Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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4',2-Dihydroxy-4,6-dimethoxydihydrochalcone
CAS:<p>4',2-Dihydroxy-4,6-dimethoxydihydrochalcone, an estrogen-like compound, binds to bovine estrogen receptors, IC50 15 μM.</p>Formula:C17H18O5Color and Shape:SolidMolecular weight:302.32PROTAC AR Degrader-4 TFA
<p>PROTAC AR Degrader-4: IAP ligand, linker, AR binder; it's a SNIPER that degrades AR non-genetically.</p>Formula:C45H68F3N3O11Color and Shape:SolidMolecular weight:884.03PD 132002
CAS:<p>PD 132002 is a renin inhibitor.</p>Formula:C31H50N4O9SColor and Shape:SolidMolecular weight:654.82BAM-22P
CAS:<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Formula:C130H184N38O31S2Purity:98%Color and Shape:SolidMolecular weight:2839.22[Orn8]-Urotensin II acetate
<p>[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.</p>Formula:C65H87N13O20S2Purity:98.63%Color and Shape:SolidMolecular weight:1434.592-Ethylhexyl trans-4-methoxycinnamate
CAS:<p>2-Ethylhexyl trans-4-methoxycinnamate is a sunscreen agent.</p>Formula:C18H26O3Purity:98.92%Color and Shape:Pale Yellow LiquidMolecular weight:290.4OT antagonist 1 demethyl derivative
<p>OT antagonist 1 demethyl derivative is the demethyl derivative of OT antagonist 1. OT antagonist 1 is a selective Oxytocin antagonist (Ki of 50 nM. )</p>Formula:C21H20N4O3Purity:98%Color and Shape:SolidMolecular weight:376.411-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone
CAS:<p>Methyl-2-quinolone from Evodia rutaecarpa blocks angiotensin II receptor with 48.2 μM IC50.</p>Formula:C25H35NOColor and Shape:SolidMolecular weight:365.55Cgp 44099
CAS:<p>Cgp 44099 is a potent plasma renin inhibitor from all subprimate species.</p>Formula:C69H104N14O13Purity:98%Color and Shape:SolidMolecular weight:1337.676Vasopressin Dimer (anti-parallel) (TFA)
<p>Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR,</p>Formula:C94H131F3N30O26S4Purity:98%Color and Shape:SolidMolecular weight:2282.49Biphalin TFA
CAS:<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Formula:C46H56N10O10·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:909.00 (free base)Olmesartan impurity
CAS:<p>Olmesartan impurity, related to parent RNH-6270, is an AT1R antagonist used for hypertension research.</p>Formula:C33H26N4OColor and Shape:SolidMolecular weight:494.598Boc-ypgflt(O-tbu)
CAS:<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Formula:C44H64N6O11Color and Shape:SolidMolecular weight:853.01Frakefamide TFA
<p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>Formula:C32H35F4N5O7Color and Shape:SolidMolecular weight:677.64Diisononyl phthalate
CAS:<p>Diisononyl phthalate (DINP), known as a plasticizer, is a phthalate. DINP is specifically a mixture of various isononyl esters of phthalic acid.</p>Formula:C26H42O4Color and Shape:Colorless Liquid In Water (Uscg 1999)Molecular weight:418.61Prednisolone farnesylate
CAS:<p>Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.</p>Formula:C36H50O6Purity:98%Color and Shape:SolidMolecular weight:578.78[Arg8]-Vasotocin
CAS:<p>[Arg8]-Vasotocin is a hormone present in the neurohypophysis of nonmammalian vertebrates that is related to vasopressin and oxytocin.</p>Formula:C43H67N15O12S2Purity:98%Color and Shape:SolidMolecular weight:1050.22DPC-AJ1951 TFA
<p>DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.</p>Formula:C78H128F3N23O21Color and Shape:SolidMolecular weight:1781.02Raloxifene 6-glucuronide
CAS:<p>Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71Gridegalutamide
CAS:<p>Gridegalutamide exhibits anti-androgen and anti-tumor activities.</p>Formula:C41H45F3N8O5SColor and Shape:SolidMolecular weight:818.9115,26-Dihydroxylanosta-7,9(11),24-trien-3-one
CAS:<p>15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is a natural product that can be used as a reference standard. The CAS number of 15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is 420781-85-7.</p>Formula:C30H46O3Color and Shape:SolidMolecular weight:454.7D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Formula:C25H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:410.98Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formula:C31H41N7O9Purity:98%Color and Shape:SolidMolecular weight:655.709Faznolutamide
CAS:<p>Faznolutamide is an antiandrogen agent [1] [2] .</p>Formula:C19H17FN4O2SColor and Shape:SolidMolecular weight:384.43[Met5]-Enkephalin, amide
CAS:<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Formula:C27H36N6O6SPurity:98%Color and Shape:SolidMolecular weight:572.68PROTAC AR-V7 degrader-1
CAS:<p>Potent, oral AR-V7 degrader (Compound 6); DC50: 0.32µM; targets AR-DBD via VHL E3; EC50: 0.88µM in 22Rv1 cells.</p>Formula:C41H52N6O6S2Color and Shape:SolidMolecular weight:789.02Bufrolin
CAS:<p>Bufrolin is a potent GPR35 agonist, mast cell stabilizer, and anti-inflammatory research agent.</p>Formula:C18H16N2O6Color and Shape:SolidMolecular weight:356.33A 779
CAS:<p>A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.</p>Formula:C39H60N12O11Purity:98%Color and Shape:SolidMolecular weight:872.97Angiotensin II (1-4), human
CAS:<p>Angiotensin II constricts blood vessels and boosts blood pressure by escalating norepinephrine release.</p>Formula:C24H37N7O8Purity:98%Color and Shape:SolidMolecular weight:551.59ICI 174,864
CAS:<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Formula:C38H53N5O7Purity:98%Color and Shape:White SolidMolecular weight:691.87PSDalpha
<p>PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.</p>Formula:C44H39N3O2SColor and Shape:SolidMolecular weight:673.86CP 85339
CAS:<p>CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.</p>Formula:C31H49ClN4O6SColor and Shape:SolidMolecular weight:641.26TF-505
CAS:<p>TF-505, a steroid 5α-reductase inhibitor, is used potentially for the treatment of benign prostatic hyperplasia.</p>Formula:C33H37NO4Purity:98%Color and Shape:SolidMolecular weight:511.65Tetrahydro Aldosterone
CAS:<p>Tetrahydro Aldosterone is a steroidal compound that inhibits the adrenal angiotensin II receptor, with an IC50 of 10 μM.</p>Formula:C21H32O5Color and Shape:SolidMolecular weight:364.48Hemorphin-7
CAS:<p>Hemorphin-7, an atypical opioid peptide from hemoglobin, may enhance memory, promote cell growth, and is a potential breast cancer biomarker.</p>Formula:C49H64N12O11Purity:98%Color and Shape:SolidMolecular weight:997.11difelikefalin acetate(1024828-77-0 Free base)
CAS:<p>is a ketone and a building block.</p>Formula:C38H57N7O8Purity:96.94%Color and Shape:SolidMolecular weight:739.9BI 653048 phosphate
CAS:<p>BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).</p>Formula:C23H28F4N3O8PSPurity:98%Color and Shape:SolidMolecular weight:613.52Estrone-N-O-C1-amido
CAS:<p>Estrone-N-O-C1-amido (ERα ligand 1) is an estrogen ligand derived from Estrone that specifically binds to estrogen receptor α (ERα).</p>Formula:C20H26N2O3Purity:98%Color and Shape:SolidMolecular weight:342.439Glucocorticoids receptor agonist 2
CAS:<p>Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.</p>Formula:C25H25FN2OColor and Shape:SolidMolecular weight:388.48PROTAC ERα Degrader-2
CAS:<p>PROTAC ERα Degrader-2 is composed of a cIAP1 ligand binding group, a linker, and an estrogen receptor α (ERα) binding group, serving as an ERα degrader.</p>Formula:C42H61N5O8Purity:98%Color and Shape:SolidMolecular weight:763.96Deacylcortivazol
CAS:<p>Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.</p>Formula:C30H36N2O4Color and Shape:SolidMolecular weight:488.62Neuropeptide EI, rat
CAS:<p>Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.</p>Formula:C63H98N16O23Purity:98%Color and Shape:SolidMolecular weight:1447.55PROTAC ERRα Degrader-3
CAS:<p>PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein.</p>Formula:C47H50F6N6O7SColor and Shape:SolidMolecular weight:957.0PL-017
CAS:<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Formula:C29H37N5O5Purity:98%Color and Shape:SolidMolecular weight:535.64GNE-502
CAS:<p>GNE-502 is an orally active and potent estrogen receptor (ER) degrader, specifically designed for research on breast cancer.</p>Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59WAY267464 HCl
CAS:<p>WAY267464: nonpeptide OT agonist, anxiolytic, modulates selectivity, improves CNS entry and oral uptake.</p>Formula:C32H37Cl2N7O4Purity:98%Color and Shape:SolidMolecular weight:654.59TD-802
CAS:<p>TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.</p>Formula:C52H61ClN10O6Color and Shape:SolidMolecular weight:957.56Chlorothiazide
CAS:<p>Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.</p>Formula:C7H6ClN3O4S2Purity:98.46% - 98.91%Color and Shape:Crystals Physical Description Crystals; White Powder (Ntp 1992)Molecular weight:295.72Arzoxifene
CAS:<p>Arzoxifene (LY353381), an oral SERM, combats breast cancer, supports bone health, and improves lipids, with few side effects.</p>Formula:C28H29NO4SColor and Shape:SolidMolecular weight:475.6PD 125967
CAS:<p>PD 125967 is a renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>Formula:C51H67N5O4Color and Shape:SolidMolecular weight:814.11Betamethasone acibutate
CAS:<p>Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.</p>Formula:C28H37FO7Purity:98%Color and Shape:SolidMolecular weight:504.59Clocinnamox mesylate
CAS:<p>Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).</p>Formula:C30H33ClN2O7SColor and Shape:SolidMolecular weight:601.11ARD-2585
CAS:<p>ARD-2585 is an orally active and selective androgen receptor PROTAC degrader with anticancer activity for the study of prostate cancer.</p>Formula:C41H43ClN8O5Color and Shape:SolidMolecular weight:763.28PROTAC ERα Y537S degrader-1
CAS:<p>PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group.</p>Formula:C46H49N5O6Color and Shape:SolidMolecular weight:767.91Raloxifene 4'-glucuronide
CAS:<p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71Osteostatin
CAS:<p>Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presenting</p>Formula:C27H41N9O8Color and Shape:SolidMolecular weight:619.67Vasopressin Dimer (parallel) (TFA)
<p>Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, and</p>Formula:C94H131F3N30O26S4Purity:98%Color and Shape:SolidMolecular weight:2282.49Dynorphin A (1-10)
CAS:<p>Dynorphin A (1-10) is an opioid peptide, binds κ-opioid receptor, blocks NMDA current, IC50: 42.0 μM.</p>Formula:C57H91N19O12Purity:98%Color and Shape:SolidMolecular weight:1234.457α-(Thiomethyl)spironolactone
CAS:<p>7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.</p>Formula:C23H32O3SPurity:>99.99%Color and Shape:SolidMolecular weight:388.56Dexamethasone cipecilate
CAS:<p>Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.</p>Formula:C33H43FO7Purity:98%Color and Shape:SolidMolecular weight:570.69Teriparatide
CAS:<p>Teriparatide is an agonist of PHT(IC50 of 2 nM in HEK293 cells).</p>Formula:C181H291N55O51S2Purity:98%Color and Shape:SolidMolecular weight:4117.72[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formula:C63H103FN22O17Purity:98.03%Color and Shape:SolidMolecular weight:1459.63ODM-204
CAS:<p>ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).</p>Formula:C20H21F3N4Purity:98%Color and Shape:SolidMolecular weight:374.40Melanin Concentrating Hormone, salmon
CAS:<p>Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>Formula:C89H139N27O24S4Purity:98%Color and Shape:White PowderMolecular weight:2099.48MT-7716 hydrochloride
CAS:<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Formula:C27H29ClN4O2Purity:98%Color and Shape:SolidMolecular weight:477Azilsartan Medoxomil Potassium
CAS:<p>Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.</p>Formula:C30H23N4O8·KPurity:98.72%Color and Shape:SolidMolecular weight:606.62Myrciacetin
CAS:<p>Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.</p>Formula:C17H16O6Color and Shape:SolidMolecular weight:316.309Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formula:C49H75N15O14Purity:98%Color and Shape:SolidMolecular weight:1098.2PROTAC ER Degrader-4
CAS:<p>PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).</p>Formula:C53H67F3N6O8SPurity:98%Color and Shape:SolidMolecular weight:1005.2NPFF1-R antagonist 1
<p>NPFF1-R antagonist 1 (compound 8b) is a piperidine analog and an effective neuropeptide FF (NPFF) receptor antagonist. It exhibits 15-fold selectivity for the NPFF1-R subtype, with Ki values of 211 nM and 3270 nM for NPFF1-R and NPFF2-R, respectively.</p>Formula:C37H44N4OMolecular weight:560.35151Epi-Cryptoacetalide
<p>Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.</p>Formula:C18H22O3Color and Shape:SolidMolecular weight:286.371ERRγ agonist-2
CAS:<p>ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a K d value of 6.5 μM.</p>Formula:C27H21N5O2Color and Shape:SolidMolecular weight:447.49(S,S)-J-113397
CAS:<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.57PIPE-3297
<p>PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.</p>Formula:C23H30N2OMolecular weight:350.23581Nurr1 agonist 9
<p>Nurr1 agonist 9 (Compound 36) acts as an agonist for Nurr1, with an EC50 of 0.090 µM and a Kd of 0.17 µM. It activates Nurr1 homodimers (NurRE, EC50 = 0.094 µM) and Nurr1-RXR heterodimers (DR5, EC50 = 0.165 µM). This compound induces the expression of Nurr1-regulated tyrosine hydroxylase (TH) in Parkinson's disease organoid models and can penetrate the human brain endothelial cell barrier.</p>Formula:C21H19ClN4O2Molecular weight:394.11965BigLEN(mouse)
CAS:<p>GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.</p>Formula:C78H130N24O22Purity:98%Color and Shape:SolidMolecular weight:1756.03NR-V04
CAS:<p>NR-V04 is a PROTAC degrader targeting NR4A1.</p>Formula:C62H87N5O11SColor and Shape:SolidMolecular weight:1110.45Antidiabetic agent 15
<p>Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.</p>Formula:C26H23NO5Color and Shape:SolidMolecular weight:429.15762THR-β agonist 8
CAS:<p>THR-β agonist 8 (Compound 1) is an orally active agonist for both TRα and TRβ. It holds potential for research into thyroid hormone-related diseases.</p>Formula:C19H12Cl2N4O4Color and Shape:SolidMolecular weight:431.23ER degrader 4
CAS:<p>ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].</p>Formula:C26H19FO4SColor and Shape:SolidMolecular weight:446.49Nurr1 agonist 12
<p>Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.</p>Formula:C18H12ClN3OColor and Shape:SolidMolecular weight:321.7611-Ketodihydrotestosterone
CAS:<p>11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).</p>Formula:C19H28O3Color and Shape:SolidMolecular weight:304.42L 363564
CAS:<p>L 363564 is a kidney renin inhibitor.</p>Formula:C54H76N12O10Color and Shape:SolidMolecular weight:1053.276Handle region peptide, rat
CAS:<p>Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.</p>Formula:C54H101N15O12SPurity:98%Color and Shape:SolidMolecular weight:1184.54LY301875
CAS:<p>LY301875 is an antagonist of nonpeptide angiotensin receptor.</p>Formula:C31H36N4O10SColor and Shape:SolidMolecular weight:656.70Koreanoside E
CAS:<p>Koreanoside E is a useful organic compound for research related to life sciences. The catalog number is T125538 and the CAS number is 1804014-67-2.</p>Formula:C27H30O11Color and Shape:SolidMolecular weight:530.526Prednicarbate
CAS:<p>Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.</p>Formula:C27H36O8Purity:99.88%Color and Shape:SolidMolecular weight:488.57(rel)-PROTAC ERRα Degrader-1
<p>(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader.</p>Formula:C54H49Cl2F6N7O8Purity:98%Color and Shape:SolidMolecular weight:1108.91GPR88 agonist 2
<p>GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].</p>Color and Shape:Odour SolidPROTAC ER Degrader-14
CAS:<p>PROTAC ER Degrader-14 (compound 86) is a PROTAC-type estrogen receptor/ERR degrader. It comprises an E3 ubiquitin ligase ligand (blue part) (S)-Deoxy-thalidomide, a PROTAC linker (black part) N-Boc-piperazine, and a target protein ligand (red part) ER ligand-6. The combination of the E3 ligase and linker forms tert-Butyl (S)-4-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)piperazine-1-carboxylate.</p>Formula:C44H46FN5O5Color and Shape:SolidMolecular weight:743.865CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formula:C34H35N5O4Color and Shape:SolidMolecular weight:577.67Bexirestrant
CAS:<p>Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.</p>Formula:C29H26F3NO2Color and Shape:SolidMolecular weight:477.527SNIPER(ER)-87
CAS:<p>SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (</p>Formula:C59H73N5O10SPurity:98%Color and Shape:SolidMolecular weight:1044.32KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Formula:C38H38N2O5Color and Shape:SolidMolecular weight:602.72Ganoderic acid Df
CAS:<p>Ganoderic acid Df, a lanostane triterpenoid from Ganoderma lucidum, inhibits aldose reductase with IC50 of 22.8 μM.</p>Formula:C30H44O7Color and Shape:SolidMolecular weight:516.67AM-5262
CAS:<p>AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.</p>Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63ZINC05925939
<p>ZINC05925939 is an estrogen receptor β (ESR2) inhibitor used in breast cancer research.</p>Formula:C17H17NO2Color and Shape:SolidMolecular weight:267.32RLA-4842
<p>RLA-4842: iron-based anti-androgen; inhibits mCRPC cell proliferation.</p>Formula:C42H46F3N5O8SColor and Shape:SolidMolecular weight:837.9PROTAC ER Degrader-15
<p>PROTAC ER Degrader-15 (Compound 40) is an orally active estrogen receptor (ER) degrader with anticancer properties, suitable for breast cancer research.</p>Formula:C47H47F4N5O5Color and Shape:SolidMolecular weight:837.9β-Endorphin, equine
CAS:<p>Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.</p>Formula:C154H248N42O44SPurity:98%Color and Shape:SolidMolecular weight:3423.94
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