Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(101 products)
- Adiponectin receptor(5 products)
- CFTR(65 products)
- CGRP Receptor(54 products)
- Calcium Channel(541 products)
- Chloride channel(53 products)
- GABA Receptor(365 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(54 products)
- Potassium Channel(280 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(209 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2512 products of "Membrane Transporter/Ion Channel"
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Benzamil
CAS:Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.75BRITE-338733
CAS:BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.Formula:C27H35N3O2Purity:99.85%Color and Shape:SolidMolecular weight:433.59Ref: TM-T22280
1mg46.00€2mg63.00€5mg97.00€10mg169.00€25mg329.00€50mg465.00€100mg655.00€200mg883.00€1mL*10mM (DMSO)105.00€Dofetilide
CAS:Dofetilide (UK 68789), a class III antiarrhythmic sulfonamide, blocks Ikr cardiac channels, prolongs action potential, and treats atrial fibrillation/flutter.Formula:C19H27N3O5S2Purity:97.85% - 99.06%Color and Shape:Off-White Or Yellowish Crystalline PowderMolecular weight:441.56Ref: TM-T6476
2mgTo inquire5mg52.00€10mg69.00€25mg114.00€50mg170.00€100mg246.00€200mg366.00€1mL*10mM (DMSO)55.00€Benzocaine xHCl(94-09-7(free base))
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).Formula:C9H11NO2·xHClPurity:99.37%Color and Shape:SolidMolecular weight:N/AEsomeprazole Sodium
CAS:Esomeprazole Sodium ((S)-Omeprazole sodium) is the S-isomer of omeprazole with selective and irreversible proton pump inhibitor activity.Formula:C17H18N3O3S·NaPurity:98.17% - >99.99%Color and Shape:SolidMolecular weight:367.4Elobixibat hydrate
CAS:Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.Formula:C36H47N3O8S2Color and Shape:SolidMolecular weight:713.9Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formula:C41H72O2Purity:99.65%Color and Shape:SolidMolecular weight:597.01AZD-9056 free base
CAS:AZD9056 is a potent, selective, orally bioavailable P2X7 receptor antagonist.Formula:C24H35ClN2O2Color and Shape:SolidMolecular weight:419Sematilide hydrochloride
CAS:Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker.Formula:C14H24ClN3O3SPurity:99.14%Color and Shape:SolidMolecular weight:349.87Lumacaftor
CAS:Lumacaftor (VRT 826809) is a CFTR modulator that corrects the folding and trafficking of CFTR protein.Formula:C24H18F2N2O5Purity:99.48% - 99.68%Color and Shape:SolidMolecular weight:452.41Zosuquidar
CAS:Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.Formula:C32H31F2N3O2Purity:99.99%Color and Shape:SolidMolecular weight:527.6Ref: TM-T6018L
1mg78.00€5mg160.00€10mg233.00€25mg378.00€50mg567.00€100mg825.00€200mg1,130.00€1mL*10mM (DMSO)180.00€DQP 1105
CAS:<p>DQP 1105 is a NMDA receptor antagonist.</p>Formula:C29H24BrN3O4Purity:98.6%Color and Shape:SolidMolecular weight:558.42Tiludronate
CAS:Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.Formula:C7H9ClO6P2SColor and Shape:SolidMolecular weight:318.61TCN 201
CAS:TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.Formula:C21H17ClFN3O4SPurity:98.5%Color and Shape:SolidMolecular weight:461.89Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Color and Shape:SolidMolecular weight:86.14Drotaverine hydrochloride
CAS:Drotaverine hydrochloride is a type 4 cyclic nucleotide phosphodiesterase (PDE4) inhibitor，and is an antispasmodic drug, used to enhance cervical dilationFormula:C24H32ClNO4Purity:99.81%Color and Shape:Pale-Yellow Crystalline SolidMolecular weight:433.968Levcromakalim
CAS:Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.Formula:C16H18N2O3Purity:99.74%Color and Shape:SolidMolecular weight:286.33Ref: TM-TQ0150
1mg52.00€2mg78.00€5mg99.00€10mg150.00€25mg335.00€50mg499.00€100mg722.00€1mL*10mM (DMSO)110.00€Felbamate
CAS:Felbamate (W-554) is an Anti-epileptic Agent.Formula:C11H14N2O4Purity:99% - >99.99%Color and Shape:White Powder SolidMolecular weight:238.24ML213
CAS:ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,Formula:C17H23NOPurity:>99.99%Color and Shape:SolidMolecular weight:257.37Amifampridine phosphate
CAS:Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.Formula:C5H10N3O4PColor and Shape:SolidMolecular weight:207.12
