Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(336 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2290 products of "Membrane Transporter/Ion Channel"
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KT-362 fumarate
CAS:<p>KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes rabbit arterial strips.</p>Formula:C26H32N2O7SPurity:99.75% - 99.98%Color and Shape:SolidMolecular weight:516.61ZM 226600
CAS:<p>ZM 226600 is an ATP-sensitive potassium channel opener with an EC50 value of 500 nM. ZM226600 has an inhibitory effect on spontaneous bladder activity.</p>Formula:C16H14F3NO4SPurity:99.87%Color and Shape:SolidMolecular weight:373.35Leminoprazole
CAS:<p>Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.</p>Formula:C19H23N3OSPurity:99.08% - 99.56%Color and Shape:SolidMolecular weight:341.47PD-118057
CAS:<p>PD-118057, a potent hERG activator, may treat long QT syndrome and heart failure without hERG activity inhibition.</p>Formula:C21H17Cl2NO2Purity:99.16% - 99.97%Color and Shape:SolidMolecular weight:386.27Orphenadrine
CAS:<p>Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner,</p>Formula:C18H23NOPurity:98.91% - 99.11%Color and Shape:SolidMolecular weight:269.38ANO1-IN-1
CAS:<p>ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.</p>Formula:C18H28N2O2SPurity:99.66%Color and Shape:SolidMolecular weight:336.49BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormula:C19H20Cl2N2OPurity:99.43% - 99.95%Color and Shape:SolidMolecular weight:363.28Coelenterazine h
CAS:<p>Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.</p>Formula:C26H21N3O2Purity:99.49%Color and Shape:Yellow To Brownish PowderMolecular weight:407.46PF-06456384
CAS:PF-06456384 is a highly potent and selective NaV1.7 inhibitor with IC50 value of 0.01 nM.Formula:C35H32F3N7O3S2Purity:98%Color and Shape:SolidMolecular weight:719.8α,β-Methylene-ATP
CAS:<p>α,β-Methylene ATP，一种ATP的膦酸酯类似物，充当P2X3和P2X7受体的配体。该化合物对P2X1和P2X3表现出高选择性激动剂活性，而在P2X2, 4, 7受体上无活性。</p>Formula:C11H18N5O12P3Color and Shape:SolidMolecular weight:505.21VU6007477
CAS:<p>VU6007477: M1 PAM, EC50=230 nM, min. agonist activity, penetrates CNS, no seizure AEs.</p>Formula:C24H26N6O2Color and Shape:SolidMolecular weight:430.5BMS-199264 hydrochloride
CAS:<p>BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.</p>Formula:C26H32Cl2N4O4SPurity:99.86%Color and Shape:SolidMolecular weight:567.53Glibornuride
CAS:<p>Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75).</p>Formula:C18H26N2O4SPurity:99.5%Color and Shape:SolidMolecular weight:366.48Piprofurol
CAS:<p>Piprofurol is used as a Calcium channel blocker.</p>Formula:C26H33NO6Purity:98%Color and Shape:SolidMolecular weight:455.54URAT1 inhibitor 6
CAS:<p>URAT1 inhibitor 6 (Compound 1h), with an IC50 of 35 nM for hURAT1, demonstrates 200-fold and 8-fold greater potency compared to Lesinurad and Benzbromarone,</p>Formula:C9H7BrN3NaO2S2Color and Shape:SolidMolecular weight:356.2RS 5773
CAS:<p>RS 5773 is a benzothiazepine derivative with antianginal effects.</p>Formula:C29H33ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:541.1PF-05241328
CAS:PF-05241328 is an effective and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (IC50: 31 nM).Formula:C19H21ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:436.91VMAT2-IN-I HCl
CAS:<p>VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.</p>Formula:C25H32ClF4NO4Purity:98%Color and Shape:SolidMolecular weight:521.97(Rac)-AMG8379
CAS:<p>(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.</p>Formula:C25H16ClF2N3O5SPurity:99.6%Color and Shape:SolidMolecular weight:543.93PF-4778574
CAS:<p>PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).</p>Formula:C19H22N2O3S2Purity:98%Color and Shape:SolidMolecular weight:390.52GNE-0723
CAS:<p>GNE-0723 is a selective positive allosteric modulator of the NMDA receptor, GluN2A.blood-brain barrier (BBB) and Dravet syndrome and Alzheimer's disease (AD).</p>Formula:C16H8ClF6N5OSPurity:97.29% - 99.91%Color and Shape:SolidMolecular weight:467.78PPADS tetrasodium
CAS:<p>PPADS tetrasodiuma is a P2X receptor antagonist and an inhibitor of the inverse mode of Na/Ca²⁺ exchange in guinea pig airway smooth muscle.</p>Formula:C14H10N3Na4O12PS2Purity:95% - ≥95%Color and Shape:SolidMolecular weight:599.3GDC-0310
CAS:<p>GDC-0310 is a selective, orally available Nav1.7 inhibitor with an IC50 of 0.6 nM for human Nav1.7, suitable for pain research.</p>Formula:C25H29Cl2FN2O4SPurity:99.877%Color and Shape:SolidMolecular weight:543.48Chromanol 293B
CAS:slow delayed rectifier K+ current (IKs) blockerFormula:C15H20N2O4SPurity:98%Color and Shape:SolidMolecular weight:324.4α,β-Methylene ATP trisodium
CAS:α,β-Methylene ATP trisodium is a ligand of P2X3 and P2X7 receptor.Formula:C11H15N5Na3O12P3Purity:99.66%Color and Shape:SolidMolecular weight:571.15KVI-020
CAS:<p>KVI-020: oral Kv1.5 blocker (IC50: 480nM), hERG inhibitor (IC50: 15100nM), potent antiarrhythmic for AF studies.</p>Formula:C20H25N3O5SColor and Shape:SolidMolecular weight:419.49CGP 55845 hydrochloride
CAS:<p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>Formula:C18H23Cl3NO3PColor and Shape:SolidMolecular weight:438.71ZM 260384
CAS:<p>ZM 260384 is a potassium channel opener.</p>Formula:C15H11F4N3O4Color and Shape:SolidMolecular weight:373.26Lingdolinurad
CAS:<p>Lingdolinurad is a uric acid transporter protein inhibitor targeting hURAT1 for the study of hyperuricemia or gout.</p>Formula:C17H12BrN3O2Purity:96.26%Color and Shape:SolidMolecular weight:370.2(R)-Elexacaftor
CAS:<p>(R)-Elexacaftor (compound 37) is the enantiomer of Elexacaftor (compound 1). (R)-Elexacaftor is a CFTR modulator with an EC50 of 0.29 μM for CFTR dF508.</p>Formula:C26H34F3N7O4SPurity:98.991%Color and Shape:SolidMolecular weight:597.65Aneratrigine
CAS:<p>Aneratrigine is a blocker of the sodium channel protein type 9 subunit alpha, utilized in research on neuropathic pain diseases [1].</p>Formula:C19H20ClF2N5O2S2Purity:98%Color and Shape:SolidMolecular weight:487.97DPO-1
CAS:<p>DPO-1 可以高效抑制电压门控钾离子通道Kv1.5，也可以阻断超快速延迟整流钾电流。它能够预防房性心律失常。</p>Formula:C22H29OPPurity:99.78%Color and Shape:SolidMolecular weight:340.44Kv3 modulator 4
CAS:<p>Kv3 modulator 4 is a Kv3.1 (pEC50=5.45) and Kv3.2 modulator .Cyclobutyl structure.</p>Formula:C20H24N2O4Purity:98%Color and Shape:SolidMolecular weight:356.42Linaprazan
CAS:<p>Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase by K+-competitive binding with an IC50 of 1.0 μM.</p>Formula:C21H26N4O2Purity:99.54%Color and Shape:SolidMolecular weight:366.46CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35(R)-3,4-DCPG
CAS:<p>AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors</p>Formula:C10H9NO6Purity:98%Color and Shape:SolidMolecular weight:239.18Sudoterb free base
CAS:<p>Sudoterb free base (Sudoterb) , also known as LL3858, is an anti-tubercular drug candidate.</p>Formula:C29H28F3N5OPurity:97.26% - 98.85%Color and Shape:SolidMolecular weight:519.56OADS
CAS:<p>OADS is an inhibitor of ClC-ec1 with low micromolar affinity. OADS has no specific effect on a CLC channel (ClC-1).</p>Formula:C30H42N2O8S2Color and Shape:SolidMolecular weight:622.79CP 154526
CAS:<p>CRF1 receptor antagonist</p>Formula:C23H33ClN4Purity:98%Color and Shape:SolidMolecular weight:400.99Dasolampanel etibutil
CAS:<p>Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).</p>Formula:C23H32ClN5O3Color and Shape:SolidMolecular weight:461.98Potassium Channel Activator 1
CAS:<p>Potassium Channel Activator 1 aids treatment of ADHD, schizophrenia, and mood disorders by targeting the dopaminergic system.</p>Formula:C19H23N3O3Purity:99.86%Color and Shape:SolidMolecular weight:341.4UBP316
CAS:GluR5-containing kainate receptor antagonistFormula:C20H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:429.45Naltiazem
CAS:<p>Naltiazem, a calcium channel antagonist, is used potentially for the treatment of arrhythmias, hypertension and myocardial infarction.</p>Formula:C26H28N2O4SPurity:98%Color and Shape:SolidMolecular weight:464.58Xeniafaraunol A
CAS:<p>Xeniafaraunol A (compound 31) is a potent inhibitor of the transient receptor potential melastatin 7 (TRPM7) channel [1].</p>Formula:C20H28O2Color and Shape:SolidMolecular weight:300.44TROX-1
CAS:<p>TROX-1 is the activation state-dependent Cav2 channel antagonist.</p>Formula:C22H16ClFN6OPurity:98%Color and Shape:SolidMolecular weight:434.85MK-2295
CAS:<p>MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.</p>Formula:C27H31FN6O2Purity:98.83% - 99.44%Color and Shape:SolidMolecular weight:490.57TRPV2-selective blocker 1
CAS:<p>TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, exhibiting an IC50 value of 6.3 μM.</p>Formula:C15H18OS2Color and Shape:SolidMolecular weight:278.43AMPA receptor modulator-2
CAS:<p>AMPA receptor modulator-2 is a modulator of AMPA receptor. The pIC50 value for TARPγ2 dependent AMPA receptor is 10.1.</p>Formula:C15H6F6N4OSPurity:99.8%Color and Shape:SolidMolecular weight:404.29BTG 502
CAS:<p>BTG 502 is an alkylamide insecticide that binds to voltage-gated sodium channels, antagonising the activation of sodium channels by Batrachotoxin (BTX).</p>Formula:C21H24BrNOPurity:99.30%Color and Shape:SolidMolecular weight:386.33XR9051
CAS:<p>XR9051, a synthetic derivative of a natural compound, potently reverses P-glycoprotein MDR (EC50 = 1.4 nM) by inhibiting cytotoxic binding.</p>Formula:C39H38N4O5Color and Shape:SolidMolecular weight:642.74Ritivixibat
CAS:<p>Ritivixibat inhibits IBAT and modulates bile acids, used in research for cardiovascular, metabolic, GI, and liver diseases.</p>Formula:C26H36N2O5S2Color and Shape:SolidMolecular weight:520.7ADCI
CAS:<p>ADCI inhibits voltage-activated sodium and NMDA channels; boosts dopamine metabolism in prefrontal cortex and nucleus accumbens.</p>Formula:C16H14N2OPurity:98%Color and Shape:SolidMolecular weight:250.3(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Formula:C21H20ClNO6Purity:98%Color and Shape:SolidMolecular weight:417.84CGP 54626 hydrochloride
CAS:<p>CGP 54626 hydrochloride is a GABAB receptor antagonist.</p>Formula:C18H29Cl3NO3PPurity:98%Color and Shape:SolidMolecular weight:444.76BMT-108908
CAS:<p>BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.</p>Formula:C22H25FN2O2Color and Shape:SolidMolecular weight:368.44Y-27152
CAS:<p>Y-27152 is a prodrug of the KATP (Kir6) channel opener Y-26763 and is a long-acting K+ channel opener.</p>Formula:C21H22N2O4Purity:98%Color and Shape:SolidMolecular weight:366.41URAT1 inhibitor 1
CAS:URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.Formula:C19H15Br2N5O2S2Purity:98%Color and Shape:SolidMolecular weight:569.29MK-8153
CAS:<p>MK-8153: Selective, potent ROMK inhibitor, orally active, IC50: ROMK EP 5 μM, hERG EP 34 μM; potential diuretic.</p>Formula:C24H28N2O6Color and Shape:SolidMolecular weight:440.4911-deoxy-PGF2a
CAS:<p>11-deoxy-PGF2a is a thromboxane A2 receptor agonist that partially alleviates crowding in Lpar3(−/−) female embryos and induces smooth muscle contraction</p>Formula:C20H34O4Color and Shape:SolidMolecular weight:338.48Zelquistinel
CAS:<p>Zelquistinel, an NMDA receptor agonist, aids research on depression, anxiety, and psychiatric disorders.</p>Formula:C15H25N3O5Color and Shape:SolidMolecular weight:327.38APS3
CAS:<p>APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].</p>Formula:C18H7Cl2F6N5O5S2Color and Shape:SolidMolecular weight:622.31JYL-1511
CAS:<p>JYL-1511 is the TRPV1 channel partial agonist.</p>Formula:C21H29N3O3S2Purity:98%Color and Shape:SolidMolecular weight:435.6GABAA receptor agent 2 TFA
CAS:<p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>Formula:C22H22F3N3O3Color and Shape:SolidMolecular weight:433.42ARN 11391
CAS:<p>ARN 11391 enhances the function of the IP3-gated calcium channel ITPR1 (Inositol 1,4,5-trisphosphate (IP3) receptor type 1), boosting intracellular calcium ion</p>Formula:C22H29N3O3Color and Shape:SolidMolecular weight:383.49D-erythro-Sphingosine hydrochloride
CAS:<p>D-erythro-Sphingosine HCl activates TRPM3 and dephosphorylates retinoblastoma protein.</p>Formula:C18H38ClNO2Color and Shape:SolidMolecular weight:335.95γ-Kainylglutamic acid
CAS:<p>gamma-Kainylglutamic acid is a selective amino acid-induced neuroexcitation antagonist.</p>Formula:C15H22N2O7Purity:98%Color and Shape:SolidMolecular weight:342.34FGIN-1-27
CAS:<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Formula:C28H37FN2OPurity:99.86%Color and Shape:SolidMolecular weight:436.6AR-C141990
CAS:<p>AR-C141990 is a lactate transporters inhibitor.</p>Formula:C26H28N4O4SColor and Shape:SolidMolecular weight:492.59BMS-986169
CAS:<p>BMS-986169 is a high-affinity and selective negative allosteric modulator of the NMDA receptor GluN2B subunit, depression.</p>Formula:C23H27FN2O2Purity:97.61%Color and Shape:SolidMolecular weight:382.47A 425619
CAS:<p>A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist</p>Formula:C18H14F3N3OPurity:99.75%Color and Shape:SolidMolecular weight:345.32Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Formula:C29H30Cl2F2N4O2Purity:98%Color and Shape:SolidMolecular weight:575.48U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Formula:C16H23N5Purity:99.62%Color and Shape:SolidMolecular weight:285.39S-Pantoprazole sodium trihydrate
CAS:<p>S-Pantoprazole (sodium trihydrate), a variant of Pantoprazole, is pivotal in managing diseases associated with gastric acid secretion disorders, serving as a</p>Formula:C16H20F2N3NaO7SPurity:98%Color and Shape:SolidMolecular weight:459.4GMA-839
CAS:<p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>Formula:C21H31F3O3Purity:98%Color and Shape:SolidMolecular weight:388.46AGN-201904Z
CAS:<p>AGN-201904Z is a slow-release, acid-resistant pro-PPI that turns into omeprazole, offering extended acid suppression.</p>Formula:C25H25N3NaO8S2Purity:98%Color and Shape:SolidMolecular weight:582.6AC-4
CAS:<p>AC-4 is a blocker of photoswitchable TRPV1 channel.</p>Formula:C26H25F3N4O2SColor and Shape:SolidMolecular weight:514.56Nepaprazole
CAS:<p>Nepaprazole (TY-11345) is a potent proton pump inhibitor; IC50: 5.8µM at pH 6.0, 9.9µM at pH 7.4. Better inhibition in weak acid.</p>Formula:C18H19N3O2SPurity:98%Color and Shape:SolidMolecular weight:341.43P-1075
CAS:<p>P-1075 activates SUR2-KIR6 channels at 45 nM; may open mitoKATP channels and protect the heart.</p>Formula:C12H17N5Purity:99.85%Color and Shape:SolidMolecular weight:231.33′-Acetate-ATP
CAS:<p>3’-Acetate-ATP, an analogue of ATP and its acetylation product, exhibits maximum ultraviolet absorption at 259 nm in neutral aqueous solutions.</p>Formula:C12H18N5O14P3Color and Shape:SolidMolecular weight:549.22NCS-382 sodium
CAS:<p>NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological disease</p>Formula:C13H13NaO3Purity:98%Color and Shape:SolidMolecular weight:240.23NPEC-caged-(S)-AMPA
CAS:<p>AMPA receptor agonist</p>Formula:C16H17N3O8Purity:98%Color and Shape:SolidMolecular weight:379.32TRPC3/6-IN-2
CAS:<p>TRPC3/6-IN-2 is a potent inhibitor of TRPC3 and TRPC6, exhibiting IC50 values of 16 nM for TRPC3 and 29.8 nM for TRPC6, respectively [1].</p>Formula:C18H23F2N5Color and Shape:SolidMolecular weight:347.41L 663581
CAS:<p>L 663581 is the benzodiazepine receptor partial agonist.</p>Formula:C17H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:357.79TPA 023
CAS:<p>TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).</p>Formula:C20H22FN7OPurity:99.75%Color and Shape:SolidMolecular weight:395.43Kv3 modulator 2
CAS:<p>Kv3 modulator 2 is a potent Kv3 channels modulator.has analgesic activity and is used in the prophylaxis or treatment of related disorders.</p>Formula:C21H21N3O4Purity:98%Color and Shape:SolidMolecular weight:379.41SLC13A5-IN-1
CAS:<p>SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5),completely blocks the uptake of 14C-citrate(IC50 : 0.022 μM in HepG2 cells).</p>Formula:C19H19Cl3N2O3SPurity:99.67%Color and Shape:SolidMolecular weight:461.79TRPC5-IN-3
CAS:<p>TRPC5-IN-3 is a potent TRPC5 inhibitor (IC50= 10.75 nM).</p>Formula:C18H15ClF3N5OColor and Shape:SolidMolecular weight:409.79VU0463271
CAS:<p>VU0463271: KCC2 antagonist, IC50 61 nM, >100x selective over NKCC1, inactive on other GPCRs, channels, transporters.</p>Formula:C19H18N4OS2Purity:97.84% - 99.55%Color and Shape:SolidMolecular weight:382.5Pristinamycin IA
CAS:<p>Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.</p>Formula:C45H54N8O10Purity:97.44%Color and Shape:SolidMolecular weight:866.96DNDS
CAS:<p>DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).</p>Formula:C14H8N2Na2O10S2Purity:99.92%Color and Shape:Physical Description White Powder (Ntp 1992)Molecular weight:474.33NS1219
CAS:<p>NS1219, an isomer of NS1209, is a selective AMPA antagonist for studying stroke, neuropathic pain, and epilepsy.</p>Formula:C24H28N4O7SColor and Shape:SolidMolecular weight:516.57Sodium Channel inhibitor 4
CAS:<p>Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].</p>Formula:C19H18ClN3O4S2Purity:98%Color and Shape:SolidMolecular weight:451.95PF 04531083
CAS:<p>PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.</p>Formula:C17H16ClN5O2Purity:99.85%Color and Shape:SolidMolecular weight:357.79(+)-Bicuculline methiodide
CAS:<p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29Budiodarone
CAS:<p>Budiodarone (ATI-2042) resembles amiodarone, potentially preventing atrial fibrillation.</p>Formula:C27H31I2NO5Color and Shape:SolidMolecular weight:703.35Piperidine-4-sulfonic acid
CAS:<p>Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].</p>Formula:C5H11NO3SPurity:98%Color and Shape:SolidMolecular weight:165.216,2'-Dihydroxyflavone
CAS:<p>6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.</p>Formula:C15H10O4Purity:99.44% - 99.67%Color and Shape:SolidMolecular weight:254.24PHP 501 trifluoroacetate
CAS:<p>GABAA antagonist</p>Formula:C20H21N3OPurity:98%Color and Shape:SolidMolecular weight:319.4ML-252 hydrochloride
CAS:<p>ML-252 is a potent, selective inhibitor of the Kv7.2 voltage-gated potassium channel, demonstrating an IC50 value of 69 nM in patch clamp assays. It exists as the (S)-enantiomer, which is significantly more effective than both its (R)-enantiomer counterpart and the racemic mixture, with respective IC50 values of 944 nM and 160 nM. ML-252 exhibits high selectivity for Kv7.2 over other potassium channel subtypes and shows minimal activity against more than 68 G protein-coupled receptors, various transporters, L- and N-type calcium channels, K_ATP, and hERG potassium channels. However, it does inhibit the melatonin MT1 receptor by 61% at a 10 µM concentration.</p>Formula:C20H24N2OHClColor and Shape:SolidMolecular weight:344.9JYL-273
CAS:<p>JYL-273 is a TRPV1 agonist.</p>Formula:C28H39NO4SColor and Shape:SolidMolecular weight:485.68
