GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(993 produtos)
- Receptor de adenosina(246 produtos)
- Receptor adrenérgico(3.004 produtos)
- Receptor de Bombesina(33 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(153 produtos)
- CaSR(33 produtos)
- Receptor de Canabinóides(212 produtos)
- Receptor de Dopamina(433 produtos)
- Receptor Endotelina(79 produtos)
- Receptor GNRH(77 produtos)
- GPCR19(32 produtos)
- GRK(32 produtos)
- GTPase(22 produtos)
- Receptor Glucagon(182 produtos)
- Hedgehog/Smoothened(47 produtos)
- Receptor de Histamina(381 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(26 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(310 produtos)
- PAFR(12 produtos)
- PKA(51 produtos)
- Receptor S1P(18 produtos)
- SGLT(31 produtos)
- Receptor Sigma(46 produtos)
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Foram encontrados 5745 produtos de "GPCR/Proteína-G"
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Neurokinin B
CAS:<p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>Fórmula:C55H79N13O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1210.42Osanetant
CAS:Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Fórmula:C35H41Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:606.62Parstatin(mouse)
CAS:Peptide inhibits endothelial migration/proliferation (IC50 ~20μM), induces cell cycle arrest, triggers apoptosis, and has cardioprotective effects.Fórmula:C189H326N58O57S3Pureza:98%Cor e Forma:SolidPeso molecular:4419.19Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Fórmula:C53H71N11O14S2Cor e Forma:SolidPeso molecular:1150.33Kisspeptin-10, rat TFA
<p>Kisspeptin-10, a rat TFA, constricts blood vessels, inhibits vessel growth, and counters Methotrexate reproductive toxicity.</p>Fórmula:C65H84F3N17O17Cor e Forma:SolidPeso molecular:1432.46Neuropeptide Y (human)
CAS:<p>Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.</p>Fórmula:C189H285N55O57SPureza:98%Cor e Forma:SolidPeso molecular:4271.68Peptide YY (PYY) (3-36), porcine TFA
Peptide YY (PYY) (3-36), porcine TFA, functions as a gut hormone that serves as a Y2 receptor agonist, effectively reducing appetite [1].Fórmula:C176H272N52O54·C2HF3O2Cor e Forma:SolidPeso molecular:4094.44Y1 receptor antagonist 1 formic
<p>H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.</p>Fórmula:C29H35N5O5Cor e Forma:SolidPeso molecular:533.62Adrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Fórmula:C248H381N77O75S5Pureza:98%Cor e Forma:SolidPeso molecular:5729.5Pemvidutide TFA
Pemvidutide (TFA), a GLP-1R/GCGR dual agonist, effectively reduces body weight, liver fat, and serum lipid levels, and is utilized in research on non-alcoholicFórmula:C182H275N39O54·xC2HF3O2Cor e Forma:SolidPeso molecular:3873.35 (free base)Albiglutide Fragment
CAS:<p>Albiglutide fragment is a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).</p>Fórmula:C148H224N40O45Pureza:98%Cor e Forma:SolidPeso molecular:3283.6CYN 154806
CAS:CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).Fórmula:C56H68N12O14S2Pureza:98%Cor e Forma:SolidPeso molecular:1197.34Amylin (8-37) (human)
CAS:Amylin (8-37) (human) is a fragment of human IAPP with a hairpin structure.Fórmula:C138H215N41O46Cor e Forma:SolidPeso molecular:3184.43PG-931 TFA
PG-931 TFA, a potent MC4 receptor agonist (IC50 0.58 nM), excels in selectivity and helps reverse hemorrhagic shock in vivo.Fórmula:C61H86F3N15O13Cor e Forma:SolidPeso molecular:1294.42PAMP-12 (unmodified) (TFA)
<p>PAMP-12 (unmodified) TFA, an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine secretion</p>Fórmula:C79H119F3N24O17Cor e Forma:SolidPeso molecular:1733.94Veldoreotide
CAS:Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Fórmula:C60H74N12O10Pureza:98%Cor e Forma:SolidPeso molecular:1123.3[D-p-Cl-Phe6,Leu17]-VIP
CAS:Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.Fórmula:C148H239ClN44O42Pureza:98%Cor e Forma:SolidPeso molecular:3342.24Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS:O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Fórmula:C11H11NO3Cor e Forma:SolidPeso molecular:205.213ELA-32(human)
CAS:Potent apelin receptor agonist with IC50 = 0.27 nM; does not bind GPR15/GPR25. Boosts hESC self-renewal and angiogenesis.Fórmula:C170H289N63O39S4Pureza:98%Cor e Forma:SolidPeso molecular:3967.8LMN-NKA acetate
LMN-NKA acetate is a modified Neurokinin A (4-10) and selective NK2R (Neurokinin 2 receptor) agonist induces bladder contraction smooth muscle contraction.Fórmula:C41H68N8O12Cor e Forma:SolidPeso molecular:865.03Pirepemat
CAS:Pirepemat (IRL752) is a cortical-preferring catecholamine agent that enhances cognition. It is utilized in the investigation of Parkinson's disease.Fórmula:C11H13F2NOCor e Forma:SolidPeso molecular:213.22MM 419447
CAS:<p>MM 419447, a linaclotide metabolite, is a guanylate cyclase-C agonist showing potential in IBS-C research.</p>Fórmula:C50H70N14O19S6Cor e Forma:SolidPeso molecular:1363.55Myristoylated ARF6 (2-13)
Myristoylated ARF6 (2-13) inhibits the MyD88–ARNO–ARF6 signaling axis by inactivating ARF6.Fórmula:C74H128N16O18Peso molecular:1528.95925VIP36
<p>VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.</p>Fórmula:C27H35FN6O4Cor e Forma:SolidPeso molecular:526.603Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Fórmula:C184H297N69O43SPureza:98%Cor e Forma:SolidPeso molecular:4195.87d[Cha4]-AVP
CAS:Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Fórmula:C50H71N13O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1094.31Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Fórmula:C14H22ClNOCor e Forma:SolidPeso molecular:255.78DSP-1053
CAS:Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.Fórmula:C26H32BrNO4Pureza:98%Cor e Forma:SolidPeso molecular:502.44Scyliorhinin II
CAS:Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.Fórmula:C77H119N21O26S3Pureza:98%Cor e Forma:SolidPeso molecular:1851.09GLP-1(9-36)amide TFA
GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.Fórmula:C142H215F3N36O45Cor e Forma:SolidPeso molecular:3203.43Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:1583.78 (free base)[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS:<p>'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.</p>Fórmula:C39H64N8O10Cor e Forma:SolidPeso molecular:804.97Thioperamide maleate
CAS:<p>Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31</p>Fórmula:C19H28N4O4SPureza:98.48%Cor e Forma:SolidPeso molecular:408.52HS014
CAS:Potent MC4 antagonist; Ki: 3.16 nM (MC4), 108 (MC1), 54.4 (MC3), 694 (MC5). Boosts rat appetite, mouse pain, blocks IL-1β Fos in hypothalamus.Fórmula:C71H94N20O17S2Pureza:98%Cor e Forma:SolidPeso molecular:1563.77Dipentylone hydrochloride
CAS:Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.Fórmula:C14H20ClNO3Pureza:99.94%Cor e Forma:SolidPeso molecular:285.77NF546
CAS:<p>NF546 is a selective agonist of non-nucleotide P2Y11(pEC50 of 6.27).</p>Fórmula:C47H44N6Na4O17P4Pureza:98%Cor e Forma:SolidPeso molecular:1180.74Apelin-17(human, bovine)
CAS:<p>Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).</p>Fórmula:C96H156N34O20SPureza:98%Cor e Forma:SolidPeso molecular:2138.5615-keto-17-phenyl trinor Prostaglandin F2α ethyl amide
CAS:Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which hasFórmula:C25H35NO4Cor e Forma:SolidPeso molecular:413.558GLP-1(7-36), amide acetate
CAS:GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.Fórmula:C151H230N40O47Pureza:99.89%Cor e Forma:SolidPeso molecular:3357.68Protease-Activated Receptor-1, PAR-1 Agonist TFA
<p>PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.</p>Cor e Forma:LiquidGalanin (2-29) (rat)
CAS:Peptide agonist for galanin receptorsFórmula:C139H208N42O40Pureza:98%Cor e Forma:SolidPeso molecular:3107.4Thielavin A
CAS:Thielavin A, from T. terricola, inhibits COX and glucose-6-phosphatase; non-competitive α-glucosidase inhibitor.Fórmula:C29H30O10Cor e Forma:SolidPeso molecular:538.549EP4-IN-1
CAS:EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.Fórmula:C27H24N2O4Pureza:99.94%Cor e Forma:SoildPeso molecular:440.49Quetiapine-d4 fumarate
CAS:Deuterium-labeled Quetiapine fumarate; an antidepressant and anxiolytic 5-HT agonist, dopamine antagonist.Fórmula:C25H29N3O6SPureza:98%Cor e Forma:SolidPeso molecular:503.61S1PR1 modulator 1
CAS:S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.Fórmula:C23H24N2O3SPureza:99.69%Cor e Forma:SolidPeso molecular:408.51Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Fórmula:C84H130F3N25O23S2Cor e Forma:SolidPeso molecular:1979.21Tetrahydro-β-carboline
CAS:<p>Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C11H12N2Pureza:96.31%Cor e Forma:Tan SolidPeso molecular:172.2264PACAP (1-38), human, ovine, rat TFA
PACAP (1-38), neuropeptide from bovine brain, surpasses VIP in adenylate cyclase activation (EC50=7 nM), alters peptide release, affects gastrin and motility.Fórmula:C203H331N63O53S·C2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:4648.28Rp-UTP-α-S tetrasodium
Rp-UTP-α-S (tetrasodium) is a nucleotide agonist of the purinergic P2Y2 and P2Y4 receptors. It can induce the accumulation of inositol phosphate in 1321N1 cells expressing P2Y2 or P2Y4, with EC50 values of 5.4 and 27 μM, respectively.Cor e Forma:Odour SolidCinnamtannin A2
CAS:<p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>Fórmula:C60H50O24Cor e Forma:SolidPeso molecular:1155.02Hemokinin 1, human
CAS:Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.Fórmula:C54H84N14O14SPureza:98%Cor e Forma:SolidPeso molecular:1185.4α1A-AR Degrader 9c
CAS:α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Fórmula:C38H43N11O11Pureza:98%Cor e Forma:SolidPeso molecular:829.82ELA-21 (human)
CAS:<p>Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.</p>Fórmula:C112H184N40O25S3Pureza:98%Cor e Forma:SolidPeso molecular:2587.12tetranor-PGJM
CAS:<p>Tetranor-PGJM is a metabolite of prostaglandin D2 and is associated with the anti-inflammatory effects of curcumin.</p>Fórmula:C16H22O6Cor e Forma:SolidPeso molecular:310.346Propranolol hydrochloride
CAS:Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverseFórmula:C16H22ClNO2Pureza:99.94% - >99.99%Cor e Forma:White Or Almost White Powder White PowderPeso molecular:295.80MR33317
<p>MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.</p>Fórmula:C22H28ClN3O2Peso molecular:401.1874-Chloromethamphetamine hydrochloride
CAS:<p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>Fórmula:C10H15Cl2NCor e Forma:SolidPeso molecular:220.14SB236057
CAS:SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.Fórmula:C33H34N4O3Pureza:98%Cor e Forma:SolidPeso molecular:534.65TDI-10229
CAS:<p>TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.</p>Fórmula:C16H16ClN5Pureza:99.85% - 99.89%Cor e Forma:SoildPeso molecular:313.78Adrenomedullin (AM) (22-52), human
CAS:<p>Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.</p>Fórmula:C159H252N46O48Pureza:98%Cor e Forma:SolidPeso molecular:3576.04Cholecystokinin (27-32)-amide
CAS:Cholecystokinin (27-32)-amide is a CCK receptor antagonist.Fórmula:C36H48N8O12S3Pureza:98%Cor e Forma:SolidPeso molecular:881.01[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.Fórmula:C82H120N20O25Cor e Forma:SolidPeso molecular:1785.95Carbazochrome salicylate
CAS:Carbazochrome salicylate can be used as a coagulant.Fórmula:C17H18N4NaO6Cor e Forma:White Crystalline PowderPeso molecular:397.343[Lys4] Sarafotoxin S6c
CAS:<p>[Lys4] Sarafotoxin S6c: potent partial endothelin receptor agonist; causes pig coronary contraction, EC50=1.5 nM.</p>Fórmula:C105H153N27O36S5Cor e Forma:SolidPeso molecular:2529.82Berobenatide
CAS:Berobenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist.Cor e Forma:SolidG-Protein antagonist peptide
CAS:<p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>Fórmula:C57H64N12O9SPureza:98%Cor e Forma:SolidPeso molecular:1093.27HCGRP-(8-37)
CAS:Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonistFórmula:C139H230N44O38Pureza:98%Cor e Forma:SolidPeso molecular:3125.59GnRH Associated Peptide (1-24), human
CAS:<p>GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.</p>Fórmula:C117H190N32O43Cor e Forma:SolidPeso molecular:2732.95Galanin (1-29)(rat, mouse)
CAS:<p>Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.</p>Fórmula:C141H211N43O41Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:3164.499Biotin-NeurokininA
Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.Fórmula:C60H94N16O16S2Cor e Forma:SolidPeso molecular:1359.61PAR650097
PAR650097 is a humanized monoclonal antibody targeting PAR2, used in migraine research.Pureza:96.67% (SEC-HPLC) - 98.83% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:145.5kDaZebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Fórmula:C58H84N16O15Cor e Forma:SolidPeso molecular:1245.39[Arg-15,20,21,Leu17]-PACAP-Gly-Lys-Arg-NH2
CAS:<p>[Arg-15,-20,-21, Leu17]-PACAP-Gly-Lys-Arg-NH2 (BM-PACAP) is a synthetic analogue of PACAP 1-27 that exhibits a relaxant effect [1].</p>Fórmula:C157H253N53O42Cor e Forma:SolidPeso molecular:3555.02BA 1
CAS:<p>Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.</p>Fórmula:C57H76N14O11Pureza:98%Cor e Forma:SolidPeso molecular:1133.32Atrial Natriuretic Peptide (ANP) (1-28), rat
CAS:Atrial Natriuretic Peptide (1-28), rat is the major circulating form of ANP in rats.Fórmula:C128H205N45O39S2Pureza:98%Cor e Forma:SolidPeso molecular:3062.41(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Fórmula:C52H74N14O12S2Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:1151.38Urocortin, rat
CAS:<p>Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.</p>Fórmula:C206H338N62O64Pureza:98%Cor e Forma:SolidPeso molecular:4707.26CYM5442 hydrochloride
CAS:<p>CYM 5442 HCl: potent, selective S1P1 agonist (EC50 = 1.35 nM), induces MAPK activation & lymphopenia, brain-penetrant.</p>Fórmula:C23H28ClN3O4Cor e Forma:SolidPeso molecular:445.94L-692429 HCl
CAS:L-692,429 is a novel non-peptide growth hormone secretagin.Fórmula:C29H32ClN7O2Cor e Forma:SolidPeso molecular:546.06CB2 receptor antagonist 2
Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 μM.Cor e Forma:Odour SolidBMS-753426
CAS:<p>BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .</p>Fórmula:C25H33F3N6O2Cor e Forma:SolidPeso molecular:506.574LY86057
CAS:LY86057 is a bioactive chemical.Fórmula:C20H26N2O3Cor e Forma:SolidPeso molecular:342.439LY-53857 free base
CAS:LY-53857 free base is a bioactive chemical.Fórmula:C23H32N2O3Cor e Forma:SolidPeso molecular:384.51Δ9-THCH
CAS:Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Fórmula:C22H32O2Cor e Forma:SolidPeso molecular:328.49CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Cor e Forma:Odour Solid16-phenoxy tetranor Prostaglandin F2α
CAS:16-phenoxy PGF2α is a metabolically stable analog of PGF2α. It binds to the FP receptor on ovine luteal cells with much greater affinity (440%) than PGF2α.Fórmula:C22H30O6Cor e Forma:SolidPeso molecular:390.47ACTH (4-11)
CAS:ACTH (4-11) is a peptide fragment of adrenocorticotropic hormone, a peptide hormone found in the brain that is involved in the biological stress response.Fórmula:C50H71N15O11SPureza:98%Cor e Forma:SolidPeso molecular:1090.265-Bromoimidazo[1,2-A]Pyrazine
CAS:5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.Fórmula:C6H4BrN3Pureza:99.92%Cor e Forma:SolidPeso molecular:198.02MGV354
MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].Fórmula:C35H37N5O3Pureza:98%Cor e Forma:SolidPeso molecular:575.7Urocortin II, human acetate
Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.Cor e Forma:Odour SolidDabelotine, (R)-
CAS:Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Fórmula:C15H22N2O2Cor e Forma:SolidPeso molecular:262.35Peptide YY (PYY), human
CAS:<p>PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.</p>Fórmula:C194H295N55O57Pureza:98%Cor e Forma:SolidPeso molecular:4309.75β2AR/M-receptor agonist-1
CAS:β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFórmula:C43H56BrN3O7Cor e Forma:SolidPeso molecular:806.82ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
CAS:<p>ACTH (3-24) is the fragment 3-24 of ACTH, used in disease research including cancer and immune disorders.</p>Fórmula:C124H196N38O27SCor e Forma:SolidPeso molecular:2683.19CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Fórmula:C74H96N14O15S2Pureza:98%Cor e Forma:SolidPeso molecular:1485.8Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Fórmula:C188H276N51F3O61Pureza:98%Cor e Forma:SolidPeso molecular:4283.5Endothelin-2 (49-69), human TFA
Endothelin-2 (49-69), human (TFA) is a 21-amino acid vasoactive peptide that binds to ET-RA and ET-RB.Fórmula:C117H161N26F3O34S4Pureza:98%Cor e Forma:SolidPeso molecular:2660.94HAEGTFTSD
CAS:<p>HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.</p>Fórmula:C40H57N11O17Pureza:98%Cor e Forma:SolidPeso molecular:963.94GB-6
CAS:<p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>Fórmula:C32H45N11O8Pureza:98%Cor e Forma:SolidPeso molecular:711.77
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