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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • CFTR corrector 6
    Targetmol
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    CFTR corrector 6

    CAS:
    <p>CFTR corrector 6, a potent CFTR potentiator, aids cystic fibrosis research and related disorders.</p>
    Formula:C22H13F4N9
    Color and Shape:Solid
    Molecular weight:479.39

    Ref: TM-T37686

  • LG 83-6-05
    Targetmol
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    LG 83-6-05

    CAS:
    <p>LG 83-6-05 is a novel kind of sodium channel blocking agent.</p>
    Formula:C21H30ClNO3S
    Color and Shape:Solid
    Molecular weight:411.99

    Ref: TM-T32731

  • TRPC5 modulator-1
    Targetmol
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    TRPC5 modulator-1

    CAS:
    <p>TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50&lt;1 nM) that can be used to study neuropsychiatric disorders.</p>
    Formula:C23H27FN2O4
    Color and Shape:Solid
    Molecular weight:414.47

    Ref: TM-T62133

  • ROMK-IN-32
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    ROMK-IN-32

    CAS:
    <p>ROMK-IN-32 is an inhibitor of the extra-renal medullary potassium channel (ROMK) (IC50: 35 nM) and also inhibits hERG (IC50: 22 μM).</p>
    Formula:C24H28N4O5
    Color and Shape:Solid
    Molecular weight:452.5

    Ref: TM-T62760

  • Dibutyryl-cGMP sodium
    Targetmol
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    Dibutyryl-cGMP sodium

    CAS:
    Bt2cGMP sodium is a cGMP analog, activates PKG, inhibits platelet [3H]-arachidonate, and induces analgesia via K+ channels.
    Formula:C18H24N5NaO9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.38

    Ref: TM-T11038

  • CGP-54626 free base
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    CGP-54626 free base

    CAS:
    CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).
    Formula:C18H28Cl2NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.3

    Ref: TM-T26998

  • GSK3395879
    Targetmol
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    GSK3395879

    CAS:
    <p>GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).</p>
    Formula:C20H15F4N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.41

    Ref: TM-T15439

  • SN40 hydrochloride
    Targetmol
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    SN40 hydrochloride

    CAS:
    <p>SN40 hydrochloride is a potent inhibitor of amino acid transport (AAT), exhibiting inhibitory constants (Kis) of 7.29 μM, 2.42 μM, 2.94 μM, 5.55 μM, 24.43 μM, and 5.55 μM for rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1, and EAAT5, respectively. It is utilized in cancer research. [1]</p>
    Formula:C18H21ClN2O2
    Color and Shape:Solid
    Molecular weight:332.82

    Ref: TM-T84754

  • AMPA-IN-1
    Targetmol
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    AMPA-IN-1

    CAS:
    <p>AMPA-IN-1: Potent AMPA receptor inhibitor; key in regulating brain excitatory transmission and plasticity.</p>
    Formula:C23H12F2N4O2
    Color and Shape:Solid
    Molecular weight:414.36

    Ref: TM-T62127

  • L-822179
    Targetmol
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    L-822179

    CAS:
    <p>L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.</p>
    Formula:C17H14N8O2
    Purity:98.5% - 99.61%
    Color and Shape:Solid
    Molecular weight:362.35

    Ref: TM-T24381

  • KCa1.1 channel activator-1
    Targetmol
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    KCa1.1 channel activator-1

    <p>A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.</p>
    Formula:C25H16O10
    Color and Shape:Solid
    Molecular weight:476.39

    Ref: TM-T72194

  • Afizagabar
    Targetmol
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    Afizagabar

    CAS:
    <p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>
    Formula:C19H12FN3O2S
    Color and Shape:Solid
    Molecular weight:365.38

    Ref: TM-T37388

  • JM-1232
    Targetmol
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    JM-1232

    CAS:
    <p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>
    Formula:C24H27N3O2
    Color and Shape:Solid
    Molecular weight:389.49

    Ref: TM-T24201

  • N-Linolenoylethanolamine
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    N-Linolenoylethanolamine

    CAS:
    <p>N-Linolenoylethanolamine (18:3 NAE), an endocannabinoid, functions as a vanillin receptor (TRPV1) agonist [1].</p>
    Formula:C20H35NO2
    Color and Shape:Solid
    Molecular weight:321.505

    Ref: TM-T84630

  • Antiarrhythmic agent-1
    Targetmol
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    Antiarrhythmic agent-1

    CAS:
    <p>Antiarrhythmic agent-1 (example I), functioning as an antiarrhythmic agent and an IKr potassium channel blocker (IC 50 &lt;1 μM), effectively inhibits cardiac</p>
    Formula:C25H27N3O4S
    Color and Shape:Solid
    Molecular weight:465.56

    Ref: TM-T72323

  • NMDA receptor modulator 4
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    NMDA receptor modulator 4

    CAS:
    <p>NMDA receptor modulator 4 (Compound 169) can be used for the research of neurological disorder that is a potent modulator of NMDA receptor [1].</p>
    Formula:C13H9F3N2O3S
    Color and Shape:Solid
    Molecular weight:330.28

    Ref: TM-T60960

  • Mesendogen
    Targetmol
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    Mesendogen

    CAS:
    <p>Mesendogen is an inhibitor of transient receptor potential cation channel, subfamily M, member 6 (TRPM6) and 7 (TRPM7) and acts by inhibiting TRPM6/TRPM7</p>
    Formula:C18H16ClF3N2OS
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:400.85

    Ref: TM-T28020

  • Biricodar
    Targetmol
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    Biricodar

    CAS:
    <p>Biricodar is a P-glycoprotein and MRP-1 modulator.</p>
    Formula:C34H41N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.71

    Ref: TM-T14616

  • Co 102862
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    Co 102862

    CAS:
    <p>Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant studies.</p>
    Formula:C14H12FN3O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:273.26

    Ref: TM-T22675

  • ADX71441
    Targetmol
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    ADX71441

    CAS:
    <p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events &amp; volume, and may aid in alcoholism and bladder pain.</p>
    Formula:C19H15ClF2N4O4
    Color and Shape:Solid
    Molecular weight:436.8

    Ref: TM-T26569

  • Cavα2δ1&NET-IN-3
    Targetmol
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    Cavα2δ1&NET-IN-3

    CAS:
    <p>Cavα2δ1&amp;NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET).</p>
    Formula:C24H30N6O2S
    Color and Shape:Solid
    Molecular weight:466.6

    Ref: TM-T72701

  • CymitQuimica logo
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    p-fin4

    CAS:
    p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.
    Formula:C39H53N8O18P
    Color and Shape:Solid
    Molecular weight:952.85

    Ref: TM-T76230

  • Adipiplon
    Targetmol
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    Adipiplon

    CAS:
    <p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>
    Formula:C18H18FN7
    Color and Shape:Solid
    Molecular weight:351.38

    Ref: TM-T29662

  • CGP 64213
    Targetmol
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    CGP 64213

    CAS:
    <p>CGP 64213 is a GABAb receptor agonist.</p>
    Formula:C26H36IN2O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:646.45

    Ref: TM-T26995

  • Etidocaine Hydrochloride
    Targetmol
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    Etidocaine Hydrochloride

    CAS:
    <p>Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.</p>
    Formula:C17H29ClN2O
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:312.88

    Ref: TM-T31716

  • VGSCs-IN-1
    Targetmol
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    VGSCs-IN-1

    CAS:
    <p>VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.</p>
    Formula:C12H12F3N3OS
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:303.3

    Ref: TM-T80626

  • L-DABA hydrobromide
    Targetmol
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    L-DABA hydrobromide

    CAS:
    <p>L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.</p>
    Formula:C4H11BrN2O2
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:199.05

    Ref: TM-T77795

  • Kv3 modulator 1
    Targetmol
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    Kv3 modulator 1

    CAS:
    <p>Kv3 modulator 1 is a voltage-gated potassium channel Kv3 modulator that can be used to study neurologic-level diseases.</p>
    Formula:C20H20N4O4
    Purity:99.41%
    Color and Shape:Solid
    Molecular weight:380.4

    Ref: TM-T11787

  • CE-224535
    Targetmol
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    CE-224535

    CAS:
    <p>CE-224535 (PF-04905428) is a selective antagonist of P2X7 receptor. CE-224535 can be used in disease-modifying antirheumatic studies.</p>
    Formula:C22H29ClN4O6
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:480.94

    Ref: TM-T14920

  • Maralixibat Chloride
    Targetmol
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    Maralixibat Chloride

    CAS:
    <p>Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation.</p>
    Formula:C40H56ClN3O4S
    Purity:99.19% - 99.65%
    Color and Shape:Solid
    Molecular weight:710.41

    Ref: TM-T32873

  • MCT1-IN-3
    Targetmol
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    MCT1-IN-3

    CAS:
    <p>MCT1-IN-3 is a monocarboxylate transporter 1 (MCT1) inhibitor.</p>
    Formula:C22H19N3O4
    Purity:99.35%
    Color and Shape:Soild
    Molecular weight:389.4

    Ref: TM-T67727

  • CFTR corrector 4
    Targetmol
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    CFTR corrector 4

    CAS:
    <p>Potent, oral CFTR corrector 4 targets cystic fibrosis, increasing cell surface CFTR levels.</p>
    Formula:C29H27F2NO7
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:539.52

    Ref: TM-T10776

  • LE135
    Targetmol
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    LE135

    CAS:
    <p>LE135: RARα/RARβ antagonist (Ki: 1.4 μM/220 nM), favors RARβ, selective vs RARγ/RXRs; also activates TRPV1/TRPA1 (EC50s: 2.5/20 μM).</p>
    Formula:C29H30N2O2
    Purity:97.94%
    Color and Shape:Solid
    Molecular weight:438.56

    Ref: TM-T22920

  • AMG-0347
    Targetmol
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    AMG-0347

    CAS:
    <p>AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.</p>
    Formula:C24H26F3N3O2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:445.48

    Ref: TM-T29968

  • Bupivacaine hydrochloride monohydrate
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    Bupivacaine hydrochloride monohydrate

    CAS:
    Bupivacaine hydrochloride monohydrate is an NMDA receptor inhibitor that inhibits SCN5A channels and is commonly used in the study of chronic pain.
    Formula:C18H31ClN2O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:342.9

    Ref: TM-T80641

  • Soraprazan
    Targetmol
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    Soraprazan

    CAS:
    BS3 Crosslinker (Bis(sulfosuccinimidyl)suberate) is an ADC linker that can be used to synthesize antibody-coupled active molecules.
    Formula:C21H25N3O3
    Purity:97.69% - 99.84%
    Color and Shape:Solid
    Molecular weight:367.44

    Ref: TM-T12977

  • EMD57033
    Targetmol
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    EMD57033

    CAS:
    <p>EMD57033 activates cardiac troponin C, enhances Ca2+ sensitivity to boost heart contraction.</p>
    Formula:C22H23N3O4S
    Purity:99.72% - >99.99%
    Color and Shape:Solid
    Molecular weight:425.5

    Ref: TM-T25372

  • C 101248
    Targetmol
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    C 101248

    CAS:
    <p>C 101248 (KCNK13-IN-1) is a selective and potent tandem pore halogen inhibitor of K+ channel 1 (THIK-1) inhibitor and a human and mouse KCNK13 inhibitor.</p>
    Formula:C15H12N6O
    Purity:99.14% - 99.31%
    Color and Shape:Solid
    Molecular weight:292.3

    Ref: TM-T83962

  • Funapide
    Targetmol
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    Funapide

    CAS:
    <p>Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.</p>
    Formula:C22H14F3NO5
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:429.35

    Ref: TM-T15358

  • Aneratrigine hydrochloride
    Targetmol
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    Aneratrigine hydrochloride

    CAS:
    <p>Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.</p>
    Formula:C19H21Cl2F2N5O2S2
    Purity:98.37% - 99.16%
    Color and Shape:Solid
    Molecular weight:524.43

    Ref: TM-T79835

  • Reldesemtiv
    Targetmol
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    Reldesemtiv

    CAS:
    <p>Reldesemtiv (CK-2127107) boosts exercise capacity, targeting fast muscle troponin, EC50 3.4 μM.</p>
    Formula:C19H18F2N6O
    Purity:97.27%
    Color and Shape:Solid
    Molecular weight:384.38

    Ref: TM-T16728

  • AMG2850
    Targetmol
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    AMG2850

    CAS:
    <p>AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).</p>
    Formula:C19H17F6N3O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:417.35

    Ref: TM-T10300

  • Metaphit methylsulfate
    Targetmol
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    Metaphit methylsulfate

    CAS:
    <p>Metaphit methylsulfate is a specific PCP antagonist and an acylating agent for the [3H] phencyclidine binding site in rat brain homogenate. It inhibits PCP-induced motor activity through a presynaptic mechanism.</p>
    Formula:C19H28N2O3S2
    Color and Shape:Solid
    Molecular weight:396.567

    Ref: TM-T204740

  • 3-Bromoamphetamine hydrochloride
    Targetmol
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    3-Bromoamphetamine hydrochloride

    CAS:
    <p>3-Bromoamphetamine hydrochloride is a para-substituted amphetamine that functions as a monoamine releaser.</p>
    Formula:C9H13BrClN
    Color and Shape:Solid
    Molecular weight:250.563

    Ref: TM-T206868

  • ML-SI1
    Targetmol
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    ML-SI1

    CAS:
    <p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>
    Formula:C23H26Cl2N2O3
    Color and Shape:Solid
    Molecular weight:449.37

    Ref: TM-T62692

  • CymitQuimica logo
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    URAT1 inhibitor 3

    <p>URAT1 inhibitor 3: potent oral URAT1 blocker, IC50=0.8 nM, for gout/hyperuricemia study.</p>
    Formula:C14H8Cl2N2O2
    Color and Shape:Solid
    Molecular weight:307.13

    Ref: TM-T60724

  • YY-23
    Targetmol
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    YY-23

    CAS:
    <p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>
    Formula:C33H54O8
    Color and Shape:Solid
    Molecular weight:578.777

    Ref: TM-T206120

  • PD-217014
    Targetmol
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    PD-217014

    CAS:
    <p>PD-217014 is an α2δ ligand that exhibits visceral analgesic activity and can suppress visceral hypersensitivity. Its antihyperalgesic effects are dose-dependent.</p>
    Formula:C10H17NO2
    Color and Shape:Solid
    Molecular weight:183.25

    Ref: TM-T200642

  • CymitQuimica logo
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    MRS4738

    <p>MRS4738 is a potent antagonist with high affinity for the P2Y14R receptor. It demonstrates in vivo anti-hyperallodynic and antiasthmatic activity [1].</p>
    Formula:C30H24F3NO2
    Color and Shape:Solid
    Molecular weight:487.51

    Ref: TM-T63242

  • ABCA1 inducer 2
    Targetmol
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    ABCA1 inducer 2

    CAS:
    <p>ABCA1 inducer 2 is a non-lipogenic inducer of ABCA1. It increases the expression of ABCA1 by targeting the LXR pathway, thereby reducing lipid accumulation induced by ox-LDL and inhibiting foam cell formation. ABCA1 inducer 2 holds potential as an anti-atherosclerotic agent.</p>
    Formula:C16H11BrN2O
    Color and Shape:Solid
    Molecular weight:327.175

    Ref: TM-T206113