Inhibitor Enzymes
Inhibitor enzymes are molecules that decrease or block the activity of enzymes, preventing them from catalyzing their specific reactions. These inhibitors can be reversible or irreversible and are crucial tools in research and drug development for studying enzyme mechanisms, controlling metabolic pathways, and developing therapeutic agents. Inhibitor enzymes are widely used to modulate biological processes and to treat various diseases by targeting specific enzymes. At CymitQuimica, we offer a comprehensive range of high-quality enzyme inhibitors to support your research and pharmaceutical development needs.
Found 123 products of "Inhibitor Enzymes"
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Nafamostat
CAS:Formula:C19H17N5O2Purity:≥ 98.0%Color and Shape:White to off-white powderMolecular weight:347.37Vildagliptin
CAS:Formula:C17H25N3O2Purity:≥ 98.0%Color and Shape:White to off-white powderMolecular weight:303.40IU1
CAS:Formula:C18H21FN2OPurity:(TLC) ≥ 98%Color and Shape:Off-white to pale brown solidMolecular weight:300.37Fumagillin
CAS:Formula:C26H34O7Purity:≥ 95.0%Color and Shape:White, off-white or pale yellow to tan powderMolecular weight:458.54Lactacystin
CAS:Formula:C15H24N2O7SPurity:≥ 95.0%Color and Shape:White solid or powderMolecular weight:376.43Nα-Tosyl-L-lysine chloromethyl ketone hydrochloride
CAS:Formula:C14H21ClN2O3S·HClPurity:(HPLC) ≥ 98.0%Color and Shape:White powderMolecular weight:369.31Bortezomib
CAS:Formula:C19H25BN4O4Purity:≥ 98.0%Color and Shape:White to off-white powder or solidMolecular weight:384.24E-64 protease inhibitor
CAS:Formula:C15H27N5O5Purity:(HPLC) ≥ 98.0%Color and Shape:White crystalline powderMolecular weight:357.40Bestatin hydrochloride
CAS:Formula:C16H24N2O4·HClPurity:≥ 98.0% (dried basis)Color and Shape:White to almost white powderMolecular weight:344.87Argatroban
CAS:Formula:C23H38N6O6SPurity:(HPLC) ≥ 98%Color and Shape:White to off-white powderMolecular weight:526.65AEBSF hydrochloride
CAS:Formula:C8H10FNO2S·HClPurity:≥ 98.0%Color and Shape:White to off-white powder or solidMolecular weight:239.69N-p-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Formula:C17H18ClNO3SPurity:(TLC) ≥ 98.0%Color and Shape:White to off-white powderMolecular weight:351.85Z-VAD-FMK, cell permeable
CAS:Formula:C22H30FN3O7Purity:≥ 95.0%Color and Shape:White to off-white solidMolecular weight:467.5Elastatinal microbial
CAS:Formula:C21H36N8O7Purity:~0.64μg/ml (IC50, pH8.8, 37°C)Color and Shape:White to light-yellow or tan powderMolecular weight:512.60Pepstatin A
CAS:Formula:C34H63N5O9Purity:≥ 98.0%Color and Shape:White to off-white powderMolecular weight:685.90Suramin sodium salt
CAS:Formula:C51H34N6Na6O23S6Purity:≥ 98%Color and Shape:White to off-white powderMolecular weight:1429.16E-64d protease inhibitor
CAS:Formula:C17H30N2O5Purity:≥ 95.0%Color and Shape:White powderMolecular weight:342.43Carfilzomib
CAS:Formula:C40H57N5O7Purity:(HPLC) ≥ 98.0%Color and Shape:White to off-white crystalline powder or crystalsMolecular weight:719.91Phosphoramidon disodium salt
CAS:Formula:C23H32N3Na2O10PPurity:≥ 97.0%Color and Shape:Colourless, transparent crystals or white to light yellow crystalline powderMolecular weight:587.47Nafamostat mesylate
CAS:Formula:C19H17N5O2Purity:≥ 99.0%Color and Shape:White to off-white or beige crystalline powderMolecular weight:347.37DAPT
CAS:Formula:C23H26F2N2O4Purity:(NMR) ≥ 98.0%Color and Shape:White to off-white solidMolecular weight:432.50Leupeptin hemisulfate
CAS:Formula:C20H38N6O4·5H2SO4Purity:≥ 95%Color and Shape:White to off-white powderMolecular weight:475.59Z-Leu-Leu-Leu-al
CAS:Formula:C26H41N3O5Purity:≥ 97.0%Color and Shape:White to off-white powder or solidMolecular weight:475.63CP-10447
CAS:<p>Applications CP-10447 is an inhibitor apolipoprotein B (apoB) and triglyceride secretion in human hepatoma cells (HepG2) by inhibiting MTP activity and stimulating the early ER degradation of apoB. It is useful tool for further study of the mechanisms of apoB secretion and triglyceride-rich lipoprotein assembly.<br>References Haghpassand, M. et al.: J. Lipid. Res., 37, 1468 (1996); Pan, M. et al.: J. Biol. chem., 275, 27399 (2000);<br></p>Formula:C16H13BrN2OColor and Shape:NeatMolecular weight:329.192-(Hydroxyamino)acetic Acid
CAS:Controlled Product<p>Applications 2-(Hydroxyamino)acetic Acid is a novel lactase inhibitor.<br>References Hattori, M., et al.: J. Insect Physiol., 51, 1359 (2005); Murao, S., et al.: Biosci. Biotech. Biochem., 56, 987 (1992)<br></p>Formula:C2H5NO3Color and Shape:NeatMolecular weight:91.07(3S,4S,3’S)-Ezetimibe
CAS:<p>Applications (3S,4S,3’S)-Ezetimbe is a 3-epimer impurity of Ezetimibe (E975000), a cholesterol absorption inhibitor.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Formula:C24H21F2NO3Color and Shape:Off-WhiteMolecular weight:409.43LCZ696
CAS:<p>Applications LCZ696 is a novel dual-acting inhibitor of angiotensin II receptor and neprilysin, which can be used for blood pressure reduction.<br>References Ruilope, L.M.; et al.: Lancet, 375, 1255 (2010)<br></p>Formula:C24H28NO5·C24H27N5O3·3Na·x(H2O)Color and Shape:MixtureMolecular weight:479.48 + (433.47) + x(18.02)Abamine
CAS:Controlled Product<p>Applications Abamine is an inhibitor of 9-Cis-Epoxycarotenoid dioxygenase (NCED), the key regulatory enzyme in the plant hormone abscisic acid (ABA) biosynthesis pathway.<br>References Kitahata, N., et al.: Bioorg. Med. Chem., 14, 5555 (2006); Han, S., et al.: Bioorg. Med. Chem. Lett., 14, 3033 (2004)<br></p>Formula:C21H24FNO4Color and Shape:NeatMolecular weight:373.423'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt (>90%)
CAS:<p>Stability Hygroscopic<br>Applications 3'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt, is a nucleotide and was proposed to be a possible inhibitor of DNA synthesis.<br>References Frederiksen, Sune.: Biochimica et Biophysica Acta, 76(3), 366-71 (1963)<br></p>Formula:C10H15N5O9P2•xC6H15NPurity:>90%Color and Shape:NeatMolecular weight:411.20 + x(101.19)Teneligliptin Hydrobromide (2:5)
CAS:Controlled Product<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formula:C22H32·5Br2·5N6OSColor and Shape:NeatMolecular weight:628.86Daidzein Diglucuronide
CAS:Controlled ProductFormula:C27H26O16Color and Shape:White To Off-WhiteMolecular weight:606.49(3S,5S)-Atorvastatin Calcium Salt
CAS:Controlled Product<p>Impurity Atorvastatin Related Compound E<br>Applications Impuritiy of Atorvaststin (A791750), a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. Atorvastatin Related Compound E<br>References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),<br></p>Formula:C33H34FN2O5·CaColor and Shape:NeatMolecular weight:1155.34N-(2-Hydroxyethyl)-1-deoxy-L-idonojirimycin Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References van de Water, F., et al.: Drug Metab. Rev., 37, 443 (2005), Koepsell, H., et al.: Pharm. Res., 24, 1227 (2007), Jappar, D., et al.: Pharm. Res., 26, 172 (2009),<br></p>Formula:C8H18ClNO5Color and Shape:NeatMolecular weight:243.69N-(2-Hydroxyethyl)-1-deoxy-L-altronojirimycin Hydrochloride Salt
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formula:C8H18ClNO5Color and Shape:NeatMolecular weight:243.6852Aprotinin Hydrochloride
CAS:<p>Applications Aprotinin is used in cardiac surgery to minimize bleeding and reduce exposure to blood products.<br>References Mangano, D. et al.: New Eng. J. Med., 354, 353 (2006); Fergusson, D. et al.: New. Eng. J. Med., 358, 2319 (2008);<br></p>Formula:C284H432N84O79S7·x(ClH)Color and Shape:White SolidMolecular weight:6511.51(free amine)Nitromifene Citrate (E/Z mixture)
CAS:Controlled Product<p>Applications Nitromifene citrate is a non-steroidal estrogen antagonist. It is structurally similar to Tamoxifen (T006000) which is a selective estrogen response modifier (SERM).<br>References Rudick, C., et al.: Endorcrinol., 144, 179 (2003); Sutherland, R., et al.: Nature, 267, 434 (1977)<br></p>Formula:C33H36N2O11Color and Shape:Yellow To OrangeMolecular weight:636.65Galacto-PUGNAc (>90%)
CAS:Controlled Product<p>Stability Moisture and Temperature Sensitive<br>Applications Galacto-PUGNAc is a highly selective inhibitor for β-hexosaminidases HEXA and HEXB is cell-permeable. Galacto-PUGNAc is able to modulate the activity of HEXA and HEXB in tissue culture, increasing ganglioside GM2 levels in neuroblastoma cells<br>References Stubbs, K.A. et al.: Angew. Chem. Int. Ed., 48, 1300 (2009);<br></p>Formula:C15H19N3O7Purity:>90%Color and Shape:NeatMolecular weight:353.332,5-Dideoxy-2,5-imino-D-mannitol
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A glucosidase inhibitor.<br>References Fellows, L.E.: Pestic. Sci., 17, 602 (1986)<br></p>Formula:C6H13NO4Color and Shape:Off White SolidMolecular weight:163.17Vitamin B12 e-Monocarboxylic Acid
CAS:<p>Stability Hygroscopic<br>Applications Vitamin B12 Monocarboxylic Acid is an impurity of Vitamin B12 (V676005) which is a water-soluble vitamin with a key role in the normal functioning of the brain and nervous system, and for the formation of blood.<br>References Rickes, et al.: Science, 107, 396 (1948); Kirschbaum, J., et al.: Anal. Profiles Drug Subs., 10, 183 (1981); Grasbeck, R., et al.: Clin. Biochem., 17, 99 (1984)<br></p>Formula:C63H87CoN13O15PColor and Shape:Dark Red SolidMolecular weight:1356.35tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate
CAS:Controlled Product<p>Applications tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate is an orally anti-diabetic agent as a inhibitors of dipeptidylpeptidase IV (DPP-4).<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705-5719 (2012);<br></p>Formula:C27H38N6O3SColor and Shape:NeatMolecular weight:526.69
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