GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.946 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(408 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5360 produtos de "GPCR/Proteína-G"
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TGR5 agonist 4
<p>TGR5 agonist 4 (compound 19), a derivative of cholic acid, selectively activates the TGR5 receptor with an effective concentration (EC50) of 4 μM [1].</p>Fórmula:C24H38F2O5Cor e Forma:SolidPeso molecular:444.55LGnRH-III, lamprey
CAS:<p>GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.</p>Fórmula:C59H74N18O14Pureza:98%Cor e Forma:SolidPeso molecular:1259.33PF-9184
CAS:<p>PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.</p>Fórmula:C21H14Cl2N2O4SPureza:97.43%Cor e Forma:SolidPeso molecular:461.32Veldoreotide
CAS:Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Fórmula:C60H74N12O10Pureza:98%Cor e Forma:SolidPeso molecular:1123.3Senktide TFA
<p>Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.</p>Cor e Forma:Odour SolidOrexin B, human
CAS:<p>Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.</p>Fórmula:C123H212N44O35SPureza:98%Cor e Forma:SolidPeso molecular:2899.34P2Y6R antagonist 1
<p>P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.</p>Cor e Forma:Odour SolidDulaglutide
CAS:<p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>Cor e Forma:SolidACT-373898
CAS:<p>ACT-373898 is a metabolite of the endothelin (ET) receptor type A (ETA) and ETBdual antagonist macitentan .1</p>Fórmula:C15H17BrN4O5SCor e Forma:SolidPeso molecular:445.29Fluphenazine free base
CAS:<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Fórmula:C22H26F3N3OSCor e Forma:SolidPeso molecular:437.52Zoliprofen
CAS:<p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.29Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Fórmula:C215H358N72O66SPureza:98%Cor e Forma:SolidPeso molecular:5039.65Cloprostenol isopropyl ester
CAS:<p>(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.</p>Fórmula:C25H35ClO6Cor e Forma:SolidPeso molecular:466.99Guanylin TFA (mouse,rat)
<p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>Fórmula:C60H90N16O22S4·xC2HF3O2Cor e Forma:SolidPeso molecular:1515.71 (free base)PACAP (6-38), human, ovine, rat TFA
<p>PACAP (6-38) is a PACAP receptor blocker with IC50s of 30, 600, 40 nM for type I, VIP1, and VIP2 receptors.</p>Fórmula:C184H301N56FO47SPureza:98%Cor e Forma:SolidPeso molecular:4138.76Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Fórmula:C19H23N3Pureza:99.88%Cor e Forma:White/Pale Yellow Crystalline SolidPeso molecular:293.41Brexpiprazole S-oxide
CAS:<p>Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).</p>Fórmula:C25H27N3O3SPureza:98%Cor e Forma:SolidPeso molecular:449.57KwFwLL-NH2
CAS:<p>KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).</p>Fórmula:C49H66N10O6Cor e Forma:SolidPeso molecular:891.11Seglitide
CAS:<p>Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.</p>Fórmula:C44H56N8O7Pureza:98%Cor e Forma:SolidPeso molecular:808.98β-CGRP (mouse)
<p>β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.</p>Fórmula:C165H265N49O55S2Cor e Forma:SolidPeso molecular:3879.29LSN3160440
CAS:<p>LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.</p>Fórmula:C27H27Cl2N3OCor e Forma:SolidPeso molecular:480.43Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Fórmula:C12H14ClN5O2SeCor e Forma:SolidPeso molecular:374.68Y1 receptor antagonist 1 formic
<p>H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.</p>Fórmula:C29H35N5O5Cor e Forma:SolidPeso molecular:533.62cAC 253 acetate
<p>cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.</p>Fórmula:C128H206N42O42S2Pureza:98.16% - 99.99%Cor e Forma:SoildPeso molecular:3069.39T-10430
<p>T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.</p>Fórmula:C17H22N6OCor e Forma:SolidPeso molecular:326.396MI 1544
CAS:<p>MI 1544 is a LHRH antagonist.</p>Fórmula:C71H94ClN17O13Cor e Forma:SolidPeso molecular:1429.09Dexchlorpheniramine free base
CAS:<p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>Fórmula:C16H19ClN2Pureza:98%Cor e Forma:Oily Liquid SolidPeso molecular:274.79Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Fórmula:C83H118N20O20S2Pureza:98.24% - 99.63%Cor e Forma:SoildPeso molecular:1780.08Adrenocorticotropic Hormone (ACTH) (1-39), rat
CAS:<p>ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.</p>Fórmula:C210H315N57O57SPureza:98%Cor e Forma:SolidPeso molecular:4582.23HDAC6-IN-49
<p>HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.</p>Cor e Forma:Odour SolidMrgprX2 antagonist-5
CAS:<p>MrgprX2 antagonist-5 from patent WO2020223255A1 inhibits MrgprX2, useful for inflammatory skin disorder studies.</p>Fórmula:C19H13ClF2N4O2SCor e Forma:SolidPeso molecular:434.85[Nle11]-Substance P
CAS:<p>'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'</p>Fórmula:C64H100N18O13Pureza:98%Cor e Forma:SolidPeso molecular:1329.59Asenapine citrate
CAS:<p>Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).</p>Fórmula:C23H24ClNO8Cor e Forma:SolidPeso molecular:477.89CB1R agonist 1
<p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>Fórmula:C20H18F3N3O3SCor e Forma:SolidPeso molecular:437.435Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:1583.78 (free base)Thioperamide maleate
CAS:<p>Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31</p>Fórmula:C19H28N4O4SPureza:98.48%Cor e Forma:SolidPeso molecular:408.52Peptide YY (PYY), human
CAS:<p>PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.</p>Fórmula:C194H295N55O57Pureza:98%Cor e Forma:SolidPeso molecular:4309.75MrgprX2 antagonist-3
CAS:<p>MrgprX2 antagonist-3 (compound E117) is a MrgprX2 antagonist applicable for investigating cutaneous inflammation.</p>Fórmula:C16H20FN3O2SPureza:98.06%Cor e Forma:SolidPeso molecular:337.41GLP-1(7-36), amide acetate
CAS:<p>GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.</p>Fórmula:C151H230N40O47Pureza:99.89%Cor e Forma:SolidPeso molecular:3357.68JNJ-10181457 (hydrochloride)
CAS:<p>JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations</p>Fórmula:C20H30Cl2N2OCor e Forma:SolidPeso molecular:385.37Lys-Bradykinin
CAS:<p>Endogenous bradykinin receptor agonist</p>Fórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38S1PR1 modulator 1
CAS:<p>S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.</p>Fórmula:C23H24N2O3SPureza:99.69%Cor e Forma:SolidPeso molecular:408.51M871
CAS:<p>GAL2 receptor antagonist; Ki: 13.1 nM (GAL2), 420 nM (GAL1); inhibits GAL2-induced pain.</p>Fórmula:C108H163N27O28Pureza:98%Cor e Forma:SolidPeso molecular:2287.64Syk Inhibitor II hydrochloride
CAS:<p>Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.</p>Fórmula:C14H16ClF3N6OPureza:99.05%Cor e Forma:SolidPeso molecular:376.77Agaridoxin
CAS:<p>Agaridoxin is a mushroom metabolite.</p>Fórmula:C11H14N2O5Cor e Forma:SolidPeso molecular:254.242Prostaglandin F1α
CAS:<p>Prostaglandin F1α (PGF1α) is a lipid mediator and an endogenous metabolite of prostacyclin, regulate smooth muscle contraction.</p>Fórmula:C20H36O5Cor e Forma:SolidPeso molecular:356.5K41498
CAS:<p>Potent CRF2α/β antagonist; Ki: 0.66/0.62 nM, weak for CRF1 (425 nM). Blocks sauvagine in hCRF2 cells and urocortin hypotension in rats.</p>Fórmula:C162H276N48O46Pureza:98%Cor e Forma:SolidPeso molecular:3632.26ALD1613
<p>ALD1613 is a potent neutralizing monoclonal antibody targeting adrenocorticotropic hormone (ACTH). It neutralizes ACTH-induced signaling and inhibits cyclic adenosine monophosphate accumulation in ACTH-stimulated Y1 (mouse adrenal cell line) via all five melanocortin receptors. ALD1613 significantly reduces plasma corticosterone levels in wild-type rats and is applicable in studies involving elevated ACTH-related conditions.</p>Cor e Forma:Odour Liquid8-iso-15-keto Prostaglandin F2α
CAS:<p>8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.</p>Fórmula:C20H32O5Cor e Forma:SolidPeso molecular:352.471Adrenomedullin (AM) (22-52), human TFA
<p>Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.</p>Fórmula:C161H253N46F3O50Pureza:98%Cor e Forma:SolidPeso molecular:3690.06LP 12 hydrochloride
CAS:<p>LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).</p>Fórmula:C32H40ClN3OCor e Forma:SolidPeso molecular:518.14PY-60
CAS:<p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>Fórmula:C16H15N3O2SPureza:99.5% - 99.67%Cor e Forma:SolidPeso molecular:313.37Scyliorhinin II
CAS:<p>Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.</p>Fórmula:C77H119N21O26S3Pureza:98%Cor e Forma:SolidPeso molecular:1851.09EP3 antagonist 4
CAS:<p>EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good bioavailability in rats, potential for diabetes research.</p>Fórmula:C22H20Cl3FN4O3S2Pureza:98%Cor e Forma:SoildPeso molecular:577.91(+)-Cloprostenol sodium
CAS:<p>Cloprostenol sodium is a water-soluble PGF2α analog and FP receptor agonist, promoting luteolysis in rats and hamsters.</p>Fórmula:C22H28ClNaO6Cor e Forma:SolidPeso molecular:446.9BIIE-0246
CAS:<p>BIIE-0246 is a potent and highly selective non-peptide neuropeptide Y (NPY) Y2 receptor antagonist. With an IC50 of 15 nM.</p>Fórmula:C49H57N11O6Pureza:98%Cor e Forma:SolidPeso molecular:896.05REGN-7544
<p>REGN-7544 is a humanised monoclonal antibody targeting NPR1, which blocks and inhibits NPR1 to increase blood pressure, hypotensione.</p>Pureza:95%Cor e Forma:Odour LiquidCagrilintide acetate
<p>.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.</p>Fórmula:C196H316N54O61S2Pureza:99.88%Cor e Forma:SolidPeso molecular:4469.06CRF, bovine
CAS:<p>CRF, bovine is a potent agonist of CRF receptor, and displaces [125I-Tyr]ovine CRF with a Ki of 3.52 nM.</p>Fórmula:C206H340N60O63SPureza:98%Cor e Forma:SolidPeso molecular:4697.34PF-07062119
<p>PF-07062119 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody designed to target and inhibit GUCY2C.</p>Cor e Forma:Odour LiquidSB-206606
CAS:<p>SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.</p>Fórmula:C19H22ClNO4Cor e Forma:SolidPeso molecular:363.83GLP-1 (9-36) amide
CAS:<p>GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.</p>Fórmula:C140H214N36O43Pureza:97%Cor e Forma:SolidPeso molecular:3089.41NF546
CAS:<p>NF546 is a selective agonist of non-nucleotide P2Y11(pEC50 of 6.27).</p>Fórmula:C47H44N6Na4O17P4Pureza:98%Cor e Forma:SolidPeso molecular:1180.74Isobutyryl-L-carnitine
CAS:<p>Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.</p>Fórmula:C11H21NO4Pureza:98%Cor e Forma:SolidPeso molecular:231.29Mosapride citrate dihydrate
CAS:<p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>Fórmula:C27H35ClFN3O11Pureza:98%Cor e Forma:SolidPeso molecular:632.04Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Cor e Forma:Odour SolidAZP-531
CAS:<p>Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.</p>Fórmula:C40H63N15O13Pureza:98%Cor e Forma:SolidPeso molecular:962.02Galanin (1-30), human
CAS:Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Fórmula:C139H210N42O43Pureza:98%Cor e Forma:SolidPeso molecular:3157.46LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Fórmula:C39H43ClN4O9S2Cor e Forma:SolidPeso molecular:811.36Quetiapine-d4 fumarate
CAS:<p>Deuterium-labeled Quetiapine fumarate; an antidepressant and anxiolytic 5-HT agonist, dopamine antagonist.</p>Fórmula:C25H29N3O6SPureza:98%Cor e Forma:SolidPeso molecular:503.61NTRC-824
CAS:<p>NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.</p>Fórmula:C25H26F3N3O6SPureza:98%Cor e Forma:SolidPeso molecular:553.55AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211Atrial natriuretic factor (1-28) (rat) TFA
<p>ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.</p>Fórmula:C130H206N45F3O41S2Pureza:98%Cor e Forma:SolidPeso molecular:3176.43Upidosin
CAS:<p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>Fórmula:C31H33N3O4Pureza:99.66%Cor e Forma:SolidPeso molecular:511.61Thielavin A
CAS:<p>Thielavin A, from T. terricola, inhibits COX and glucose-6-phosphatase; non-competitive α-glucosidase inhibitor.</p>Fórmula:C29H30O10Cor e Forma:SolidPeso molecular:538.5498-iso Prostaglandin E1
CAS:<p>8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.</p>Fórmula:C20H34O5Cor e Forma:Light Yellow Crystalline SolidPeso molecular:354.48Adrenomedullin (AM) (22-52), human
CAS:<p>Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.</p>Fórmula:C159H252N46O48Pureza:98%Cor e Forma:SolidPeso molecular:3576.04GLP-1 receptor agonist 13
<p>Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].</p>Fórmula:C25H23ClF2N6OCor e Forma:SolidPeso molecular:496.94JNJ-39933673
CAS:<p>JNJ-39933673 is a bio-active chemical.</p>Fórmula:C48H54F2N2O11Cor e Forma:SolidPeso molecular:872.96Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Fórmula:C21H26Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:433.4PAR-4 Agonist Peptide, amide
CAS:<p>PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).</p>Fórmula:C34H48N8O7Pureza:98%Cor e Forma:SolidPeso molecular:680.79Calcitonin (8-32), salmon
CAS:<p>Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.</p>Fórmula:C119H198N36O37Pureza:98%Cor e Forma:SolidPeso molecular:2725.06(Ala13)-Apelin-13 TFA
<p>'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].'</p>Fórmula:C63H107N23O16S·xC2HF3O2Cor e Forma:SolidPeso molecular:1474.73 (free acid)Colulintide
CAS:<p>Colulintide is an analog of amylin, utilized in obesity research.</p>Cor e Forma:SolidMRS 2365
CAS:<p>Highly potent, selective P2Y1 receptor agonist</p>Fórmula:C13H19N5O9P2SPureza:98%Cor e Forma:SolidPeso molecular:483.33Sarafotoxin S6a
CAS:<p>Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo.</p>Fórmula:C105H156N28O34S5Pureza:98%Cor e Forma:SolidPeso molecular:2514.85Eledoisin Related Peptide
CAS:<p>Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.</p>Fórmula:C34H58N8O6SPureza:98%Cor e Forma:SolidPeso molecular:706.94J-115814
CAS:<p>J-115814 is a potent feeding stimulant.</p>Fórmula:C29H38ClN5O3SCor e Forma:SolidPeso molecular:572.16PF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Fórmula:C36H50Cl2N4O7SPureza:98.81%Cor e Forma:SolidPeso molecular:753.78Hemopressin (human, mouse)
CAS:<p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>Fórmula:C50H79N13O12Pureza:98%Cor e Forma:SolidPeso molecular:1054.26Atrial Natriuretic Peptide (ANP) (1-28), rat
CAS:<p>Atrial Natriuretic Peptide (1-28), rat is the major circulating form of ANP in rats.</p>Fórmula:C128H205N45O39S2Pureza:98%Cor e Forma:SolidPeso molecular:3062.4112-epi Leukotriene B4
CAS:<p>LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.472IRL-1620 acetate
<p>IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a Ki of 16 pM which is more selective than ETA with a Ki of 19 μM.</p>Fórmula:C88H121N17O29Pureza:96.64%Cor e Forma:SolidPeso molecular:1881MCUF-651
CAS:<p>MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.</p>Fórmula:C17H22F2N4OSPureza:99.83%Cor e Forma:SoildPeso molecular:368.44Neuropeptide S(Mouse)
CAS:<p>Endogenous NPSR agonist, EC50 = 3 nM. Boosts Ca2+ levels, activity, wakefulness, reduces anxiety in mice.</p>Fórmula:C93H156N34O27Pureza:98%Cor e Forma:SolidPeso molecular:2182.47Spantide acetate
<p>Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.</p>Fórmula:C77H112N20O15Pureza:98.9200%Cor e Forma:SolidPeso molecular:1557.84PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44MrgprX2 antagonist-2
CAS:<p>MrgprX2 antagonist-2, from patent WO2021092262A1 E163, is potent for skin inflammation studies.</p>Fórmula:C17H16F5N3O3Cor e Forma:SolidPeso molecular:405.32517-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS:<p>17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.</p>Fórmula:C26H37NO4Cor e Forma:SolidPeso molecular:427.585Linzagolix choline
CAS:<p>Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.</p>Fórmula:C27H28F3N3O8SPureza:99.64%Cor e Forma:SolidPeso molecular:611.59
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