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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • HENA

    CAS:
    <p>HENA is a novel activator of large conductance, voltage- and Ca2+-gated K+ (BK) channels.</p>
    Formula:C30H48NaO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.701
  • Lanceotoxin A

    CAS:
    <p>Lanceotoxin A is a potent Ip blocker.</p>
    Formula:C32H44O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:620.68
  • Dopropidil hydrochloride

    CAS:
    <p>Dopropidil, a calcium channel antagonist, is used potentially for the treatment of arrhymia and angina pectoris.</p>
    Formula:C20H36ClNO2
    Color and Shape:Solid
    Molecular weight:357.96
  • SCH00013

    CAS:
    <p>SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.</p>
    Formula:C18H20N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.38
  • GZ4

    CAS:
    <p>GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.</p>
    Formula:C11H17NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:195.26
  • AFD-21

    CAS:
    <p>AFD-21 is a class I antiarrhythmic that inhibits sodium channels with moderate kinetics.</p>
    Formula:C28H39NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.61
  • Hexadecylphosphoserine

    CAS:
    <p>Hexadecylphosphoserine is a representative growth inhibitor.</p>
    Formula:C19H40NO6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.5
  • Metaphit

    CAS:
    <p>Acylator of PCP and σ-receptors</p>
    Formula:C18H24N2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:300.46
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Formula:C10H12ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:213.66
  • AMG7905

    CAS:
    AMG7905 is a modulator of transient receptor potential vanilloid type 1.
    Formula:C25H24F3N5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:483.55
  • Ro18-5362

    CAS:
    <p>Ro18-5362 is the less active prodrug of Ro 18-5364.</p>
    Formula:C22H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.52
  • Ceefourin-2

    CAS:
    <p>Ceefourin-2 is a highly selective multidrug resistance protein 4 inhibitor.</p>
    Formula:C15H9ClF3N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.7
  • BDF 9148

    CAS:
    BDF 9148, a Na(+)-channel modulator, increases the contractile force of guinea-pig atria and papillary muscles.
    Formula:C28H27N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.53
  • EO-122

    CAS:
    <p>EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.</p>
    Formula:C16H23ClN2O
    Color and Shape:Solid
    Molecular weight:294.82
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Formula:C24H24ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.91
  • Levamlodipine gentisate

    CAS:
    <p>Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.</p>
    Formula:C27H31ClN2O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:563
  • JTT-552

    CAS:
    <p>JTT-552, a uric acid transporter 1 (URAT1) inhibitor, is used potentially for the treatment of hyperuricemia.</p>
    Formula:C15H12ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:289.71
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17
  • TAS-4

    CAS:
    <p>TAS-4 is a modulator of metabotropic glutamate receptor 4-positive allosteric.</p>
    Formula:C12H8Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.11
  • Hydroflumethiazide

    CAS:
    <p>Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.</p>
    Formula:C8H8F3N3O4S2
    Color and Shape:Crystals Solid
    Molecular weight:331.29
  • Lombazole

    CAS:
    <p>Lombazole is an antimicrobial agent in the class of imidazole.</p>
    Formula:C22H17ClN2
    Color and Shape:Solid
    Molecular weight:344.84
  • Aladorian

    CAS:
    <p>Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.</p>
    Formula:C12H13NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.3
  • Arginylproline

    CAS:
    <p>Arginylproline is a dipeptide composed of arginine and proline. It is an incomplete breakdown product of protein digestion or protein catabolism.</p>
    Formula:C11H21N5O3
    Color and Shape:Solid
    Molecular weight:271.32
  • Ro 8-4304

    CAS:
    Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM
    Formula:C21H23FN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.42
  • CS476

    CAS:
    <p>CS476 is a potent drug of hypoglycaemic.</p>
    Formula:C24H29N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.57
  • Fluzinamide

    CAS:
    <p>Fluzinamide (AHR-8559) has anticonvulsant effects on ignited amygdala seizures.</p>
    Formula:C12H13F3N2O2
    Purity:99.38% - >99.99%
    Color and Shape:Solid
    Molecular weight:274.24
  • Laurinterol

    CAS:
    <p>Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.</p>
    Formula:C15H19BrO
    Color and Shape:Solid
    Molecular weight:295.21
  • BRL 55834

    CAS:
    <p>BRL 55834, a potassium channel activator, has shown to relax airways and vasculature in vivo.</p>
    Formula:C18H20F5NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.35
  • S-312-d

    CAS:
    <p>S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.</p>
    Formula:C20H22N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.46
  • Niguldipine Free Base

    CAS:
    <p>Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.</p>
    Formula:C36H39N3O6
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:609.71
  • CGP 28392

    CAS:
    <p>CGP 28392 is used as a partial calcium channel agonist.</p>
    Formula:C18H17F2NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:365.33
  • RH01617

    CAS:
    <p>RH01617 possesses potent inhibitory activities against Kv1.5.</p>
    Formula:C22H26N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.52
  • Glypromate

    CAS:
    <p>Glypromate (Gly-Pro-Glu) is a neuroprotective agent, is a weak NMDA receptor agonist</p>
    Formula:C12H19N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.3
  • SR57227A

    CAS:
    <p>SR 57227A: Selective 5-HT3 receptor inhibitor, affects NMDA responses, has anti-depressant effects and reduces aggression in rats.</p>
    Formula:C10H14ClN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.69
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Formula:C18H23ClN6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.87
  • Guanosine 5'-diphosphate ditromethamine

    CAS:
    Guanosine 5'-diphosphate ditromethamine (GDP ditromethamine) is a nucleoside diphosphate that activates ATP-sensitive K+ channels. It acts as a potential iron mobilizer, inhibiting the interaction between hepcidin and ferroportin, and modulating the IL-6/STAT-3 pathway. This compound finds application in inflammation research, such as studying anemia of inflammation (AI).
    Formula:C18H37N7O17P2
    Molecular weight:685.47
  • GSK1702934A

    CAS:
    GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in the study of diabetes mellitus.
    Formula:C22H25N3O2S
    Purity:98.15%
    Color and Shape:Solid
    Molecular weight:395.52
  • N-Oleoyl Valine

    CAS:
    N-Oleoyl valine, an N-acyl amine, antagonizes TRPV3 for thermoregulation; rises post-cold exposure; elevates in mouse lung injury.
    Formula:C23H43NO3
    Molecular weight:381.59
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Formula:C15H23N5O2S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:337.44
  • SM-6586

    CAS:
    SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular
    Formula:C26H27N5O5
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:489.52
  • (5R)-BW-4030W92

    CAS:
    <p>(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.</p>
    Formula:C11H9Cl2FN4
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:287.12
  • MDL-29951

    CAS:
    MDL-29951 is a novel glycine antagonist of NMDA receptor activation.
    Formula:C12H9Cl2NO4
    Purity:98.79% - 99.49%
    Color and Shape:Solid
    Molecular weight:302.11
  • YM-900

    CAS:
    YM-900, an AMPA receptor antagonist and glutamate receptor antagonist, is used potentially for the treatment of stroke.
    Formula:C11H7N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.2
  • AM12

    CAS:
    AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).
    Formula:C15H9BrO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.13
  • ML402

    CAS:
    <p>ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM.</p>
    Formula:C14H14ClNO2S
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:295.78
  • Zatebradine hydrochloride

    CAS:
    <p>Zatebradine hydrochloride (UL-FS-49CL) inhibits HCN channels (IC50: ~1.9 µM) blocking human HCN1-4 currents effectively.</p>
    Formula:C26H37ClN2O5
    Purity:97%
    Color and Shape:Solid
    Molecular weight:493.04
  • Cyclic ADP-ribose

    CAS:
    <p>cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.</p>
    Formula:C15H21N5O13P2
    Purity:98%
    Color and Shape:Lyophilized Powder
    Molecular weight:541.3
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Formula:C17H20N2O3
    Purity:99.62%
    Color and Shape:Solid Crystalline
    Molecular weight:300.35
  • BMS-919373

    CAS:
    <p>BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.</p>
    Formula:C25H20N6O2S
    Purity:98.51% - 99.01%
    Color and Shape:Solid
    Molecular weight:468.53
  • McN5691

    CAS:
    McN5691 is a voltage sensitive calcium channel blocker.
    Formula:C30H35NO3
    Purity:98.93% - 99.38%
    Color and Shape:Solid
    Molecular weight:457.6
  • Levosemotiadil

    CAS:
    <p>Levosemotiadil(SA 3212) is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to prevent</p>
    Formula:C29H32N2O6S
    Purity:98.53% - 99.47%
    Color and Shape:Solid
    Molecular weight:536.64
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Formula:C10H13Cl2NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:250.12
  • Vernakalant

    CAS:
    <p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>
    Formula:C20H31NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.46
  • Amsacrine

    CAS:
    <p>Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.</p>
    Formula:C21H19N3O3S
    Purity:99.2%
    Color and Shape:Yellow Crystalline Powder Solid
    Molecular weight:393.46
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Formula:C8H15NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:173.21
  • Phenamil

    CAS:
    <p>Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.</p>
    Formula:C12H12ClN7O
    Purity:99.07%
    Color and Shape:Solid
    Molecular weight:305.72
  • B-TPMF

    CAS:
    <p>B-TPMF is a highly efficient and selective KCa2.1 channel inhibitor with an IC50 of 31 nM, interacting with serine residue at position 293 to inhibit KCa2.1.</p>
    Formula:C19H24N6O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:368.43
  • CM-TPMF

    CAS:
    <p>CM-TPMF is a highly efficient and potent activator of the K(Ca)2.1 channel, Ser293 in the transmembrane segment 5, neurological disorders.</p>
    Formula:C16H17ClN6O2
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:360.8
  • TTA-Q6

    CAS:
    <p>TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.</p>
    Formula:C20H15ClF3N3O
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:405.8
  • 18:0 LYSO-PE

    CAS:
    <p>18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.</p>
    Formula:C23H48NO7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.6
  • ABCG2-IN-1

    CAS:
    <p>ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with an inhibitory concentration (IC50) of 0.13 μM.</p>
    Formula:C26H36N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.59
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Formula:C9H8F4N2O2S
    Purity:98.22% - 98.54%
    Color and Shape:Solid
    Molecular weight:284.23
  • TWIK-1/TREK-1-IN-2

    CAS:
    <p>TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 values</p>
    Formula:C20H29F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.45
  • ABCG2-IN-2

    CAS:
    <p>ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrug</p>
    Formula:C25H34N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.56
  • U-89843A

    CAS:
    <p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>
    Formula:C16H24ClN5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.85
  • TWIK-1/TREK-1-IN-1

    CAS:
    <p>Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and</p>
    Formula:C21H24F3NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.42
  • D-3263 hydrochloride

    CAS:
    <p>D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 (TRPM8) agonist.</p>
    Formula:C21H32ClN3O3
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:409.95
  • Vernakalant Hydrochloride

    CAS:
    <p>Vernakalant Hydrochloride (RSD1235 hydrochloride) is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel blocker.</p>
    Formula:C20H32ClNO4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:385.93
  • YHO-13351 free base

    CAS:
    <p>YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .</p>
    Formula:C26H33N3O4S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:483.62
  • Pinacidil

    CAS:
    <p>Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and</p>
    Formula:C13H19N5
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:245.32
  • TRPV4 agonist-1

    CAS:
    TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).
    Formula:C25H23ClF2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:484.93
  • PF 05089771 tosylate

    CAS:
    <p>PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x affinity for half-inactivated state.</p>
    Formula:C18H12Cl2FN5O3S2·C7H8O3S
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:672.56
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Formula:C3H9FNO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:141.08
  • UK 78282 hydrochloride

    CAS:
    UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T cell activation.
    Formula:C29H36ClNO2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:466.05
  • Puliginurad

    CAS:
    <p>Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad is used in the treatment of gout.</p>
    Formula:C19H16N2O2S
    Purity:99.96% - 99.96%
    Color and Shape:Solid
    Molecular weight:336.41
  • GX-674

    CAS:
    <p>GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an IC50 value of 0.1 nM measured at -40 mV for the study of</p>
    Formula:C21H13ClF2N6O3S2
    Purity:98.60%
    Color and Shape:Solid
    Molecular weight:534.95
  • TRAM 39

    CAS:
    <p>TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.</p>
    Formula:C20H14ClN
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:303.78
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Formula:C16H25ClN4O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:340.85
  • TRPM4-IN-2

    CAS:
    NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.
    Formula:C19H14ClNO4
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:355.77
  • RO 4938581

    CAS:
    RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).
    Formula:C13H8BrF2N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.14
  • JYL 1421

    CAS:
    <p>JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).</p>
    Formula:C20H26FN3O2S2
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:423.57
  • GDC-0276

    CAS:
    <p>GDC-0276 is an orally active, selective, and potent NaV1.7 inhibitor that can be used for the study of pain-related diseases.</p>
    Formula:C24H31FN2O4S
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:462.58
  • RY796

    CAS:
    <p>RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.</p>
    Formula:C21H27N3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:353.46
  • RN9893

    CAS:
    RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.
    Formula:C21H23F3N4O5S
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:500.49
  • ATX-II TFA


    <p>ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).</p>
    Purity:98%
    Color and Shape:Odour Solid
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Formula:C19H29NO5
    Purity:98.19% - 99.55%
    Color and Shape:Solid
    Molecular weight:351.44
  • E 0747

    CAS:
    <p>E 0747 is an antiarrhythmic agent of class 1C type. E-0747 suppresses arrhythmia by inhibiting the Na channels of cardiac cells.</p>
    Formula:C21H28ClN3O4
    Purity:95.17%
    Color and Shape:Solid
    Molecular weight:421.92
  • TRPV3 antagonist 74a

    CAS:
    <p>TRPV3 antagonist 74a (TRPV3 74a) is a specific TRPV3 antagonist for the study of neurological disorders.</p>
    Formula:C17H17F3N2O2
    Purity:≥98.0%
    Color and Shape:Solid
    Molecular weight:338.32
  • AVE1231

    CAS:
    AVE1231 is a TASK-1 channel blocker that inhibits TASK-1 and can be used in the study of atrial fibrillation.
    Formula:C20H27N3O4S
    Purity:98.03%
    Color and Shape:Solid
    Molecular weight:405.51
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Formula:C9H13ClNO3P
    Purity:99.32%
    Color and Shape:White Solid
    Molecular weight:249.63
  • GAL-021 sulfate

    CAS:
    GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.
    Formula:C11H24N6O5S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:352.41
  • Istaroxime hydrochloride

    CAS:
    <p>Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.</p>
    Formula:C21H33ClN2O3
    Color and Shape:Solid
    Molecular weight:396.95
  • GX-585

    CAS:
    <p>GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.</p>
    Formula:C24H25Cl2FN4O3S
    Purity:99.02% - 99.03%
    Color and Shape:Solid
    Molecular weight:539.45
  • SRI-37240

    CAS:
    SRI-37240 suppresses CFTR nonsense mutations, aids in fixing premature termination codons, works with G418.
    Formula:C24H23N3O2
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:385.46
  • AGN-201904

    CAS:
    AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.
    Formula:C25H25N3O8S2
    Purity:97.32%
    Color and Shape:Solid
    Molecular weight:559.61
  • Ani9

    CAS:
    <p>Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating cancer, hypertension, pain, diarrhea, asthma.</p>
    Formula:C17H17ClN2O3
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:332.78
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Formula:C20H20ClN5O3S2
    Purity:99.21% - 99.73%
    Color and Shape:Solid
    Molecular weight:477.99
  • S 18986

    CAS:
    <p>S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, showcasing cognitive-enhancing properties in</p>
    Formula:C10H12N2O2S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:224.28
  • Quinabactin

    CAS:
    <p>Quinabactin (LC-66C6): ABA agonist, induces guard cell closure, reduces water loss, hinders germination, boosts drought resistance in Arabidopsis/soybean.</p>
    Formula:C20H24N2O3S
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:372.48
  • AV-101

    CAS:
    <p>AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with antidepressant activity that reduces dyskinesia.</p>
    Formula:C10H11ClN2O3
    Purity:97.78% - 98.27%
    Color and Shape:Solid
    Molecular weight:242.66