GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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Xaliproden hydrochloride
CAS:<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Fórmula:C24H23ClF3NPureza:99.99%Cor e Forma:SolidPeso molecular:417.89Antalarmin
CAS:<p>Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.</p>Fórmula:C24H34N4Cor e Forma:SolidPeso molecular:378.55Diquafosol tetrasodium
CAS:<p>Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear film</p>Fórmula:C18H22N4Na4O23P4Pureza:98.25% - 99.97%Cor e Forma:SolidPeso molecular:878.23H2L 5765834
CAS:<p>H2L 5765834 is a lysophosphatidic acid receptors antagonist</p>Fórmula:C21H12N2O7Pureza:98.25% - 99.47%Cor e Forma:SolidPeso molecular:404.33Bradykinin (2-9)
CAS:<p>Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.</p>Fórmula:C44H61N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:904.02PAR-4 Agonist Peptide, amide TFA
CAS:<p>PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.</p>Fórmula:C36H49F3N8O9Pureza:99.72%Cor e Forma:SolidPeso molecular:794.82Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Cor e Forma:SolidPeso molecular:575.61Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSCor e Forma:SolidPeso molecular:340.48BMS-986020
CAS:BMS-986020 (AM152) is a selective antagonist of LPA1.Fórmula:C29H26N2O5Pureza:98.82% - >99.99%Cor e Forma:SolidPeso molecular:482.53Derenofylline
CAS:<p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>Fórmula:C18H20N4OPureza:98.09%Cor e Forma:SolidPeso molecular:308.384F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Cor e Forma:SolidPeso molecular:429.49Parmodulin 2
CAS:<p>ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).</p>Fórmula:C17H17BrN2O2Pureza:97.35% - 99.95%Cor e Forma:SolidPeso molecular:361.23Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Fórmula:C46H60F3N13O12SPureza:98.49%Cor e Forma:SolidPeso molecular:1076.12Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.41[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Fórmula:C81H113N19O14Pureza:97.68%Cor e Forma:SolidPeso molecular:1576.91Pramlintide acetate(151126-32-8 free base)
CAS:<p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>Fórmula:C173H271N51O55S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:4009Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Fórmula:C15H19NO2Pureza:98.93% - 99.93%Cor e Forma:SolidPeso molecular:245.32Norfluoxetine Hydrochloride
CAS:<p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>Fórmula:C16H17ClF3NOPureza:99.71%Cor e Forma:SolidPeso molecular:331.76RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.Fórmula:C69H105N19O16SPureza:96.84%Cor e Forma:SolidPeso molecular:1488.77Chemerin-9 (149-157) acetate
<p>Chemerin-9 (149-157) acetate, a nonapeptide C-terminal fragment of chemerin, retains full protein's activity as chemerinR agonist.</p>Fórmula:C56H70N10O15Pureza:99.93%Cor e Forma:SolidPeso molecular:1123.23ABT-702 dihydrochloride
CAS:<p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>Fórmula:C22H21BrCl2N6OPureza:98.42% - 98.98%Cor e Forma:SolidPeso molecular:536.25GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Cor e Forma:SolidPeso molecular:415.53Anisotropine Methylbromide
CAS:<p>Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.</p>Fórmula:C17H32BrNO2Pureza:99.73%Cor e Forma:Crystals From Acetone SolidPeso molecular:362.35Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Fórmula:C19H25N5O4·HCl·2H2OPureza:99.81%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:459.92Cinaciguat
CAS:<p>Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.</p>Fórmula:C36H39NO5Pureza:98% - 99.18%Cor e Forma:SolidPeso molecular:565.7Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Fórmula:C19H23NO3·CH4O3SPureza:99.18% - 99.87%Cor e Forma:Tan Or Off-White Cyrstalline SolidPeso molecular:409.5PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:301.21Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Fórmula:C26H31N3O4Pureza:98.13% - 99.66%Cor e Forma:SolidPeso molecular:449.54Cetirizine Impurity B dihydrochloride
CAS:<p>Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.</p>Fórmula:C19H23Cl3N2O2Pureza:99.24%Cor e Forma:SolidPeso molecular:417.76α-MSH, amide Acetate
<p>a-MSH, amide Acetate as an endogenous neuropeptide.</p>Fórmula:C79H113N21O21SPureza:98.67%Cor e Forma:SolidPeso molecular:1724.94Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Fórmula:C40H55N7O11SPureza:99.84% - >99.99%Cor e Forma:White PowderPeso molecular:841.97Relenopride hydrochloride
CAS:<p>Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.</p>Fórmula:C24H31Cl2FN4O4Cor e Forma:SolidPeso molecular:529.43Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Fórmula:C68H87N17O15Pureza:99.98%Cor e Forma:SolidPeso molecular:1382.55Aprocitentan
CAS:<p>Aprocitentan (ACT-132577) is ETA and ETB antagonist .</p>Fórmula:C16H14Br2N6O4SPureza:99.17%Cor e Forma:SolidPeso molecular:546.19S 38093 HCl
CAS:<p>S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.</p>Fórmula:C17H25ClN2O2Pureza:97.91%Cor e Forma:SolidPeso molecular:324.85Bremelanotide Acetate
CAS:<p>Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .</p>Fórmula:C52H72N14O12Pureza:96.72% - >99.99%Cor e Forma:SolidPeso molecular:1085.22Vilazodone Hydrochloride
CAS:<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Fórmula:C26H27N5O2·HClPureza:99.56% - >99.99%Cor e Forma:SolidPeso molecular:477.99BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Fórmula:C34H51N5NaO7Cor e Forma:SolidPeso molecular:664.8ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Fórmula:C16H15N7O2Pureza:97.02% - 99.69%Cor e Forma:SolidPeso molecular:337.34Doxazosin
CAS:<p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>Fórmula:C23H25N5O5Pureza:99.47% - 99.87%Cor e Forma:SolidPeso molecular:451.48Peptide YY (PYY) (3-36), human
CAS:<p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>Fórmula:C176H272N52O54Pureza:97.76%Cor e Forma:SolidPeso molecular:3980.42lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Fórmula:C30H27BrN4O3Pureza:98.12%Cor e Forma:SolidPeso molecular:571.46Pridopidine
CAS:<p>Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.</p>Fórmula:C15H23NO2SPureza:95.2% - 99.89%Cor e Forma:SolidPeso molecular:281.41Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS:<p>Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-</p>Fórmula:C24H35ClO9Pureza:99.88% - 99.94%Cor e Forma:SolidPeso molecular:502.98Naluzotan
CAS:<p>Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>Fórmula:C23H38N4O3SPureza:>99.99%Cor e Forma:SolidPeso molecular:450.64PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47Hydroxyzine dihydrochloride
CAS:<p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>Fórmula:C21H27ClN2O2·2HClPureza:99.46% - 99.79%Cor e Forma:Oil PowderPeso molecular:447.83Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Fórmula:C25H25Cl2N7OPureza:99.43%Cor e Forma:SolidPeso molecular:510.42Antazoline
CAS:<p>Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.</p>Fórmula:C17H19N3Pureza:≥95%Cor e Forma:White Crystalline Powder SolidPeso molecular:265.35Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Fórmula:C18H24ClN3O2Cor e Forma:SolidPeso molecular:349.86VKGILS-NH2 Acetate
<p>VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.</p>Fórmula:C30H58N8O9Pureza:98.83%Cor e Forma:SolidPeso molecular:674.83ELA-11 (human) acetate(1784687-32-6 free base)
<p>ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.</p>Fórmula:C60H94N16O15S2Pureza:99.53%Cor e Forma:SolidPeso molecular:1343.611-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:<p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>Fórmula:C9H15N3OPureza:95%Cor e Forma:SolidPeso molecular:181.23Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Fórmula:C19H16F2N8O2Pureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:426.38Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Fórmula:C21H20O9Pureza:98.90% - 99.21%Cor e Forma:Yellow Brown Fine PowderPeso molecular:416.38SBI-553
CAS:<p>SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).</p>Fórmula:C26H31FN4O2Pureza:99.33%Cor e Forma:SolidPeso molecular:450.55CYM5442
CAS:<p>CYM5442 is an S1P agonist, targeting to Sphingosine.</p>Fórmula:C23H27N3O4Pureza:98.02% - 99.48%Cor e Forma:SolidPeso molecular:409.48Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Fórmula:C21H25ClN2O3·C6H6O3SPureza:99.83% - 99.9%Cor e Forma:Brown Viscous LiquidPeso molecular:547.06Tetradecyl Phosphonate
CAS:<p>Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。</p>Fórmula:C14H31O3PPureza:99.95%Cor e Forma:White To Off-White PowderPeso molecular:278.37Ditolylguanidine
CAS:<p>Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).</p>Fórmula:C15H17N3Pureza:98.42%Cor e Forma:White To Pinkish Solid PowderPeso molecular:239.32Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Fórmula:C21H26ClNPureza:99.99%Cor e Forma:Crystalline SolidPeso molecular:327.90PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Fórmula:C26H32O4Pureza:98.53%Cor e Forma:SolidPeso molecular:408.53S 38093
CAS:<p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>Fórmula:C17H24N2O2Pureza:99.95%Cor e Forma:SolidPeso molecular:288.38MK-0557
CAS:<p>MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).</p>Fórmula:C22H19FN4O3Pureza:99.88%Cor e Forma:SolidPeso molecular:406.41Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Fórmula:C26H29N5O3SPureza:99.49% - 99.843%Cor e Forma:SolidPeso molecular:491.61OXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Fórmula:C79H125N23O22Pureza:98.52%Cor e Forma:SolidPeso molecular:1748.98Lofexidine
CAS:<p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>Fórmula:C11H12Cl2N2OPureza:98.78%Cor e Forma:SolidPeso molecular:259.13Protease-Activated Receptor-2, amide
CAS:<p>Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)</p>Fórmula:C28H54N8O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:614.78Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Fórmula:C17H25N3O2S·HClPureza:99.17% - 99.93%Cor e Forma:Beige SolidPeso molecular:371.93Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Fórmula:C28H33ClN2·2HClPureza:98.05%Cor e Forma:Off-White PowderPeso molecular:505.95SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:319.32Atrasentan
CAS:Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.Fórmula:C29H38N2O6Pureza:97.65% - 99.08%Cor e Forma:SolidPeso molecular:510.62Fenspiride
CAS:<p>Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.</p>Fórmula:C15H20N2O2Cor e Forma:SolidPeso molecular:260.33Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Fórmula:C18H19ClN4OPureza:98.65% - 99.94%Cor e Forma:SolidPeso molecular:342.82SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Cor e Forma:SolidPeso molecular:324.24Ibutamoren Mesylate
CAS:<p>Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.</p>Fórmula:C28H40N4O8S2Pureza:97.98% - ≥98%Cor e Forma:SolidPeso molecular:624.77Talinolol
CAS:(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Fórmula:C20H33N3O3Pureza:98.8%Cor e Forma:SolidPeso molecular:363.49Gadolinium chloride
CAS:<p>Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist</p>Fórmula:Cl3GdPureza:98%Cor e Forma:White Crystalline SolidPeso molecular:263.61LML134
CAS:<p>LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).</p>Fórmula:C19H29N5O3Pureza:99.36%Cor e Forma:SolidPeso molecular:375.47Thonzylamine
CAS:<p>Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.</p>Fórmula:C16H22N4OPureza:99.45%Cor e Forma:SolidPeso molecular:286.37ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Fórmula:C29H29ClN4O2Pureza:99.88%Cor e Forma:SolidPeso molecular:501.02Tavapadon
CAS:<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Fórmula:C19H16F3N3O3Pureza:99.33% - 99.8%Cor e Forma:SolidPeso molecular:391.34Betaxolol
CAS:<p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>Fórmula:C18H29NO3Pureza:99.01%Cor e Forma:White Crystalline SolidPeso molecular:307.43Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Fórmula:C14H22ClNO2Pureza:97.63%Cor e Forma:SolidPeso molecular:271.78Mizagliflozin
CAS:<p>Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.</p>Fórmula:C28H44N4O8Pureza:98.66% - 99.67%Cor e Forma:SolidPeso molecular:564.67GLP-1 receptor agonist 9
CAS:<p>1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.</p>Fórmula:C32H31ClFN3O5Pureza:98%Cor e Forma:SolidPeso molecular:592.06Eformoterol Hemifumarate
CAS:<p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>Fórmula:C19H24N2O4C4H4O4Pureza:99.86% - >99.99%Cor e Forma:White PowderPeso molecular:402.4Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Fórmula:C22H32ClN3O2Cor e Forma:SolidPeso molecular:405.96Medetomidine hydrochloride
CAS:<p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>Fórmula:C13H16N2·HClPureza:99.96%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.74Fluorogestone acetate
CAS:<p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>Fórmula:C23H31FO5Pureza:99.47%Cor e Forma:CoaPeso molecular:406.49Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Fórmula:C32H51F3N8O9Pureza:99.88%Cor e Forma:SolidPeso molecular:748.79RO 46-8443
CAS:<p>RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.</p>Fórmula:C31H35N3O8SPureza:98.77% - 99.77%Cor e Forma:SolidPeso molecular:609.69Rimegepant
CAS:<p>View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.</p>Fórmula:C28H28F2N6O3Pureza:99.1% - 99.99%Cor e Forma:SolidPeso molecular:534.56AdipoRon
CAS:<p>AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: 1.8/3.1 μM).</p>Fórmula:C27H28N2O3Pureza:97.90% - 99.86%Cor e Forma:SolidPeso molecular:428.52YIL781 hydrochloride
CAS:<p>YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).</p>Fórmula:C24H29ClFN3O2Cor e Forma:SolidPeso molecular:445.96RTICBM-189
CAS:<p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>Fórmula:C15H14Cl2N2OPureza:99.96%Cor e Forma:SolidPeso molecular:309.19L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Fórmula:C18H20Cl2N4Pureza:97.36%Cor e Forma:SolidPeso molecular:363.28Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Fórmula:C80H115N21O21Pureza:98% - 99.494%Cor e Forma:SolidPeso molecular:1706.9Naftopidil hydrochloride
CAS:<p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>Fórmula:C24H29ClN2O3Pureza:99.5%Cor e Forma:SolidPeso molecular:428.951-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Fórmula:C6H9N3O2Pureza:99.29%Cor e Forma:SolidPeso molecular:155.15Tripelennamine citrate
CAS:<p>Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.</p>Fórmula:C22H29N3O7Cor e Forma:SolidPeso molecular:447.488Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Fórmula:C21H24Cl2FNO2Cor e Forma:SolidPeso molecular:412.33Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:White SolidPeso molecular:506.47cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Fórmula:C16H14O2Pureza:98.15%Cor e Forma:SolidPeso molecular:238.2812Veralipride
CAS:<p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>Fórmula:C17H25N3O5SPureza:99.65%Cor e Forma:SolidPeso molecular:383.46Canagliflozin
CAS:<p>Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.</p>Fórmula:C24H25FO5SPureza:98.01% - >99.99%Cor e Forma:SolidPeso molecular:444.52Dobutamine
CAS:<p>Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.</p>Fórmula:C18H23NO3Cor e Forma:SolidPeso molecular:301.38AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Fórmula:C20H20N4O4Pureza:99.92%Cor e Forma:SolidPeso molecular:380.4Cinacalcet
CAS:<p>Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .</p>Fórmula:C22H22F3NPureza:99.48%Cor e Forma:Yellow OilPeso molecular:357.41BAR 501 impurity
CAS:<p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>Fórmula:C26H46O3Pureza:98.78%Cor e Forma:SolidPeso molecular:406.64LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Fórmula:C24H27FN2O2·HClPureza:99.8%Cor e Forma:SolidPeso molecular:430.94Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Cor e Forma:White SolidPeso molecular:238.24BD1063 dhydrochloride
CAS:BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).Fórmula:C13H20Cl4N2Pureza:99.52% - ≥95%Cor e Forma:SolidPeso molecular:346.12Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Fórmula:C172H265N43O51Pureza:97.65% - 99.04%Cor e Forma:SolidPeso molecular:3751.25Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Fórmula:C149H234N40O47SPureza:98% - 99.65%Cor e Forma:SolidPeso molecular:3369.76Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Cor e Forma:SolidPeso molecular:336.38SB756050
CAS:<p>SB756050 is a specific TGR5 agonist.</p>Fórmula:C21H28N2O8S2Pureza:98.78% - >99.99%Cor e Forma:SolidPeso molecular:500.59[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Fórmula:C46H62F3N11O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1018.05(S)-Amisulpride
CAS:(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Fórmula:C17H27N3O4SPureza:98.38%Cor e Forma:SolidPeso molecular:369.48Urantide acetate(669089-53-6 free base)
<p>Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in Ca²⁺ assay.</p>Fórmula:C53H70N10O14S2Pureza:99.22%Cor e Forma:SolidPeso molecular:1135.31Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Fórmula:C32H34N4O5SPureza:98.26% - 99.43%Cor e Forma:SolidPeso molecular:586.7Fenoprofen Calcium
CAS:<p>Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.</p>Fórmula:C30H26CaO6Pureza:99.24% - 99.66%Cor e Forma:SolidPeso molecular:522.62-Methoxyidazoxan monohydrochloride
CAS:<p>L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.</p>Fórmula:C12H14N2O3·HClPureza:98.99%Cor e Forma:SolidPeso molecular:270.72AZD1283
CAS:AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).Fórmula:C23H26N4O5SPureza:98.37% - 99.63%Cor e Forma:SolidPeso molecular:470.54Tecadenoson
CAS:<p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>Fórmula:C14H19N5O5Pureza:98.83%Cor e Forma:SolidPeso molecular:337.33IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Fórmula:C23H27N5O2Pureza:97.05%Cor e Forma:SolidPeso molecular:405.49Ralmitaront
CAS:<p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>Fórmula:C17H22N4O2Pureza:99.71% - 99.79%Cor e Forma:SolidPeso molecular:314.38Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Cor e Forma:SolidPeso molecular:438.49[D-Phe12]-Bombesin acetate
<p>[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Fórmula:C76H116N22O20SPureza:99.81%Cor e Forma:SolidPeso molecular:1689.94BQU57
CAS:<p>BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.</p>Fórmula:C16H13F3N4OPureza:97.45% - 98.72%Cor e Forma:SolidPeso molecular:334.3Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Fórmula:C16H19ClN2Cor e Forma:SolidPeso molecular:274.79Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Fórmula:C14H20F6N4O7Pureza:98.18%Cor e Forma:SolidPeso molecular:470.32Talnetant hydrochloride
CAS:<p>Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.</p>Fórmula:C25H23ClN2O2Cor e Forma:SolidPeso molecular:418.92BMY-25368
CAS:<p>BMY-25368 is a long-acting antagonist of the H2-receptor.</p>Fórmula:C19H25N3O3Cor e Forma:SolidPeso molecular:343.42m-Chlorophenylbiguanide hydrochloride
CAS:<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Fórmula:C8H11Cl2N5Pureza:99.43% - 99.87%Cor e Forma:SolidPeso molecular:248.11tcY-NH2 TFA(327177-34-4 free base)
<p>tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.</p>Fórmula:C42H50F3N7O9Pureza:>99.99%Cor e Forma:SolidPeso molecular:853.9PD 117519
CAS:<p>PD 117519 (CI947) is an agonist of adenosine receptor</p>Fórmula:C19H21N5O4Pureza:99.98%Cor e Forma:SolidPeso molecular:383.4Poloxamer 407
CAS:<p>Poloxamer 407 is a nonionic surfactant.</p>Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:7700(Average)Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Fórmula:C22H25ClN2OSPureza:98.9% - 99.82%Cor e Forma:SolidPeso molecular:400.963-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Fórmula:C21H25Cl2NOPureza:99.03%Cor e Forma:SolidPeso molecular:378.33JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Fórmula:C20H32N2OPureza:97.19%Cor e Forma:SolidPeso molecular:316.48Empagliflozin
CAS:<p>Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.</p>Fórmula:C23H27ClO7Pureza:98% - 99.98%Cor e Forma:SolidPeso molecular:450.91Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Fórmula:C23H29Cl2N3O3Cor e Forma:SolidPeso molecular:466.4Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Fórmula:C28H42F2N2O12S2Pureza:99.98%Cor e Forma:SolidPeso molecular:700.77Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Fórmula:C18H19N3O·HClPureza:99.78%Cor e Forma:White PowderPeso molecular:329.82Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Fórmula:C21H25ClN2O3Pureza:99.75%Cor e Forma:SolidPeso molecular:388.89Siponimod hemifumarate
CAS:<p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>Fórmula:C62H74F6N4O10Cor e Forma:SolidPeso molecular:1149.282Fertirelin
CAS:<p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>Fórmula:C55H76N16O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1153.29SKF38393 hydrobromide
CAS:<p>SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;</p>Fórmula:C16H18BrNO2Pureza:98.99%Cor e Forma:SolidPeso molecular:336.22Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:463RO1138452
CAS:<p>RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).</p>Fórmula:C19H23N3OPureza:97.01% - 99.34%Cor e Forma:SolidPeso molecular:309.41Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Fórmula:C23H23ClN2O5SPureza:97.6% - 97.78%Cor e Forma:SolidPeso molecular:474.96BAY 41-8543
CAS:<p>BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).</p>Fórmula:C21H21FN8OPureza:99.86%Cor e Forma:SolidPeso molecular:420.44Icatibant Acetate
CAS:<p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>Fórmula:C61H93N19O15SPureza:99.68%Cor e Forma:SolidPeso molecular:1364.57MK-2894 sodium salt
CAS:MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.Fórmula:C25H22F3NNaO3SPureza:98%Cor e Forma:SolidPeso molecular:496.5Terazosin
CAS:<p>Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43Guanabenz Acetate
CAS:<p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>Fórmula:C8H8Cl2N4·C2H4O2Pureza:99% - 99.66%Cor e Forma:White Solid From Acetonitrile White SolidPeso molecular:291.13Melanotan I
CAS:<p>Melanotan I is a non-specific melanocortin receptor (MCR) agonist, an α-melanocyte-stimulating hormone (α-MSH) analog, which is injected subcutaneously to</p>Fórmula:C78H111N21O19Pureza:>99.99%Cor e Forma:SolidPeso molecular:1646.85Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Fórmula:C25H34FN3O2Pureza:97.84% - 99.69%Cor e Forma:Pale Yellow To Pale Orange SolidPeso molecular:427.55SB-222200
CAS:<p>SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).</p>Fórmula:C26H24N2OPureza:97.13%Cor e Forma:SolidPeso molecular:380.48HS024
CAS:<p>HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.</p>Fórmula:C58H79N19O10S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1266.5M617 acetate
<p>M617 acetate is a selective agonist of galanin receptor 1 (GAL1).</p>Fórmula:C112H161N29O28Pureza:96.02%Cor e Forma:SolidPeso molecular:2361.65Sotagliflozin
CAS:<p>Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potential</p>Fórmula:C21H25ClO5SPureza:99% - 99.86%Cor e Forma:SolidPeso molecular:424.94Cinacalcet hydrochloride
CAS:<p>Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-</p>Fórmula:C22H23ClF3NPureza:99.96% - >99.99%Cor e Forma:Off-White To Tan SolidPeso molecular:393.87AnaMorelin hydrochloride
CAS:<p>AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).</p>Fórmula:C31H43ClN6O3Pureza:99.18% - ≥98%Cor e Forma:SolidPeso molecular:583.16Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Fórmula:C8H12N2Pureza:99.87% - 99.87%Cor e Forma:Yellowish Liquid Liquid LiquidPeso molecular:136.19Octreotide Acetate
CAS:<p>Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.</p>Fórmula:C51H70N10O12S2Pureza:99.03% - 99.87%Cor e Forma:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidPeso molecular:1079.3Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Fórmula:C29H33FN2O4Pureza:98.77% - 99.93%Cor e Forma:SolidPeso molecular:492.58Montelukast dicyclohexylamine
CAS:<p>Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.</p>Fórmula:C47H59ClN2O3SCor e Forma:SolidPeso molecular:767.5Clozapine HCl
CAS:<p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>Fórmula:C18H20Cl2N4Cor e Forma:SolidPeso molecular:363.29ML-191
CAS:<p>ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.</p>Fórmula:C24H25N3O3Pureza:99.58%Cor e Forma:SolidPeso molecular:403.47Hemopressin (human, mouse) acetate
<p>Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.</p>Fórmula:C52H83N13O14Pureza:99.86%Cor e Forma:SolidPeso molecular:1114.29UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Fórmula:C52H68N10O14S2Pureza:99.78%Cor e Forma:SolidPeso molecular:1121.29SKF-83566
CAS:<p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>Fórmula:C17H18BrNOPureza:95.00% - 99.82%Cor e Forma:SolidPeso molecular:332.23Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Fórmula:C12H17NO9Pureza:97.32% - 99.97%Cor e Forma:SolidPeso molecular:319.27Bavisant dihydrochloride hydrate
CAS:Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.Fórmula:C19H31Cl2N3O3Cor e Forma:SolidPeso molecular:420.38Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Fórmula:C18H22ClNOPureza:99.44% - 99.85%Cor e Forma:SolidPeso molecular:303.83Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3Pureza:99.85% - >99.99%Cor e Forma:SolidPeso molecular:387.48d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Fórmula:C52H75N13O13S2Pureza:99.86%Cor e Forma:SolidPeso molecular:1154.37Frovatriptan Succinate
CAS:<p>Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.</p>Fórmula:C18H25N3O6Cor e Forma:SolidPeso molecular:379.41PF-04418948
CAS:<p>PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.</p>Fórmula:C23H20FNO5Pureza:98.67% - 99.45%Cor e Forma:SolidPeso molecular:409.41SLF1081851 TFA
CAS:<p>SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.</p>Fórmula:C23H34F3N3O3Cor e Forma:SolidPeso molecular:457.538Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Fórmula:C37H56F7N6O16PPureza:98% - 99.03%Cor e Forma:SolidPeso molecular:1004.83Bretylium tosylate
CAS:<p>Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.</p>Fórmula:C18H24BrNO3SPureza:>99.99%Cor e Forma:SolidPeso molecular:414.36Ornipressin Acetate(3397-23-7,free)
CAS:<p>Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent.</p>Fórmula:C47H67N13O124S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1102.25Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Fórmula:C15H19Cl2N3O3SPureza:98.48%Cor e Forma:SolidPeso molecular:392.3Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Fórmula:C40H67N7O10Pureza:99.95%Cor e Forma:SolidPeso molecular:805.9Quipazine
CAS:<p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>Fórmula:C13H15N3Cor e Forma:SolidPeso molecular:213.28FSLLRY-NH2 TFA(245329-02-6 free base)
<p>FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.</p>Fórmula:C41H61F3N10O10Pureza:99.32%Cor e Forma:SolidPeso molecular:910.99Brefonalol
CAS:<p>Brefonalol is a vasodilating beta-adrenergic receptor blocker.</p>Fórmula:C22H28N2O2Cor e Forma:SolidPeso molecular:352.47Reboxetine
CAS:<p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>Fórmula:C19H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:313.39Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Cor e Forma:SolidPeso molecular:507.96SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Cor e Forma:SolidPeso molecular:394.85Ambrisentan
CAS:<p>Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.</p>Fórmula:C22H22N2O4Pureza:99.65% - 99.86%Cor e Forma:SolidPeso molecular:378.42Endothelin-2 (49-69), human
CAS:Endothelin-2 (49-69), human (Human endothelin-2) is a 21-amino acid vasoactive peptide that binds to G-protein-linked transmembrane receptors, ET-RA and ET-RB.Fórmula:C115H160N26O32S4Pureza:98.26%Cor e Forma:SolidPeso molecular:2546.92Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Fórmula:C21H28N2O2Pureza:99.53%Cor e Forma:White Or Similar To White PowderPeso molecular:340.46Raclopride tartrate
CAS:<p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>Fórmula:C19H26Cl2N2O9Cor e Forma:SolidPeso molecular:497.32
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