mg1.103,00€500mg2.205,00€1mL*10mM (DMSO)301,00€Torsemide
CAS:<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Formula:C16H20N4O3SPurezza:99.81%Colore e forma:Crystalline SolidPeso molecolare:348.42NMDA-IN-1
CAS:<p>NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).</p>Formula:C20H23ClFN3OPurezza:99.57%Colore e forma:SolidPeso molecolare:375.87EN6
CAS:EN6, a small molecule, activates autophagy by modifying ATP6V1A, inhibiting mTORC1 and enhancing lysosomal function to clear TDP-43 aggregates.Formula:C19H14F2N4O2Purezza:95.74% - 97.04%Colore e forma:SolidPeso molecolare:368.34Ref: TM-T11191
1mg47,00€5mg88,00€10mg137,00€25mg205,00€50mg264,00€100mg400,00€500mg909,00€1mL*10mM (DMSO)70,00€Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purezza:99.96%Colore e forma:Crystals From Benzene SolidPeso molecolare:241.24Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Formula:C21H28ClNOPurezza:99.15% - 99.33%Colore e forma:Crystals Soluble In Methanol WaterPeso molecolare:345.91Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purezza:99.49%Colore e forma:SolidPeso molecolare:474.26γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purezza:99.95%Colore e forma:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecolare:103.12NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Formula:C17H16ClN7Purezza:99.55%Colore e forma:SolidPeso molecolare:353.81Flindokalner
CAS:Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.Formula:C16H10ClF4NO2Purezza:99.96%Colore e forma:SolidPeso molecolare:359.7Devapamil
CAS:Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.Formula:C26H36N2O3Purezza:99.63%Colore e forma:SolidPeso molecolare:424.58Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Formula:C17H27NO3·HClPurezza:99.15% - 99.61%Colore e forma:Crystals White Or Off White Crystalline PowderPeso molecolare:329.86Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Formula:C21H29N3OPurezza:99.62%Colore e forma:SolidPeso molecolare:339.47Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Formula:C13H9Cl2N3OSPurezza:98.87% - 99.74%Colore e forma:SolidPeso molecolare:326.2Ref: TM-T11076
1mg46,00€2mg59,00€5mg87,00€10mg140,00€25mg274,00€50mg510,00€100mg735,00€1mL*10mM (DMSO)96,00€Ciclopirox olamine
CAS:Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.Formula:C14H24N2O3Purezza:99.16% - >99.99%Colore e forma:White To Yellow Solid Solid Particulate/PowderPeso molecolare:268.353,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormula:C12H14O5Purezza:98.91%Colore e forma:SolidPeso molecolare:238.241-EBIO
CAS:1-EBIO (1-EBIO) is a calium channel agonist.Formula:C9H10N2OPurezza:98.75%Colore e forma:SolidPeso molecolare:162.19Manidipine dihydrochloride
CAS:Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Formula:C35H40Cl2N4O6Purezza:99.76% - 99.86%Colore e forma:SolidPeso molecolare:683.62NBQX disodium
CAS:NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.Formula:C12H6N4Na2O6SPurezza:97.32% - 97.6%Colore e forma:SolidPeso molecolare:380.2415Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurezza:98.97% - 99.83%Colore e forma:SolidPeso molecolare:365.83Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Formula:C13H21ClN2OPurezza:99.97%Colore e forma:Needles White Or Off White Crystalline PowderPeso molecolare:256.77Tocainide hydrochloride
CAS:<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Formula:C11H17ClN2OPurezza:97%Colore e forma:SolidPeso molecolare:228.72Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Formula:C18H28N2O·HClPurezza:99.89% - 99.9%Colore e forma:SolidPeso molecolare:324.89Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Formula:C16H17N2NaO4SPurezza:98.11%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:356.37Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purezza:99.89%Colore e forma:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Peso molecolare:155.19IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFormula:C31H32N4O2Purezza:98.9%Colore e forma:SolidPeso molecolare:492.61Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purezza:97.37%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:246.3BMS-394136
CAS:BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.Formula:C24H21Cl2FN4OPurezza:98.59% - 99.95%Colore e forma:SolidPeso molecolare:471.35T16Ainh-A01
CAS:T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.Formula:C19H20N4O3S2Purezza:97.18% - 98.15%Colore e forma:SolidPeso molecolare:416.52Ref: TM-T13059
1mg35,00€5mg66,00€10mg97,00€25mg183,00€50mg280,00€100mg425,00€200mg615,00€1mL*10mM (DMSO)87,00€Z433927330
CAS:<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Formula:C20H20N4O3Purezza:99.78%Colore e forma:SolidPeso molecolare:364.4Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurezza:99.56%Colore e forma:SolidPeso molecolare:596.76Ref: TM-T15775
1mg44,00€2mg58,00€5mg94,00€10mg144,00€25mg335,00€50mg550,00€100mg882,00€200mg1.188,00€1mL*10mM (DMSO)111,00€Moxidectin
CAS:Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.Formula:C37H53NO8Purezza:97.38%Colore e forma:Appearance White Or Pale Yellow Amorphous PowderPeso molecolare:639.82Dibucaine
CAS:Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.Formula:C20H29N3O2Purezza:99.698% - 99.88%Colore e forma:Colorless Or Almost Colorless Powder SolidPeso molecolare:343.46FFN 206 dihydrochloride
CAS:<p>FFN 206 dihydrochloride: fluorescent VMAT2 marker, detects subcellular sites, non-inhibitory to DAT.</p>Formula:C12H15ClN2O2Purezza:98.96% - >99.99%Colore e forma:SolidPeso molecolare:254.71Ethosuximide
CAS:Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied byFormula:C7H11NO2Purezza:98.87% - 99.72%Colore e forma:Crystals From Acetone And Ether SolidPeso molecolare:141.17Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Formula:C9H17NO3Purezza:99.87%Colore e forma:SolidPeso molecolare:187.24DMT1 blocker 2
CAS:Compound 12f, a DMT1 blocker, inhibits DMT1 with a 0.83 IC50, potentially blocking intestinal iron absorption.Formula:C16H13N3OPurezza:99.68%Colore e forma:SolidPeso molecolare:263.29Ref: TM-T11064
1mg92,00€5mg188,00€10mg354,00€25mg597,00€50mg852,00€100mg1.159,00€1mL*10mM (DMSO)215,00€Domperidone EP Impurity A
CAS:Domperidone EP Impurity A is used as pharmaceutical intermediates.Formula:C12H14ClN3OPurezza:99.97%Colore e forma:SolidPeso molecolare:251.71Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:179.22γ-DGG acetate(6729-55-1 free base)
CAS:gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.Formula:C9H16N2O7Purezza:99.81%Colore e forma:SolidPeso molecolare:264.23GET73
CAS:GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.Formula:C13H16F3NO2Purezza:99.54%Colore e forma:SolidPeso molecolare:275.27Ref: TM-T11393
5mg42,00€10mg59,00€25mg110,00€50mg166,00€100mg243,00€200mg359,00€1mL*10mM (DMSO)47,00€Etimizol
CAS:Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.Formula:C9H14N4O2Purezza:99%Colore e forma:SolidPeso molecolare:210.23Oxybuprocaine hydrochloride
CAS:Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.Formula:C17H29ClN2O3Purezza:>99.99%Colore e forma:White Crystalline PowderPeso molecolare:344.88Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Formula:C106H175N35O24S4Purezza:98.06% - 98.09%Colore e forma:SolidPeso molecolare:2452Glimepiride
CAS:Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.Formula:C24H34N4O5SPurezza:97.84% - 98.87%Colore e forma:White Cyrstalline SolidPeso molecolare:490.62CGP37157
CAS:CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release fromFormula:C15H11Cl2NOSPurezza:99.92%Colore e forma:SolidPeso molecolare:324.22Butamben
CAS:Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Formula:C11H15NO2Purezza:99.43%Colore e forma:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Peso molecolare:193.24Trichlormethiazide
CAS:Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.Formula:C8H8Cl3N3O4S2Purezza:98.8% - 99.54%Colore e forma:SolidPeso molecolare:380.66D-AP5
CAS:D-AP5 (D-APV) is a NMDA receptor antagonist.Formula:C5H12NO5PPurezza:98.77% - >99.99%Colore e forma:White Fine Crystalline PowderPeso molecolare:197.13N-Acetylprocainamide
CAS:N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmicFormula:C15H23N3O2Purezza:99.65% - 99.74%Colore e forma:SolidPeso molecolare:277.36AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Formula:C23H34N4O5Purezza:98.42% - 98.51%Colore e forma:SoildPeso molecolare:446.54GsMTx4
CAS:GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).Formula:C185H273N49O45S6Purezza:98%Colore e forma:SolidPeso molecolare:4095.84AChE/Aβ-IN-1
AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting theFormula:C20H25BrN4Colore e forma:SolidPeso molecolare:401.34EVT-401
EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].Formula:C22H20F4N2O3Colore e forma:SolidPeso molecolare:436.4Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formula:C17H13N5O2Colore e forma:SolidPeso molecolare:319.32Elgodipine
CAS:Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formula:C29H33FN2O6Purezza:99.84% - 99.98%Colore e forma:SolidPeso molecolare:524.58Apamin acetate
Apamin acetate: Selective Ca2+-activated K+ channel blocker, 18-amino acid bee venom peptide, promotes synapse repair, anti-inflammatory.Purezza:96.97%Colore e forma:SolidMambalgin 1
CAS:ASIC1a inhibitor; IC50: 192 nM (human), 72 nM (dimer); inactive channel binding; selective; pain response delay.Formula:C272H429N85O84S10Purezza:98%Colore e forma:SolidPeso molecolare:6554.51(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Formula:C6H11NO2Colore e forma:SolidPeso molecolare:129.163-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Formula:C3H10NO2PColore e forma:SolidPeso molecolare:123.092Leptomycin A
CAS:<p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>Formula:C32H46O6Purezza:98%Colore e forma:SolidPeso molecolare:526.7Cavα2δ-IN-1
CAS:Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a KiFormula:C18H27N5OColore e forma:SolidPeso molecolare:329.448TRPA1-IN-1
CAS:TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.Formula:C19H17ClN6O3Colore e forma:SolidPeso molecolare:412.83CHET3
CAS:CHET3 is a highly selective allosteric activator for TASK-3-containing K2P channels. CHET3 has shown potent in vivo analgesic effects. Cost-effective and quality-assured.Formula:C21H21N5O3SPurezza:98.28% - 99.92%Colore e forma:SoildPeso molecolare:423.49LY-466195
CAS:LY-466195 is a competitive antagonist of GLUK5 receptor.Formula:C16H24F2N2O4Colore e forma:SolidPeso molecolare:346.37BeKm-1
CAS:Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.Formula:C174H261N51O52S6Purezza:98%Colore e forma:SolidPeso molecolare:4091.65Huwentoxin I
CAS:Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.Formula:C161H246N48O44S6Purezza:98%Colore e forma:SolidPeso molecolare:3750.36GpTx-1 TFA
GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.Colore e forma:Odour SolidWAY-326766
CAS:WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).Formula:C21H23N3O5Purezza:99.87%Colore e forma:SolidPeso molecolare:397.42TP-050
CAS:TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.Formula:C16H15ClF2N6OColore e forma:SolidPeso molecolare:380.78Cevadine
Cevadine is a natural product that can be used as a reference standard.Formula:C32H49NO9Colore e forma:SolidPeso molecolare:591.742Atagabalin
CAS:Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Formula:C10H19NO2Colore e forma:SolidPeso molecolare:185.26TRPA1 Antagonist 3
CAS:TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.Formula:C11H8ClN3Colore e forma:SolidPeso molecolare:217.6617α-Hydroxywithanolide D
<p>17alpha-Hydroxywithanolide D is an allosteric modulator of the NMDA receptor, with an IC50 of 44.24 nM. This compound exhibits neuroprotective properties and can be utilized in Alzheimer's disease research.</p>Formula:C28H46O7Colore e forma:SolidPeso molecolare:494.661Chlorotoxin TFA
Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.Formula:C160H250F3N53O49S11Colore e forma:SolidPeso molecolare:4109.74Hyp9
CAS:Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].Formula:C18H26O5Colore e forma:SolidPeso molecolare:322.40Homocarnosine
CAS:Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.Formula:C10H16N4O3Colore e forma:SolidPeso molecolare:240.26JAMI1001A
CAS:JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.Formula:C16H17F3N4O3SColore e forma:SolidPeso molecolare:402.39AChE/Aβ-IN-2
AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.Formula:C20H25ClN4Colore e forma:SolidPeso molecolare:356.89SLC26A3-IN-2
CAS:Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.Formula:C19H13ClN2O2SPurezza:99.86%Colore e forma:SolidPeso molecolare:368.8417(S)-HETE
CAS:<p>Arachidonic acid and its CYP450 metabolite, 17(S)-HETE, regulate kidney electrolytes; 17(S)-HETE reduces proximal tubule ATPase activity by 70% at 2 μM.</p>Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.473Anticonvulsant agent 9
Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.Formula:C22H24N4O2Colore e forma:SolidPeso molecolare:376.45Crofelemer
CAS:Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.Colore e forma:SolidIdactamab
CAS:Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.Purezza:> 95%Colore e forma:LiquidPeso molecolare:146.2 kDaAmpullosporin A
CAS:Ampullosporin A is a peptaibol-type polypeptide isolated from the fungus Sepedonium ampullosporum (HKI-0053), exhibiting neuromodulatory activity. It inhibits hyperactivity induced by the NMDA receptor antagonist MK-801 and ameliorates social behavior abnormalities caused by subchronic ketamine treatment. Ampullosporin A modulates glutamate receptor activity without affecting dopamine D1 and D2 receptors.Formula:C77H127N19O19Colore e forma:SolidPeso molecolare:1622.95Levamlodipine besylate Hemipentahydrate
CAS:<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formula:C20H25ClN2O5·C6H6O3SH2OColore e forma:SolidPeso molecolare:1224.18Analgesic/antidepressant agent-1
<p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>Formula:C22H25ClN2O2Colore e forma:SolidPeso molecolare:384.9α,β-Methylene-ATP dilithium
CAS:α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.Formula:C11H16Li2N5O12P3Colore e forma:SolidPeso molecolare:517.07
