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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

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  • Fluralaner

    CAS:
    <p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>
    Formula:C22H17Cl2F6N3O3
    Purity:99.72% - 99.90%
    Color and Shape:Solid Powder
    Molecular weight:556.29
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Formula:C4H10N2O2
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:118.13
  • ONO-8590580

    CAS:
    <p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>
    Formula:C21H21FN6
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:376.43
  • Kavain

    CAS:
    <p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>
    Formula:C14H14O3
    Purity:99.93% - ≥95%
    Color and Shape:Solid
    Molecular weight:230.26
  • Isoflurane

    CAS:
    <p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>
    Formula:C3H2ClF5O
    Purity:98%
    Color and Shape:Clear Colorless Liquid Liquid
    Molecular weight:184.49
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Formula:C53H90O22
    Purity:98.83% - 99.56%
    Color and Shape:White Powder
    Molecular weight:1079.27
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Formula:C16H14O4
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:270.28
  • NS11394

    CAS:
    <p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) &gt; α(3) &gt; α(2) &gt; α(</p>
    Formula:C23H19N3O
    Purity:99.44% - 99.86%
    Color and Shape:Solid
    Molecular weight:353.42
  • Afloqualone

    CAS:
    <p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>
    Formula:C16H14FN3O
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:283.3
  • Songorine

    CAS:
    <p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>
    Formula:C22H31NO3
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:357.49
  • Pikamilone

    CAS:
    <p>Pikamilone (Picamilon) is an intelligent medicine.</p>
    Formula:C10H12N2O3
    Purity:99.38%
    Color and Shape:White Crystalline Powder
    Molecular weight:208.21
  • AZD-6280

    CAS:
    <p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>
    Formula:C20H22N4O3
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:366.41
  • (-)-Securinine

    CAS:
    <p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>
    Formula:C13H15NO2
    Purity:99.58% - 99.87%
    Color and Shape:Solid
    Molecular weight:217.26
  • Thiocolchicoside

    CAS:
    <p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>
    Formula:C27H33NO10S
    Purity:99.11% - 99.39%
    Color and Shape:Solid
    Molecular weight:563.62
  • Loreclezole

    CAS:
    <p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>
    Formula:C10H6Cl3N3
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:274.53
  • Bicuculline

    CAS:
    <p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>
    Formula:C20H17NO6
    Purity:98% - 99.99%
    Color and Shape:Light Yellow Powder
    Molecular weight:367.35
  • Baclofen hydrochloride

    CAS:
    <p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>
    Formula:C10H13Cl2NO2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:250.122
  • γ-Acetylenic GABA

    CAS:
    <p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>
    Formula:C6H9NO2
    Color and Shape:Solid
    Molecular weight:127.143
  • Tiagabine hydrochloride

    CAS:
    <p>Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.</p>
    Formula:C20H25NO2S2·HCl
    Purity:99.09% - 99.77%
    Color and Shape:White To Off-White Solid
    Molecular weight:412.01
  • Dihydroergotoxine mesylate

    CAS:
    <p>Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.</p>
    Formula:C20H29N3O5S
    Purity:99.39% - ≥95%
    Color and Shape:Solid
    Molecular weight:423.53
  • 6-Methylflavone

    CAS:
    <p>6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.</p>
    Formula:C16H12O2
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:236.27
  • Basmisanil

    CAS:
    <p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>
    Formula:C21H20FN3O5S
    Purity:99.21% - 99.42%
    Color and Shape:Solid
    Molecular weight:445.46
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Formula:C15H17N3O3
    Color and Shape:Solid
    Molecular weight:287.31
  • rac-BHFF

    CAS:
    <p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency &gt;15x, efficacy &gt;149%, has anxiolytic effects, and is orally active.</p>
    Formula:C17H21F3O3
    Purity:99.69% - >99.99%
    Color and Shape:Solid
    Molecular weight:330.34
  • Acamprosate calcium

    CAS:
    <p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>
    Formula:C10H20CaN2O8S2
    Purity:98% - 99.93%
    Color and Shape:White Odorless Or Nearly Odorless Powder
    Molecular weight:400.48
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Formula:C6H6N2O2
    Purity:99.94%
    Color and Shape:Soild
    Molecular weight:138.1238
  • DL-Menthol

    CAS:
    <p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>
    Formula:C10H20O
    Purity:99.74%
    Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)
    Molecular weight:156.27
  • Lorediplon

    CAS:
    <p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>
    Formula:C20H15FN4O2S
    Purity:99.12% - 99.19%
    Color and Shape:Solid
    Molecular weight:394.42
  • Suritozole

    CAS:
    <p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>
    Formula:C10H10FN3S
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:223.27
  • CL 218872

    CAS:
    <p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>
    Formula:C13H9F3N4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:278.23
  • Imidazenil

    CAS:
    <p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>
    Formula:C18H12BrFN4O
    Purity:98.4%
    Color and Shape:Solid
    Molecular weight:399.22
  • (E)-3,4,5-Trimethoxycinnamic acid

    CAS:
    <p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>
    Formula:C12H14O5
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:238.24
  • CGP52432

    CAS:
    <p>CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).</p>
    Formula:C15H24Cl2NO4P
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:384.24
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Formula:C6H11NO3
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:145.16
  • Cholesterol myristate

    CAS:
    <p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>
    Formula:C41H72O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:597.01
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Formula:C6H10ClNO2
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:163.602
  • α-Thujone

    CAS:
    <p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>
    Formula:C10H16O
    Purity:97.02% - 98.41%
    Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)
    Molecular weight:152.23
  • (2S)-6-Prenylnaringenin

    CAS:
    <p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>
    Formula:C20H20O5
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:340.37
  • Piperazine citrate

    CAS:
    <p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>
    Formula:C24H46N6O14
    Purity:99.8%
    Color and Shape:Crystals Indication
    Molecular weight:642.65
  • (+)-Kavain

    CAS:
    <p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>
    Formula:C14H14O3
    Purity:97% - ≥95%
    Color and Shape:White Fine Powder
    Molecular weight:230.26
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Formula:C12H16O3
    Purity:99.64% - 99.64%
    Color and Shape:Monoclinic Needles From Water Monoclinic Needles From Water
    Molecular weight:208.25
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Formula:C18H21ClF3N3O
    Purity:99.03% - 99.95%
    Color and Shape:Solid
    Molecular weight:387.83
  • Loreclezole hydrochloride

    CAS:
    <p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>
    Formula:C10H7Cl4N3
    Color and Shape:Solid
    Molecular weight:310.99
  • Temgicoluril

    CAS:
    <p>Temgicoluril (mebikar) acts on GABA Receptor.</p>
    Formula:C8H14N4O2
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:198.22
  • Phenibut (hydrochloride)

    CAS:
    <p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>
    Formula:C10H14ClNO2
    Purity:99.93%
    Color and Shape:White Crystalline Powder
    Molecular weight:215.68
  • Saclofen

    CAS:
    <p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>
    Formula:C9H12ClNO3S
    Purity:99.17%
    Color and Shape:White Crystalline Solid
    Molecular weight:249.71
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Formula:C19H19FN4O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:354.38
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Formula:C20H28ClNO3S2
    Color and Shape:Solid
    Molecular weight:430.02
  • 2'MeO6MF

    CAS:
    <p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>
    Formula:C17H14O3
    Purity:99.28% - 99.63%
    Color and Shape:Solid
    Molecular weight:266.29
  • Jujuboside A

    CAS:
    <p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>
    Formula:C58H94O26
    Purity:98% - >99.99%
    Color and Shape:Solid
    Molecular weight:1207.35
  • Miltirone

    CAS:
    <p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>
    Formula:C19H22O2
    Purity:99.22% - 99.66%
    Color and Shape:Solid
    Molecular weight:282.38
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Formula:C22H26ClNO2
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:371.9
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Formula:C4H10N2
    Color and Shape:Solid
    Molecular weight:86.14
  • Ginkgolide A

    CAS:
    <p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>
    Formula:C20H24O9
    Purity:98.76% - 99.81%
    Color and Shape:White Powder
    Molecular weight:408.4
  • Imepitoin

    CAS:
    <p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>
    Formula:C13H14ClN3O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:279.72
  • Isonipecotic acid

    CAS:
    <p>Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.</p>
    Formula:C6H11NO2
    Purity:99.82%
    Color and Shape:White To Faint Pink-Beige Powder
    Molecular weight:129.16
  • Gabazine

    CAS:
    <p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>
    Formula:C15H18BrN3O3
    Purity:98.51% - 99.24%
    Color and Shape:Solid
    Molecular weight:368.23
  • Tiagabine

    CAS:
    <p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>
    Formula:C20H25NO2S2
    Purity:99.25%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:375.55
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Formula:C17H24O4
    Purity:98.22%
    Color and Shape:Solid
    Molecular weight:292.37
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Formula:C30H18O10
    Purity:98.21% - 99.22%
    Color and Shape:Odourless Whitish Solid
    Molecular weight:538.46
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Formula:C2H5NO3·5HCl
    Purity:98.03%
    Color and Shape:Light Beige Crystalline Powder
    Molecular weight:109.3
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Formula:C11H11N3O
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:201.22
  • Fipronil

    CAS:
    <p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>
    Formula:C12H4Cl2F6N4OS
    Purity:97.21%
    Color and Shape:Solid Powder
    Molecular weight:437.15
  • Darigabat

    CAS:
    <p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>
    Formula:C22H21FN4O3S
    Purity:98.42% - 99.29%
    Color and Shape:Solid
    Molecular weight:440.49
  • Riluzole

    CAS:
    <p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>
    Formula:C8H5F3N2OS
    Purity:99.71% - 99.88%
    Color and Shape:Powder
    Molecular weight:234.2
  • CGP 36216 hydrochloride

    CAS:
    <p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>
    Formula:C5H14NO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:151.14
  • β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Formula:C16H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.31
  • NO 711

    CAS:
    <p>NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>
    Formula:C21H22N2O3
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:350.41
  • (±)-Homoproline Hydrochloride

    CAS:
    <p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>
    Formula:C6H12ClNO2
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:165.62
  • CP-457920

    CAS:
    <p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>
    Formula:C18H17N3O3
    Purity:99.06% - 99.74%
    Color and Shape:Solid
    Molecular weight:323.35
  • Ro 41-3290

    CAS:
    <p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>
    Formula:C24H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.89
  • PF-0713

    CAS:
    <p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>
    Formula:C14H22O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:206.32
  • HZ166

    CAS:
    <p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>
    Formula:C21H16N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.38
  • Pregabalin arenacarbil

    CAS:
    <p>Pregabalin arenacarbil is a gabamimetic.</p>
    Formula:C15H27NO6
    Color and Shape:Solid
    Molecular weight:317.38
  • NCS-382

    CAS:
    <p>γ-Hydroxybutyric acid antagonist</p>
    Formula:C13H14O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:218.25
  • Ro 19-4603

    CAS:
    <p>Benzodiazepine inverse agonist</p>
    Formula:C15H17N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.38
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Formula:C17H24N2O
    Color and Shape:Solid
    Molecular weight:272.39
  • mGAT3/4-IN-1

    CAS:
    <p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>
    Formula:C26H31ClN2O2S2
    Color and Shape:Solid
    Molecular weight:503.12
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Formula:C21H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:446.33
  • 17-PA

    CAS:
    <p>17-PA is a GABAA receptor antagonist.</p>
    Formula:C25H34O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.54
  • MK-0343

    CAS:
    <p>MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.</p>
    Formula:C19H17F2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:397.38
  • DS2

    CAS:
    <p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>
    Formula:C18H12ClN3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.83
  • CGS8216

    CAS:
    <p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>
    Formula:C16H11N3O
    Purity:98.53%
    Color and Shape:Solid
    Molecular weight:261.28
  • BHF-177

    CAS:
    <p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>
    Formula:C19H20F3N3
    Color and Shape:Solid
    Molecular weight:347.38
  • SKF 97541

    CAS:
    <p>GABAB agonist</p>
    Formula:C4H12NO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:137.12
  • CGP 7930

    CAS:
    <p>Positive allosteric modulator of GABAB receptors</p>
    Formula:C19H32O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.46
  • TPA-023B

    CAS:
    <p>TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.</p>
    Formula:C21H15F2N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.37
  • U-101017

    CAS:
    <p>U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.</p>
    Formula:C23H27ClN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.94
  • Org 20599

    CAS:
    <p>GABAA receptor agonist</p>
    Formula:C25H40ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.04
  • SX-3228

    CAS:
    <p>SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).</p>
    Formula:C18H18N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.36
  • CGS 20625

    CAS:
    <p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>
    Formula:C18H19N3O2
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:309.36
  • 2-Hydroxysaclofen

    CAS:
    <p>2-Hydroxysaclofen is a GABAB receptor antagonist.</p>
    Formula:C9H12ClNO4S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:265.71
  • Ro15-4513

    CAS:
    <p>Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.</p>
    Formula:C15H14N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.31
  • 3-Methyl-GABA

    CAS:
    <p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>
    Formula:C20H30N2O10S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:522.59
  • DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Formula:C18H10Br2ClN3OS
    Color and Shape:Solid
    Molecular weight:511.62
  • Cyprodenate

    CAS:
    <p>Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.</p>
    Formula:C13H25NO2
    Color and Shape:Solid
    Molecular weight:227.34
  • Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Formula:C18H13ClN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.83
  • U-7524

    CAS:
    <p>U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.</p>
    Formula:C2H5NO3
    Color and Shape:Solid
    Molecular weight:91.07
  • Ethyl dirazepate

    CAS:
    <p>Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.</p>
    Formula:C18H14Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.22
  • Arbaclofen placarbil

    CAS:
    <p>Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.</p>
    Formula:C19H26ClNO6
    Color and Shape:Solid
    Molecular weight:399.87