Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(207 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(296 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3178 products of "Endocrinology/Hormones"
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VPC-3033
CAS:<p>VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.</p>Formula:C21H14O2Purity:98%Color and Shape:SolidMolecular weight:298.33Dup 747
CAS:<p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>Formula:C24H28Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:447.4Carbazole derivative 1
CAS:<p>Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.</p>Formula:C18H13FN2Purity:98%Color and Shape:SolidMolecular weight:276.31TUG-424
CAS:<p>TUG-424 boosts insulin secretion, is a selective FFAR1 agonist with an EC50 of 32 nM.</p>Formula:C18H16O2Purity:98.94%Color and Shape:SolidMolecular weight:264.32Fenhexamid
CAS:<p>Fenhexamid (Elevate), a sterol biosynthesis inhibitor, shows antifungal activity against the plant pathogenic fungus.</p>Formula:C14H17Cl2NO2Purity:99.56%Color and Shape:SolidMolecular weight:302.20CPSA
CAS:<p>CPSA is an effective and selective AKR1C1 inhibitor.</p>Formula:C13H9ClO3Color and Shape:SolidMolecular weight:248.66SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Formula:C25H37FN4Purity:98%Color and Shape:SolidMolecular weight:412.59ALR1/2-IN-1
CAS:<p>ALR1/2-IN-1 (Compound 6e) is an aldehyde reductase (ALR1) (IC50: 3.26 μM) and aldose reductase (ALR2) (IC50: 3.06 μM) inhibitor with anticancer effects.</p>Formula:C18H18N4O5S2Color and Shape:SolidMolecular weight:434.49ES 6864
CAS:<p>ES 6864 is an orally active inhibitor of renin.</p>Formula:C42H58N6O7SColor and Shape:SolidMolecular weight:791.01CFMB
CAS:<p>CFMB is the FFA2 receptor agonist.</p>Formula:C21H21ClN2OSPurity:98%Color and Shape:SolidMolecular weight:384.92L162441
CAS:<p>L162441 is an antagonist of Angiotensin type 1 receptor.</p>Formula:C34H43N5O5SPurity:98%Color and Shape:SolidMolecular weight:633.8WAY-267464
CAS:<p>oxytocin receptor (OTR) agonist</p>Formula:C32H35N7O4Purity:98%Color and Shape:SolidMolecular weight:581.66NGD-4715
CAS:<p>NGD-4715 is a selective and orally active antagonist of melanin-concentrating hormone receptor 1.</p>Formula:C19H24BrN3O3Purity:98%Color and Shape:SolidMolecular weight:422.32TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Formula:C37H38N4O6Purity:98%Color and Shape:SolidMolecular weight:634.72Milfasartan
CAS:<p>Milfasartan: Potent AT1 antagonist, oral, effectively reduces blood pressure in hypertensive rats.</p>Formula:C30H30N6O3SColor and Shape:SolidMolecular weight:554.66RU 25055
CAS:<p>RU 25055 is a synthetic antiglucocorticoid.</p>Formula:C24H26O2SPurity:98%Color and Shape:SolidMolecular weight:378.53Ralaniten
CAS:<p>Ralaniten (EPI-002), a potent AR-NTD antagonist, inhibits AR with IC50 of 7.4 μM, for CRPC study.</p>Formula:C21H27ClO5Purity:99.77%Color and Shape:SolidMolecular weight:394.89AS-1669058 oxalate
CAS:<p>AS-1669058 is a G-protein-coupled receptor 119 (GPR119) agonist for the treatment of type 2 diabetes mellitus.</p>Formula:C20H17BrF2N4O5Color and Shape:SolidMolecular weight:511.27SC 46944
CAS:<p>SC 46944 is a highly potent human renin inhibitor.</p>Formula:C34H55N3O7Color and Shape:SolidMolecular weight:617.82Honokiol DCA
CAS:<p>Honokiol DCA inhibits DRP1, enhances respiration via mitochondrial repair, and is active against Vemurafenib-resistant melanoma.</p>Formula:C22H18Cl4O4Color and Shape:SolidMolecular weight:488.19AL 4114
CAS:<p>AL 4114 is used as an aldose reductase inhibitor.</p>Formula:C17H12F2N2O4Purity:98%Color and Shape:SolidMolecular weight:346.29DK1
CAS:<p>DK1: potent ERRα modulator, lowers blood glucose, promising for diabetes research.</p>Formula:C16H13ClN2O2Color and Shape:SolidMolecular weight:300.74Isoflupredone
CAS:<p>Isoflupredone, a synthetic corticosteroid, inhibits inflammation and immune response in animals.</p>Formula:C21H27FO5Purity:97.62% - 99.85%Color and Shape:SolidMolecular weight:378.43LY191704
CAS:<p>LY 191704 is a 5α-reductase type 1 inhibitor.</p>Formula:C14H16ClNOColor and Shape:SolidMolecular weight:249.74NXT629
CAS:<p>NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.</p>Formula:C35H39N5O3SPurity:99.07% - 99.07%Color and Shape:SolidMolecular weight:609.78GSK9027
CAS:<p>GSK9027, a nonsteroidal GR agonist, is a partial 2×GRE reporter gene activator, less potent than dexamethasone.</p>Formula:C27H19F4N3O2SPurity:99.36%Color and Shape:SolidMolecular weight:525.526-Raloxifene-β-D-glucopyranoside
CAS:<p>6-Raloxifene-β-D-glucopyranoside is a benzothiophene glucuronidated at the 6' position.</p>Formula:C34H37NO9SPurity:98%Color and Shape:SolidMolecular weight:635.72LGD-2226
CAS:<p>LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.</p>Formula:C14H9F9N2OPurity:98%Color and Shape:SolidMolecular weight:392.22SC 51316
CAS:<p>SC 51316 is a nonpeptidic angiotensin II (AII) receptor antagonist.</p>Formula:C24H29N7OColor and Shape:SolidMolecular weight:431.53Estrogen receptor-IN-1
CAS:<p>Estrogen receptor-IN-1 (compound 16) is an effective estrogen receptor (ER) inhibitor with IC 50 s of 13, 5μM for ERα and Erβ, respectively [1].</p>Formula:C14H16OSiColor and Shape:SolidMolecular weight:228.365-bromo-3-phenyl Salicylic Acid
CAS:<p>AKR1C1 inhibitor</p>Formula:C13H9BrO3Purity:98%Color and Shape:SolidMolecular weight:293.11Pipendoxifene hydrochloride
CAS:<p>Pipendoxifene hydrochloride is a selective modulator of estrogen receptor.</p>Formula:C29H33ClN2O3Purity:99.56%Color and Shape:SolidMolecular weight:493.04Erteberel
CAS:<p>Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.</p>Formula:C18H18O3Purity:99.46%Color and Shape:SolidMolecular weight:282.33Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Formula:C36H42N6O7Color and Shape:SolidMolecular weight:670.75GPR40 agonist 1
CAS:<p>GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40).</p>Formula:C27H30FN3O4Purity:98%Color and Shape:SolidMolecular weight:479.54Bromopropylate
CAS:<p>Bromopropylate is an insecticide. Bromopropylate is the active substance in fumigant strips for mites.</p>Formula:C17H16Br2O3Purity:98%Color and Shape:White Crystalline Solid Yellowish CrystalsMolecular weight:428.11CR-665 Acetate
CAS:<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Formula:C38H53N9O6Color and Shape:SolidMolecular weight:731.899Paramethasone Acetate
CAS:<p>Paramethasone Acetate is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive effects that can be used in the treatment of systemic lupus</p>Formula:C24H31FO6Purity:98.1%Color and Shape:SolidMolecular weight:434.50BMS-819881
CAS:<p>BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for</p>Formula:C24H21ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:468.95TRβ agonist 2
CAS:<p>TRβ agonist 2 (Compound 1) is a highly potent agonist of TRβ.</p>Formula:C22H27NO4Color and Shape:SolidMolecular weight:369.45Androgen receptor antagonist 3
CAS:<p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84KB-141
CAS:<p>KB-141 is an agonist of thyroid hormone receptor.</p>Formula:C17H16Cl2O4Purity:98%Color and Shape:SolidMolecular weight:355.21L-366509
CAS:<p>L-366,509 is an antagonist of oxytocin.</p>Formula:C25H33NO5SPurity:98%Color and Shape:SolidMolecular weight:459.6RU 43044
CAS:<p>RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.</p>Formula:C29H34O2Purity:98%Color and Shape:SolidMolecular weight:414.58DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Formula:C20H20N2Purity:98%Color and Shape:SolidMolecular weight:288.39KB-130015
CAS:<p>KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.</p>Formula:C18H14I2O4Purity:98%Color and Shape:SolidMolecular weight:548.1127-Hydroxycholesterol
CAS:<p>27-Hydroxycholesterol (25(R)-27-hydroxy Cholesterol) is a selective modulator of estrogen receptor and an agonist of the liver X receptor.</p>Formula:C27H46O2Purity:99.45% - 99.82%Color and Shape:SolidMolecular weight:402.65(Rac)-Acolbifene
CAS:<p>(Rac)-Acolbifene (EM-343) is the racemic form of Acolbifene.</p>Formula:C29H31NO4Purity:99.7%Color and Shape:SolidMolecular weight:457.56AM-4668
CAS:<p>AM-4668, a GPR40 (FFA1) agonist with oral availability, was optimized to reduce central nervous system (CNS) permeability, and reduced blood glucose level.</p>Formula:C24H19F3N2O4SPurity:99.32% - 99.92%Color and Shape:SolidMolecular weight:488.48JHU-083
CAS:<p>JHU-083 is a glutaminase antagonist that improves cognition and normalizes aberrant hippocampal glutaminase activity in APOE4 mice.</p>Formula:C14H24N4O4Purity:97.89% - 99.53%Color and Shape:SolidMolecular weight:312.37MK-4541
CAS:<p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>Formula:C22H31F3N2O3Color and Shape:SolidMolecular weight:428.49GSK 1562590 hydrochloride
CAS:<p>urotensin II (UT) receptor antagonist</p>Formula:C30H31Cl3N4O4Purity:98%Color and Shape:SolidMolecular weight:617.95BTI-A-404
CAS:<p>BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43.</p>Formula:C22H26N4O2Color and Shape:SolidMolecular weight:378.47D36
CAS:<p>D36 is an androgen receptor allosteric antagonist. It also has inverse agonist properties.</p>Formula:C21H24N2O2Purity:98%Color and Shape:SolidMolecular weight:336.43VPC-13789
CAS:<p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>Formula:C21H16F3N3OColor and Shape:SolidMolecular weight:383.37Glutaurine aceate
<p>Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid.</p>Formula:C9H18N2O8SPurity:98%Color and Shape:SoildMolecular weight:314.31OT antagonist 1
CAS:<p>OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)</p>Formula:C22H22N4O3Purity:98%Color and Shape:SolidMolecular weight:390.44L 366682
CAS:<p>L 366682 is an oxytocin antagonist.</p>Formula:C40H53N9O6Purity:98%Color and Shape:SolidMolecular weight:755.91NCG21
CAS:<p>NCG21, a GPR120 agonist, boosts ERK, Ca²⁺ responses, and GLP-1 in GPR120-expressing cells; raises GLP-1 in mice.</p>Formula:C23H24N2O3Purity:98%Color and Shape:SolidMolecular weight:376.45MCH-1 antagonist 1
CAS:<p>MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).</p>Formula:C25H26N4O2Purity:98%Color and Shape:SolidMolecular weight:414.5Fidarestat
CAS:<p>Fidarestat (SNK 860),Aldose reductase inhibitor (IC50=26 nM). Targets AKR1B10 (33 μM) and V301L AKR1B10 (1.8 μM). Potential diabetes treatment.</p>Formula:C12H10FN3O4Purity:98%Color and Shape:SolidMolecular weight:279.22ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49Dimethomorph
CAS:<p>Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .</p>Formula:C21H22ClNO4Purity:99.2%Color and Shape:Solid CrystallineMolecular weight:387.86EM-800
CAS:<p>EM-800, an ERα ligand & prodrug of EM-652, inhibits E1-stimulated ZR-75-1 tumor growth in mice.</p>Formula:C39H47NO6Color and Shape:SolidMolecular weight:625.79PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Formula:C21H29ClN2O2SPurity:99.59%Color and Shape:SolidMolecular weight:408.99Androgen receptor antagonist 1
CAS:<p>Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.</p>Formula:C21H25ClN4O3Purity:99.054%Color and Shape:SolidMolecular weight:416.9Capesaris
CAS:<p>Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.</p>Formula:C19H13F2NO3Purity:99.65%Color and Shape:SolidMolecular weight:341.31(R)-Bicalutamide
CAS:<p>(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.</p>Formula:C18H14F4N2O4SColor and Shape:SolidMolecular weight:430.37Norethisterone enanthate
CAS:<p>Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.</p>Formula:C27H38O3Purity:99.23%Color and Shape:SolidMolecular weight:410.59SHR1653
CAS:<p>SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).</p>Formula:C21H21ClFN5O2Purity:98%Color and Shape:SolidMolecular weight:429.88(±)-AC 7954 hydrochloride
CAS:<p>(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.</p>Formula:C19H21Cl2NO2Purity:99.42%Color and Shape:White SolidMolecular weight:366.28Diallyl G
CAS:<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Formula:C38H53N5O8Color and Shape:SolidMolecular weight:707.86BMS 183920
CAS:<p>BMS 183920 is a potent Angiotensin II Receptor antagonist that improves improves Caco-2 cell permeability in vivo.</p>Formula:C26H19N5O3Purity:98.92%Color and Shape:SolidMolecular weight:449.46A 81282
CAS:<p>A 81282 is a selective antagonist of angiotensin receptors. It has the activity of lowering blood pressure.</p>Formula:C23H23N7O2Purity:98%Color and Shape:SolidMolecular weight:429.47AR antagonist 5
CAS:<p>Compound 30a, known as AR Antagonist 5, is a selective androgen receptor (AR) antagonist that demonstrates an IC 50 value of 134.8 nM. It exhibits favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure [1].</p>Formula:C23H21F3N6O2Color and Shape:SolidMolecular weight:470.45OBHS
CAS:<p>OBHS is an inhibitor of estrogen receptor alpha (ERα).</p>Formula:C24H20O6SColor and Shape:SolidMolecular weight:436.48OT antagonist 3
CAS:<p>OT antagonist 3 is an antagonist of oxytocin (OT).</p>Formula:C21H20N6O2Purity:98%Color and Shape:SolidMolecular weight:388.42OP-1074
CAS:<p>OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.</p>Formula:C29H31NO4Purity:98%Color and Shape:SolidMolecular weight:457.56D-Methionine sulfoxide
CAS:<p>D-Methionine sulfoxide inhibits peptide methionine sulfoxide reductase and can be used to inhibit ochre mites.D-Methionine sulfoxide can be added to chicken</p>Formula:C5H11NO3SPurity:99.54%Color and Shape:SolidMolecular weight:165.21SB 611812
CAS:<p>SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.</p>Formula:C17H16Cl3F3N2O3SPurity:99.34%Color and Shape:SolidMolecular weight:491.74LY117018
CAS:<p>LY117018 shows antiproliferative effects on breast cancer cell lines. LY117018 is a Raloxifene analog and is a selective estrogen receptor modulator.</p>Formula:C27H25NO4SPurity:98%Color and Shape:SolidMolecular weight:459.56MK-3984
CAS:<p>MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.</p>Formula:C17H12F7NO2Purity:99.91%Color and Shape:SolidMolecular weight:395.27Pratosartan
CAS:<p>Pratosartan is a selective antagonist of angiotensin II receptor.</p>Formula:C25H26N6OPurity:98%Color and Shape:SolidMolecular weight:426.51TUG-905
CAS:<p>TUG-905 is an agonist for free fatty acid receptor 4 (FFA4/GPR120), and TUG-905 has the potential to treat agitation.</p>Formula:C27H30FNO5SColor and Shape:SolidMolecular weight:499.59MK181
CAS:<p>MK181 is an inhibitor of AKR1B10, a tumor marker and promising antineoplastic target.</p>Formula:C16H13BrClNO4Purity:98%Color and Shape:SolidMolecular weight:398.64Methylprednisolone Aceponate
CAS:<p>Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.</p>Formula:C27H36O7Purity:99.00% - 99.61%Color and Shape:SolidMolecular weight:472.57DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Formula:C22H24Cl3N3OSPurity:98%Color and Shape:SolidMolecular weight:484.87FFA3 agonist 1
CAS:<p>FFA3 Agonist 1, a potent agonist of the free fatty acid receptor 3 (FFA3), plays a crucial role in mediating the health-promoting effects of the intestinal</p>Formula:C22H22N2O3Color and Shape:SolidMolecular weight:362.42Dehydro Olmesartan
CAS:<p>Dehydro Olmesartan, from Olmesartan, is an AT1R blocker for researching hypertension.</p>Formula:C24H24N6O2Color and Shape:SolidMolecular weight:428.49Dunnione
CAS:<p>Dunnione is an antifungal agent exerting its action primarily through initiation of redox cycling.</p>Formula:C15H14O3Color and Shape:SolidMolecular weight:242.27LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7Idoxifene
CAS:<p>Idoxifene is a tissue-specific selective estrogen receptor modulator.</p>Formula:C28H30INOColor and Shape:SolidMolecular weight:523.45Aldose reductase-IN-3
CAS:<p>Aldose reductase-IN-3 (Compound 5) is a moderately selective AR inhibitor with IC50 of 3.99 μM, potential for sepsis research.</p>Formula:C18H12ClN3O2S2Color and Shape:SolidMolecular weight:401.89Cyprodinil
CAS:<p>Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.</p>Formula:C14H15N3Color and Shape:SolidMolecular weight:225.29Aldose reductase-IN-4
CAS:<p>Aldose reductase-IN-4 (compund IIc) is an inhibitor of aldose reductase with IC50s of 11.70 μM and 0.98 μM for ALR1 and ALR2, respectively [1].</p>Formula:C14H10FNO3SColor and Shape:SolidMolecular weight:291.3Aldose reductase-IN-6
CAS:<p>AR inhibitor Aldose reductase-IN-6: IC50 3.164 μM, Ki 0.018 μM, non-toxic to normal cells.</p>Formula:C20H16N4O2SColor and Shape:SolidMolecular weight:376.43BHPI
CAS:<p>BHPI is a potent ERα inhibitor, activating UPR and blocking protein synthesis with an IC50 value. It depletes EnR Ca(2+) via PLCγ in ERα(+) cancer cells.</p>Formula:C21H17NO3Color and Shape:SolidMolecular weight:331.36Olmesartan methyl ester
CAS:<p>Olmesartan methyl ester: an intermediate for synthesizing Olmesartan medoxomil, a strong AT1 receptor blocker.</p>Formula:C25H28N6O3Color and Shape:SolidMolecular weight:460.53SIM-688
CAS:<p>SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).</p>Formula:C34H31F3N2O2Purity:99.56%Color and Shape:SolidMolecular weight:556.62ORL1 antagonist 1
CAS:<p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>Formula:C20H22ClN5Purity:98.92%Color and Shape:SolidMolecular weight:367.88Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38Zuclomiphene citrate
CAS:<p>Zuclomiphene citrate, a cis isomer of Clomiphene, has stronger antiestrogenic effects and better inhibits LH secretion.</p>Formula:C32H36ClNO8Purity:98%Color and Shape:SolidMolecular weight:598.08Estrogen receptor β antagonist 2
CAS:<p>Estrogen receptor β antagonist 2 is a selective, potent estrogen receptor β (ERβ) antagonist that acts on Erα (IC50: 109.10 μM) and Erβ (IC50: 0.63 μM).</p>Formula:C23H26N2O6Color and Shape:SolidMolecular weight:426.46Anordiol
CAS:<p>Anordiol is an antiestrogen with estrogenic activity. It also is known to inhibit fertility.</p>Formula:C22H30O2Purity:98%Color and Shape:SolidMolecular weight:326.47(R)-DPN
CAS:<p>estrogen receptor (ER) β agonist</p>Formula:C15H13NO2Purity:98%Color and Shape:SolidMolecular weight:239.27RU 28318, potassium salt
CAS:<p>mineralocorticoid receptor (MR) antagonist</p>Formula:C25H38KO4Purity:98%Color and Shape:SolidMolecular weight:441.67JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Formula:C26H25N3O2Purity:98%Color and Shape:SolidMolecular weight:411.5Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94Lubabegron fumarate
CAS:<p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66GSK706
CAS:<p>GSK706 is a novel effective agonist of the GPR119.</p>Formula:C23H29N5O4SPurity:98%Color and Shape:SolidMolecular weight:471.57GPR35 agonist 3
CAS:<p>GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.</p>Formula:C12H9NO5SPurity:98.80%Color and Shape:SolidMolecular weight:279.27L 156373
CAS:<p>L 156373 is an oxytocin antagonist.</p>Formula:C40H54N8O7Purity:98%Color and Shape:SolidMolecular weight:758.91LY88074 Trimethyl ether
CAS:<p>LY88074 Trimethyl ether inhibits conditions like osteoporosis and hyperlipidemia caused by low estrogen.</p>Formula:C24H20O4SPurity:98%Color and Shape:SolidMolecular weight:404.48FK-739 free acid
CAS:<p>FK-739, an angiotensin II receptor blocker, inhibits rat aorta binding (IC50=8.6 nM) but not bovine cerebellum.</p>Formula:C24H23N7Purity:98%Color and Shape:SolidMolecular weight:409.49CAY10595
CAS:<p>CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.</p>Formula:C20H13Cl2FN2O5Purity:99.95% - 99.97%Color and Shape:SolidMolecular weight:451.23Aldose reductase-IN-2
CAS:<p>Aldose reductase-IN-2 (5f) inhibits AR with antioxidant effects; potential anti-diabetic drug.</p>Formula:C25H28N4O5Color and Shape:SolidMolecular weight:464.51Ici 174865
CAS:<p>Ici 174865 is a delta opioid receptor antagonist agent.</p>Formula:C38H53N5O7Color and Shape:SolidMolecular weight:691.86LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Formula:C28H41N5O4Color and Shape:SolidMolecular weight:511.66CRTh2 antagonist 1
CAS:<p>CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).</p>Formula:C23H25N3O5SPurity:97.24%Color and Shape:SolidMolecular weight:455.53Pivalopril
CAS:<p>Pivalopril is a new orally active inhibitor of angiotensin-converting enzyme.</p>Formula:C16H27NO4SPurity:98%Color and Shape:SolidMolecular weight:329.45HG122
CAS:<p>HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.</p>Formula:C15H13N5O5Color and Shape:SolidMolecular weight:343.29FR 62765
CAS:<p>FR 62765 is a derivative of WF-3681, an aldose reductase inhibitor.</p>Formula:C16H18O5Color and Shape:SolidMolecular weight:290.31D 15413
CAS:<p>D 15413 is an inhibitor of estrogen-dependent mammary tumors.</p>Formula:C16H12Cl3NO2Purity:98%Color and Shape:SolidMolecular weight:356.63LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Formula:C24H22F2N2O2Purity:99.18%Color and Shape:SolidMolecular weight:408.44TUG-469
CAS:<p>TUG-469 is an agonist of free fatty acid 1(FFA) receptor.</p>Formula:C23H23NO2Purity:99.73%Color and Shape:SolidMolecular weight:345.43BMS-564929
CAS:<p>BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.</p>Formula:C14H12ClN3O3Purity:98.17%Color and Shape:SolidMolecular weight:305.72Omapatrilat
CAS:<p>Omapatrilat is a metalloprotease ACE and NEP dual inhibitor (Ki: 0.64 and 0.45 nM, respectively).</p>Formula:C19H24N2O4S2Purity:98%Color and Shape:SolidMolecular weight:408.53Desketoraloxifene
CAS:<p>Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).</p>Formula:C27H27NO3SPurity:98%Color and Shape:SolidMolecular weight:445.57Org-34517
CAS:<p>Org-34517, a glucocorticoid receptor (GR) antagonist, is used potentially for the treatment of depression.</p>Formula:C28H30O4Purity:98%Color and Shape:SolidMolecular weight:430.54GW7604
CAS:<p>GW7604 is an antiestrogen and it also is the metabolite of GW5638. GW5638 is an antagonist of high-affinity estrogen receptor (ER).</p>Formula:C25H22O3Purity:98%Color and Shape:SolidMolecular weight:370.44ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Formula:C34H46N4O6SPurity:98%Color and Shape:SolidMolecular weight:638.82Prednisolone Tebutate
CAS:<p>Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.</p>Formula:C27H38O6Purity:98%Color and Shape:SolidMolecular weight:458.59Renin inhibitor-1
CAS:<p>Renin inhibitor-1 (compound 26) is a potent, orally active renin inhibitor capable of acting on rh-renin (IC50: 0.9 nM) and hPRA (IC50: 1.8 nM). renal disease.</p>Formula:C22H30N4O4Color and Shape:SolidMolecular weight:414.5Fispemifene
CAS:<p>Fispemifene (HM-101) is an estrogen receptor modulator (SERM) used to treat genitourinary syndromes and vaginal atrophy.</p>Formula:C26H27ClO3Purity:98.74% - 99.67%Color and Shape:SolidMolecular weight:422.94Etacstil
CAS:<p>GW5638, a prodrug of GW7604, is a unique estrogen receptor antagonist & a pseudo-SERD with potential in breast cancer therapy.</p>Formula:C25H22O2Color and Shape:SolidMolecular weight:354.449L-159282
CAS:<p>L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.</p>Formula:C30H28N4O3SPurity:98%Color and Shape:SolidMolecular weight:524.63(S)-Baxdrostat
CAS:<p>(S)-Baxdrostat is an S-enantiomer of Baxdrostat, which functions as an inhibitor of aldosterone synthase [1].</p>Formula:C22H25N3O2Color and Shape:SolidMolecular weight:363.45Bopindolol fumarate
CAS:<p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>Formula:C27H32N2O7Color and Shape:SolidMolecular weight:496.56SB-436811
CAS:<p>SB-436811 is an antagonist of human urotensin-II receptor.</p>Formula:C23H29Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:450.4(1R,2R)-2-PCCA hydrochloride
CAS:<p>(1R,2R)-2-PCCA HCl: Potent, selective GPR88 agonist, crosses BBB, EC50 1140 nM in mouse striatum. Useful for CNS research.</p>Formula:C30H39Cl2N3OPurity:98.75% - 99.67%Color and Shape:SolidMolecular weight:528.56L 364918
CAS:<p>L 364918 is an oxytocin antagonist.</p>Formula:C40H54N8O6Purity:98%Color and Shape:SolidMolecular weight:742.91Rentiapril
CAS:<p>Rentiapril is an orally active inhibitor of angiotensin converting enzyme (ACE), with antihypertensive activity.</p>Formula:C13H15NO4S2Purity:98%Color and Shape:SolidMolecular weight:313.39(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Formula:C13H20ClNO3Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:273.76AZ12216052
CAS:<p>AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to study obesity and metabolic disorders.</p>Formula:C19H22BrNOSPurity:99.29%Color and Shape:SolidMolecular weight:392.35PF-3882845
CAS:<p>PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).</p>Formula:C24H22ClN3O2Purity:99.63%Color and Shape:SolidMolecular weight:419.9AZD2906
CAS:<p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>Formula:C26H25FN4O3Color and Shape:SolidMolecular weight:460.5Zenarestat
CAS:<p>Zenarestat is an orally active aldose reductase inhibitor capable of ameliorating diabetic peripheral neuropathy in rats with type 2 diabetes.</p>Formula:C17H11BrClFN2O4Purity:99.51% - 99.51%Color and Shape:SolidMolecular weight:441.64Iodothiouracil
CAS:<p>Iodothiouracil is a uracil derivative. It was used as a thyroid antagonist.</p>Formula:C4H3IN2OSPurity:98%Color and Shape:SolidMolecular weight:254.05NNC45-0781
CAS:<p>NNC45-0781 is a tissue-selective partial-agonist of estrogen.</p>Formula:C27H29NO3Purity:98%Color and Shape:SolidMolecular weight:415.52AT2R antagonist 1
CAS:<p>AT2R antagonist 1: potent, selective ligand, Ki 29 nM, inhibits CYP enzymes, stable in liver microsomes.</p>Formula:C23H30N4O4S2Color and Shape:SolidMolecular weight:490.64Fludrocortisone
CAS:<p>Fludrocortisone （Florinef） is a synthetic corticosteroid with moderate glucocorticoid potency and greater mineralocorticoid potency.Cost-effective and quality-assured.</p>Formula:C21H29FO5Purity:98.56% - 98.66%Color and Shape:White SolidMolecular weight:380.45Alrestatin Sodium
CAS:<p>Alrestatin is a specific inhibitor of the aldose reductase enzyme.</p>Formula:C14H9NNaO4Purity:98%Color and Shape:SolidMolecular weight:278.219μ opioid receptor agonist 2
CAS:<p>μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>Formula:C25H34N4OColor and Shape:SolidMolecular weight:406.56Ono-3805 sodium
CAS:<p>Ono-3805 is an inhibitor of nonsteroidal 5 alpha-reductase.</p>Formula:C31H37NNaO5Purity:98%Color and Shape:SolidMolecular weight:526.629LG-121071
CAS:<p>LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.</p>Formula:C15H15F3N2OPurity:98%Color and Shape:SolidMolecular weight:296.29ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Formula:C25H29BrF3N5OColor and Shape:SolidMolecular weight:552.43AS1907417
CAS:<p>AS1907417 is a GPR119 agonist.</p>Formula:C19H27N3O4SColor and Shape:SolidMolecular weight:393.5ALR2-IN-3
<p>ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.</p>Formula:C17H12N2O3S2Color and Shape:SolidMolecular weight:356.42EMD 66684
CAS:<p>angiotensin AT1 receptor antagonist</p>Formula:C28H31ClN8O2Purity:98%Color and Shape:SolidMolecular weight:547.06TCS 3035
CAS:<p>GPR35 agonist 4 (compound 10), pEC50 5.86, potent in human/rat but inactive with R3.36 mutation.</p>Formula:C12H9NO5SColor and Shape:SolidMolecular weight:279.27Liothyronine HCl
CAS:<p>Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.</p>Formula:C15H13ClI3NO4Purity:98%Color and Shape:SolidMolecular weight:687.43Androgen receptor antagonist 4
CAS:<p>Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84RU 752
CAS:<p>RU 752 is an antagonist of mineralocorticoid receptor that inhibits aldosterone synthesis.</p>Formula:C22H30O4Purity:98%Color and Shape:SolidMolecular weight:358.47TFM-4AS-1
CAS:<p>androgen receptor modulator</p>Formula:C27H33F3N2O2Purity:98%Color and Shape:SolidMolecular weight:474.56Tolonidine
CAS:<p>Tolonidine is orally active and has been shown to possess hypotensive. Tolonidine is a derivative of imidazoline.</p>Formula:C10H12ClN3Purity:98%Color and Shape:SolidMolecular weight:209.68FFA1 agonist-1
CAS:<p>FFA1 agonist-1 (Compound 17a) is an orally active fatty acid receptor (FFA1) agonist (EC50: 0.75 μM).</p>Formula:C27H36ClNO3Color and Shape:SolidMolecular weight:458.04GPR4 antagonist 1
CAS:<p>GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).</p>Formula:C27H37N5Purity:98%Color and Shape:SolidMolecular weight:431.62GPR81 agonist 1
CAS:<p>GPR81 agonist 1 is a GPR81 agonist that improves glycaemic control in insulin-resistant mouse models for the study of diabetes and obesity.</p>Formula:C22H30N4O2S2Purity:99.68%Color and Shape:SolidMolecular weight:446.63Chlorothiazide Sodium
CAS:<p>diuretic and antihypertensive</p>Formula:C7H6ClN3NaO4S2Purity:98%Color and Shape:SolidMolecular weight:318.71Tranilast Sodium
CAS:<p>Tranilast Sodium has been used for the treatment of bronchial asthma. Tranilast is also used to autoimmune diseases, atopic and fibrotic pat.</p>Formula:C18H17NNaO5Purity:98%Color and Shape:SolidMolecular weight:350.32ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Formula:C19H14Cl2N4OSColor and Shape:SolidMolecular weight:417.31Estrogen receptor antagonist 2
CAS:<p>ER antagonist 2 selectively suppresses ERα, a key breast cancer driver, with research potential in the disease.</p>Formula:C26H31F4N5Color and Shape:SolidMolecular weight:489.55Xelaglifam
CAS:<p>Xelaglifam is a potent agonist of G protein-coupled receptor 40 (GPR40) and exhibits hypoglycemic effects.</p>Formula:C30H28FNO5Color and Shape:SolidMolecular weight:501.55GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Formula:C24H20F2N4Purity:99.85%Color and Shape:SolidMolecular weight:402.44SQ 30774
CAS:<p>SQ 30774 is a representative of the imidazole alcohols-a novel class of renin inhibitors.</p>Formula:C32H45N7O5Purity:98%Color and Shape:SolidMolecular weight:607.74GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9TAK-875 Hemihydrate
CAS:<p>TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.</p>Formula:C29H32O7SH2OPurity:98%Color and Shape:SolidMolecular weight:533.63RU 45144
CAS:<p>RU 45144 is an estradiol derivative with antiestrogenic activity.</p>Formula:C28H37NO3Purity:98%Color and Shape:SolidMolecular weight:435.6AC-7954
CAS:<p>AC-7954 is a potent and efficacious agonist of urotensin II receptor.</p>Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82GPR40 Activator 1
CAS:GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes.Formula:C31H31NO3SPurity:98%Color and Shape:SolidMolecular weight:497.65GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43Org30958
CAS:<p>Org30958 is a potent inhibitor of aromatase in vivo.</p>Formula:C21H30O2S2Purity:98%Color and Shape:SolidMolecular weight:378.59Estrogen receptor antagonist 1
CAS:<p>"Potent estrogen receptor blocker with promise for breast cancer treatment per WO2021249533A1."</p>Formula:C28H33F4N5Color and Shape:SolidMolecular weight:515.59AMG-076
CAS:<p>AMG-076 is an antagonist of melanin-concentrating hormone receptor 1. It also reduced hERG inhibition.</p>Formula:C32H39F3N2O5SPurity:98%Color and Shape:SolidMolecular weight:620.72LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41GSK1104252A
CAS:<p>GSK1104252A is a potent and selective agonist of GPR119.</p>Formula:C22H27FN4O5SPurity:98%Color and Shape:SolidMolecular weight:478.54DS20362725
CAS:<p>DS20362725 is a selective estrogen-related receptor alpha (ERRα) agonist, commonly used in the study of metabolic disorders.</p>Formula:C19H22N2O2Purity:99.34%Color and Shape:SolidMolecular weight:310.39Gumelutamide
CAS:<p>Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.</p>Formula:C22H21ClN6OColor and Shape:SolidMolecular weight:420.89AZD7268
CAS:<p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64J 628
CAS:<p>J 628 is a synthetic "impeded" estrogen derivative. It also has some postcoital antifertility activity.</p>Formula:C23H31NO4SColor and Shape:SolidMolecular weight:417.56Aldose reductase-IN-5
CAS:<p>Aldose reductase-IN-5 inhibits ALR2, boosts inhibitory response and antioxidants, slowing diabetes complications.</p>Formula:C18H15NO5Color and Shape:SolidMolecular weight:325.32ALR2-IN-2
<p>ALR2-IN-2 inhibits ALR2 (27 nM IC50) & ALR1 (228 nM IC50), used in diabetes complication research.</p>Formula:C17H11FN2O2S2Color and Shape:SolidMolecular weight:358.41AT1R antagonist 1
CAS:<p>AT1R Antagonist 1 (compound 10) serves as a potent, selective ligand for AT1R with considerable affinity, demonstrated by a K i value of 8.5 nM [1].</p>Formula:C28H32F3N5O4S2Color and Shape:SolidMolecular weight:623.71Paraprost
CAS:<p>Paraprost consists of 1-glutamic acid, alanine, and glycine. It was used in prostate hypertrophy drug therapy.</p>Formula:C10H21N3O8Purity:98%Color and Shape:SolidMolecular weight:311.291Glucocorticoid receptor-IN-2
CAS:<p>Glucocorticoid receptor-IN-2 selectively targets GR with anti-inflammatory effects (IC50: 0.171 nM) and activates MMTV (EC50: 0.94 nM).</p>Formula:C25H20F4N6O2Color and Shape:SolidMolecular weight:512.46AT-076
CAS:<p>AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.</p>Formula:C26H35N3O3Color and Shape:SolidMolecular weight:437.57Levormeloxifene
CAS:<p>Levormeloxifene is a selective modulator of the estrogen receptor. It inhibits the production of vaginal tropoelastin and transforming growth factor-beta 1.</p>Formula:C30H35NO3Purity:98%Color and Shape:SolidMolecular weight:457.6Nitromifene
CAS:<p>Nitromifene is the estrogen receptor antagonist.</p>Formula:C27H28N2O4Purity:98%Color and Shape:SolidMolecular weight:444.52VPC-14449
CAS:<p>VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.</p>Formula:C10H10Br2N4OSPurity:99.56%Color and Shape:SolidMolecular weight:394.09DK3
CAS:<p>DK3 is a potent and selective agonist of estrogen-related receptor alpha (ERRα). ERRα is a potential drug target for cancer and metabolic diseases [1].</p>Formula:C16H14N2O2Color and Shape:SolidMolecular weight:266.29
