GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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Linaclotide acetate
CAS:<p>Linaclotide acetate, an oral guanylate cyclase C agonist with 14 amino acids, treats constipation-predominant IBS and chronic constipation.</p>Fórmula:C61H83N15O23S6Pureza:98%Cor e Forma:SolidPeso molecular:1586.79GLP-1R agonist 16
CAS:<p>Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].</p>Fórmula:C50H58FN10O6PCor e Forma:SolidPeso molecular:945.03Prostaglandin D2 methyl ester
CAS:<p>PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.</p>Fórmula:C21H34O5Cor e Forma:SolidPeso molecular:366.498GRL093-22
<p>GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.</p>Fórmula:C33H29FN6O3Cor e Forma:SolidPeso molecular:576.62Amylin (8-37), rat
CAS:<p>Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.</p>Fórmula:C140H227N43O43Pureza:98%Cor e Forma:SolidPeso molecular:3200.61Albiglutide fragment TFA
<p>Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as a</p>Fórmula:C148H224N40O45·xC2HF3O2Cor e Forma:SolidBIBP3226
CAS:<p>BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.</p>Fórmula:C27H31N5O3Cor e Forma:SolidPeso molecular:473.57CCR4 antagonist 3 hydrochloride
CAS:<p>Orally active CCR4 antagonist 3 hydrochloride with potent selectivity, IC50s: 22/50 nM; has antitumor properties.</p>Fórmula:C24H27Cl2N7O·xHClCor e Forma:SolidImnopitant dihydrochloride
CAS:<p>Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .</p>Fórmula:C28H30Cl2F6N4OCor e Forma:SolidPeso molecular:623.46Lys-γ3-MSH(human)
CAS:<p>Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysis</p>Fórmula:C128H193N45O39SPureza:98%Cor e Forma:SolidPeso molecular:3018.25Neuropeptide Y 13-36 (porcine)
CAS:<p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>Fórmula:C135H209N41O36Cor e Forma:SolidPeso molecular:2982.408Khusimol
CAS:Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Fórmula:C15H24OPureza:98%Cor e Forma:SolidPeso molecular:220.35Ramelteon metabolite M-II
CAS:<p>Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.</p>Fórmula:C16H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:275.34Alverine hydrochloride
CAS:<p>Alverine hydrochloride is a parasympatholytic.</p>Fórmula:C20H28ClNCor e Forma:SolidPeso molecular:317.9HTL22562
CAS:<p>HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.</p>Fórmula:C40H49N11O5Cor e Forma:SolidPeso molecular:763.904(S)-V-0219 hydrochloride
<p>(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.</p>Fórmula:C20H26ClF3N4O2Cor e Forma:SolidPeso molecular:446.89PACAP (6-38), human, ovine, rat
CAS:<p>PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.</p>Fórmula:C182H300N56O45SPureza:98%Cor e Forma:SolidPeso molecular:4024.74Orexin B, rat, mouse
CAS:<p>Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.</p>Fórmula:C126H215N45O34SPureza:98%Cor e Forma:SolidPeso molecular:2936.45Metaraminol
CAS:<p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Fórmula:C9H13NO2Cor e Forma:SolidPeso molecular:167.21Bodilisant
CAS:<p>Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.</p>Fórmula:C27H34BF2N3OCor e Forma:SolidPeso molecular:465.4Hemokinin 1 (mouse)
CAS:<p>Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.</p>Fórmula:C61H100N22O15SPureza:98%Cor e Forma:White PowderPeso molecular:1413.65Neuropeptide FF
CAS:<p>Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).</p>Fórmula:C54H76N14O10Pureza:98%Cor e Forma:SolidPeso molecular:1081.27Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Fórmula:C23H27N5O3Cor e Forma:SolidPeso molecular:421.501Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Fórmula:C14H20ClN3SCor e Forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85Plecanatide acetate
CAS:Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Fórmula:C67H108N18O28S4Pureza:98%Cor e Forma:SolidPeso molecular:1741.94d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Fórmula:C47H67N11O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1026.2FXR/TGR5 agonist 1
CAS:<p>FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.</p>Fórmula:C31H32ClN3O3Cor e Forma:SolidPeso molecular:530.07[D-Trp8]-γ-MSH
CAS:<p>[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).</p>Fórmula:C74H99N21O16SPureza:98%Cor e Forma:SolidPeso molecular:1570.798-iso Prostaglandin E2
CAS:<p>"8-iso PGE2: Isoprostane from arachidonic acid, potent rat renal vasoconstrictor, reduces GFR and renal flow by 80%, no BP effect."</p>Fórmula:C20H32O5Cor e Forma:SolidPeso molecular:352.47Neuropeptide Y5 receptor ligand-1
CAS:<p>Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].</p>Fórmula:C19H17N3O2Cor e Forma:SolidPeso molecular:319.36Neurokinin B
CAS:<p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>Fórmula:C55H79N13O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1210.4217-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:<p>Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.</p>Fórmula:C27H39NO4Cor e Forma:SolidPeso molecular:441.612Bz-Dab(nbd)-awfpp-nle-NH2
CAS:<p>Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.</p>Fórmula:C56H65N13O11Cor e Forma:SolidPeso molecular:1096.2L-797,591
CAS:<p>L-797,591 is a selective agonist of somatostatin receptor subtype 1.</p>Fórmula:C38H49N5O2Cor e Forma:SolidPeso molecular:607.83dCNP
<p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>Fórmula:C141H248N38O36S3Cor e Forma:SolidPeso molecular:3147.91RGS2-Galpha-q interaction-IN-1
RGS2–Galpha-q interaction-IN-1 (Compound AJ-3) is an inhibitor of the RGS2-Galpha-q interaction. It inhibits the growth of cancer cell lines that express RGS2 and has anti-cell migration properties.Fórmula:C30H30ClN7O3Cor e Forma:SolidPeso molecular:572.06Apelin-12 acetate
<p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>Fórmula:C66H107N21O16SPureza:98.82%Cor e Forma:SolidPeso molecular:1482.7517-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Fórmula:C25H37NO5Cor e Forma:SolidPeso molecular:431.573Avorelin
CAS:<p>Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.</p>Fórmula:C65H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1296.48NI-0701
<p>NI-0701 is a humanized antibody targeting CCL5/RANTES.</p>Pureza:95.4% (SDS-PAGE); 99.4% (SEC-HPLC) - 95.4% (SDS-PAGE); 99.4% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:145.5kDaM40
CAS:<p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>Fórmula:C94H145N23O24Pureza:98%Cor e Forma:SolidPeso molecular:1981.33[Nle11]-Substance P
CAS:<p>'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'</p>Fórmula:C64H100N18O13Pureza:98%Cor e Forma:SolidPeso molecular:1329.59Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Fórmula:C163H267N51O50S2Pureza:98%Cor e Forma:SolidPeso molecular:3805.31Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29Cloprostenol isopropyl ester
CAS:<p>(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.</p>Fórmula:C25H35ClO6Cor e Forma:SolidPeso molecular:466.99Bertilimumab
CAS:<p>Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].</p>Cor e Forma:LiquidGalanin (1-16), mouse, porcine, rat TFA
<p>Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.</p>Fórmula:C80H117F3N20O23Pureza:98%Cor e Forma:SolidPeso molecular:1783.917-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS:<p>17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.</p>Fórmula:C26H37NO4Cor e Forma:SolidPeso molecular:427.585Dehydro Aripiprazole (hydrochloride)
CAS:<p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>Fórmula:C23H26Cl3N3O2Cor e Forma:SolidPeso molecular:482.83[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Fórmula:C74H112N22O18SPureza:98%Cor e Forma:SolidPeso molecular:1629.88GLP-1R Antagonist 1
CAS:<p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>Fórmula:C16H11ClF6N4O2Pureza:99.84%Cor e Forma:SolidPeso molecular:440.73Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Fórmula:C22H15ClFN7OCor e Forma:SolidPeso molecular:447.86Adenosine 2',5'-diphosphate sodium
CAS:<p>Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.</p>Fórmula:C10H15N5NaO10P2Cor e Forma:SolidPeso molecular:450.192Antipsychotic agent-2
<p>Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.</p>Fórmula:C22H26FN5OCor e Forma:SolidPeso molecular:395.47Glucagon receptor antagonists-1
CAS:<p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>Fórmula:C29H34FNO2Pureza:98%Cor e Forma:SolidPeso molecular:447.58Somatostatin-28 (1-14)
CAS:<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Fórmula:C61H105N23O21SPureza:98%Cor e Forma:SolidPeso molecular:1528.71[Ala1,3,11,15]-Endothelin
CAS:<p>Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).</p>Fórmula:C109H163N25O32SPureza:98%Cor e Forma:SolidPeso molecular:2368Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Fórmula:C24H21N5O5SCor e Forma:SolidPeso molecular:491.52Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Fórmula:C74H92ClN17O13Pureza:98%Cor e Forma:SolidPeso molecular:1463.08IRL-1620
CAS:<p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>Fórmula:C86H117N17O27Pureza:98%Cor e Forma:SolidPeso molecular:1820.974Dipentylone hydrochloride
CAS:<p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>Fórmula:C14H20ClNO3Pureza:99.94%Cor e Forma:SolidPeso molecular:285.77α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFórmula:C162H262N50O52S2Pureza:98%Cor e Forma:SolidPeso molecular:3806.25Vapiprost hydrochloride
CAS:<p>Vapiprost hydrochloride is a biochemicla.</p>Fórmula:C30H40ClNO4Cor e Forma:SolidPeso molecular:514.117-phenyl trinor Prostaglandin E2 ethyl amide
CAS:<p>17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.</p>Fórmula:C25H35NO4Cor e Forma:SolidPeso molecular:413.5516-phenoxy tetranor Prostaglandin F2α methyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Fórmula:C23H32O6Cor e Forma:SolidPeso molecular:404.503GB-110 hydrochloride
<p>GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.</p>Fórmula:C33H49ClN6O5Cor e Forma:SolidPeso molecular:645.23Rubraxanthone
CAS:<p>Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.</p>Fórmula:C24H26O6Cor e Forma:SolidPeso molecular:410.466β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Fórmula:C162H267N51O48S3Pureza:98%Cor e Forma:SolidPeso molecular:3793.41Gulgafafusp alfa
CAS:<p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>Cor e Forma:LiquidApelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Fórmula:C185H304N68O43SPureza:98%Cor e Forma:SolidPeso molecular:4200.93S(-)-Bisoprolol fumarate
CAS:<p>S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.</p>Fórmula:C18H31NO4·xC4H4O4Cor e Forma:SolidPeso molecular:441.521Eletriptan
CAS:<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Fórmula:C22H26N2O2SCor e Forma:SolidPeso molecular:382.52Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Fórmula:C21H26Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:433.4Vicasinabin
CAS:<p>Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.</p>Fórmula:C15H22N10OCor e Forma:SolidPeso molecular:358.4115-keto Latanoprost
CAS:<p>Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.</p>Fórmula:C26H38O5Cor e Forma:SolidPeso molecular:430.58Substance P (1-9)
CAS:<p>Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.</p>Fórmula:C52H77N15O12Pureza:98%Cor e Forma:SolidPeso molecular:1104.26(S, R)-LSN 3318839
CAS:<p>(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.</p>Fórmula:C26H23Cl2N3O2Pureza:99.57%Cor e Forma:SoildPeso molecular:480.39Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Fórmula:C16H18ClN3Pureza:98.45%Cor e Forma:SoildPeso molecular:287.79THX-B
CAS:<p>THX-B, a potent non-peptidic p75 NTR antagonist, aids in researching diabetic kidney disease and neurodegenerative and inflammatory disorders.</p>Fórmula:C16H24N6O4Cor e Forma:SolidPeso molecular:364.4Spantide II
CAS:<p>Spantide II is an antagonist of tachykinin.</p>Fórmula:C86H104Cl2N18O13Pureza:98%Cor e Forma:SolidPeso molecular:1668.77LHRH, Ala(6)-
CAS:<p>LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.</p>Fórmula:C56H77N17O13Cor e Forma:SolidPeso molecular:1196.32Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Fórmula:C27H22F4N4O3SPureza:98.83%Cor e Forma:SolidPeso molecular:558.55PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Fórmula:C142H224N40O39SPureza:98%Cor e Forma:SolidPeso molecular:3147.66{Val1}-Exendin-3/4
{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.Fórmula:NAPureza:98%Cor e Forma:SolidPeso molecular:3241.7Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Fórmula:C184H297N69O43SPureza:98%Cor e Forma:SolidPeso molecular:4195.87PF-03382792
CAS:<p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>Fórmula:C23H32FN3O4Pureza:99.64%Cor e Forma:SolidPeso molecular:433.52A71378
CAS:<p>A71378 is a high potency, selectivity CCK-A receptors agonist.</p>Fórmula:C48H62N8O13SPureza:98%Cor e Forma:SolidPeso molecular:991.12(R)-CJ 11974
CAS:<p>(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.</p>Fórmula:C31H38N2OPureza:97.15%Cor e Forma:SoildPeso molecular:454.65RWJ 676070
CAS:<p>RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.</p>Fórmula:C30H26ClFN2O5Cor e Forma:SolidPeso molecular:548.99Chemerin-9 (149-157) TFA
<p>Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.</p>Fórmula:C56H67F3N10O15Pureza:99.77%Cor e Forma:SolidPeso molecular:1177.18FR190997
CAS:<p>FR190997 is an agonist of bradykinin B2 receptor.</p>Fórmula:C37H33Cl2N5O5Cor e Forma:SolidPeso molecular:698.59Ecraprost
CAS:<p>Ecraprost is used as a prodrug of prostaglandin E1.</p>Fórmula:C28H48O6Cor e Forma:SolidPeso molecular:480.68Enuvaptan
CAS:<p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>Fórmula:C21H15ClF6N8O3Cor e Forma:SolidPeso molecular:576.84I-BOP
CAS:<p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>Fórmula:C23H29IO5Cor e Forma:SolidPeso molecular:512.384CRL-42872 free base
CAS:<p>CRL-42872 free base is a bioactive chemical.</p>Fórmula:C22H26N6O6SCor e Forma:SolidPeso molecular:502.54AB21 HCl
<p>AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces mechanical hypersensitivity.</p>Fórmula:C23H29ClN2OPureza:99.91%Cor e Forma:SolidPeso molecular:384.2NF157
CAS:<p>NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.</p>Fórmula:C49H28F2N6Na6O23S6Pureza:98%Cor e Forma:SolidPeso molecular:1437.1(R)-V-0219 hydrochloride
<p>(R)-V-0219 hydrochloride: Oral GLP-1R PAM, enantiomer of V-0219, triggers Ca2+ flux in hGLP-1R HEK cells.</p>Fórmula:C20H26ClF3N4O2Cor e Forma:SolidPeso molecular:446.89Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Fórmula:C22H37NO4Cor e Forma:SolidPeso molecular:379.541GLP-1R agonist 27
<p>GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).</p>Fórmula:C32H33N5O4SeCor e Forma:SolidPeso molecular:630.6
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