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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2280 products of "Membrane Transporter/Ion Channel"

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  • LY 215490
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    LY 215490

    CAS:
    <p>LY 215490 is a selective AMPA receptor antagonist with neuroprotective properties in rat ischemia.</p>
    Formula:C13H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.34

    Ref: TM-T27897

  • SOAT-IN-1
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    SOAT-IN-1

    CAS:
    <p>SOAT-IN-1 (compound 40) is a potent and selective inhibitor targeting the sodium-dependent organic anion transporter (SOAT), exhibiting IC50 values of 1.6 µM for SOAT and 14.3 µM for NTCP.</p>
    Formula:C20H16ClN3O6S
    Color and Shape:Solid
    Molecular weight:461.88

    Ref: TM-T201002

  • Coleon-U-quinone
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    Coleon-U-quinone

    CAS:
    <p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>
    Formula:C20H24O5
    Color and Shape:Solid
    Molecular weight:344.4

    Ref: TM-T72735

  • TRPV1 antagonist 10
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    TRPV1 antagonist 10

    CAS:
    <p>TRPV1 antagonist 10 is a potent, orally active TRPV1 antagonist with an IC50 of 33.06 nM and serves as a moderate to weak inhibitor of URAT1 (IC50 = 22.51 μM) and GLUT9 (inhibition of 60.25% at 50 μM). It exhibits analgesic and urate-lowering properties and is applicable for research in hyperuricemia and inflammatory pain.</p>
    Formula:C16H14N2O5
    Color and Shape:Solid
    Molecular weight:314.293

    Ref: TM-T207037

  • CFTR corrector 16
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    CFTR corrector 16

    CAS:
    <p>CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), utilized in the research of cystic fibrosis disease.</p>
    Formula:C27H26ClN5O2S
    Color and Shape:Solid
    Molecular weight:520.05

    Ref: TM-T200113

  • Ro-51
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    Ro-51

    CAS:
    <p>dual P2X3 and P2X2/3 antagonist</p>
    Formula:C17H23IN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.29

    Ref: TM-T23245

  • Quinacainol dihydrochloride
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    Quinacainol dihydrochloride

    CAS:
    <p>Quinacainol dihydrochloride (PK 10139 dihydrochloride) is the bis(2 hydrochloride) salt form of Quinacainol. It acts as an inhibitor of the sodium current, with an EC50 of 95 µM. This compound displays antiarrhythmic activity by modulating the electrophysiological properties of the heart.</p>
    Formula:C21H32Cl2N2O
    Color and Shape:Solid
    Molecular weight:399.398

    Ref: TM-T204878

  • Butein tetramethyl ether
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    Butein tetramethyl ether

    CAS:
    <p>Butein tetramethyl ether (Compound 20) is a potent and selective inhibitor of breast cancer resistance protein / ATP-binding cassette sub-family G member 2 (BCRP/ABCG2). It inhibits MCF-7 MX and MDCKBCRP cells with IC50 values of 2.2 μM and 1.03 μM, respectively. Butein tetramethyl ether holds potential for cancer research.</p>
    Formula:C19H20O5
    Color and Shape:Solid
    Molecular weight:328.359

    Ref: TM-T204268

  • Olisutrigine bromide
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    Olisutrigine bromide

    CAS:
    <p>Olisutrigine bromide is a sodium channel blocker used as an analgesic.</p>
    Formula:C25H35BrN2
    Color and Shape:Solid
    Molecular weight:443.463

    Ref: TM-T205479

  • CymitQuimica logo
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    DAD dichloride

    <p>DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.</p>
    Formula:C26H42Cl2N6O
    Color and Shape:Solid
    Molecular weight:525.56

    Ref: TM-T63684

  • P-gp inhibitor 2
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    P-gp inhibitor 2

    CAS:
    <p>Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.</p>
    Formula:C29H26N2O6
    Color and Shape:Solid
    Molecular weight:498.53

    Ref: TM-T72739

  • ICA-105665
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    ICA-105665

    CAS:
    <p>ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.</p>
    Formula:C19H15F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.34

    Ref: TM-T11606

  • CymitQuimica logo
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    DAD

    <p>DAD is an ion channel blocker (blocks voltage-gated potassium channels) and is a third generation photoelectric switch that responds to visible light.</p>
    Formula:C26H40N6O
    Color and Shape:Solid
    Molecular weight:452.64

    Ref: TM-T62770

  • TRPA1 Antagonist 1
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    TRPA1 Antagonist 1

    CAS:
    <p>TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.</p>
    Formula:C24H20F6N5Na2O7PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:713.45

    Ref: TM-T13212

  • (RS)-AMPA hydrobromide
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    (RS)-AMPA hydrobromide

    CAS:
    AMPAR agonist
    Formula:C7H11BrN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.08

    Ref: TM-T23267

  • SR 33805 oxalate
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    SR 33805 oxalate

    CAS:
    <p>Ca2+ channel antagonist</p>
    Formula:C34H42N2O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.77

    Ref: TM-T23391

  • cis-KV1.3-IN-1
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    cis-KV1.3-IN-1

    CAS:
    <p>cis-KV1.3-IN-1, also known as Compound cis-18, is the cis-isomer of KV1.3-IN-1 and functions as an inhibitor of the KV1.3 channel. In Xenopus laevis oocytes expressing human hKV1.3, cis-KV1.3-IN-1 (10 μM) achieves an inhibition rate of 25.53% against KV1.3.</p>
    Formula:C23H30N2O4S
    Color and Shape:Solid
    Molecular weight:430.56

    Ref: TM-T201783

  • Dehydroindapamide
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    Dehydroindapamide

    CAS:
    <p>Dehydroindapamide, an indole form of Indapamide, is utilized to quantify the turnover rate of Indapamide in CYP3A4, which is approximately 10 times higher than that of Indoline, with slightly enhanced affinity for CYP3A4.</p>
    Formula:C16H14ClN3O3S
    Color and Shape:Solid
    Molecular weight:363.82

    Ref: TM-T200811

  • Cyazofamid
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    Cyazofamid

    CAS:
    <p>Cyazofamid functions as a fungicide by impairing the production of ATP. It inhibits Organic Cation Transporter 3 (OCT3) and OAT1 with IC50 values of 1.54 and 17.3 μM, respectively.</p>
    Formula:C13H13ClN4O2S
    Color and Shape:Solid
    Molecular weight:324.79

    Ref: TM-T201605

  • CFTR corrector 18
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    CFTR corrector 18

    CAS:
    <p>CFTRcorrector 18 (Compound I-99) acts as a modulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It enhances the processing and trafficking of CFTR, thereby increasing the amount of CFTR present on the cell surface. CFTRcorrector 18 holds potential for research in cystic fibrosis (CF).</p>
    Formula:C38H40N6O5S
    Color and Shape:Solid
    Molecular weight:692.826

    Ref: TM-T206874