Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(101 products)
- Adiponectin receptor(5 products)
- CFTR(65 products)
- CGRP Receptor(54 products)
- Calcium Channel(541 products)
- Chloride channel(53 products)
- GABA Receptor(365 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(54 products)
- Potassium Channel(280 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(209 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2512 products of "Membrane Transporter/Ion Channel"
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ML277
CAS:ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).Formula:C23H25N3O4S2Purity:99.35%Color and Shape:SolidMolecular weight:471.59Indecainide hydrochloride
CAS:Indecainide hydrochloride is a cardiac depressant.Formula:C20H25ClN2OColor and Shape:SolidMolecular weight:344.88CX614
CAS:CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.Formula:C13H13NO4Purity:97.37%Color and Shape:SolidMolecular weight:247.25Ref: TM-T19698
5mg55.00€10mg82.00€25mg126.00€50mg182.00€100mg273.00€200mg409.00€1mL*10mM (DMSO)58.00€TC-I2000
CAS:TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.Formula:C23H18F4N2OPurity:99.778%Color and Shape:SolidMolecular weight:414.4Ref: TM-T8449
5mg35.00€10mg50.00€25mg88.00€50mg119.00€100mg173.00€200mg259.00€1mL*10mM (DMSO)To inquireVU590 HCl
CAS:VU590 is a small molecule inhibitor of KCNJ1 (IC50 = 294 nM).Formula:C24H34Cl2N4O7Color and Shape:SolidMolecular weight:561.457PF-01247324
CAS:PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).Formula:C13H10Cl3N3OPurity:99.22%Color and Shape:SolidMolecular weight:330.6IDRA-21
CAS:IDRA-21 is a positive AMPA receptor modulator.Formula:C8H9ClN2O2SPurity:99.73%Color and Shape:SolidMolecular weight:232.69(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37Nisoxetine
CAS:Nisoxetine is a selective NET (noradrenaline transporter) inhibitor (Kd=0.76 nM) capable of blocking voltage-gated sodium channels.Formula:C17H21NO2Purity:98.71%Color and Shape:SolidMolecular weight:271.35cim0216
CAS:CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.Formula:C21H21N3O2Purity:99.87%Color and Shape:SolidMolecular weight:347.41Ref: TM-T9263
1mg47.00€2mg59.00€5mg92.00€10mg145.00€25mg298.00€50mg465.00€100mg702.00€500mg1,454.00€1mL*10mM (DMSO)92.00€VX-150
CAS:VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).Formula:C21H17F4N2O7PPurity:97.58%Color and Shape:SolidMolecular weight:516.34Ref: TM-T9683
1mg66.00€5mg144.00€10mg235.00€25mg472.00€50mg755.00€100mg1,206.00€1mL*10mM (DMSO)164.00€Delucemine Free Base
CAS:Delucemine Free Base is an NMDA Receptor AntagonistFormula:C16H17F2NColor and Shape:SolidMolecular weight:261.31Pyr10
CAS:Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.Formula:C18H13F6N3O2SPurity:99.69% - 99.7%Color and Shape:SolidMolecular weight:449.37Zosuquidar
CAS:Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.Formula:C32H31F2N3O2Purity:99.99%Color and Shape:SolidMolecular weight:527.6Ref: TM-T6018L
1mg78.00€5mg160.00€10mg233.00€25mg378.00€50mg567.00€100mg825.00€200mg1,130.00€1mL*10mM (DMSO)180.00€Sematilide hydrochloride
CAS:Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker.Formula:C14H24ClN3O3SPurity:99.14%Color and Shape:SolidMolecular weight:349.87α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:97.02% - 98.41%Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Molecular weight:152.23Benzamil
CAS:Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.75BRITE-338733
CAS:BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.Formula:C27H35N3O2Purity:99.85%Color and Shape:SolidMolecular weight:433.59Ref: TM-T22280
1mg46.00€2mg63.00€5mg97.00€10mg169.00€25mg329.00€50mg465.00€100mg655.00€200mg883.00€1mL*10mM (DMSO)105.00€CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurity:98.75%Color and Shape:SolidMolecular weight:384.24Benzocaine xHCl(94-09-7(free base))
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).Formula:C9H11NO2·xHClPurity:99.37%Color and Shape:SolidMolecular weight:N/A
