GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 371 products of "GABA Receptor"
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Primidone (Standard)
CAS:Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Formula:C12H14N2O2Color and Shape:Crystals (Ntp 1992)Molecular weight:218.25Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formula:C6H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:165.62CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColor and Shape:SolidMolecular weight:179.2MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formula:C17H20N8O2Purity:99.76%Color and Shape:SolidMolecular weight:368.39L-655708
CAS:L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Formula:C18H19N3O4Purity:99.36%Color and Shape:PowderMolecular weight:341.36Furosemide-d5
CAS:Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.Formula:C12H11ClN2O5SColor and Shape:SolidMolecular weight:335.78(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purity:98% - 99.93%Color and Shape:White Odorless Or Nearly Odorless PowderMolecular weight:400.48Acetoxyvalerensre
CAS:Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.
Formula:C17H24O4Purity:98.22%Color and Shape:SolidMolecular weight:292.37Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Formula:C24H46N6O14Purity:99.8%Color and Shape:Crystals IndicationMolecular weight:642.65AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
Formula:C19H19FN4O2Purity:99.83%Color and Shape:SolidMolecular weight:354.38Ginkgolide A
CAS:Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Formula:C20H24O9Purity:98.76% - 99.81%Color and Shape:White PowderMolecular weight:408.40Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Formula:C6H10ClNO2Purity:98.42%Color and Shape:SolidMolecular weight:163.602CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formula:C13H9F3N4Purity:99.92%Color and Shape:SolidMolecular weight:278.23Pipequaline hydrochloride
CAS:Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formula:C22H25ClN2Purity:99.46%Color and Shape:SolidMolecular weight:352.9Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:177.63Ref: TM-T5799
2mg34.00€5mg48.00€10mg67.00€25mg100.00€50mg149.00€100mg213.00€200mg316.00€1mL*10mM (DMSO)49.00€(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formula:C10H12ClNO2Purity:97.20% - 98.94%Color and Shape:SolidMolecular weight:213.66Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.3L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormula:C14H14O3Purity:99.93% - ≥95%Color and Shape:SolidMolecular weight:230.26Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:357.49AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purity:98.99%Color and Shape:SolidMolecular weight:366.41Ref: TM-T7136
1mg215.00€5mg439.00€10mg640.00€25mg1,018.00€50mg1,423.00€100mg1,935.00€1mL*10mM (DMSO)484.00€Cholesterol myristate
CAS:Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.
Formula:C41H72O2Purity:99.65%Color and Shape:SolidMolecular weight:597.01α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:97.02% - 98.41%Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Molecular weight:152.23Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purity:99.8%Color and Shape:SolidMolecular weight:198.226-Aminonicotinic acid
CAS:6-Aminonicotinic acid is a natural product.
Formula:C6H6N2O2Purity:99.94%Color and Shape:SoildMolecular weight:138.1238rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formula:C17H21F3O3Purity:99.69% - >99.99%Color and Shape:SolidMolecular weight:330.34Ref: TM-T4176
2mg43.00€5mg60.00€10mg96.00€25mg187.00€50mg311.00€100mg472.00€200mg657.00€1mL*10mM (DMSO)71.00€α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purity:99.64% - 99.64%Color and Shape:Monoclinic Needles From Water Monoclinic Needles From WaterMolecular weight:208.25Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurity:97.21%Color and Shape:Solid PowderMolecular weight:437.15Thiocolchicoside
CAS:Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.Formula:C27H33NO10SPurity:99.11% - 99.39%Color and Shape:SolidMolecular weight:563.62γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.143Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurity:99.09% - 99.77%Color and Shape:White To Off-White SolidMolecular weight:412.01Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formula:C15H17N3O3Color and Shape:SolidMolecular weight:287.31Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formula:C20H15FN4O2SPurity:99.12% - 99.19%Color and Shape:SolidMolecular weight:394.42Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Color and Shape:SolidMolecular weight:310.99Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.022'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purity:99.28% - 99.63%Color and Shape:SolidMolecular weight:266.29Ref: TM-T8887
1mg49.00€5mg102.00€10mg152.00€25mg243.00€50mg340.00€100mg460.00€200mg627.00€1mL*10mM (DMSO)96.00€Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Color and Shape:SolidMolecular weight:86.14Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.26(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purity:99.58% - 99.87%Color and Shape:SolidMolecular weight:217.26Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Formula:C6H11NO2Purity:99.82%Color and Shape:White To Faint Pink-Beige PowderMolecular weight:129.16SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormula:C22H26ClNO2Purity:98.02%Color and Shape:SolidMolecular weight:371.9Ref: TM-T12930
1mg34.00€5mg65.00€10mg89.00€25mg167.00€50mg264.00€100mg409.00€200mg590.00€1mL*10mM (DMSO)71.00€Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purity:99.93%Color and Shape:White Crystalline PowderMolecular weight:215.684-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formula:C6H11NO3Purity:98.51%Color and Shape:SolidMolecular weight:145.16CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurity:98.75%Color and Shape:SolidMolecular weight:384.24(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24Imidazenil
CAS:Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.Formula:C18H12BrFN4OPurity:98.4%Color and Shape:SolidMolecular weight:399.22Isoflurane
CAS:Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.Formula:C3H2ClF5OPurity:98%Color and Shape:Clear Colorless Liquid LiquidMolecular weight:184.49Cyclothiazide
CAS:Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Formula:C14H16ClN3O4S2Purity:98.23% - 99.49%Color and Shape:Crystals From Dilute Alcohol SolidMolecular weight:389.88SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurity:99.03% - 99.95%Color and Shape:SolidMolecular weight:387.83Ref: TM-T4522
2mg34.00€5mg50.00€10mg75.00€25mg111.00€50mg172.00€100mg290.00€200mg419.00€1mL*10mM (DMSO)46.00€p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purity:99.05% - 99.86%Color and Shape:SolidMolecular weight:122.12Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurity:98.03%Color and Shape:Light Beige Crystalline PowderMolecular weight:109.3Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purity:98.21% - 99.22%Color and Shape:Odourless Whitish SolidMolecular weight:538.46Ref: TM-T3417
2mg34.00€5mg50.00€10mg80.00€25mg126.00€50mg215.00€100mg349.00€200mg512.00€1mL*10mM (DMSO)59.00€Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purity:99.25% - 99.67%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formula:C6H9ClN2O2Purity:99.39%Molecular weight:176.601SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Color and Shape:SolidMolecular weight:335.44Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purity:98.51% - 99.24%Color and Shape:SolidMolecular weight:368.236-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurity:99.03%Color and Shape:SolidMolecular weight:201.22L-838417 D9
CAS:L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formula:C19H10D9F2N7OPurity:99.65%Color and Shape:SolidMolecular weight:408.45Ref: TM-T22301
2mg34.00€5mg52.00€10mg71.00€25mg128.00€50mg200.00€100mg323.00€200mg447.00€1mL*10mM (DMSO)58.00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:99.55%Color and Shape:SolidMolecular weight:250.1226-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurity:99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurity:99.17%Color and Shape:White Crystalline SolidMolecular weight:249.71Ref: TM-T4440
1mg52.00€5mg113.00€10mg177.00€25mg340.00€50mg550.00€100mg860.00€200mg1,161.00€1mL*10mM (DMSO)108.00€Imepitoin
CAS:Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Formula:C13H14ClN3O2Purity:99.82%Color and Shape:SolidMolecular weight:279.72U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purity:99.72% - 99.99%Color and Shape:Solid PowderMolecular weight:556.29Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
Formula:C53H90O22Purity:98.83% - 99.56%Color and Shape:White PowderMolecular weight:1079.27NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurity:99.44% - 99.86%Color and Shape:SolidMolecular weight:353.42Ref: TM-T2067
2mg34.00€5mg50.00€10mg80.00€25mg131.00€50mg212.00€100mg321.00€200mg460.00€1mL*10mM (DMSO)58.00€ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formula:C21H21FN6Purity:99.43%Color and Shape:SolidMolecular weight:376.43Ref: TM-TQ0040
1mg57.00€5mg119.00€10mg166.00€25mg356.00€50mg532.00€100mg760.00€1mL*10mM (DMSO)133.00€Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purity:98% - >99.99%Color and Shape:SolidMolecular weight:1207.35Suritozole
CAS:Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptorFormula:C10H10FN3SPurity:99.25%Color and Shape:SolidMolecular weight:223.27Ref: TM-T8568
1mg58.00€5mg116.00€10mg172.00€25mg281.00€50mg396.00€100mg537.00€200mg712.00€1mL*10mM (DMSO)104.00€Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFormula:C21H20FN3O5SPurity:99.21% - 99.42%Color and Shape:SolidMolecular weight:445.46Ref: TM-T7165
2mg35.00€5mg52.00€10mg74.00€25mg116.00€50mg187.00€100mg356.00€500mg802.00€1mL*10mM (DMSO)49.00€Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:423.53Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Formula:C20H17NO6Purity:98% - 99.99%Color and Shape:Light Yellow PowderMolecular weight:367.35Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Formula:C10H6Cl3N3Purity:99.78%Color and Shape:SolidMolecular weight:274.53Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formula:C16H14FN3OPurity:99.72%Color and Shape:SolidMolecular weight:283.3Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurity:98.42% - 99.29%Color and Shape:SolidMolecular weight:440.49Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.
Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:PowderMolecular weight:234.2GABAA receptor agent 5
CAS:Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.Formula:C21H25N3O2SPurity:99.39%Color and Shape:SolidMolecular weight:383.51ABP-700
CAS:ABP-700 is a positive allosteric modulator of the GABAA receptor.Formula:C17H18N2O4Purity:98%Color and Shape:SolidMolecular weight:314.34RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Formula:C13H8BrF2N5Purity:98%Color and Shape:SolidMolecular weight:352.14DAA-1097
CAS:DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Formula:C24H24ClNO3Purity:98%Color and Shape:SolidMolecular weight:409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:group I metabotropic glutamate receptor antagonist and group II mGlu agonistFormula:C9H9NO5Purity:98%Color and Shape:SolidMolecular weight:211.17BGT1-IN-9
CAS:BGT1-IN-9 is an M1 muscarinic agonist.Formula:C5H10ClN3O2Color and Shape:SolidMolecular weight:179.605PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purity:98%Color and Shape:SolidMolecular weight:358.87CGP 46381
CAS:CGP 46381 is a GABAB receptor antagonist.Formula:C10H22NO2PPurity:98%Color and Shape:White SolidMolecular weight:219.26PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formula:C14H22OPurity:98%Color and Shape:SolidMolecular weight:206.32GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormula:C15H23N5O2SPurity:99.92%Color and Shape:SolidMolecular weight:337.44Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Formula:C24H21ClN2O3Purity:98%Color and Shape:SolidMolecular weight:420.89SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formula:C8H15NO3Purity:98%Color and Shape:SolidMolecular weight:173.21Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purity:98.61%Color and Shape:SolidMolecular weight:337.33Ref: TM-T23445
1mg64.00€2mg96.00€5mg115.00€10mg150.00€25mg330.00€50mg472.00€100mg655.00€500mg1,293.00€CP-409092 hydrochloride
CAS:CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.Formula:C17H20ClN3O2Color and Shape:SolidMolecular weight:333.81Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formula:C20H18BrClN4SColor and Shape:SolidMolecular weight:461.81Arbaclofen placarbil
CAS:Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Formula:C19H26ClNO6Color and Shape:SolidMolecular weight:399.87SH-053-S-CH3-2'F
CAS:SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Formula:C23H18FN3O2Color and Shape:SolidMolecular weight:387.41Ethyl dirazepate
CAS:Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Formula:C18H14Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:377.22
