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Apoptose

Apoptose

Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.

Subcategorias de "Apoptose"

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Foram encontrados 5599 produtos de "Apoptose"

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  • Mocetinostat

    CAS:
    <p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>
    Fórmula:C23H20N6O
    Pureza:99% - 99.21%
    Cor e Forma:Solid
    Peso molecular:396.44
  • AG1024

    CAS:
    <p>AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).</p>
    Fórmula:C14H13BrN2O
    Pureza:98% - 99.37%
    Cor e Forma:Solid
    Peso molecular:305.17
  • WHI-P154

    CAS:
    <p>WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.</p>
    Fórmula:C16H14BrN3O3
    Pureza:98% - 99.67%
    Cor e Forma:Solid
    Peso molecular:376.2
  • Taurolidine

    CAS:
    <p>Taurolidine is a synthetic taurine analog with antimicrobial and anti-neoplastic actions. It displays broad bactericidal and fungicidal activity.</p>
    Fórmula:C7H16N4O4S2
    Pureza:99.79% - 99.81%
    Cor e Forma:Solid
    Peso molecular:284.36
  • Topotecan

    CAS:
    <p>Topotecan (NSC-609669) is a Topoisomerase I inhibitor,and is an antineoplastic agent used to treat ovarian cancer that works by inhibiting DNA topoisomerases.</p>
    Fórmula:C23H23N3O5
    Pureza:96.14% - 98.23%
    Cor e Forma:Light Yellow Needle Crystal Or Crystalline Powder
    Peso molecular:421.45
  • Inauhzin

    CAS:
    <p>Inauhzin (INZ) reactivates p53, inhibits SIRT1, induces Y cell apoptosis without genotoxic stress (IC50=3 uM in A549).</p>
    Fórmula:C25H19N5OS2
    Pureza:98% - 99.36%
    Cor e Forma:Solid
    Peso molecular:469.58
  • Bafetinib

    CAS:
    <p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>
    Fórmula:C30H31F3N8O
    Pureza:94.16% - 99.68%
    Cor e Forma:Solid
    Peso molecular:576.62
  • Sertaconazole

    CAS:
    <p>Sertaconazole is a broad-spectrum antifungal.</p>
    Fórmula:C20H15Cl3N2OS
    Pureza:99.483%
    Cor e Forma:Solid
    Peso molecular:437.77
  • Azoramide

    CAS:
    <p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>
    Fórmula:C15H17ClN2OS
    Pureza:99.08% - 99.85%
    Cor e Forma:Solid
    Peso molecular:308.83
  • Thalidomide-5-methyl

    CAS:
    <p>Thalidomide-5-methyl is the Thalidomide-based cereblon (CRBN) ligand. Thalidomide-5-methyl is used in the recruitment of CRBN protein.</p>
    Fórmula:C14H12N2O4
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:272.26
  • S63845

    CAS:
    <p>S63845 is a selective myeloid leukemia 1(MCL1) inhibitor that binds to human MCL1 with a Kd of 0.19 nM.Cost-effective and quality-assured.</p>
    Fórmula:C39H37ClF4N6O6S
    Pureza:97.7% - ≥98%
    Cor e Forma:Solid
    Peso molecular:829.26
  • Ciprofloxacin hydrochloride monohydrate

    CAS:
    <p>Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) is a fluoroquinolone antibiotic with potent antibacterial activity.</p>
    Fórmula:C17H21ClFN3O4
    Pureza:99.23% - 99.85%
    Cor e Forma:White Or Yellowish Crystalline Powder
    Peso molecular:385.82
  • Y-27632 dihydrochloride

    CAS:
    <p>View and buy Y-27632 dihydrochloride from TargetMol.Y-27632 is a selective inhibitor of ROCKs.Cited in 10 publications.</p>
    Fórmula:C14H21N3O·2HCl
    Pureza:97.96% - 99.98%
    Cor e Forma:Solid
    Peso molecular:320.26
  • Tenovin-3

    CAS:
    <p>Tenovin-3 acts as a p53 activator.</p>
    Fórmula:C18H21N3OS
    Pureza:99.72% - ≥95%
    Cor e Forma:Solid
    Peso molecular:327.44
  • Rigosertib

    CAS:
    <p>Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by disrupting PI3K/Akt.</p>
    Fórmula:C21H25NO8S
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:451.49
  • Dapivirine

    CAS:
    <p>Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>
    Fórmula:C20H19N5
    Pureza:98% - 99.77%
    Cor e Forma:Solid
    Peso molecular:329.4
  • Demethoxycurcumin

    CAS:
    <p>Demethoxycurcumin: antioxidant, anti-inflammatory, anti-proliferative, anti-acanthamoebic, enhances chemo for resistant cancers, inhibits cancer pathways.</p>
    Fórmula:C20H18O5
    Pureza:94.54% - 99.86%
    Cor e Forma:Solid
    Peso molecular:338.35
  • A-419259

    CAS:
    <p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>
    Fórmula:C29H34N6O
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:482.62
  • PI-103

    CAS:
    <p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>
    Fórmula:C19H16N4O3
    Pureza:97.79% - 99.3%
    Cor e Forma:Solid
    Peso molecular:348.36
  • PKD-IN-1 dihydrochloride (956121-30-5 free base)

    CAS:
    <p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>
    Fórmula:C18H21Cl3N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:415.75
  • ML311

    CAS:
    <p>ML311 is a selective inhibitor of the Mcl-1/Bim interaction.</p>
    Fórmula:C23H24F3N3O
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:415.45
  • Tauroursodeoxycholate

    CAS:
    <p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>
    Fórmula:C26H45NO6S
    Pureza:98.77% - 99.93%
    Cor e Forma:White Solid
    Peso molecular:499.7
  • PEAQX

    CAS:
    <p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>
    Fórmula:C17H17BrN3O5P
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:454.21
  • AR42

    CAS:
    <p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>
    Fórmula:C18H20N2O3
    Pureza:98.46% - 98.96%
    Cor e Forma:Solid
    Peso molecular:312.36
  • Asiaticoside

    CAS:
    <p>Asiaticoside, in Centella asiatica, may treat wounds/burns.</p>
    Fórmula:C48H78O19
    Pureza:98% - 99.96%
    Cor e Forma:Powder
    Peso molecular:959.12
  • Emricasan

    CAS:
    <p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>
    Fórmula:C26H27F4N3O7
    Pureza:98.13% - 99%
    Cor e Forma:Solid
    Peso molecular:569.5
  • Aloperine

    CAS:
    <p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>
    Fórmula:C15H24N2
    Pureza:98% - 99.88%
    Cor e Forma:Yellow Crystalline Powder
    Peso molecular:232.36
  • 1400W dihydrochloride

    CAS:
    <p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>
    Fórmula:C10H17Cl2N3
    Pureza:98% - 99.94%
    Cor e Forma:Solid
    Peso molecular:250.17
  • SC66

    CAS:
    <p>SC66 is a AKT inhibitor in HepG2, HA22T/VGH, and PLC/PRF/5 cells (IC50: about 0.75 μg/ml, at 72 h).</p>
    Fórmula:C18H16N2O
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:276.33
  • Bilobalide

    CAS:
    <p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>
    Fórmula:C15H18O8
    Pureza:98.81% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:326.3
  • Rhosin hydrochloride

    CAS:
    <p>Rhosin hydrochloride is a specific inhibitor of the RhoA subfamily Rho GTPases.Cost-effective and quality-assured.</p>
    Fórmula:C20H20Cl2N6O
    Pureza:97.33% - 98.92%
    Cor e Forma:Solid
    Peso molecular:431.318
  • Nω-Hydroxy-nor-L-Arginine Dihydrochloride

    CAS:
    <p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>
    Fórmula:C5H14Cl2N4O3
    Pureza:99.12% - 99.84%
    Cor e Forma:Solid
    Peso molecular:249.10
  • Thalidomide-NH-PEG1-NH2 hydrochloride

    CAS:
    <p>Thalidomide-NH-PEG1-NH2 hydrochloride (4-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione HCl) is a synthetic E3 ligase ligand-</p>
    Fórmula:C17H21ClN4O5
    Pureza:97.13%
    Cor e Forma:Solid
    Peso molecular:396.83
  • UTL-5g

    CAS:
    <p>UTL-5g is a chemoprotective TNF-α inhibitor reducing cisplatin side effects and toxicity in liver, kidneys, and blood.</p>
    Fórmula:C11H8Cl2N2O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:271.1
  • Tetrahydroxyquinone monohydrate

    CAS:
    <p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>
    Fórmula:C6H6O7
    Cor e Forma:Solid
    Peso molecular:190.11
  • Nobiletin

    CAS:
    <p>Nobiletin: a citrus-derived flavone with anti-inflammatory and anti-cancer properties; water-insoluble, very weak acid.</p>
    Fórmula:C21H22O8
    Pureza:98.65% - 99.76%
    Cor e Forma:Solid
    Peso molecular:402.39
  • Alda-1

    CAS:
    <p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>
    Fórmula:C15H11Cl2NO3
    Pureza:98.5% - 99.63%
    Cor e Forma:Solid
    Peso molecular:324.16
  • CCCP

    CAS:
    <p>CCCP blocks STING activation, TBK1, IRF3 signaling, and IFN-β production by disrupting MMP.</p>
    Fórmula:C9H5ClN4
    Pureza:97.15% - 99.64%
    Cor e Forma:Yellow To Orange Powder
    Peso molecular:204.62
  • PD173955

    CAS:
    <p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>
    Fórmula:C21H16Cl2N4OS
    Pureza:98.52% - 98.99%
    Cor e Forma:Solid
    Peso molecular:443.35
  • RGX-202

    CAS:
    <p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>
    Fórmula:C4H9N3O2
    Pureza:99.67% - 99.8%
    Cor e Forma:Solid
    Peso molecular:131.13
  • Neobavaisoflavone

    CAS:
    <p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>
    Fórmula:C20H18O4
    Pureza:99.31% - 99.87%
    Cor e Forma:Solid
    Peso molecular:322.35
  • Ibandronate sodium monohydrate

    CAS:
    <p>Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.</p>
    Fórmula:C9H24NNaO8P2
    Pureza:99.62%
    Cor e Forma:White Crystalline Powder
    Peso molecular:359.23
  • HA15

    CAS:
    <p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>
    Fórmula:C23H22N4O3S2
    Pureza:99.77% - 99.86%
    Cor e Forma:Solid
    Peso molecular:466.58
  • NADPH tetracyclohexanamine

    CAS:
    <p>NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.</p>
    Fórmula:C45H82N11O17P3
    Pureza:98.73% - 99.05%
    Cor e Forma:Solid
    Peso molecular:1142.12
  • Obatoclax Mesylate

    CAS:
    Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, and
    Fórmula:C20H19N3O·CH4O3S
    Pureza:99.58% - 99.88%
    Cor e Forma:Solid
    Peso molecular:413.49
  • Idasanutlin

    CAS:
    <p>Idasanutlin (Ro 5503781) (RG-7388) is an effective and specific p53-MDM2 inhibitor (IC50: 6 nM).</p>
    Fórmula:C31H29Cl2F2N3O4
    Pureza:99.13% - 99.88%
    Cor e Forma:Solid
    Peso molecular:616.48
  • Eriocitrin

    CAS:
    <p>Eriocitrin: an antioxidative flavonoid; reduces exercise-induced oxidative damage and lipids; fights fatty liver and inhibits carbonic anhydrase VA.</p>
    Fórmula:C27H32O15
    Pureza:98.41% - 99.11%
    Cor e Forma:Solid
    Peso molecular:596.53
  • CHR-6494 TFA

    CAS:
    <p>CHR-6494 TFA: potent haspin inhibitor (IC50=2 nM), blocks H3T3 phosphorylation, triggers apoptosis in cancer cells. Used for cancer research.</p>
    Fórmula:C18H17F3N6O2
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:406.36
  • CA-4948

    CAS:
    <p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>
    Fórmula:C24H25N7O5
    Pureza:99.35% - 99.88%
    Cor e Forma:Solid
    Peso molecular:491.5
  • Tenovin-6

    CAS:
    <p>Tenovin-6 is a p53 transcriptional activity agonist.</p>
    Fórmula:C25H34N4O2S
    Pureza:97.71% - >99.99%
    Cor e Forma:Solid
    Peso molecular:454.63
  • Trabectedin

    CAS:
    <p>Trabectedin (Ecteinascidin 743) has potent antitumor activity and the potential for soft tissue sarcoma and ovarian cancer research.</p>
    Fórmula:C39H43N3O11S
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:761.84
  • CPTH2

    CAS:
    <p>CPTH2 is a histone acetyltransferase inhibitor modulating Gcn5 network.</p>
    Fórmula:C14H14ClN3S
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:291.8
  • ZMC1

    CAS:
    <p>NSC-319726 (ZMC1), a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).</p>
    Fórmula:C11H14N4S
    Pureza:98.97% - 99.76%
    Cor e Forma:Solid
    Peso molecular:234.32
  • MPTP hydrochloride

    CAS:
    <p>MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.</p>
    Fórmula:C12H16ClN
    Pureza:96.35% - >99.99%
    Cor e Forma:Solid
    Peso molecular:209.72
  • FOXO4-DRI acetate


    <p>FOXO4-DRI acetate is a bioactive chemical.</p>
    Fórmula:C36H64N14O14S
    Pureza:99.10%
    Cor e Forma:Solid
    Peso molecular:5358.06
  • Choline

    CAS:
    <p>Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins</p>
    Fórmula:C5H15NO2
    Pureza:99.97% - ≥98%
    Cor e Forma:Liquid
    Peso molecular:121.18
  • Periplocin

    CAS:
    <p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>
    Fórmula:C36H56O13
    Pureza:99.66% - 99.74%
    Cor e Forma:Solid
    Peso molecular:696.82
  • RAD51 Inhibitor B02

    CAS:
    <p>RAD51 Inhibitor B02 (B02) (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM.</p>
    Fórmula:C22H17N3O
    Pureza:99.72% - 99.89%
    Cor e Forma:Solid
    Peso molecular:339.39
  • Salubrinal

    CAS:
    <p>Salubrinal, a phosphatases (PP1) inhibitor(IC50=1.7 μM), exhibits function on the eukaryotic translation initiation factor 2 subunit (eIF2α).</p>
    Fórmula:C21H17Cl3N4OS
    Pureza:97.25% - >99.99%
    Cor e Forma:Solid
    Peso molecular:479.81
  • Bendamustine

    CAS:
    <p>Bendamustine (SDX105) for the treatment of Non-Hodgkin Lymphomas and Chronic Lymphocytic Leukemia</p>
    Fórmula:C16H21Cl2N3O2
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:358.26
  • TrxR1-IN-B19

    CAS:
    <p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>
    Fórmula:C21H22O5
    Pureza:98.6%
    Cor e Forma:Solid
    Peso molecular:354.4
  • Sertaconazole nitrate

    CAS:
    <p>Sertaconazole nitrate, a broad-spectrum topical antifungal, treats skin and mucosal infections.</p>
    Fórmula:C20H15Cl3N2OS·HNO3
    Pureza:98.66% - 99.65%
    Cor e Forma:Solid
    Peso molecular:500.78
  • Thalidomide-O-amido-C3-NH2 TFA

    CAS:
    <p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>
    Fórmula:C20H21F3N4O8
    Pureza:98.47%
    Cor e Forma:Solid
    Peso molecular:502.4
  • Thalidomide-O-COOH

    CAS:
    <p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>
    Fórmula:C15H12N2O7
    Pureza:98% - 98.29%
    Cor e Forma:Solid
    Peso molecular:332.27
  • Polygalacin D

    CAS:
    <p>Polygalacin D shows anti- proliferation, anti-inflammary, and hepatoprotective activities, it can inhibit the expression of lipopolysaccharide (LPS)-induced</p>
    Fórmula:C57H92O27
    Pureza:98.95% - ≥98%
    Cor e Forma:Solid
    Peso molecular:1209.4
  • Almorexant

    CAS:
    <p>Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for OX1 and 0.17 nM for OX2.</p>
    Fórmula:C29H31F3N2O3
    Pureza:97.75% - 98.02%
    Cor e Forma:Solid
    Peso molecular:512.56
  • m-3M3FBS

    CAS:
    <p>m-3M3FBS is a phospholipase C (PLC) activator.</p>
    Fórmula:C16H16F3NO2S
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:343.36
  • Grape Seed Extract

    CAS:
    <p>Grape Seed Extract (Grape Seed P.E.) is exudate from seeds of the grape plant Vitis vinifera, composed of oils and secondary plant metabolites.</p>
    Fórmula:C32H30O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:590.581
  • ENMD-2076

    CAS:
    <p>ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.</p>
    Fórmula:C21H25N7
    Pureza:97.63% - ≥95%
    Cor e Forma:Solid
    Peso molecular:375.47
  • CVT-11127

    CAS:
    <p>CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.</p>
    Fórmula:C25H23Cl2N5O3
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:512.39
  • Vesatolimod

    CAS:
    <p>Vesatolimod (GS-9620) is an effective and specific orally active agonist of Toll-like receptor 7.</p>
    Fórmula:C22H30N6O2
    Pureza:97.46% - 99.03%
    Cor e Forma:Solid
    Peso molecular:410.51
  • IC261

    CAS:
    <p>IC261 (SU-5607) is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for Cdk5 is 4.5 mM.</p>
    Fórmula:C18H17NO4
    Pureza:99.45% - 99.91%
    Cor e Forma:Solid
    Peso molecular:311.33
  • Methoxychlor

    CAS:
    <p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>
    Fórmula:C16H15Cl3O2
    Pureza:98.82% - ≥95%
    Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment If
    Peso molecular:345.65
  • Delanzomib

    CAS:
    <p>Delanzomib (CEP-18770) is an oral proteasome inhibitor with an IC50 of 3.8 nM, targeting chymotrypsin-like activity with minimal effect on other activities.</p>
    Fórmula:C21H28BN3O5
    Pureza:95.52% - 99.46%
    Cor e Forma:Solid
    Peso molecular:413.28
  • Gardenin B

    CAS:
    <p>Gardenin B exhibits superior antiproliferative activity against lung, breast, colon, hepatic and leukaemia cell lines as well as in keratinocytes .</p>
    Fórmula:C19H18O7
    Pureza:98.80% - 99.74%
    Cor e Forma:Solid
    Peso molecular:358.34
  • N-Ethylmaleimide

    CAS:
    <p>N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor. Cost-effective and quality-assured.</p>
    Fórmula:C6H7NO2
    Pureza:99.50%
    Cor e Forma:White Solid
    Peso molecular:125.13
  • Salvigenin

    CAS:
    <p>Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.</p>
    Fórmula:C18H16O6
    Pureza:99.17% - 99.78%
    Cor e Forma:Solid
    Peso molecular:328.32
  • Cucurbitacin IIA

    CAS:
    <p>1.</p>
    Fórmula:C32H50O8
    Pureza:98.62% - 99.87%
    Cor e Forma:Solid
    Peso molecular:562.73
  • Infigratinib

    CAS:
    <p>Infigratinib (NVP-BGJ398) (BGJ398) is an orally bioavailable pan FGFR inhibitor (IC50: 0.9/1.4/1 nM for FGFR1/2/3), &gt;40-fold selective for FGFR versus FGFR4 and</p>
    Fórmula:C26H31Cl2N7O3
    Pureza:98% - 98.97%
    Cor e Forma:Solid
    Peso molecular:560.48
  • CCPA

    CAS:
    <p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>
    Fórmula:C15H20ClN5O4
    Pureza:99.1%
    Cor e Forma:Off-White To Light Yellow Solid
    Peso molecular:369.8
  • OSI-930

    CAS:
    <p>OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.</p>
    Fórmula:C22H16F3N3O2S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:443.44
  • GSK778 hydrochloride

    CAS:
    <p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>
    Fórmula:C30H34ClN5O3
    Pureza:97.26% - 98.35%
    Cor e Forma:Solid
    Peso molecular:548.08
  • Thalidomide-4-OH

    CAS:
    <p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>
    Fórmula:C13H10N2O5
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:274.23
  • Difurazon hydrochloride

    CAS:
    <p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>
    Fórmula:C14H13ClN6O6
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:396.74
  • Methoxyamine HCl

    CAS:
    <p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>
    Fórmula:CH6ClNO
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:83.51
  • Sal003

    CAS:
    <p>Sal003, an effective cell-permeable analog, inhibitis the eIF2α phosphatase.</p>
    Fórmula:C18H15Cl4N3OS
    Pureza:99.17% - 99.77%
    Cor e Forma:Solid
    Peso molecular:463.21
  • Momordin Ic

    CAS:
    <p>Momordin Ic (Momordin 1c) might represent a potential anticancer activity, by inducing apoptosis through oxidative stress-regulated mitochondrial dysfunction</p>
    Fórmula:C41H64O13
    Pureza:98% - 99.69%
    Cor e Forma:Solid
    Peso molecular:764.94
  • Neferine

    CAS:
    <p>Neferine: anti-tumor, enhances DOX efficacy, prevents diabetic vasculopathy; mediates via CYP3A4, GSH depletion, blocks ROS/Akt/NF-κB.</p>
    Fórmula:C38H44N2O6
    Pureza:98.81% - 99.65%
    Cor e Forma:Solid
    Peso molecular:624.77
  • PKR-IN-C16

    CAS:
    <p>PKR-IN-C16: inhibits PKR autophosphorylation and translation blockade; binds ATP site; IC50 of 186-210 nM; protects cells from ER stress damage.</p>
    Fórmula:C13H8N4OS
    Pureza:97.8%
    Cor e Forma:Solid
    Peso molecular:268.29
  • Alogliptin Benzoate

    CAS:
    <p>Alogliptin Benzoate, a potent DPP-4 inhibitor with &gt;10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>
    Fórmula:C25H27N5O4
    Pureza:99.94% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:461.51
  • Levomenol

    CAS:
    <p>Levomenol, or (-)-α-Bisabolol, is a sesquiterpene in aromatic plant oils with antioxidant, anti-inflammatory, and anti-apoptotic properties.</p>
    Fórmula:C15H26O
    Pureza:96.01%
    Cor e Forma:Clear To Yellowish Liquid
    Peso molecular:222.37
  • SC144

    CAS:
    <p>SC144 is an orally active small-molecule gp130 inhibitor.</p>
    Fórmula:C16H11FN6O
    Pureza:99.20%
    Cor e Forma:Solid
    Peso molecular:322.3
  • PIK-75

    CAS:
    <p>PIK-75, a DNA-PK and PI3K inhibitor, suppresses DNA-PK(IC50=2 nM), p110α(IC50=5.8 nM) and p110γ(IC50=76 nM).</p>
    Fórmula:C16H14BrN5O4S
    Pureza:98.52% - >99.99%
    Cor e Forma:Solid
    Peso molecular:452.28
  • Pectolinarin

    CAS:
    <p>Pectolinarin is a Cirsium isolate with anti-inflammatory activity.</p>
    Fórmula:C29H34O15
    Pureza:98% - 99.79%
    Cor e Forma:Solid
    Peso molecular:622.57
  • Epibrassinolide

    CAS:
    <p>Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator with</p>
    Fórmula:C28H48O6
    Pureza:97.57% - 98.11%
    Cor e Forma:Solid
    Peso molecular:480.68
  • KRCA-0008

    CAS:
    <p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>
    Fórmula:C30H37ClN8O4
    Pureza:96.19%
    Cor e Forma:Solid
    Peso molecular:609.12
  • Perhexiline

    CAS:
    <p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>
    Fórmula:C19H35N
    Cor e Forma:Solid
    Peso molecular:277.49
  • Ketorolac hemicalcium

    CAS:
    <p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation &amp; pain, used in cancer research.</p>
    Fórmula:C30H24CaN2O6
    Cor e Forma:Solid
    Peso molecular:548.608
  • Thalidomide-propargyl

    CAS:
    <p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>
    Fórmula:C16H12N2O5
    Pureza:95.14%
    Cor e Forma:Solid
    Peso molecular:312.28
  • Thalidomide-NH-C6-NH2 hydrochloride

    CAS:
    <p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>
    Fórmula:C19H25ClN4O4
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:408.88
  • Britannin

    CAS:
    <p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>
    Fórmula:C19H26O7
    Pureza:98% - 99.98%
    Cor e Forma:Solid
    Peso molecular:366.41
  • PK11000

    CAS:
    <p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>
    Fórmula:C6H5ClN2O4S
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:236.63
  • Abacavir monosulfate

    CAS:
    <p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>
    Fórmula:C14H20N6O5S
    Cor e Forma:Solid
    Peso molecular:384.41
  • Tanespimycin

    CAS:
    <p>Tanespimycin (KOS 953) is an Hsp90 inhibitor (IC50=5 nM) and is selective. Tanespimycin depletes intracellular STK38/NDR1. High-Quality, Low-Cost!</p>
    Fórmula:C31H43N3O8
    Pureza:99.07% - 99.83%
    Cor e Forma:Dark Purple Solid
    Peso molecular:585.69
  • Benidipine hydrochloride

    CAS:
    <p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>
    Fórmula:C28H32ClN3O6
    Pureza:99.80%
    Cor e Forma:Solid
    Peso molecular:542.03
  • 2-tert-Butyl-1,4-benzoquinone

    CAS:
    <p>TBQ, a BHA metabolite, activates Nrf2 and S-arylates Keap1 in RAW264.7 cells.</p>
    Fórmula:C10H12O2
    Pureza:97.19%
    Cor e Forma:Solid
    Peso molecular:164.2
  • Thalidomide-O-amido-PEG2-C2-NH2 TFA

    CAS:
    <p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>
    Fórmula:C23H27F3N4O10
    Pureza:95.74% - 99%
    Cor e Forma:Solid
    Peso molecular:576.48
  • Tasisulam

    CAS:
    <p>Tasisulam (LY573636) is an apoptosis inducer and an antitumor agent via the intrinsic pathway.</p>
    Fórmula:C11H6BrCl2NO3S2
    Pureza:99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:415.11
  • MS7972

    CAS:
    <p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>
    Fórmula:C14H13NO2
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:227.26
  • RO8994

    CAS:
    <p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>
    Fórmula:C31H31Cl2FN4O4
    Pureza:99.31% - 99.44%
    Cor e Forma:Solid
    Peso molecular:613.51
  • KX2-361

    CAS:
    <p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>
    Fórmula:C24H24FN3O2
    Pureza:99.64% - 99.68%
    Cor e Forma:Solid
    Peso molecular:405.46
  • AZ 628

    CAS:
    <p>AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM, 34 nM and 29 nM, also inhibits VEGFR2, DDR2, Lyn, Flt1, FMS, etc.</p>
    Fórmula:C27H25N5O2
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:451.52
  • Capsazepine

    CAS:
    <p>Capsazepine, a TRPV1 antagonist (IC50: 562 nM), blocks capsaicin-induced heat pain.</p>
    Fórmula:C19H21ClN2O2S
    Pureza:98% - 99.78%
    Cor e Forma:White To Off-White Powder
    Peso molecular:376.9
  • Quizartinib

    CAS:
    <p>Quizartinib (AC220) is an inhibitor of FLT3 (Kd: 1.6 nM) and demonstrates high selectivity for FLT3 when tested against a panel of 227 additional kinases.</p>
    Fórmula:C29H32N6O4S
    Pureza:98% - 99.42%
    Cor e Forma:Solid
    Peso molecular:560.67
  • Ralimetinib dimesylate

    CAS:
    <p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>
    Fórmula:C24H29FN6·2CH4O3S
    Pureza:98% - 99.38%
    Cor e Forma:Solid
    Peso molecular:612.74
  • (1E,6E)-Bis(demethoxy)curcumin

    CAS:
    <p>(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) is a natural demethoxy derivative of curcumin,with anti-inflammatory and anti-cancer activities.</p>
    Fórmula:C19H16O4
    Pureza:97.45%
    Cor e Forma:Solid
    Peso molecular:308.33
  • Genistein

    CAS:
    <p>Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has antitumor effects. Cost effective and quality assured.</p>
    Fórmula:C15H10O5
    Pureza:98.22% - 99.64%
    Cor e Forma:Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether Solid
    Peso molecular:270.24
  • Crebanine

    CAS:
    <p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>
    Fórmula:C20H21NO4
    Pureza:99.17% - 99.77%
    Cor e Forma:Solid
    Peso molecular:339.39
  • DEL-22379

    CAS:
    <p>DEL-22379 is a water-soluble ERK dimerization inhibitor with IC50 of ~0.5 μM.</p>
    Fórmula:C26H28N4O3
    Pureza:99.3% - 99.53%
    Cor e Forma:Solid
    Peso molecular:444.53
  • Caudatin

    CAS:
    <p>Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.</p>
    Fórmula:C28H42O7
    Pureza:98.83% - 99.9%
    Cor e Forma:Solid
    Peso molecular:490.63
  • Rabeprazole sodium

    CAS:
    <p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>
    Fórmula:C18H20N3NaO3S
    Pureza:98% - 99.912%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:381.42
  • Taurochenodeoxycholic acid sodium

    CAS:
    <p>Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).</p>
    Fórmula:C26H44NNaO6S
    Pureza:98.23% - 99.45%
    Cor e Forma:White To Off-White Powder
    Peso molecular:521.68
  • Pifithrin-α hydrobromide

    CAS:
    <p>Pifithrin-α hydrobromide (Pifithrin-α hydrobromide) is a p53 inhibitor, inhibiting p53-dependent transactivation of p53-responsive genes.</p>
    Fórmula:C16H18N2OS·HBr
    Pureza:97.71% - >99.99%
    Cor e Forma:Solid
    Peso molecular:367.3
  • Stattic

    CAS:
    <p>Stattic (STAT3 Inhibitor V) is a STAT3 inhibitor (IC50=5.1 μM) that selectively inhibits STAT3 activation, dimerization, and nuclear translocation.</p>
    Fórmula:C8H5NO4S
    Pureza:98.32% - 99.76%
    Cor e Forma:Solid
    Peso molecular:211.19
  • GSK-J4

    CAS:
    <p>GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.</p>
    Fórmula:C24H27N5O2
    Pureza:98.24% - 99.98%
    Cor e Forma:Solid
    Peso molecular:417.5
  • Mitochonic acid 5

    CAS:
    <p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>
    Fórmula:C18H13F2NO3
    Pureza:98.85%
    Cor e Forma:Solid
    Peso molecular:329.3
  • Angelicin

    CAS:
    <p>Angelicin (Isopsoralen), is a furanocoumarin with anti-Y, antiviral, anti-inflammatory activity.</p>
    Fórmula:C11H6O3
    Pureza:99.86% - 99.89%
    Cor e Forma:White Solid
    Peso molecular:186.16
  • Mdivi-1

    CAS:
    <p>Mdivi-1 (Mitochondrial division inhibitor 1) is a mitochondrial division inhibitor that inhibits DRP1 and Dynamin I (IC50=1-10 μM).</p>
    Fórmula:C15H10Cl2N2O2S
    Pureza:96.57% - 99.23%
    Cor e Forma:Solid
    Peso molecular:353.22
  • D4476

    CAS:
    <p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>
    Fórmula:C23H18N4O3
    Pureza:99.7% - 99.96%
    Cor e Forma:Solid
    Peso molecular:398.41
  • Nutlin-3

    CAS:
    <p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C30H30Cl2N4O4
    Pureza:98.13% - 99.89%
    Cor e Forma:Solid
    Peso molecular:581.49
  • Avadomide HCl

    CAS:
    <p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>
    Fórmula:C14H15ClN4O3
    Cor e Forma:Solid
    Peso molecular:322.75
  • Cyasterone

    CAS:
    <p>Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via regulating EGFR signaling pathway, it may be a promising</p>
    Fórmula:C29H44O8
    Pureza:99.32% - 99.70%
    Cor e Forma:Solid
    Peso molecular:520.65
  • NAE-IN-M22

    CAS:
    <p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>
    Fórmula:C20H24Cl2N2
    Pureza:97.65%
    Cor e Forma:Solid
    Peso molecular:363.32
  • NSC622608

    CAS:
    <p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>
    Fórmula:C9H12BrN3OS2
    Pureza:98.48%
    Cor e Forma:Solid
    Peso molecular:322.24
  • Formosanin C

    CAS:
    <p>Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity.</p>
    Fórmula:C51H82O20
    Pureza:99.75% - >99.99%
    Cor e Forma:Solid
    Peso molecular:1015.18
  • Fimasartan

    CAS:
    <p>Fimasartan (BR-A-657), an ARB, treats hypertension and heart failure; safe with hydrochlorothiazide.</p>
    Fórmula:C27H31N7OS
    Pureza:98.96%
    Cor e Forma:Solid
    Peso molecular:501.65
  • Wogonin

    CAS:
    <p>Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.</p>
    Fórmula:C16H12O5
    Pureza:98% - 99.8%
    Cor e Forma:Yellow Crystal
    Peso molecular:284.26
  • LW6

    CAS:
    <p>LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.</p>
    Fórmula:C26H29NO5
    Pureza:98.1% - 98.22%
    Cor e Forma:Solid
    Peso molecular:435.51
  • Atractylenolide II

    CAS:
    <p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>
    Fórmula:C15H20O2
    Pureza:99.89% - 99.93%
    Cor e Forma:Solid
    Peso molecular:232.32
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:248.75
  • Bardoxolone Methyl

    CAS:
    <p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>
    Fórmula:C32H43NO4
    Pureza:97.81% - 99.09%
    Cor e Forma:Solid
    Peso molecular:505.69
  • CHS-828

    CAS:
    <p>CHS-828 (GMX1778), a pyridyl cyanoguanidine, is an effective inhibitor of NAD+ biosynthesis enzyme NAMPT (IC50 &lt;25 nM).</p>
    Fórmula:C19H22ClN5O
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:371.86
  • MSC 2032964A

    CAS:
    <p>MSC 2032964A: Potent, selective ASK1 inhibitor, IC50=93 nM, oral, brain-permeable, curbs neuroinflammation, blocks LPS-induced ASK1/p38 activation.</p>
    Fórmula:C16H13F3N6O
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:362.31
  • Lenalidomide hemihydrate

    CAS:
    <p>Lenalidomide hemihydrate inhibits TNF-α (IC50=13nM) and binds CRBN/DDB1 complexes.</p>
    Fórmula:C13H13N3O3H2O
    Pureza:96.22%
    Cor e Forma:Solid
    Peso molecular:268.28
  • Saquinavir

    CAS:
    <p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>
    Fórmula:C38H50N6O5
    Pureza:99.50% - >99.99%
    Cor e Forma:Solid
    Peso molecular:670.84
  • MG 149

    CAS:
    <p>MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).</p>
    Fórmula:C22H28O3
    Pureza:98.69% - 99.86%
    Cor e Forma:Solid
    Peso molecular:340.46
  • SRT 2183

    CAS:
    <p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>
    Fórmula:C27H24N4O2S
    Pureza:97.86%
    Cor e Forma:Solid
    Peso molecular:468.57
  • ASTX660

    CAS:
    <p>Tolinapant (ASTX660) is an orally bioavailable cIAP1/2 and XIAP antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C30H42FN5O3
    Pureza:98.33% - 99.85%
    Cor e Forma:Solid
    Peso molecular:539.68
  • Mycophenolic acid sodium

    CAS:
    <p>Mycophenolic acid sodium inhibits IMPDH with EC50 of 0.24 μM, has antiviral, immunosuppressive, antiangiogenic, and antitumor properties.</p>
    Fórmula:C17H19NaO6
    Cor e Forma:Solid
    Peso molecular:342.323
  • Deguelin

    CAS:
    <p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>
    Fórmula:C23H22O6
    Pureza:96.39% - 99.29%
    Cor e Forma:Solid
    Peso molecular:394.42
  • GSK 3 Inhibitor IX

    CAS:
    <p>GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex.</p>
    Fórmula:C16H10BrN3O2
    Pureza:98% - 99.72%
    Cor e Forma:Solid
    Peso molecular:356.17
  • VER-50589

    CAS:
    <p>VER-50589 is a potent HSP90 inhibitor.</p>
    Fórmula:C19H17ClN2O5
    Pureza:99.96% - >99.99%
    Cor e Forma:Solid
    Peso molecular:388.8
  • JQ-1 (carboxylic acid)

    CAS:
    <p>JQ-1 (carboxylic acid) is a cell-permeable BRD4 inhibitor with IC50s of 77 nM for BRD4(1) and 33 nM for BRD4(2)</p>
    Fórmula:C19H17ClN4O2S
    Pureza:99.14% - 99.9%
    Cor e Forma:Solid
    Peso molecular:400.88
  • Palomid 529

    CAS:
    <p>Palomid 529 (SG 00529) has been used in trials studying the treatment of Age-Related Macular Degeneration.</p>
    Fórmula:C24H22O6
    Pureza:98.40% - 98.59%
    Cor e Forma:Solid
    Peso molecular:406.43
  • BI-6C9

    CAS:
    <p>BI-6C9 is an inhibitor of tBid (Kd = 20 μM).BI-6c9 prevented MOMP and mitochondrial fission, and protected the cells from cell death.</p>
    Fórmula:C23H25N3O4S2
    Pureza:98.39%
    Cor e Forma:Solid
    Peso molecular:471.59
  • GW779439X

    CAS:
    <p>GW779439X is an inhibitor of CDK.</p>
    Fórmula:C22H21F3N8
    Pureza:97.87%
    Cor e Forma:Solid
    Peso molecular:454.45
  • Alogliptin

    CAS:
    <p>Alogliptin (SYR-322)(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of &lt;10 nM, exhibits greater than 10, 000-fold selectivity over DPP-8 and DPP-9</p>
    Fórmula:C18H21N5O2
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:339.39
  • Embelin

    CAS:
    <p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>
    Fórmula:C17H26O4
    Pureza:97.07% - 99.88%
    Cor e Forma:Solid
    Peso molecular:294.39
  • Takinib

    CAS:
    <p>Takinib (EDHS-206) is a specific and effective TAK1 inhibitor(IC50= 9.5 nM).</p>
    Fórmula:C18H18N4O2
    Pureza:98.29% - 99.35%
    Cor e Forma:Solid
    Peso molecular:322.36
  • ML-210

    CAS:
    <p>ML-210 (CID 49766530) is a glutathione peroxidase 4 (GPX4) inhibitor. ML-210 has antitumor activity and induces ferroptosis. Cost-effective and quality-assured.</p>
    Fórmula:C22H20Cl2N4O4
    Pureza:97% - 99.03%
    Cor e Forma:Solid
    Peso molecular:475.32
  • ATH686

    CAS:
    <p>ATH686 is an potent and selective Inhibitor of FLT3.</p>
    Fórmula:C25H28F3N7O2
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:515.53
  • Pantoprazole

    CAS:
    <p>Pantoprazole (BY1023) is a proton pump inhibitor used for short-term treatment of erosion and ulceration of the esophagus caused by gastroesophageal reflux</p>
    Fórmula:C16H15F2N3O4S
    Pureza:99.28% - 99.63%
    Cor e Forma:Almost White Solid
    Peso molecular:383.37
  • UMI-77

    CAS:
    <p>UMI-77 is a selective Mcl-1 inhibitor. UMI-77 binds to the BH3-binding groove of Mcl-1.Cost-effective and quality-assured.</p>
    Fórmula:C18H14BrNO5S2
    Pureza:96% - 99.57%
    Cor e Forma:Solid
    Peso molecular:468.34
  • Larotrectinib sulfate

    CAS:
    <p>Larotrectinib sulfate (LOXO-101 sulfate) is an oral active and specific ATP-competitive inhibitor of tropomyosin receptor kinases (TRK).</p>
    Fórmula:C21H22F2N6O2·H2O4S
    Pureza:98.62% - 99.76%
    Cor e Forma:Solid
    Peso molecular:526.51
  • ACBI1

    CAS:
    <p>ACBI1 is a potent PROTAC degrader of BAF ATPase subunits SMARCA2 and SMARCA4, also degrades the polybromo-associated BAF (PBAF) complex member PBRM1, with DC50s</p>
    Fórmula:C49H58FN9O7S
    Pureza:97.54% - 98.15%
    Cor e Forma:Solid
    Peso molecular:936.1
  • Pantoprazole sodium

    CAS:
    <p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>
    Fórmula:C16H14F2N3NaO4S
    Pureza:96.92% - 99.81%
    Cor e Forma:White To Off-White Solid
    Peso molecular:405.35
  • [8]-Shogaol

    CAS:
    <p>[8]-Shogaol is a component of ginger and maintains anti-inflammatory activity as a cyclooxygenase-2 inhibitor.</p>
    Fórmula:C19H28O3
    Pureza:97.01%
    Cor e Forma:Solid
    Peso molecular:304.42
  • R-7050

    CAS:
    <p>R-7050 (TNF-α Antagonist III), a tumor necrosis factor receptor (TNFR) antagonist, exhibits heightened selectivity for TNFα.</p>
    Fórmula:C16H8ClF3N4S
    Pureza:98.64% - 99.8%
    Cor e Forma:Solid
    Peso molecular:380.77
  • Soyasapogenol B

    CAS:
    <p>Soyasapogenol B has anti-cancer, hypocholesterolemic, anticomplementary, hepatoprotective effects, it inhibits proliferation of cultured Hep-G2.</p>
    Fórmula:C30H50O3
    Pureza:99.51% - 99.81%
    Cor e Forma:Solid
    Peso molecular:458.72
  • (+)-Nortrachelogenin

    CAS:
    <p>(+)-Nortrachelogenin is a lignan isolated from Wikstroemia indica C.A. Meyer (Thymelaeaceae). (+)-Nortrachelogenin possesses antileukemic activity.</p>
    Fórmula:C20H22O7
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:374.38
  • Cidofovir dihydrate

    CAS:
    <p>Cidofovir dihydrate: Injectable anti-CMV; suppresses CMV by inhibiting viral DNA polymerase; treats CMV retinitis in AIDS.</p>
    Fórmula:C8H18N3O8P
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:315.22
  • Cynaroside

    CAS:
    <p>Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.</p>
    Fórmula:C21H20O11
    Pureza:98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:448.38
  • PI-1840

    CAS:
    <p>PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.</p>
    Fórmula:C22H26N4O3
    Pureza:98.82%
    Cor e Forma:Solid
    Peso molecular:394.47
  • Darapladib

    CAS:
    <p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>
    Fórmula:C36H38F4N4O2S
    Pureza:99.82% - >99.99%
    Cor e Forma:Solid
    Peso molecular:666.77
  • Capmatinib xHCl

    CAS:
    <p>Capmatinib xHCl (INCB28060) is a potent, orally active, selective, and ATP competitive c-Met kinase inhibitor, potently blocking in vitro kinase activity (IC50</p>
    Fórmula:C23H18ClFN6O
    Pureza:98.62% - 99.81%
    Cor e Forma:Solid
    Peso molecular:448.89
  • A-1155463

    CAS:
    <p>A-1155463, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and &gt;1000-fold weaker binding to BCL-2, BCL-W and MCL-1.</p>
    Fórmula:C35H32FN5O4S2
    Pureza:96.1% - 99%
    Cor e Forma:Solid
    Peso molecular:669.79
  • Sinomenine

    CAS:
    <p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>
    Fórmula:C19H23NO4
    Pureza:99.02% - 99.73%
    Cor e Forma:White Powder
    Peso molecular:329.39
  • Zinc Protoporphyrin

    CAS:
    <p>Zinc Protoporphyrin is an oral HO-1 inhibitor that reduces PG's protection against H2O2 and has anti-cancer properties.</p>
    Fórmula:C34H32N4O4Zn
    Pureza:95.43% - 99.27%
    Cor e Forma:Solid
    Peso molecular:626.02
  • Picrocrocin

    CAS:
    <p>Picrocrocin is a natural product</p>
    Fórmula:C16H26O7
    Pureza:98.4%
    Cor e Forma:Solid
    Peso molecular:330.37
  • Erdafitinib

    CAS:
    <p>Erdafitinib (JNJ-42756493) is a quinoxaline derivative compound, acts on FGFR1/2/3/4.</p>
    Fórmula:C25H30N6O2
    Pureza:97.00% - 99.07%
    Cor e Forma:Solid
    Peso molecular:446.54
  • 4-Methylbenzylidene camphor

    CAS:
    <p>4-Methylbenzylidene camphor: UVB blocker in sunscreens, cosmetics; exhibits estrogenic activity.</p>
    Fórmula:C18H22O
    Pureza:99.92%
    Cor e Forma:White Solid
    Peso molecular:254.37
  • L524-0366

    CAS:
    <p>L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.</p>
    Fórmula:C13H13ClN4OS
    Pureza:98.6% - 99.13%
    Cor e Forma:Solid
    Peso molecular:308.79
  • ASK1-IN-1

    CAS:
    <p>ASK1-IN-1 inhibits apoptosis kinase 1, crucial in cell stress responses, with 21 nM IC50.</p>
    Fórmula:C19H19N9O2
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:405.41
  • Tacedinaline

    CAS:
    <p>Tacedinaline (CI994) is a selective class I HDAC inhibitor with potential antineoplastic activity.</p>
    Fórmula:C15H15N3O2
    Pureza:96.83% - 99.15%
    Cor e Forma:White
    Peso molecular:269.3
  • Anagrelide

    CAS:
    <p>Anagrelide (Xagrid) is a Platelet-reducing Agent.</p>
    Fórmula:C10H7Cl2N3O
    Pureza:99.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:256.09
  • Diallyl Trisulfide

    CAS:
    <p>Diallyl Trisulfide is an organic polysulfide compound found in garlic that acts as an H2S donor.</p>
    Fórmula:C6H10S3
    Pureza:95% - ≥98%
    Cor e Forma:Liquid
    Peso molecular:178.34
  • Taurochenodeoxycholic Acid

    CAS:
    <p>Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.</p>
    Fórmula:C26H45NO6S
    Pureza:99.53% - 99.86%
    Cor e Forma:Solid
    Peso molecular:499.7
  • W-7 hydrochloride

    CAS:
    <p>W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride</p>
    Fórmula:C16H22Cl2N2O2S
    Pureza:99.63%
    Cor e Forma:White Crystalline Solid
    Peso molecular:377.32
  • MGH-CP1

    CAS:
    <p>MGH-CP1 inhibits TEAD2/4 auto-palmitoylation with IC50 of 710 and 672 nM, respectively.</p>
    Fórmula:C20H24N4OS
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:368.5
  • Levobupivacaine hydrochloride

    CAS:
    <p>Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.</p>
    Fórmula:C18H28N2O·HCl
    Pureza:99.74%
    Cor e Forma:White Crystalline Powder
    Peso molecular:324.89
  • CBL0137

    CAS:
    <p>CBL0137 (Curaxin 137), a metabolically stable curaxin, activates p53 (EC50: 0.37 μM) and inhibits NF-κB (EC50: 0.47 μM).</p>
    Fórmula:C21H24N2O2
    Pureza:99.57% - 99.68%
    Cor e Forma:Solid
    Peso molecular:336.43
  • BAY 61-3606 dihydrochloride

    CAS:
    <p>BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).</p>
    Fórmula:C20H18N6O3·2HCl
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:463.32
  • L-Ascorbic acid sodium salt

    CAS:
    <p>L-Ascorbic acid sodium salt (Vitamin C sodium salt) is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.</p>
    Fórmula:C6H7NaO6
    Pureza:98.73% - 99.75%
    Cor e Forma:Less Solid Powder
    Peso molecular:198.11
  • ISOGINKGETIN

    CAS:
    <p>ISOGINKGETIN (4',4'''-Dimethylamentoflavone), a compound derived from the leaves of Ginkgo biloba, to up-regulate adiponectin secretion.</p>
    Fórmula:C32H22O10
    Pureza:98% - 99.72%
    Cor e Forma:Solid
    Peso molecular:566.51
  • Lycorine

    CAS:
    <p>Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.</p>
    Fórmula:C16H17NO4
    Pureza:98.60% - 99.95%
    Cor e Forma:Solid
    Peso molecular:287.31
  • Alemtuzumab

    CAS:
    <p>Alemtuzumab is a humanized monoclonal antibody against CD52 an antigen found on the surface of normal and malignant lymphocytes.</p>
    Pureza:97.2% (SDS-PAGE); 96.7% (SEC-HPLC) - 98.00%
    Cor e Forma:Liquid
    Peso molecular:146.04 kDa
  • PKCβ inhibitor 1

    CAS:
    <p>PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,</p>
    Fórmula:C24H21N5O2
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:411.46
  • 2BAct

    CAS:
    <p>2BAct is a novel eif2b activator, preventing neurological defects caused by a chronic integrated stress response</p>
    Fórmula:C19H16ClF3N4O3
    Pureza:97.97% - 99.04%
    Cor e Forma:Solid
    Peso molecular:440.8
  • Ganoderic acid A

    CAS:
    <p>Ganoderic acid A fights tumors, suppresses gene regulators, induces cancer cell death, and enhances cisplatin efficacy.</p>
    Fórmula:C30H44O7
    Pureza:99.31% - ≥95%
    Cor e Forma:Solid
    Peso molecular:516.67
  • Cysteamine hydrochloride

    CAS:
    <p>Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant.</p>
    Fórmula:C2H7NS·HCl
    Pureza:99.34% - 99.87%
    Cor e Forma:White Crystalline Powder With A Strong And Disagreeable Smell
    Peso molecular:113.61