Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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Ethyl tosylcarbamate
CAS:Gliclazide blocks beta-cell ATP-sensitive K+ currents, IC50: 184 nM. Ethyl tosylcarbamate is a synthesis intermediate.Formula:C10H13NO4SColor and Shape:SolidMolecular weight:243.28H-D-Allo-Ile-OH
CAS:<p>H-D-Allo-Ile-OH inhibits 3[H] gabapentin binding/voltage-dependent L-type calcium channels and can be used for studying neurological and psychiatric disorders.</p>Formula:C6H13NO2Purity:99.92%Color and Shape:SolidMolecular weight:131.17Mepivacaine
CAS:<p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>Formula:C15H22N2OPurity:99.35%Color and Shape:SolidMolecular weight:246.35(+)-SJ733
CAS:<p>(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.</p>Formula:C24H16F4N4O2Purity:99.21%Color and Shape:SolidMolecular weight:468.4GYKI 53655 hydrochloride
CAS:GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the study of neurological disorders.Formula:C19H21ClN4O3Purity:98.02%Color and Shape:SolidMolecular weight:388.85β-Cyfluthrin
CAS:<p>β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.</p>Formula:C22H18Cl2FNO3Color and Shape:SolidMolecular weight:434.29Lubiprostone hemiketal
CAS:Lubiprostone (hemiketal) (RU-0211 (hemiketal)), a selective activator of the chloride channel 2 (CLCN2), facilitates the treatment of chronic idiopathic constipation and opioid-induced constipation. It functions by enhancing CLCN2 channel activity, which boosts chloride ion secretion in the intestines, subsequently increasing fluid secretion and improving intestinal peristalsis. Additionally, Lubiprostone (hemiketal) may be utilized in research related to chronic constipation and cancer.Formula:C20H32F2O5Color and Shape:SolidMolecular weight:390.46(R)-BPO-27
CAS:(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.Formula:C26H18BrN3O6Purity:99.1%Color and Shape:SolidMolecular weight:548.34Crinecerfont hydrochloride
CAS:<p>SSR-125543, a potent CRF1 receptor non-peptide antagonist, effective in CAH research, taken orally.</p>Formula:C27H29Cl2FN2OSColor and Shape:SolidMolecular weight:519.5Flumazenil acid
CAS:<p>Flumazenil is an antagonist of GABAA receptor. Flumazenil acid is a metabolite of Flumazenil.</p>Formula:C13H10FN3O3Color and Shape:SolidMolecular weight:275.24Tetrabenazine-d6
CAS:Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder.Formula:C19H27NO3Purity:98%Color and Shape:SolidMolecular weight:323.46L-Palmitoylcarnitine
CAS:<p>L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.</p>Formula:C23H45NO4Purity:97% - 99.81%Color and Shape:SolidMolecular weight:399.61VU041
CAS:VU041 inhibits mosquito Kir1 channels (IC50: An. gambiae 2.5μM, Ae. aegypti 1.7μM), less on mammalian Kir2.1 (12.7μM), and minimally on other Kir channels.Formula:C19H20F3N3OPurity:98%Color and Shape:SolidMolecular weight:363.38YM-244769 dihydrochloride
CAS:YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.Formula:C26H24Cl2FN3O3Purity:98%Color and Shape:SolidMolecular weight:516.39(R)-Tegoprazan
CAS:<p>(R)-Tegoprazan, a benzimidazole derivative, inhibits kidney H+/K+-ATPase (IC50: 98 nM). Potential in GI disease research.</p>Formula:C20H19F2N3O3Color and Shape:SolidMolecular weight:387.38PF-04856264
CAS:<p>PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.</p>Formula:C20H15N5O3S2Purity:97.43%Color and Shape:SolidMolecular weight:437.5(R)-Lercanidipine-d3 hydrochloride
CAS:(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.Formula:C36H42ClN3O6Purity:98%Color and Shape:SolidMolecular weight:651.21Leptin (22-56), human
CAS:Leptin(22-56),human is a peptide fragment of Leptin, which ACTS through a variety of subtypes of Ob-Rs.Formula:C171H298N50O56Color and Shape:SolidMolecular weight:3950.52Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Formula:C22H31ClN2OColor and Shape:SolidMolecular weight:374.95MRS1845
CAS:MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).Formula:C21H22N2O6Purity:99.69%Color and Shape:SolidMolecular weight:398.41Clamikalant sodium
CAS:<p>Clamikalant sodium (HMR 1098) is an ATP-dependent potassium channel (KATP) cardiac-selective blocker, used in the study of arrhythmias.</p>Formula:C19H21ClN3NaO5S2Purity:99.95%Color and Shape:SolidMolecular weight:493.96GI-530159
CAS:<p>TREK1/2 activator, selective over TRAAK/TASK3; hyperpolarizes neurons, depresses activity (EC50 = 0.76 μM).</p>Formula:C27H20F6N2O2Color and Shape:White CrystalsMolecular weight:518.45(-)-α-Pinene
CAS:<p>(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,</p>Formula:C10H16Purity:98.02% - 98.60%Color and Shape:Colourless LiquidMolecular weight:136.23QO-58
CAS:<p>QO-58 is a novel Kv7 activator (opener) that activates neuronal Kv7/KCNQ/M channels, danti-nociceptive effects on inflammatory pain</p>Formula:C18H8Cl2F4N4OPurity:99.17%Color and Shape:SolidMolecular weight:443.18Luciferase, firefly
CAS:<p>Luciferase, firefly is a reporter gene in cellular imaging studies to quantify target gene expression levels and measure intracellular ATP content,</p>Purity:98%Color and Shape:SolidMolecular weight:N/ABenzocaine hydrochloride
CAS:<p>Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and</p>Formula:C9H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:201.65Triamterene D5
CAS:Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.Formula:C12H11N7Purity:98%Color and Shape:SolidMolecular weight:258.29Tetramethrin
CAS:<p>Tetramethrin is a type I pyrethroid insecticide that affects the inactivation process of sodium channels in insect neurons, prolonged sodium currents.</p>Formula:C19H25NO4Purity:98.85%Color and Shape:White Crystals Or PowderMolecular weight:331.41Poneratoxin acetate
<p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>Formula:C129H215N33O31S·xC2H4O2Color and Shape:SolidMolecular weight:2756.35 (free base)L-364,373
CAS:KV7.1 (KCNQ1) channel activatorFormula:C25H20FN3OColor and Shape:SolidMolecular weight:397.44SDZ 220-581 hydrochloride
CAS:SDZ 220-581 hydrochloride is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).Formula:C16H18Cl2NO5PPurity:98%Color and Shape:SolidMolecular weight:406.2BI-9627 hydrochloride
CAS:<p>BIX HCl is a sodium-hydrogen exchange type 1 inhibitor.</p>Formula:C16H20ClF3N4O2Color and Shape:SolidMolecular weight:392.8HSK16149
CAS:<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Formula:C12H19NO2Color and Shape:SolidMolecular weight:209.28SDZ 220-581 Ammonium salt
CAS:<p>SDZ 220-581 Ammonium salt is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Formula:C16H20ClN2O5PPurity:98%Color and Shape:SolidMolecular weight:386.77TACA
CAS:<p>GABAA agonist</p>Formula:C4H7NO2Purity:98%Color and Shape:White SolidMolecular weight:101.1Dibucaine hydrochloride
CAS:<p>Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.</p>Formula:C20H30ClN3O2Purity:99.66%Color and Shape:White PowderMolecular weight:379.92Lansoprazole-d4
CAS:Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid.Formula:C16H14F3N3O2SPurity:98%Color and Shape:SolidMolecular weight:373.39(R)-Nicardipine
CAS:<p>(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formula:C26H29N3O6Color and Shape:SolidMolecular weight:479.53Cabotegravir sodium
CAS:<p>Cabotegravir sodium inhibits HIV integrase (IC50: 2.5 nM), metabolized by UGT1A1, with minimal ARV interaction.</p>Formula:C19H16F2N3NaO5Color and Shape:SolidMolecular weight:427.34TGN-073
CAS:<p>TGN-073 is an enhancer of aquaporin 4 (AQP4), a water channel in astrocytes. It shows an increase in lymphatic transport in the rat brain by up to 41%.</p>Formula:C18H16N2O3SColor and Shape:SolidMolecular weight:340.396SDZ 220-581
CAS:<p>SDZ 220-581 is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Formula:C16H17ClNO5PPurity:98%Color and Shape:SolidMolecular weight:369.74Nateglinide D5
CAS:<p>Nateglinide D5 is a deuterium labeled Nateglinide.</p>Formula:C19H27NO3Purity:98%Color and Shape:SolidMolecular weight:322.4517β-Estradiol sulfate sodium
CAS:<p>17β-Estradiol sulfate sodium (17β-Estradiol 3-sulfate sodium) is a neuroactive estrogen with vasoprotective properties that inhibits the growth of Neisseria brasiliensis and disrupts aquatic ecosystems.</p>Formula:C18H23NaO5SPurity:99%Color and Shape:SolidMolecular weight:374.43SKA-121
CAS:<p>SKA-121 is a selective KCa3.1 activator (EC50s: 109 nM and 4.4 μM for KCa3.1 and KCa2.3, respectively).</p>Formula:C12H10N2OPurity:98%Color and Shape:SolidMolecular weight:198.22Mexiletine-d6 hydrochloride
CAS:<p>Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.</p>Formula:C11H18ClNOPurity:98%Color and Shape:SolidMolecular weight:221.76N-Methyl-DL-aspartic acid
CAS:<p>N-Methyl-DL-aspartic acid, a glutamate analogue and NMDA receptor agonist, is utilized in neurological disease research.</p>Formula:C5H9NO4Purity:99.85%Color and Shape:SolidMolecular weight:147.13UBP608
CAS:<p>UBP608 selectively inhibits NMDA GluN1/GluN2A receptors, 23x more than GluN1/GluN2D.</p>Formula:C10H5BrO4Color and Shape:SolidMolecular weight:269.05YM-244769
CAS:<p>YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)</p>Formula:C26H22FN3O3Purity:95.62%Color and Shape:SolidMolecular weight:443.473,3-Diethylthiacarbocyanine iodide
CAS:<p>3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.</p>Formula:C21H21IN2S2Purity:99.79%Color and Shape:SolidMolecular weight:492.44Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formula:C17H26ClNOPurity:99.80%Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMolecular weight:295.85Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Formula:C18H12ClF4N5O2Purity:98.6%Color and Shape:SolidMolecular weight:441.77YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Formula:C20H22N2O3SPurity:98.78%Color and Shape:SolidMolecular weight:370.47HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Formula:C18H21N5O3Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:355.39CCTA-1523
CAS:<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Formula:C16H15Cl2NO3Purity:99.71%Color and Shape:SolidMolecular weight:340.2VU0134992
CAS:<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Formula:C20H31BrN2O2Purity:99.86%Color and Shape:SolidMolecular weight:411.38Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.77%Color and Shape:SolidMolecular weight:159.14Omecamtiv mecarbil
CAS:<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Formula:C20H24FN5O3Purity:98% - 99.23%Color and Shape:SolidMolecular weight:401.43Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Formula:C14H9Cl2NO4SPurity:97.43% - 98.04%Color and Shape:SolidMolecular weight:358.2BzATP triethylammonium salt
CAS:<p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>Formula:C30H39N6O15P3Purity:95% - 99.57%Color and Shape:SolidMolecular weight:816.59(S)-ATPO
CAS:<p>(S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.</p>Formula:C11H19N2O7PPurity:98.37% - 99.41%Color and Shape:SolidMolecular weight:322.25Procyclidine hydrochloride
CAS:<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Formula:C19H30ClNOPurity:99.24% - 99.88%Color and Shape:Crystals From Petroleum Ether White PowderMolecular weight:323.9DL-Menthol
CAS:<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Formula:C10H20OPurity:99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27γ-Acetylenic GABA
CAS:<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.143Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21UBP551
CAS:<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Formula:C11H8O4Purity:98.69%Color and Shape:SolidMolecular weight:204.18DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Formula:C7H5FN2OPurity:97.84%Color and Shape:SolidMolecular weight:152.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formula:C34H60N14O12SPurity:96.79% - 99.65%Color and Shape:White PowderMolecular weight:888.99OAC3
CAS:<p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>Formula:C15H11FN2OPurity:97.13%Color and Shape:SolidMolecular weight:254.26Myomodulin acetate(110570-93-9 free base)
Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.Formula:C38H71N11O10S2Purity:99.24%Color and Shape:SolidMolecular weight:906.17Raxatrigine
CAS:Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.Formula:C18H19FN2O2Purity:98% - 99.43%Color and Shape:SolidMolecular weight:314.35Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formula:C38H52CaN2O8Purity:98.97% - 99.96%Color and Shape:White SolidMolecular weight:704.91HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purity:99.95%Color and Shape:SolidMolecular weight:507.98Ivacaftor
CAS:<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Formula:C24H28N2O3Purity:99% - 99.98%Color and Shape:SolidMolecular weight:392.49NPPB
CAS:<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Formula:C16H16N2O4Purity:99.95%Color and Shape:Light Yellow To Yellow SolidMolecular weight:300.31NBQX
CAS:<p>NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.</p>Formula:C12H8N4O6SPurity:97.66% - 99.42%Color and Shape:SolidMolecular weight:336.286-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Formula:C15H14O4Purity:98.06%Color and Shape:SolidMolecular weight:258.27Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Formula:C17H16FN3O2SPurity:99.87% - 99.92%Color and Shape:SolidMolecular weight:345.39TRPM8 antagonist WS-3
CAS:TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).Formula:C13H25NOPurity:97.64%Color and Shape:DrypowderMolecular weight:211.34SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Formula:C10H12N2O3Purity:99.84%Color and Shape:SolidMolecular weight:208.21AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Formula:C34H31F2N3O3Purity:99.61%Color and Shape:SolidMolecular weight:567.62ICA-121431
CAS:<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Formula:C23H19N3O3S2Purity:98.06%Color and Shape:SolidMolecular weight:449.55SAR7334 hydrochloride
CAS:<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formula:C21H24Cl3N3OPurity:98%Color and Shape:SolidMolecular weight:440.79Selinexor (KPT-330)
CAS:<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Formula:C17H11F6N7OPurity:98% - 99.97%Color and Shape:SolidMolecular weight:443.31Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Formula:C15H17FN4O2·C4H4O4Purity:99.5% - 99.9%Color and Shape:Off-White Crystalline PowderMolecular weight:420.39Homo-VK-II-36
CAS:<p>Homo-VK-II-36 (Homo-V-II-36) is a carvedilol analogue that acts by inhibiting store- overload-induced calcium release through the RyR2 channel.</p>Formula:C27H28N2O5Purity:99.26%Color and Shape:SolidMolecular weight:460.527-Chlorokynurenic acid sodium salt
CAS:<p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>Formula:C10H6ClNNaO3Color and Shape:SolidMolecular weight:246.6α-Cyano-4-hydroxycinnamic acid
CAS:<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Formula:C10H7NO3Purity:99.8% - 99.86%Color and Shape:PowderMolecular weight:189.17Thonzonium Bromide
CAS:<p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>Formula:C32H55BrN4OPurity:98.48% - 99.94%Color and Shape:SolidMolecular weight:591.71Linerixibat
CAS:<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Formula:C28H38N2O7SPurity:98.5% - 99.98%Color and Shape:SolidMolecular weight:546.68ML365
CAS:<p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>Formula:C22H20N2O3Purity:98.78%Color and Shape:SolidMolecular weight:360.41Vanilloid receptor antagonist 1
CAS:<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Formula:C18H15N3O2Purity:98.14%Color and Shape:SolidMolecular weight:305.33Zoniporide hydrochloride hydrate
CAS:Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.Formula:C17H19ClN6O2Purity:98%Color and Shape:SolidMolecular weight:374.83SB-366791
CAS:<p>SB-366791 is a new and selective cinnamide TRPV1 antagonist.</p>Formula:C16H14ClNO2Purity:99.51%Color and Shape:SolidMolecular weight:287.74Optovin
CAS:<p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>Formula:C15H13N3OS2Purity:99.47% - 99.67%Color and Shape:SolidMolecular weight:315.41Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formula:C24H32NO6ClPurity:99.9%Color and Shape:SolidMolecular weight:465.97Methyl homoveratrate
CAS:<p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>Formula:C11H14O4Purity:99.48%Color and Shape:SolidMolecular weight:210.23Vocacapsaicin
CAS:<p>Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.</p>Formula:C26H41N3O4Color and Shape:SolidMolecular weight:459.631N-Me-aminopyrimidinone9
CAS:<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Formula:C16H21N3OSPurity:99.21%Color and Shape:SolidMolecular weight:303.42SKA-31
CAS:<p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>Formula:C11H8N2SPurity:99.38%Color and Shape:SolidMolecular weight:200.26
