Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Read more
Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
PF 05089771 tosylate
CAS:1430806-04-4
PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x …
Formula:
C18H12Cl2FN5O3S2·C7H8O3S
Purity:
97.76%
Color and Shape:
Solid
Molecular weight:
672.56
Ref: TM-T7502
| 1mg | 62.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 381.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
DFP00173
CAS:672286-03-2
DFP00173: Potent, selective AQP3 inhibitor; IC50 ~0.1-0.4 μM; less effective on AQP7, AQP9.
Formula:
C11H7Cl2N3O3S
Purity:
99.15% - 99.55%
Color and Shape:
Solid
Molecular weight:
332.16
Ref: TM-T11014
| 1mg | 75.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 765.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 177.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
SCH-23390 maleate
CAS:87134-87-0
SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 …
Formula:
C21H22ClNO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
403.86
Ref: TM-T12865
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Ru-32514
CAS:90807-98-0
Ru-32514 is a benzodiazepine receptor agonist.
Formula:
C18H17N3O2
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T12779
| 1mg | 274.00 € | ||
| 2mg | 408.00 € | ||
| 5mg | 675.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
TRPV4 agonist-1
CAS:2314467-60-0
TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).
Formula:
C25H23ClF2N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
484.93
Ref: TM-T13214
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
MSP3
CAS:1820968-63-5
MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective …
Formula:
C16H19NO3S
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
305.39
Ref: TM-T28118
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Golexanolone
CAS:2089238-18-4
Golexanolone can be used to study neurological diseases.
Formula:
C21H31NO2
Purity:
98.81% - 99.98%
Color and Shape:
Solid
Molecular weight:
329.48
Ref: TM-T25458
| 1mg | 273.00 € | ||
| 5mg | 672.00 € | ||
| 10mg | 918.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
HC-070
CAS:1628291-95-1
HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).
Formula:
C22H20Cl2N4O4
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
475.32
Ref: TM-T15465
| 1mg | 131.00 € | ||
| 5mg | 271.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 707.00 € | ||
| 50mg | 994.00 € | ||
| 100mg | 1,341.00 € | ||
| 200mg | 1,052.00 € | ||
| 1mL*10mM (DMSO) | 277.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Abeprazan hydrochloride
CAS:1902954-87-3
Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting …
Formula:
C19H18ClF3N2O3S
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
446.87
Ref: TM-T10221
| 1mg | 91.00 € | ||
| 5mg | 221.00 € | ||
| 10mg | 328.00 € | ||
| 25mg | 527.00 € | ||
| 50mg | 713.00 € | ||
| 100mg | 917.00 € | ||
| 500mg | 1,838.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
CyPPA
CAS:73029-73-9
CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.
Formula:
C16H23N5
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
285.39
Ref: TM-T20968
| 2mg | 43.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 458.00 € | ||
| 500mg | 1,009.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
RL648_81
CAS:1919050-87-5
RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be …
Formula:
C17H17F4N3O2
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
371.33
Ref: TM-T28544
| 2mg | 43.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 467.00 € | ||
| 200mg | 633.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
WY-47766
CAS:134217-27-9
WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.
Formula:
C14H13N3O2S
Purity:
98.11% - 99.75%
Color and Shape:
Solid
Molecular weight:
287.34
Ref: TM-T29164
| 1mg | 275.00 € | ||
| 5mg | 676.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,572.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
NS-2710
CAS:184220-36-8
NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.
Formula:
C22H20N4O
Purity:
98.10% - 99.82%
Color and Shape:
Solid
Molecular weight:
356.42
Ref: TM-T28197
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
FR-167356
CAS:174185-16-1
FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone …
Formula:
C19H17Cl2NO3
Purity:
98.44% - 99.19%
Color and Shape:
Solid
Molecular weight:
378.25
Ref: TM-T27371
| 1mg | 184.00 € | ||
| 5mg | 445.00 € | ||
| 10mg | 609.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,238.00 € | ||
| 100mg | 1,629.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
E 0747
CAS:99599-78-7
E 0747 is an antiarrhythmic agent of class 1C type. E-0747 suppresses arrhythmia by inhibiting …
Formula:
C21H28ClN3O4
Purity:
95.01%
Color and Shape:
Solid
Molecular weight:
421.92
Ref: TM-T24021
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 671.00 € | ||
| 10mg | 917.00 € | ||
| 25mg | 1,410.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Mavatrep
CAS:956274-94-5
Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can …
Formula:
C25H21F3N2O
Purity:
98.01% - 98.38%
Color and Shape:
Solid
Molecular weight:
422.44
Ref: TM-T16014
| 1mg | 65.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 449.00 € | ||
| 50mg | 724.00 € | ||
| 100mg | 1,154.00 € | ||
| 200mg | 897.00 € | ||
| 500mg | 2,312.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
UK 78282 hydrochloride
CAS:136647-02-4
UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T …
Formula:
C29H36ClNO2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
466.05
Ref: TM-T23497
| 1mg | 91.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 325.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,019.00 € | ||
| 500mg | 2,083.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Puliginurad
CAS:2013582-27-7
Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad …
Formula:
C19H16N2O2S
Purity:
99.96% - 99.96%
Color and Shape:
Liquid
Molecular weight:
336.41
Ref: TM-T61048
| 1mg | 66.00 € | ||
| 5mg | 142.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ZTZ240
CAS:325457-98-5
ZTZ240 is a KCNQ2 channel activator used in the study of epilepsy.
Formula:
C12H8ClFN2O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
250.66
Ref: TM-T29236
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
