Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
DMCM hydrochloride
CAS:1215833-62-7
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.
Formula:
C17H19ClN2O4
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T11061
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 650.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Sarmazenil
CAS:78771-13-8
Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used …
Formula:
C15H14ClN3O3
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
319.74
Ref: TM-T16844
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
TWIK-1/TREK-1-IN-1
CAS:1440532-30-8
Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain …
Formula:
C21H24F3NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
395.42
Ref: TM-T78868
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
TWIK-1/TREK-1-IN-3
CAS:1440532-33-1
TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used …
Formula:
C19H27F3N2O2
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
372.43
Ref: TM-T78870
| 1mg | 86.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 509.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 984.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
UK 66914
CAS:113049-11-9
UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.
Formula:
C18H24N4O3S
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
376.47
Ref: TM-T29050
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
NC-1300-B
CAS:104340-52-5
NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.
Formula:
C17H19N3OS
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
313.42
Ref: TM-T28136
| 1mg | 276.00 € | ||
| 5mg | 680.00 € | ||
| 10mg | 930.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Riluzole hydrochloride
CAS:850608-87-6
Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).
Formula:
C8H6ClF3N2OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
270.66
Ref: TM-T41265
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GX-585
CAS:2098540-08-8
GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited …
Formula:
C24H25Cl2FN4O3S
Purity:
100% - 99.18%
Color and Shape:
Liquid
Molecular weight:
539.45
Ref: TM-T69915
| 1mg | 274.00 € | ||
| 5mg | 666.00 € | ||
| 10mg | 914.00 € | ||
| 25mg | 1,379.00 € | ||
| 50mg | 1,869.00 € | ||
| 100mg | 2,545.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
XE991
CAS:122955-42-4
XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and …
Formula:
C26H20N2O
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
376.45
Ref: TM-T78570
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 824.00 € | ||
| 500mg | 1,651.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ABCG2-IN-2
CAS:2559759-59-8
ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and …
Formula:
C25H34N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
454.56
Ref: TM-T79514
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
TRPM4-IN-2
CAS:667411-04-3
NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in …
Formula:
C19H14ClNO4
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
355.77
Ref: TM-T61275
| 2mg | To inquire |
Estimated delivery in United States, on Thursday 16 Jan 2025
TWIK-1/TREK-1-IN-2
CAS:1440532-32-0
TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 …
Formula:
C20H29F3N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.45
Ref: TM-T78869
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Lirequinil
CAS:143943-73-1
Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.
Formula:
C26H25ClN2O3
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
448.94
Ref: TM-T27838
| 1mg | 155.00 € | ||
| 5mg | 372.00 € | ||
| 10mg | 561.00 € | ||
| 25mg | 891.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,635.00 € | ||
| 500mg | 3,240.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
RO 4938581
CAS:883093-10-5
RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, …
Formula:
C13H8BrF2N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T16794
| 25mg | 1,141.00 € | ||
| 50mg | 1,499.00 € | ||
| 100mg | 2,468.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
E2730
CAS:1520073-91-9
E2730 is a selective and noncompetitive inhibitor of the gamma-aminobutyric acid (GABA) transporter 1 (GAT1) …
Formula:
C9H8F4N2O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
284.23
Ref: TM-T79399
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
KT-362 fumarate
CAS:105394-80-7
KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes …
Formula:
C26H32N2O7S
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
516.61
Ref: TM-T27753
| 1mg | 300.00 € | ||
| 5mg | 694.00 € | ||
| 10mg | 981.00 € | ||
| 25mg | 1,449.00 € | ||
| 50mg | 1,930.00 € | ||
| 100mg | 2,627.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
JYL 1421
CAS:401907-26-4
JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).
Formula:
C20H26FN3O2S2
Color and Shape:
Solid
Molecular weight:
423.57
Ref: TM-T15634
| 25mg | 710.00 € | ||
| 50mg | 934.00 € | ||
| 100mg | 1,470.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ABCG2-IN-1
CAS:2559759-40-7
ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with …
Formula:
C26H36N4O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
468.59
Ref: TM-T79513
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
CBS9106
CAS:1076235-04-5
CBS9106 (SL-801) is a CRM1 inhibitor with CRM1-degrading and anti-tumor activity that inhibits CRM1-dependent nuclear …
Formula:
C18H21ClF3N3O3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
419.83
Ref: TM-T14885
| 1mg | 247.00 € | ||
| 5mg | 605.00 € | ||
| 10mg | 836.00 € | ||
| 25mg | 1,293.00 € | ||
| 50mg | 1,761.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
