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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • Levcromakalim

    CAS:
    <p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>
    Formula:C16H18N2O3
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:286.33
  • Felbamate

    CAS:
    Felbamate (W-554) is an Anti-epileptic Agent.
    Formula:C11H14N2O4
    Purity:99% - >99.99%
    Color and Shape:White Powder Solid
    Molecular weight:238.24
  • N-Me-aminopyrimidinone9

    CAS:
    <p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>
    Formula:C16H21N3OS
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:303.42
  • Vocacapsaicin

    CAS:
    <p>Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.</p>
    Formula:C26H41N3O4
    Color and Shape:Solid
    Molecular weight:459.631
  • Zoniporide hydrochloride hydrate

    CAS:
    Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.
    Formula:C17H19ClN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.83
  • OAC3

    CAS:
    <p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>
    Formula:C15H11FN2O
    Purity:97.13%
    Color and Shape:Solid
    Molecular weight:254.26
  • SKA-31

    CAS:
    <p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>
    Formula:C11H8N2S
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:200.26
  • Thonzonium Bromide

    CAS:
    <p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>
    Formula:C32H55BrN4O
    Purity:98.48% - 99.94%
    Color and Shape:Solid
    Molecular weight:591.71
  • ML213

    CAS:
    <p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>
    Formula:C17H23NO
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:257.37
  • TCN 201

    CAS:
    TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.
    Formula:C21H17ClFN3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:461.89
  • A2764 dihydrochloride

    CAS:
    <p>A2764 dihydrochloride is a highly selective inhibitor of TRESK.</p>
    Formula:C15H21Cl3N2O
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:351.7
  • Nav1.8-IN-1

    CAS:
    <p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>
    Formula:C20H15ClF3N3O2
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:421.8
  • Methyl homoveratrate

    CAS:
    <p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>
    Formula:C11H14O4
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:210.23
  • WS-12

    CAS:
    WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)
    Formula:C18H27NO2
    Purity:99.99%
    Color and Shape:Whitish To White Solid Crystalline
    Molecular weight:289.41
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Formula:C11H11N3O
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:201.22
  • Pirmenol

    CAS:
    <p>Pirmenol is a new antiarrhythmic drug</p>
    Formula:C22H30N2O
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:338.49
  • HBT1

    CAS:
    <p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>
    Formula:C16H17F3N4O2S
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:386.39
  • Tulrampator

    CAS:
    Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.
    Formula:C20H17FN4O3
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:380.37
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Formula:C17H24O4
    Purity:98.22%
    Color and Shape:Solid
    Molecular weight:292.37
  • Tricaine methanesulfonate

    CAS:
    <p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>
    Formula:C10H15NO5S
    Purity:99.259% - 99.86%
    Color and Shape:White Powder
    Molecular weight:261.30
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Formula:C10H20CaN2O8S2
    Purity:98% - 99.93%
    Color and Shape:White Odorless Or Nearly Odorless Powder
    Molecular weight:400.48
  • O4I1

    CAS:
    <p>O4I1 is an effective Oct3/4 inducer.</p>
    Formula:C16H15NO2
    Purity:96.25% - 99.47%
    Color and Shape:Solid
    Molecular weight:253.3
  • 9-Phenanthrol

    CAS:
    <p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>
    Formula:C14H10O
    Purity:98.48%
    Color and Shape:Solid
    Molecular weight:194.23
  • Neramexane HCl

    CAS:
    PAC is a cyclic amine used as a chiral auxiliary in various asymmetric syntheses.
    Formula:C11H24ClN
    Purity:95.00%
    Color and Shape:Solid
    Molecular weight:205.768
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Formula:C10H12ClNO2
    Purity:97.20% - 98.94%
    Color and Shape:Solid
    Molecular weight:213.66
  • CL 218872

    CAS:
    <p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>
    Formula:C13H9F3N4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:278.23
  • Revaprazan

    CAS:
    <p>Revaprazan: novel, K⁺-competitive acid blocker; reversibly halts gastric H⁺/K⁺-ATPase; rivals PPIs in acid reduction.</p>
    Formula:C22H23FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.44
  • TGN-020

    CAS:
    <p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>
    Formula:C8H6N4OS
    Purity:99.54% - 99.99%
    Color and Shape:Solid
    Molecular weight:206.22
  • BzATP triethylammonium salt

    CAS:
    <p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>
    Formula:C30H39N6O15P3
    Purity:95% - 99.57%
    Color and Shape:Solid
    Molecular weight:816.59
  • Ko 143

    CAS:
    <p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>
    Formula:C26H35N3O5
    Purity:99.01% - 99.89%
    Color and Shape:Solid
    Molecular weight:469.57
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Formula:C18H21ClF3N3O
    Purity:99.03% - 99.95%
    Color and Shape:Solid
    Molecular weight:387.83
  • MK6-83

    CAS:
    <p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>
    Formula:C16H20N2O2S2
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:336.47
  • TRPM4-IN-1

    CAS:
    <p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>
    Formula:C15H11Cl2NO4
    Purity:97.22%
    Color and Shape:Solid
    Molecular weight:340.16
  • ML204

    CAS:
    <p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>
    Formula:C15H18N2
    Purity:98.1% - 99.72%
    Color and Shape:Solid
    Molecular weight:226.32
  • DHQ

    CAS:
    <p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>
    Formula:C8H6N2O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:162.15
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Formula:C6H6N2O2
    Purity:99.94%
    Color and Shape:Soild
    Molecular weight:138.1238
  • Guanosine 5'-diphosphate

    CAS:
    <p>Guanosine 5'-diphosphate (GDP) as Potential Iron Mobilizer, Preventing the Hepcidin-Ferroportin Interaction and Modulating the Interleukin-6/Stat-3 Pathway.</p>
    Formula:C10H15N5O11P2
    Purity:98.46% - 99.52%
    Color and Shape:Solid
    Molecular weight:443.2
  • M8-B Hydrochloride

    CAS:
    <p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>
    Formula:C22H25ClN2O3S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:432.96
  • Rufinamide

    CAS:
    <p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>
    Formula:C10H8F2N4O
    Purity:99.77% - >99.99%
    Color and Shape:White Powder
    Molecular weight:238.19
  • Caroverine hydrochloride

    CAS:
    Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.
    Formula:C22H28ClN3O2
    Purity:98.37% - 98.75%
    Color and Shape:Solid
    Molecular weight:401.9
  • Phenyl benzoate

    CAS:
    <p>Phenyl benzoate is a benzoate ester obtained by the formal condensation of phenol with benzoic acid.It is an important organic synthesis intermediate.</p>
    Formula:C13H10O2
    Purity:99.63%
    Color and Shape:White Crystalline Powder
    Molecular weight:198.22
  • Pico145

    CAS:
    <p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>
    Formula:C23H20ClF3N4O5
    Purity:99.06%
    Color and Shape:Solid
    Molecular weight:524.88
  • RN-1734

    CAS:
    <p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>
    Formula:C14H22Cl2N2O2S
    Purity:99.1% - 99.3%
    Color and Shape:Solid
    Molecular weight:353.31
  • Chloroprocaine hydrochloride

    CAS:
    Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.
    Formula:C13H20Cl2N2O2
    Purity:99.65%
    Color and Shape:White Crystalline Powder
    Molecular weight:307.22
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Formula:C19H19FN4O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:354.38
  • BZAD01

    CAS:
    <p>BZAD01 is a selective NMDA NR1A/2B receptor antagonist.</p>
    Formula:C16H12F6N2O
    Purity:99.61% - 99.70%
    Color and Shape:Solid
    Molecular weight:362.27
  • Polyoxyethylene stearate

    CAS:
    <p>Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.</p>
    Formula:C20H40O3
    Purity:n~9-10
    Color and Shape:Light Amber Semisolid
    Molecular weight:328.29775
  • Blebbistatin

    CAS:
    <p>Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.</p>
    Formula:C18H16N2O2
    Purity:99.88% - 99.97%
    Color and Shape:Bright Yellow Solid
    Molecular weight:292.33
  • DS-1971a

    CAS:
    <p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>
    Formula:C20H21ClFN5O3S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:465.93
  • Tenatoprazole sodium

    CAS:
    <p>Tenatoprazole sodium is a potent proton pump inhibitor with an IC50 of 6.2 μM against hog gastric H+/K+-ATPase.</p>
    Formula:C16H17N4NaO3S
    Color and Shape:Solid
    Molecular weight:368.39
  • HC067047 Hydrochloride(883031-03-6 free base)

    CAS:
    HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.
    Formula:C26H29ClF3N3O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:507.98
  • O4I2

    CAS:
    <p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>
    Formula:C12H11ClN2O2S
    Purity:97.97% - 99.84%
    Color and Shape:Solid
    Molecular weight:282.75
  • A2793

    CAS:
    <p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>
    Formula:C13H12ClNO3
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:265.69
  • Dotinurad

    CAS:
    Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).
    Formula:C14H9Cl2NO4S
    Purity:97.43% - 98.04%
    Color and Shape:Solid
    Molecular weight:358.2
  • Lorediplon

    CAS:
    <p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>
    Formula:C20H15FN4O2S
    Purity:99.12% - 99.19%
    Color and Shape:Solid
    Molecular weight:394.42
  • Parimifasor

    CAS:
    <p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>
    Formula:C18H11Cl2F4N5O
    Purity:96.77% - 98.97%
    Color and Shape:Solid
    Molecular weight:460.21
  • DL-Willardiine

    CAS:
    <p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>
    Formula:C7H9N3O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:199.16
  • Tirofiban hydrochloride monohydrate

    CAS:
    <p>Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>
    Formula:C22H39ClN2O6S
    Purity:98.81% - >99.99%
    Color and Shape:White Solid
    Molecular weight:495.07
  • Vanillyl butyl ether

    CAS:
    <p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>
    Formula:C12H18O3
    Purity:99.57%
    Color and Shape:Yellowish Liquid Liquid
    Molecular weight:210.27
  • HC-056456

    CAS:
    <p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>
    Formula:C12H6N2O4S2
    Purity:99.62% - 99.65%
    Color and Shape:Solid
    Molecular weight:306.32
  • Vonoprazan fumarate

    CAS:
    <p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>
    Formula:C17H16FN3O2S·C4H4O4
    Purity:99.16% - 99.98%
    Color and Shape:Solid
    Molecular weight:461.46
  • Cis-ACBD

    CAS:
    <p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>
    Formula:C6H9NO4
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:159.14
  • Azimilide Dihydrochloride

    CAS:
    Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.
    Formula:C23H30Cl3N5O3
    Purity:97.59% - ≥95%
    Color and Shape:Solid
    Molecular weight:530.88
  • Guan-fu base A hydrochloride(1394-48-5 free base)

    CAS:
    <p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>
    Formula:C24H32NO6Cl
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:465.97
  • S107

    CAS:
    <p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>
    Formula:C11H15NOS
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:209.31
  • L-Phenylalanine-15N

    CAS:
    L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.
    Formula:C9H11NO2
    Purity:98.98%
    Color and Shape:Solid
    Molecular weight:166.18
  • QX-222 chloride

    CAS:
    <p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>
    Formula:C13H21ClN2O
    Purity:97.37%
    Color and Shape:Solid
    Molecular weight:256.77
  • SB-705498

    CAS:
    <p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>
    Formula:C17H16BrF3N4O
    Purity:99.57% - ≥95%
    Color and Shape:Solid
    Molecular weight:429.23
  • Quadrol

    CAS:
    <p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>
    Formula:C14H32N2O4
    Purity:99.91% - 99.92%
    Color and Shape:Viscous Liquid Liquid Viscous
    Molecular weight:292.41
  • (E)-KPT330

    CAS:
    <p>(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.</p>
    Formula:C17H11F6N7O
    Purity:98.69% - 99.49%
    Color and Shape:Solid
    Molecular weight:443.31
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Formula:C4H10N2O2
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:118.13
  • AMG9810

    CAS:
    <p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>
    Formula:C21H23NO3
    Purity:99.79% - 99.95%
    Color and Shape:Solid
    Molecular weight:337.41
  • Eperisone hydrochloride

    CAS:
    <p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>
    Formula:C17H26ClNO
    Purity:99.80%
    Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter Taste
    Molecular weight:295.85
  • Mitiglinide calcium hydrate

    CAS:
    <p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>
    Formula:C38H52CaN2O8
    Purity:98.97% - 99.96%
    Color and Shape:White Solid
    Molecular weight:704.91
  • TCN 213

    CAS:
    <p>TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2B</p>
    Formula:C18H24N4OS2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:376.54
  • Flecainide acetate

    CAS:
    <p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>
    Formula:C19H24F6N2O5
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:474.39
  • Selamectin

    CAS:
    <p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>
    Formula:C43H63NO11
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:769.96
  • DAAO inhibitor-1

    CAS:
    <p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>
    Formula:C7H5FN2O
    Purity:97.84%
    Color and Shape:Solid
    Molecular weight:152.13
  • Argireline

    CAS:
    <p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>
    Formula:C34H60N14O12S
    Purity:96.79% - 99.65%
    Color and Shape:White Powder
    Molecular weight:888.99
  • VK-II-36

    CAS:
    <p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>
    Formula:C26H26N2O5
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:446.49
  • ICA-069673

    CAS:
    <p>ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).</p>
    Formula:C11H6ClF2N3O
    Purity:99.04% - 99.68%
    Color and Shape:Solid
    Molecular weight:269.63
  • ML133 hydrochloride

    CAS:
    <p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>
    Formula:C19H19NO·HCl
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:313.82
  • TKIM

    CAS:
    <p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>
    Formula:C18H14ClN3O2S
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:371.84
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Formula:C10H12N2O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:208.21
  • Budipine

    CAS:
    Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.
    Formula:C21H27N
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:293.45
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Formula:C16H14O4
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:270.28
  • AER-271

    CAS:
    <p>AER-271 is an inhibitor of aquaporin-4.</p>
    Formula:C15H9ClF6NO5P
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:463.65
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Formula:C34H31F2N3O3
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:567.62
  • Ilaprazole sodium

    CAS:
    <p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>
    Formula:C19H17N4NaO2S
    Purity:99.06%
    Color and Shape:Solid
    Molecular weight:388.42
  • Tariquidar dihydrochloride

    CAS:
    Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).
    Formula:C38H40Cl2N4O6
    Color and Shape:Solid
    Molecular weight:719.65
  • Trofinetide

    CAS:
    Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.
    Formula:C13H21N3O6
    Purity:98.70% - 99.50%
    Color and Shape:Solid
    Molecular weight:315.32
  • YHO-13351

    CAS:
    YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.
    Formula:C27H37N3O7S2
    Purity:97.88%
    Color and Shape:Solid
    Molecular weight:579.73
  • Rimeporide hydrochloride

    CAS:
    <p>Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>
    Formula:C11H16ClN3O5S2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:369.84
  • Verinurad

    CAS:
    <p>Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.</p>
    Formula:C20H16N2O2S
    Purity:97.36% - 99.22%
    Color and Shape:Solid
    Molecular weight:348.42
  • SN 2

    CAS:
    <p>SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.</p>
    Formula:C17H21NO
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:255.35
  • Ocinaplon

    CAS:
    <p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>
    Formula:C17H11N5O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:301.3
  • (-)-Blebbistatin

    CAS:
    <p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>
    Formula:C18H16N2O2
    Purity:99.38% - 99.61%
    Color and Shape:Solid
    Molecular weight:292.33
  • Metaflumizone

    CAS:
    <p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>
    Formula:C24H16F6N4O2
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:506.40
  • LY 303511 hydrochloride

    CAS:
    <p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>
    Formula:C19H19ClN2O2
    Purity:98.47%
    Color and Shape:Solid
    Molecular weight:342.82
  • NBI-98782

    CAS:
    <p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>
    Formula:C19H29NO3
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:319.44