
Apoptose
Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.
Subcategorias de "Apoptose"
- ASK(6 produtos)
- BCL(11 produtos)
- Caspase(125 produtos)
- FOXO1(3 produtos)
- IAP(66 produtos)
- Mdm2(12 produtos)
- PD-1/PD-L1(125 produtos)
- PDK(9 produtos)
- PERK(25 produtos)
- Serina/treonina quinase(15 produtos)
- Survivina(13 produtos)
- TNF(92 produtos)
- c-RET(51 produtos)
- p53(62 produtos)
Exibir 6 mais subcategorias
Foram encontrados 5599 produtos de "Apoptose"
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Mocetinostat
CAS:<p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>Fórmula:C23H20N6OPureza:99% - 99.21%Cor e Forma:SolidPeso molecular:396.44AG1024
CAS:<p>AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).</p>Fórmula:C14H13BrN2OPureza:98% - 99.37%Cor e Forma:SolidPeso molecular:305.17WHI-P154
CAS:<p>WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.</p>Fórmula:C16H14BrN3O3Pureza:98% - 99.67%Cor e Forma:SolidPeso molecular:376.2Taurolidine
CAS:<p>Taurolidine is a synthetic taurine analog with antimicrobial and anti-neoplastic actions. It displays broad bactericidal and fungicidal activity.</p>Fórmula:C7H16N4O4S2Pureza:99.79% - 99.81%Cor e Forma:SolidPeso molecular:284.36Topotecan
CAS:<p>Topotecan (NSC-609669) is a Topoisomerase I inhibitor,and is an antineoplastic agent used to treat ovarian cancer that works by inhibiting DNA topoisomerases.</p>Fórmula:C23H23N3O5Pureza:96.14% - 98.23%Cor e Forma:Light Yellow Needle Crystal Or Crystalline PowderPeso molecular:421.45Inauhzin
CAS:<p>Inauhzin (INZ) reactivates p53, inhibits SIRT1, induces Y cell apoptosis without genotoxic stress (IC50=3 uM in A549).</p>Fórmula:C25H19N5OS2Pureza:98% - 99.36%Cor e Forma:SolidPeso molecular:469.58Bafetinib
CAS:<p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>Fórmula:C30H31F3N8OPureza:94.16% - 99.68%Cor e Forma:SolidPeso molecular:576.62Sertaconazole
CAS:<p>Sertaconazole is a broad-spectrum antifungal.</p>Fórmula:C20H15Cl3N2OSPureza:99.483%Cor e Forma:SolidPeso molecular:437.77Azoramide
CAS:<p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>Fórmula:C15H17ClN2OSPureza:99.08% - 99.85%Cor e Forma:SolidPeso molecular:308.83Thalidomide-5-methyl
CAS:<p>Thalidomide-5-methyl is the Thalidomide-based cereblon (CRBN) ligand. Thalidomide-5-methyl is used in the recruitment of CRBN protein.</p>Fórmula:C14H12N2O4Pureza:99.48%Cor e Forma:SolidPeso molecular:272.26S63845
CAS:<p>S63845 is a selective myeloid leukemia 1(MCL1) inhibitor that binds to human MCL1 with a Kd of 0.19 nM.Cost-effective and quality-assured.</p>Fórmula:C39H37ClF4N6O6SPureza:97.7% - ≥98%Cor e Forma:SolidPeso molecular:829.26Ciprofloxacin hydrochloride monohydrate
CAS:<p>Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) is a fluoroquinolone antibiotic with potent antibacterial activity.</p>Fórmula:C17H21ClFN3O4Pureza:99.23% - 99.85%Cor e Forma:White Or Yellowish Crystalline PowderPeso molecular:385.82Y-27632 dihydrochloride
CAS:<p>View and buy Y-27632 dihydrochloride from TargetMol.Y-27632 is a selective inhibitor of ROCKs.Cited in 10 publications.</p>Fórmula:C14H21N3O·2HClPureza:97.96% - 99.98%Cor e Forma:SolidPeso molecular:320.26Tenovin-3
CAS:<p>Tenovin-3 acts as a p53 activator.</p>Fórmula:C18H21N3OSPureza:99.72% - ≥95%Cor e Forma:SolidPeso molecular:327.44Rigosertib
CAS:<p>Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by disrupting PI3K/Akt.</p>Fórmula:C21H25NO8SPureza:99.53%Cor e Forma:SolidPeso molecular:451.49Dapivirine
CAS:<p>Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C20H19N5Pureza:98% - 99.77%Cor e Forma:SolidPeso molecular:329.4Demethoxycurcumin
CAS:<p>Demethoxycurcumin: antioxidant, anti-inflammatory, anti-proliferative, anti-acanthamoebic, enhances chemo for resistant cancers, inhibits cancer pathways.</p>Fórmula:C20H18O5Pureza:94.54% - 99.86%Cor e Forma:SolidPeso molecular:338.35A-419259
CAS:<p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>Fórmula:C29H34N6OPureza:99.48%Cor e Forma:SolidPeso molecular:482.62PI-103
CAS:<p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>Fórmula:C19H16N4O3Pureza:97.79% - 99.3%Cor e Forma:SolidPeso molecular:348.36PKD-IN-1 dihydrochloride (956121-30-5 free base)
CAS:<p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>Fórmula:C18H21Cl3N4OPureza:99.5%Cor e Forma:SolidPeso molecular:415.75ML311
CAS:<p>ML311 is a selective inhibitor of the Mcl-1/Bim interaction.</p>Fórmula:C23H24F3N3OPureza:99.75%Cor e Forma:SolidPeso molecular:415.45Tauroursodeoxycholate
CAS:<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Fórmula:C26H45NO6SPureza:98.77% - 99.93%Cor e Forma:White SolidPeso molecular:499.7PEAQX
CAS:<p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>Fórmula:C17H17BrN3O5PPureza:98% - 99.9%Cor e Forma:SolidPeso molecular:454.21AR42
CAS:<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Fórmula:C18H20N2O3Pureza:98.46% - 98.96%Cor e Forma:SolidPeso molecular:312.36Asiaticoside
CAS:<p>Asiaticoside, in Centella asiatica, may treat wounds/burns.</p>Fórmula:C48H78O19Pureza:98% - 99.96%Cor e Forma:PowderPeso molecular:959.12Emricasan
CAS:<p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>Fórmula:C26H27F4N3O7Pureza:98.13% - 99%Cor e Forma:SolidPeso molecular:569.5Aloperine
CAS:<p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>Fórmula:C15H24N2Pureza:98% - 99.88%Cor e Forma:Yellow Crystalline PowderPeso molecular:232.361400W dihydrochloride
CAS:<p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>Fórmula:C10H17Cl2N3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:250.17SC66
CAS:<p>SC66 is a AKT inhibitor in HepG2, HA22T/VGH, and PLC/PRF/5 cells (IC50: about 0.75 μg/ml, at 72 h).</p>Fórmula:C18H16N2OPureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:276.33Bilobalide
CAS:<p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>Fórmula:C15H18O8Pureza:98.81% - 99.92%Cor e Forma:White SolidPeso molecular:326.3Rhosin hydrochloride
CAS:<p>Rhosin hydrochloride is a specific inhibitor of the RhoA subfamily Rho GTPases.Cost-effective and quality-assured.</p>Fórmula:C20H20Cl2N6OPureza:97.33% - 98.92%Cor e Forma:SolidPeso molecular:431.318Nω-Hydroxy-nor-L-Arginine Dihydrochloride
CAS:<p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>Fórmula:C5H14Cl2N4O3Pureza:99.12% - 99.84%Cor e Forma:SolidPeso molecular:249.10Thalidomide-NH-PEG1-NH2 hydrochloride
CAS:<p>Thalidomide-NH-PEG1-NH2 hydrochloride (4-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione HCl) is a synthetic E3 ligase ligand-</p>Fórmula:C17H21ClN4O5Pureza:97.13%Cor e Forma:SolidPeso molecular:396.83UTL-5g
CAS:<p>UTL-5g is a chemoprotective TNF-α inhibitor reducing cisplatin side effects and toxicity in liver, kidneys, and blood.</p>Fórmula:C11H8Cl2N2O2Pureza:99.83%Cor e Forma:SolidPeso molecular:271.1Tetrahydroxyquinone monohydrate
CAS:<p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>Fórmula:C6H6O7Cor e Forma:SolidPeso molecular:190.11Nobiletin
CAS:<p>Nobiletin: a citrus-derived flavone with anti-inflammatory and anti-cancer properties; water-insoluble, very weak acid.</p>Fórmula:C21H22O8Pureza:98.65% - 99.76%Cor e Forma:SolidPeso molecular:402.39Alda-1
CAS:<p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>Fórmula:C15H11Cl2NO3Pureza:98.5% - 99.63%Cor e Forma:SolidPeso molecular:324.16CCCP
CAS:<p>CCCP blocks STING activation, TBK1, IRF3 signaling, and IFN-β production by disrupting MMP.</p>Fórmula:C9H5ClN4Pureza:97.15% - 99.64%Cor e Forma:Yellow To Orange PowderPeso molecular:204.62PD173955
CAS:<p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>Fórmula:C21H16Cl2N4OSPureza:98.52% - 98.99%Cor e Forma:SolidPeso molecular:443.35RGX-202
CAS:<p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>Fórmula:C4H9N3O2Pureza:99.67% - 99.8%Cor e Forma:SolidPeso molecular:131.13Neobavaisoflavone
CAS:<p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>Fórmula:C20H18O4Pureza:99.31% - 99.87%Cor e Forma:SolidPeso molecular:322.35Ibandronate sodium monohydrate
CAS:<p>Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.</p>Fórmula:C9H24NNaO8P2Pureza:99.62%Cor e Forma:White Crystalline PowderPeso molecular:359.23HA15
CAS:<p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>Fórmula:C23H22N4O3S2Pureza:99.77% - 99.86%Cor e Forma:SolidPeso molecular:466.58NADPH tetracyclohexanamine
CAS:<p>NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.</p>Fórmula:C45H82N11O17P3Pureza:98.73% - 99.05%Cor e Forma:SolidPeso molecular:1142.12Obatoclax Mesylate
CAS:Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, andFórmula:C20H19N3O·CH4O3SPureza:99.58% - 99.88%Cor e Forma:SolidPeso molecular:413.49Idasanutlin
CAS:<p>Idasanutlin (Ro 5503781) (RG-7388) is an effective and specific p53-MDM2 inhibitor (IC50: 6 nM).</p>Fórmula:C31H29Cl2F2N3O4Pureza:99.13% - 99.88%Cor e Forma:SolidPeso molecular:616.48Eriocitrin
CAS:<p>Eriocitrin: an antioxidative flavonoid; reduces exercise-induced oxidative damage and lipids; fights fatty liver and inhibits carbonic anhydrase VA.</p>Fórmula:C27H32O15Pureza:98.41% - 99.11%Cor e Forma:SolidPeso molecular:596.53CHR-6494 TFA
CAS:<p>CHR-6494 TFA: potent haspin inhibitor (IC50=2 nM), blocks H3T3 phosphorylation, triggers apoptosis in cancer cells. Used for cancer research.</p>Fórmula:C18H17F3N6O2Pureza:99.50%Cor e Forma:SolidPeso molecular:406.36CA-4948
CAS:<p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>Fórmula:C24H25N7O5Pureza:99.35% - 99.88%Cor e Forma:SolidPeso molecular:491.5Tenovin-6
CAS:<p>Tenovin-6 is a p53 transcriptional activity agonist.</p>Fórmula:C25H34N4O2SPureza:97.71% - >99.99%Cor e Forma:SolidPeso molecular:454.63Trabectedin
CAS:<p>Trabectedin (Ecteinascidin 743) has potent antitumor activity and the potential for soft tissue sarcoma and ovarian cancer research.</p>Fórmula:C39H43N3O11SPureza:≥98%Cor e Forma:SolidPeso molecular:761.84CPTH2
CAS:<p>CPTH2 is a histone acetyltransferase inhibitor modulating Gcn5 network.</p>Fórmula:C14H14ClN3SPureza:99.81%Cor e Forma:SolidPeso molecular:291.8ZMC1
CAS:<p>NSC-319726 (ZMC1), a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).</p>Fórmula:C11H14N4SPureza:98.97% - 99.76%Cor e Forma:SolidPeso molecular:234.32MPTP hydrochloride
CAS:<p>MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.</p>Fórmula:C12H16ClNPureza:96.35% - >99.99%Cor e Forma:SolidPeso molecular:209.72FOXO4-DRI acetate
<p>FOXO4-DRI acetate is a bioactive chemical.</p>Fórmula:C36H64N14O14SPureza:99.10%Cor e Forma:SolidPeso molecular:5358.06Choline
CAS:<p>Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins</p>Fórmula:C5H15NO2Pureza:99.97% - ≥98%Cor e Forma:LiquidPeso molecular:121.18Periplocin
CAS:<p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>Fórmula:C36H56O13Pureza:99.66% - 99.74%Cor e Forma:SolidPeso molecular:696.82RAD51 Inhibitor B02
CAS:<p>RAD51 Inhibitor B02 (B02) (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM.</p>Fórmula:C22H17N3OPureza:99.72% - 99.89%Cor e Forma:SolidPeso molecular:339.39Salubrinal
CAS:<p>Salubrinal, a phosphatases (PP1) inhibitor(IC50=1.7 μM), exhibits function on the eukaryotic translation initiation factor 2 subunit (eIF2α).</p>Fórmula:C21H17Cl3N4OSPureza:97.25% - >99.99%Cor e Forma:SolidPeso molecular:479.81Bendamustine
CAS:<p>Bendamustine (SDX105) for the treatment of Non-Hodgkin Lymphomas and Chronic Lymphocytic Leukemia</p>Fórmula:C16H21Cl2N3O2Pureza:≥98%Cor e Forma:SolidPeso molecular:358.26TrxR1-IN-B19
CAS:<p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>Fórmula:C21H22O5Pureza:98.6%Cor e Forma:SolidPeso molecular:354.4Sertaconazole nitrate
CAS:<p>Sertaconazole nitrate, a broad-spectrum topical antifungal, treats skin and mucosal infections.</p>Fórmula:C20H15Cl3N2OS·HNO3Pureza:98.66% - 99.65%Cor e Forma:SolidPeso molecular:500.78Thalidomide-O-amido-C3-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>Fórmula:C20H21F3N4O8Pureza:98.47%Cor e Forma:SolidPeso molecular:502.4Thalidomide-O-COOH
CAS:<p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>Fórmula:C15H12N2O7Pureza:98% - 98.29%Cor e Forma:SolidPeso molecular:332.27Polygalacin D
CAS:<p>Polygalacin D shows anti- proliferation, anti-inflammary, and hepatoprotective activities, it can inhibit the expression of lipopolysaccharide (LPS)-induced</p>Fórmula:C57H92O27Pureza:98.95% - ≥98%Cor e Forma:SolidPeso molecular:1209.4Almorexant
CAS:<p>Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for OX1 and 0.17 nM for OX2.</p>Fórmula:C29H31F3N2O3Pureza:97.75% - 98.02%Cor e Forma:SolidPeso molecular:512.56m-3M3FBS
CAS:<p>m-3M3FBS is a phospholipase C (PLC) activator.</p>Fórmula:C16H16F3NO2SPureza:99.66%Cor e Forma:SolidPeso molecular:343.36Grape Seed Extract
CAS:<p>Grape Seed Extract (Grape Seed P.E.) is exudate from seeds of the grape plant Vitis vinifera, composed of oils and secondary plant metabolites.</p>Fórmula:C32H30O11Pureza:98%Cor e Forma:SolidPeso molecular:590.581ENMD-2076
CAS:<p>ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.</p>Fórmula:C21H25N7Pureza:97.63% - ≥95%Cor e Forma:SolidPeso molecular:375.47CVT-11127
CAS:<p>CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.</p>Fórmula:C25H23Cl2N5O3Pureza:98.32%Cor e Forma:SolidPeso molecular:512.39Vesatolimod
CAS:<p>Vesatolimod (GS-9620) is an effective and specific orally active agonist of Toll-like receptor 7.</p>Fórmula:C22H30N6O2Pureza:97.46% - 99.03%Cor e Forma:SolidPeso molecular:410.51IC261
CAS:<p>IC261 (SU-5607) is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for Cdk5 is 4.5 mM.</p>Fórmula:C18H17NO4Pureza:99.45% - 99.91%Cor e Forma:SolidPeso molecular:311.33Methoxychlor
CAS:<p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>Fórmula:C16H15Cl3O2Pureza:98.82% - ≥95%Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment IfPeso molecular:345.65Delanzomib
CAS:<p>Delanzomib (CEP-18770) is an oral proteasome inhibitor with an IC50 of 3.8 nM, targeting chymotrypsin-like activity with minimal effect on other activities.</p>Fórmula:C21H28BN3O5Pureza:95.52% - 99.46%Cor e Forma:SolidPeso molecular:413.28Gardenin B
CAS:<p>Gardenin B exhibits superior antiproliferative activity against lung, breast, colon, hepatic and leukaemia cell lines as well as in keratinocytes .</p>Fórmula:C19H18O7Pureza:98.80% - 99.74%Cor e Forma:SolidPeso molecular:358.34N-Ethylmaleimide
CAS:<p>N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor. Cost-effective and quality-assured.</p>Fórmula:C6H7NO2Pureza:99.50%Cor e Forma:White SolidPeso molecular:125.13Salvigenin
CAS:<p>Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.</p>Fórmula:C18H16O6Pureza:99.17% - 99.78%Cor e Forma:SolidPeso molecular:328.32Cucurbitacin IIA
CAS:<p>1.</p>Fórmula:C32H50O8Pureza:98.62% - 99.87%Cor e Forma:SolidPeso molecular:562.73Infigratinib
CAS:<p>Infigratinib (NVP-BGJ398) (BGJ398) is an orally bioavailable pan FGFR inhibitor (IC50: 0.9/1.4/1 nM for FGFR1/2/3), >40-fold selective for FGFR versus FGFR4 and</p>Fórmula:C26H31Cl2N7O3Pureza:98% - 98.97%Cor e Forma:SolidPeso molecular:560.48CCPA
CAS:<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Fórmula:C15H20ClN5O4Pureza:99.1%Cor e Forma:Off-White To Light Yellow SolidPeso molecular:369.8OSI-930
CAS:<p>OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.</p>Fórmula:C22H16F3N3O2SPureza:99.67%Cor e Forma:SolidPeso molecular:443.44GSK778 hydrochloride
CAS:<p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>Fórmula:C30H34ClN5O3Pureza:97.26% - 98.35%Cor e Forma:SolidPeso molecular:548.08Thalidomide-4-OH
CAS:<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Fórmula:C13H10N2O5Pureza:99.59%Cor e Forma:SolidPeso molecular:274.23Difurazon hydrochloride
CAS:<p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>Fórmula:C14H13ClN6O6Pureza:98.51%Cor e Forma:SolidPeso molecular:396.74Methoxyamine HCl
CAS:<p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>Fórmula:CH6ClNOPureza:≥98%Cor e Forma:SolidPeso molecular:83.51Sal003
CAS:<p>Sal003, an effective cell-permeable analog, inhibitis the eIF2α phosphatase.</p>Fórmula:C18H15Cl4N3OSPureza:99.17% - 99.77%Cor e Forma:SolidPeso molecular:463.21Momordin Ic
CAS:<p>Momordin Ic (Momordin 1c) might represent a potential anticancer activity, by inducing apoptosis through oxidative stress-regulated mitochondrial dysfunction</p>Fórmula:C41H64O13Pureza:98% - 99.69%Cor e Forma:SolidPeso molecular:764.94Neferine
CAS:<p>Neferine: anti-tumor, enhances DOX efficacy, prevents diabetic vasculopathy; mediates via CYP3A4, GSH depletion, blocks ROS/Akt/NF-κB.</p>Fórmula:C38H44N2O6Pureza:98.81% - 99.65%Cor e Forma:SolidPeso molecular:624.77PKR-IN-C16
CAS:<p>PKR-IN-C16: inhibits PKR autophosphorylation and translation blockade; binds ATP site; IC50 of 186-210 nM; protects cells from ER stress damage.</p>Fórmula:C13H8N4OSPureza:97.8%Cor e Forma:SolidPeso molecular:268.29Alogliptin Benzoate
CAS:<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Fórmula:C25H27N5O4Pureza:99.94% - >99.99%Cor e Forma:White PowderPeso molecular:461.51Levomenol
CAS:<p>Levomenol, or (-)-α-Bisabolol, is a sesquiterpene in aromatic plant oils with antioxidant, anti-inflammatory, and anti-apoptotic properties.</p>Fórmula:C15H26OPureza:96.01%Cor e Forma:Clear To Yellowish LiquidPeso molecular:222.37SC144
CAS:<p>SC144 is an orally active small-molecule gp130 inhibitor.</p>Fórmula:C16H11FN6OPureza:99.20%Cor e Forma:SolidPeso molecular:322.3PIK-75
CAS:<p>PIK-75, a DNA-PK and PI3K inhibitor, suppresses DNA-PK(IC50=2 nM), p110α(IC50=5.8 nM) and p110γ(IC50=76 nM).</p>Fórmula:C16H14BrN5O4SPureza:98.52% - >99.99%Cor e Forma:SolidPeso molecular:452.28Pectolinarin
CAS:<p>Pectolinarin is a Cirsium isolate with anti-inflammatory activity.</p>Fórmula:C29H34O15Pureza:98% - 99.79%Cor e Forma:SolidPeso molecular:622.57Epibrassinolide
CAS:<p>Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator with</p>Fórmula:C28H48O6Pureza:97.57% - 98.11%Cor e Forma:SolidPeso molecular:480.68KRCA-0008
CAS:<p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>Fórmula:C30H37ClN8O4Pureza:96.19%Cor e Forma:SolidPeso molecular:609.12Perhexiline
CAS:<p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>Fórmula:C19H35NCor e Forma:SolidPeso molecular:277.49Ketorolac hemicalcium
CAS:<p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation & pain, used in cancer research.</p>Fórmula:C30H24CaN2O6Cor e Forma:SolidPeso molecular:548.608Thalidomide-propargyl
CAS:<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Fórmula:C16H12N2O5Pureza:95.14%Cor e Forma:SolidPeso molecular:312.28Thalidomide-NH-C6-NH2 hydrochloride
CAS:<p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>Fórmula:C19H25ClN4O4Pureza:99.27%Cor e Forma:SolidPeso molecular:408.88Britannin
CAS:<p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>Fórmula:C19H26O7Pureza:98% - 99.98%Cor e Forma:SolidPeso molecular:366.41PK11000
CAS:<p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>Fórmula:C6H5ClN2O4SPureza:99.70%Cor e Forma:SolidPeso molecular:236.63Abacavir monosulfate
CAS:<p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>Fórmula:C14H20N6O5SCor e Forma:SolidPeso molecular:384.41Tanespimycin
CAS:<p>Tanespimycin (KOS 953) is an Hsp90 inhibitor (IC50=5 nM) and is selective. Tanespimycin depletes intracellular STK38/NDR1. High-Quality, Low-Cost!</p>Fórmula:C31H43N3O8Pureza:99.07% - 99.83%Cor e Forma:Dark Purple SolidPeso molecular:585.69Benidipine hydrochloride
CAS:<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Fórmula:C28H32ClN3O6Pureza:99.80%Cor e Forma:SolidPeso molecular:542.032-tert-Butyl-1,4-benzoquinone
CAS:<p>TBQ, a BHA metabolite, activates Nrf2 and S-arylates Keap1 in RAW264.7 cells.</p>Fórmula:C10H12O2Pureza:97.19%Cor e Forma:SolidPeso molecular:164.2Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Fórmula:C23H27F3N4O10Pureza:95.74% - 99%Cor e Forma:SolidPeso molecular:576.48Tasisulam
CAS:<p>Tasisulam (LY573636) is an apoptosis inducer and an antitumor agent via the intrinsic pathway.</p>Fórmula:C11H6BrCl2NO3S2Pureza:99% - >99.99%Cor e Forma:SolidPeso molecular:415.11MS7972
CAS:<p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>Fórmula:C14H13NO2Pureza:99.78%Cor e Forma:SolidPeso molecular:227.26RO8994
CAS:<p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>Fórmula:C31H31Cl2FN4O4Pureza:99.31% - 99.44%Cor e Forma:SolidPeso molecular:613.51KX2-361
CAS:<p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>Fórmula:C24H24FN3O2Pureza:99.64% - 99.68%Cor e Forma:SolidPeso molecular:405.46AZ 628
CAS:<p>AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM, 34 nM and 29 nM, also inhibits VEGFR2, DDR2, Lyn, Flt1, FMS, etc.</p>Fórmula:C27H25N5O2Pureza:99.50%Cor e Forma:SolidPeso molecular:451.52Capsazepine
CAS:<p>Capsazepine, a TRPV1 antagonist (IC50: 562 nM), blocks capsaicin-induced heat pain.</p>Fórmula:C19H21ClN2O2SPureza:98% - 99.78%Cor e Forma:White To Off-White PowderPeso molecular:376.9Quizartinib
CAS:<p>Quizartinib (AC220) is an inhibitor of FLT3 (Kd: 1.6 nM) and demonstrates high selectivity for FLT3 when tested against a panel of 227 additional kinases.</p>Fórmula:C29H32N6O4SPureza:98% - 99.42%Cor e Forma:SolidPeso molecular:560.67Ralimetinib dimesylate
CAS:<p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>Fórmula:C24H29FN6·2CH4O3SPureza:98% - 99.38%Cor e Forma:SolidPeso molecular:612.74(1E,6E)-Bis(demethoxy)curcumin
CAS:<p>(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) is a natural demethoxy derivative of curcumin,with anti-inflammatory and anti-cancer activities.</p>Fórmula:C19H16O4Pureza:97.45%Cor e Forma:SolidPeso molecular:308.33Genistein
CAS:<p>Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has antitumor effects. Cost effective and quality assured.</p>Fórmula:C15H10O5Pureza:98.22% - 99.64%Cor e Forma:Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether SolidPeso molecular:270.24Crebanine
CAS:<p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>Fórmula:C20H21NO4Pureza:99.17% - 99.77%Cor e Forma:SolidPeso molecular:339.39DEL-22379
CAS:<p>DEL-22379 is a water-soluble ERK dimerization inhibitor with IC50 of ~0.5 μM.</p>Fórmula:C26H28N4O3Pureza:99.3% - 99.53%Cor e Forma:SolidPeso molecular:444.53Caudatin
CAS:<p>Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.</p>Fórmula:C28H42O7Pureza:98.83% - 99.9%Cor e Forma:SolidPeso molecular:490.63Rabeprazole sodium
CAS:<p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>Fórmula:C18H20N3NaO3SPureza:98% - 99.912%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:381.42Taurochenodeoxycholic acid sodium
CAS:<p>Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).</p>Fórmula:C26H44NNaO6SPureza:98.23% - 99.45%Cor e Forma:White To Off-White PowderPeso molecular:521.68Pifithrin-α hydrobromide
CAS:<p>Pifithrin-α hydrobromide (Pifithrin-α hydrobromide) is a p53 inhibitor, inhibiting p53-dependent transactivation of p53-responsive genes.</p>Fórmula:C16H18N2OS·HBrPureza:97.71% - >99.99%Cor e Forma:SolidPeso molecular:367.3Stattic
CAS:<p>Stattic (STAT3 Inhibitor V) is a STAT3 inhibitor (IC50=5.1 μM) that selectively inhibits STAT3 activation, dimerization, and nuclear translocation.</p>Fórmula:C8H5NO4SPureza:98.32% - 99.76%Cor e Forma:SolidPeso molecular:211.19GSK-J4
CAS:<p>GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.</p>Fórmula:C24H27N5O2Pureza:98.24% - 99.98%Cor e Forma:SolidPeso molecular:417.5Mitochonic acid 5
CAS:<p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>Fórmula:C18H13F2NO3Pureza:98.85%Cor e Forma:SolidPeso molecular:329.3Angelicin
CAS:<p>Angelicin (Isopsoralen), is a furanocoumarin with anti-Y, antiviral, anti-inflammatory activity.</p>Fórmula:C11H6O3Pureza:99.86% - 99.89%Cor e Forma:White SolidPeso molecular:186.16Mdivi-1
CAS:<p>Mdivi-1 (Mitochondrial division inhibitor 1) is a mitochondrial division inhibitor that inhibits DRP1 and Dynamin I (IC50=1-10 μM).</p>Fórmula:C15H10Cl2N2O2SPureza:96.57% - 99.23%Cor e Forma:SolidPeso molecular:353.22D4476
CAS:<p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>Fórmula:C23H18N4O3Pureza:99.7% - 99.96%Cor e Forma:SolidPeso molecular:398.41Nutlin-3
CAS:<p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C30H30Cl2N4O4Pureza:98.13% - 99.89%Cor e Forma:SolidPeso molecular:581.49Avadomide HCl
CAS:<p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>Fórmula:C14H15ClN4O3Cor e Forma:SolidPeso molecular:322.75Cyasterone
CAS:<p>Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via regulating EGFR signaling pathway, it may be a promising</p>Fórmula:C29H44O8Pureza:99.32% - 99.70%Cor e Forma:SolidPeso molecular:520.65NAE-IN-M22
CAS:<p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>Fórmula:C20H24Cl2N2Pureza:97.65%Cor e Forma:SolidPeso molecular:363.32NSC622608
CAS:<p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>Fórmula:C9H12BrN3OS2Pureza:98.48%Cor e Forma:SolidPeso molecular:322.24Formosanin C
CAS:<p>Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity.</p>Fórmula:C51H82O20Pureza:99.75% - >99.99%Cor e Forma:SolidPeso molecular:1015.18Fimasartan
CAS:<p>Fimasartan (BR-A-657), an ARB, treats hypertension and heart failure; safe with hydrochlorothiazide.</p>Fórmula:C27H31N7OSPureza:98.96%Cor e Forma:SolidPeso molecular:501.65Wogonin
CAS:<p>Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.</p>Fórmula:C16H12O5Pureza:98% - 99.8%Cor e Forma:Yellow CrystalPeso molecular:284.26LW6
CAS:<p>LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.</p>Fórmula:C26H29NO5Pureza:98.1% - 98.22%Cor e Forma:SolidPeso molecular:435.51Atractylenolide II
CAS:<p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>Fórmula:C15H20O2Pureza:99.89% - 99.93%Cor e Forma:SolidPeso molecular:232.321-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.75Bardoxolone Methyl
CAS:<p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>Fórmula:C32H43NO4Pureza:97.81% - 99.09%Cor e Forma:SolidPeso molecular:505.69CHS-828
CAS:<p>CHS-828 (GMX1778), a pyridyl cyanoguanidine, is an effective inhibitor of NAD+ biosynthesis enzyme NAMPT (IC50 <25 nM).</p>Fórmula:C19H22ClN5OPureza:98% - 99.9%Cor e Forma:SolidPeso molecular:371.86MSC 2032964A
CAS:<p>MSC 2032964A: Potent, selective ASK1 inhibitor, IC50=93 nM, oral, brain-permeable, curbs neuroinflammation, blocks LPS-induced ASK1/p38 activation.</p>Fórmula:C16H13F3N6OPureza:99.76%Cor e Forma:SolidPeso molecular:362.31Lenalidomide hemihydrate
CAS:<p>Lenalidomide hemihydrate inhibits TNF-α (IC50=13nM) and binds CRBN/DDB1 complexes.</p>Fórmula:C13H13N3O3H2OPureza:96.22%Cor e Forma:SolidPeso molecular:268.28Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Fórmula:C38H50N6O5Pureza:99.50% - >99.99%Cor e Forma:SolidPeso molecular:670.84MG 149
CAS:<p>MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).</p>Fórmula:C22H28O3Pureza:98.69% - 99.86%Cor e Forma:SolidPeso molecular:340.46SRT 2183
CAS:<p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>Fórmula:C27H24N4O2SPureza:97.86%Cor e Forma:SolidPeso molecular:468.57ASTX660
CAS:<p>Tolinapant (ASTX660) is an orally bioavailable cIAP1/2 and XIAP antagonist.Cost-effective and quality-assured.</p>Fórmula:C30H42FN5O3Pureza:98.33% - 99.85%Cor e Forma:SolidPeso molecular:539.68Mycophenolic acid sodium
CAS:<p>Mycophenolic acid sodium inhibits IMPDH with EC50 of 0.24 μM, has antiviral, immunosuppressive, antiangiogenic, and antitumor properties.</p>Fórmula:C17H19NaO6Cor e Forma:SolidPeso molecular:342.323Deguelin
CAS:<p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>Fórmula:C23H22O6Pureza:96.39% - 99.29%Cor e Forma:SolidPeso molecular:394.42GSK 3 Inhibitor IX
CAS:<p>GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex.</p>Fórmula:C16H10BrN3O2Pureza:98% - 99.72%Cor e Forma:SolidPeso molecular:356.17VER-50589
CAS:<p>VER-50589 is a potent HSP90 inhibitor.</p>Fórmula:C19H17ClN2O5Pureza:99.96% - >99.99%Cor e Forma:SolidPeso molecular:388.8JQ-1 (carboxylic acid)
CAS:<p>JQ-1 (carboxylic acid) is a cell-permeable BRD4 inhibitor with IC50s of 77 nM for BRD4(1) and 33 nM for BRD4(2)</p>Fórmula:C19H17ClN4O2SPureza:99.14% - 99.9%Cor e Forma:SolidPeso molecular:400.88Palomid 529
CAS:<p>Palomid 529 (SG 00529) has been used in trials studying the treatment of Age-Related Macular Degeneration.</p>Fórmula:C24H22O6Pureza:98.40% - 98.59%Cor e Forma:SolidPeso molecular:406.43BI-6C9
CAS:<p>BI-6C9 is an inhibitor of tBid (Kd = 20 μM).BI-6c9 prevented MOMP and mitochondrial fission, and protected the cells from cell death.</p>Fórmula:C23H25N3O4S2Pureza:98.39%Cor e Forma:SolidPeso molecular:471.59GW779439X
CAS:<p>GW779439X is an inhibitor of CDK.</p>Fórmula:C22H21F3N8Pureza:97.87%Cor e Forma:SolidPeso molecular:454.45Alogliptin
CAS:<p>Alogliptin (SYR-322)(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of <10 nM, exhibits greater than 10, 000-fold selectivity over DPP-8 and DPP-9</p>Fórmula:C18H21N5O2Pureza:99.63%Cor e Forma:SolidPeso molecular:339.39Embelin
CAS:<p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>Fórmula:C17H26O4Pureza:97.07% - 99.88%Cor e Forma:SolidPeso molecular:294.39Takinib
CAS:<p>Takinib (EDHS-206) is a specific and effective TAK1 inhibitor(IC50= 9.5 nM).</p>Fórmula:C18H18N4O2Pureza:98.29% - 99.35%Cor e Forma:SolidPeso molecular:322.36ML-210
CAS:<p>ML-210 (CID 49766530) is a glutathione peroxidase 4 (GPX4) inhibitor. ML-210 has antitumor activity and induces ferroptosis. Cost-effective and quality-assured.</p>Fórmula:C22H20Cl2N4O4Pureza:97% - 99.03%Cor e Forma:SolidPeso molecular:475.32ATH686
CAS:<p>ATH686 is an potent and selective Inhibitor of FLT3.</p>Fórmula:C25H28F3N7O2Pureza:98.07%Cor e Forma:SolidPeso molecular:515.53Pantoprazole
CAS:<p>Pantoprazole (BY1023) is a proton pump inhibitor used for short-term treatment of erosion and ulceration of the esophagus caused by gastroesophageal reflux</p>Fórmula:C16H15F2N3O4SPureza:99.28% - 99.63%Cor e Forma:Almost White SolidPeso molecular:383.37UMI-77
CAS:<p>UMI-77 is a selective Mcl-1 inhibitor. UMI-77 binds to the BH3-binding groove of Mcl-1.Cost-effective and quality-assured.</p>Fórmula:C18H14BrNO5S2Pureza:96% - 99.57%Cor e Forma:SolidPeso molecular:468.34Larotrectinib sulfate
CAS:<p>Larotrectinib sulfate (LOXO-101 sulfate) is an oral active and specific ATP-competitive inhibitor of tropomyosin receptor kinases (TRK).</p>Fórmula:C21H22F2N6O2·H2O4SPureza:98.62% - 99.76%Cor e Forma:SolidPeso molecular:526.51ACBI1
CAS:<p>ACBI1 is a potent PROTAC degrader of BAF ATPase subunits SMARCA2 and SMARCA4, also degrades the polybromo-associated BAF (PBAF) complex member PBRM1, with DC50s</p>Fórmula:C49H58FN9O7SPureza:97.54% - 98.15%Cor e Forma:SolidPeso molecular:936.1Pantoprazole sodium
CAS:<p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>Fórmula:C16H14F2N3NaO4SPureza:96.92% - 99.81%Cor e Forma:White To Off-White SolidPeso molecular:405.35[8]-Shogaol
CAS:<p>[8]-Shogaol is a component of ginger and maintains anti-inflammatory activity as a cyclooxygenase-2 inhibitor.</p>Fórmula:C19H28O3Pureza:97.01%Cor e Forma:SolidPeso molecular:304.42R-7050
CAS:<p>R-7050 (TNF-α Antagonist III), a tumor necrosis factor receptor (TNFR) antagonist, exhibits heightened selectivity for TNFα.</p>Fórmula:C16H8ClF3N4SPureza:98.64% - 99.8%Cor e Forma:SolidPeso molecular:380.77Soyasapogenol B
CAS:<p>Soyasapogenol B has anti-cancer, hypocholesterolemic, anticomplementary, hepatoprotective effects, it inhibits proliferation of cultured Hep-G2.</p>Fórmula:C30H50O3Pureza:99.51% - 99.81%Cor e Forma:SolidPeso molecular:458.72(+)-Nortrachelogenin
CAS:<p>(+)-Nortrachelogenin is a lignan isolated from Wikstroemia indica C.A. Meyer (Thymelaeaceae). (+)-Nortrachelogenin possesses antileukemic activity.</p>Fórmula:C20H22O7Pureza:99.88%Cor e Forma:SolidPeso molecular:374.38Cidofovir dihydrate
CAS:<p>Cidofovir dihydrate: Injectable anti-CMV; suppresses CMV by inhibiting viral DNA polymerase; treats CMV retinitis in AIDS.</p>Fórmula:C8H18N3O8PPureza:99.44%Cor e Forma:SolidPeso molecular:315.22Cynaroside
CAS:<p>Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.</p>Fórmula:C21H20O11Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:448.38PI-1840
CAS:<p>PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.</p>Fórmula:C22H26N4O3Pureza:98.82%Cor e Forma:SolidPeso molecular:394.47Darapladib
CAS:<p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>Fórmula:C36H38F4N4O2SPureza:99.82% - >99.99%Cor e Forma:SolidPeso molecular:666.77Capmatinib xHCl
CAS:<p>Capmatinib xHCl (INCB28060) is a potent, orally active, selective, and ATP competitive c-Met kinase inhibitor, potently blocking in vitro kinase activity (IC50</p>Fórmula:C23H18ClFN6OPureza:98.62% - 99.81%Cor e Forma:SolidPeso molecular:448.89A-1155463
CAS:<p>A-1155463, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2, BCL-W and MCL-1.</p>Fórmula:C35H32FN5O4S2Pureza:96.1% - 99%Cor e Forma:SolidPeso molecular:669.79Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Cor e Forma:White PowderPeso molecular:329.39Zinc Protoporphyrin
CAS:<p>Zinc Protoporphyrin is an oral HO-1 inhibitor that reduces PG's protection against H2O2 and has anti-cancer properties.</p>Fórmula:C34H32N4O4ZnPureza:95.43% - 99.27%Cor e Forma:SolidPeso molecular:626.02Picrocrocin
CAS:<p>Picrocrocin is a natural product</p>Fórmula:C16H26O7Pureza:98.4%Cor e Forma:SolidPeso molecular:330.37Erdafitinib
CAS:<p>Erdafitinib (JNJ-42756493) is a quinoxaline derivative compound, acts on FGFR1/2/3/4.</p>Fórmula:C25H30N6O2Pureza:97.00% - 99.07%Cor e Forma:SolidPeso molecular:446.544-Methylbenzylidene camphor
CAS:<p>4-Methylbenzylidene camphor: UVB blocker in sunscreens, cosmetics; exhibits estrogenic activity.</p>Fórmula:C18H22OPureza:99.92%Cor e Forma:White SolidPeso molecular:254.37L524-0366
CAS:<p>L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.</p>Fórmula:C13H13ClN4OSPureza:98.6% - 99.13%Cor e Forma:SolidPeso molecular:308.79ASK1-IN-1
CAS:<p>ASK1-IN-1 inhibits apoptosis kinase 1, crucial in cell stress responses, with 21 nM IC50.</p>Fórmula:C19H19N9O2Pureza:99.92%Cor e Forma:SolidPeso molecular:405.41Tacedinaline
CAS:<p>Tacedinaline (CI994) is a selective class I HDAC inhibitor with potential antineoplastic activity.</p>Fórmula:C15H15N3O2Pureza:96.83% - 99.15%Cor e Forma:WhitePeso molecular:269.3Anagrelide
CAS:<p>Anagrelide (Xagrid) is a Platelet-reducing Agent.</p>Fórmula:C10H7Cl2N3OPureza:99.53% - >99.99%Cor e Forma:SolidPeso molecular:256.09Diallyl Trisulfide
CAS:<p>Diallyl Trisulfide is an organic polysulfide compound found in garlic that acts as an H2S donor.</p>Fórmula:C6H10S3Pureza:95% - ≥98%Cor e Forma:LiquidPeso molecular:178.34Taurochenodeoxycholic Acid
CAS:<p>Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.</p>Fórmula:C26H45NO6SPureza:99.53% - 99.86%Cor e Forma:SolidPeso molecular:499.7W-7 hydrochloride
CAS:<p>W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride</p>Fórmula:C16H22Cl2N2O2SPureza:99.63%Cor e Forma:White Crystalline SolidPeso molecular:377.32MGH-CP1
CAS:<p>MGH-CP1 inhibits TEAD2/4 auto-palmitoylation with IC50 of 710 and 672 nM, respectively.</p>Fórmula:C20H24N4OSPureza:98.66%Cor e Forma:SolidPeso molecular:368.5Levobupivacaine hydrochloride
CAS:<p>Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.</p>Fórmula:C18H28N2O·HClPureza:99.74%Cor e Forma:White Crystalline PowderPeso molecular:324.89CBL0137
CAS:<p>CBL0137 (Curaxin 137), a metabolically stable curaxin, activates p53 (EC50: 0.37 μM) and inhibits NF-κB (EC50: 0.47 μM).</p>Fórmula:C21H24N2O2Pureza:99.57% - 99.68%Cor e Forma:SolidPeso molecular:336.43BAY 61-3606 dihydrochloride
CAS:<p>BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).</p>Fórmula:C20H18N6O3·2HClPureza:99.46%Cor e Forma:SolidPeso molecular:463.32L-Ascorbic acid sodium salt
CAS:<p>L-Ascorbic acid sodium salt (Vitamin C sodium salt) is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.</p>Fórmula:C6H7NaO6Pureza:98.73% - 99.75%Cor e Forma:Less Solid PowderPeso molecular:198.11ISOGINKGETIN
CAS:<p>ISOGINKGETIN (4',4'''-Dimethylamentoflavone), a compound derived from the leaves of Ginkgo biloba, to up-regulate adiponectin secretion.</p>Fórmula:C32H22O10Pureza:98% - 99.72%Cor e Forma:SolidPeso molecular:566.51Lycorine
CAS:<p>Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.</p>Fórmula:C16H17NO4Pureza:98.60% - 99.95%Cor e Forma:SolidPeso molecular:287.31Alemtuzumab
CAS:<p>Alemtuzumab is a humanized monoclonal antibody against CD52 an antigen found on the surface of normal and malignant lymphocytes.</p>Pureza:97.2% (SDS-PAGE); 96.7% (SEC-HPLC) - 98.00%Cor e Forma:LiquidPeso molecular:146.04 kDaPKCβ inhibitor 1
CAS:<p>PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,</p>Fórmula:C24H21N5O2Pureza:99.33%Cor e Forma:SolidPeso molecular:411.462BAct
CAS:<p>2BAct is a novel eif2b activator, preventing neurological defects caused by a chronic integrated stress response</p>Fórmula:C19H16ClF3N4O3Pureza:97.97% - 99.04%Cor e Forma:SolidPeso molecular:440.8Ganoderic acid A
CAS:<p>Ganoderic acid A fights tumors, suppresses gene regulators, induces cancer cell death, and enhances cisplatin efficacy.</p>Fórmula:C30H44O7Pureza:99.31% - ≥95%Cor e Forma:SolidPeso molecular:516.67Cysteamine hydrochloride
CAS:<p>Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant.</p>Fórmula:C2H7NS·HClPureza:99.34% - 99.87%Cor e Forma:White Crystalline Powder With A Strong And Disagreeable SmellPeso molecular:113.61

