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PDE
THPP-1
CAS:1257051-63-0
THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 …
Formula:
C23H21ClN6O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
464.9
Estimated delivery in United States, on Monday 7 Feb 2022
Rolipram
CAS:61413-54-5
Rolipram is a phosphodiesterase 4 inhibitor with antidepressant properties.
Formula:
C16H21NO3
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
275.34
Estimated delivery in United States, on Monday 7 Feb 2022
GSK256066
CAS:801312-28-7
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, …
Formula:
C27H26N4O5S
Purity:
98.0%
Color and Shape:
solid
Molecular weight:
518.58
Estimated delivery in United States, on Monday 7 Feb 2022
Deltarasin
CAS:1440898-61-2
Deltarasin is a small molecular inhibitor of KRAS-PDE interaction with Kd of 38 nM for …
Formula:
C40H37N5O
Purity:
98.0%
Color and Shape:
solid
Molecular weight:
603.75
Estimated delivery in United States, on Monday 7 Feb 2022
Mirodenafil dihydrochloride
CAS:862189-96-6
Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.
Formula:
C26H39Cl2N5O5S
Purity:
99.46%
Color and Shape:
solid
Molecular weight:
604.59
Estimated delivery in United States, on Monday 7 Feb 2022
DprE1-IN-1
CAS:1494675-86-3
DprE1-IN-1 is a potent inhibitor of DprE1 and PDE6.
Formula:
C18H21N5O3
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
355.39
Estimated delivery in United States, on Monday 7 Feb 2022
Amrinone
CAS:60719-84-8
Amrinone is a positive inotropic cardiotonic (cardiotonic agent) with vasodilator properties, phosphodiesterase 3 inhibitory activity.
Formula:
C10H9N3O
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
187.2
Estimated delivery in United States, on Monday 7 Feb 2022
Triflusal
CAS:322-79-2
Triflusal is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a …
Formula:
C10H7F3O4
Purity:
93.15%
Color and Shape:
solid
Molecular weight:
248.16
Estimated delivery in United States, on Monday 7 Feb 2022
Roflumilast
CAS:162401-32-3
Roflumilast is an orally available, long-acting inhibitor of phosphodiesterase (PDE) type 4 (PDE4), with anti-inflammatory …
Formula:
C17H14Cl2F2N2O3
Purity:
99.64%
Color and Shape:
solid
Molecular weight:
403.21
Estimated delivery in United States, on Monday 7 Feb 2022
Doxofylline
CAS:69975-86-6
Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. …
Formula:
C11H14N4O4
Purity:
99.98%
Color and Shape:
solid
Molecular weight:
266.26
Estimated delivery in United States, on Monday 7 Feb 2022
Aminophylline
CAS:317-34-0
Aminophylline is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.
Formula:
C7H8O2·C2H8N2
Purity:
99.94%
Color and Shape:
White Or Slightly Yellowish Granules Or Powder Solid
Molecular weight:
420.43
Estimated delivery in United States, on Monday 7 Feb 2022
Vesnarinone
CAS:81840-15-5
Vesnarinone (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, …
Formula:
C22H25N3O4
Purity:
96.69%
Color and Shape:
solid
Molecular weight:
395.46
Estimated delivery in United States, on Monday 7 Feb 2022
Avanafil
CAS:330784-47-9
Avanafil is a selective inhibitor of phosphodiesterase type 5 (PDE5) and is used as therapy …
Formula:
C23H26ClN7O3
Purity:
98.00%
Color and Shape:
White Solid
Molecular weight:
483.95
Estimated delivery in United States, on Monday 7 Feb 2022
Pentoxifylline
CAS:6493-05-6
Pentoxifylline modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits …
Formula:
C13H18N4O3
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
278.31
Estimated delivery in United States, on Monday 7 Feb 2022
Dypyridamole
CAS:58-32-2
Dipyridamole is a Platelet Aggregation Inhibitor. The physiologic effect of dipyridamole is by means of …
Formula:
C24H40N8O4
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
504.63
Estimated delivery in United States, on Monday 7 Feb 2022
Diprophylline
CAS:479-18-5
Dyphylline is a xanthine derivative. Dyphilline exerts bronchodilator effects and to a lesser extent vasodilator …
Formula:
C10H14N4O4
Purity:
99.10%
Color and Shape:
Crystals From Alcohol Solid
Molecular weight:
254.25
Estimated delivery in United States, on Monday 7 Feb 2022
Pimobendan
CAS:74150-27-9
Pimobendan is a selective inhibitor of PDE3 (IC50: 0.32 μM).
Formula:
C19H18N4O2
Purity:
99.84%
Color and Shape:
solid
Molecular weight:
334.37
Estimated delivery in United States, on Monday 7 Feb 2022
Indometacin
CAS:53-86-1
Indomethacin is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of indomethacin is as a …
Formula:
C19H16ClNO4
Purity:
99.27%
Color and Shape:
Pale-Yellow To Yellow-Tan Crystalline Powder Physical Description Crystals (Ntp 1992)
Molecular weight:
357.79
Estimated delivery in United States, on Monday 7 Feb 2022
Heptaminol hydrochloride
CAS:543-15-7
Heptaminol hydrochloride, a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.
Formula:
C8H20ClNO
Purity:
98.00%
Color and Shape:
White Crystalline Powder
Molecular weight:
181.71
Estimated delivery in United States, on Monday 7 Feb 2022
Trapidil
CAS:15421-84-8
Trapidil is a coronary vasodilator agent. It was originally developed as a vasodilator and anti-platelet …
Formula:
C10H15N5
Purity:
99.96%
Color and Shape:
solid
Molecular weight:
205.26
Estimated delivery in United States, on Monday 7 Feb 2022
2-(Hydroxymethyl)pyridine
CAS:586-98-1
2-Pyridinylmethanol is an organic compound.
Formula:
C6H7NO
Purity:
99.79%
Color and Shape:
Clear Light Yellow To Orange Liquid Liquid
Molecular weight:
109.13
Estimated delivery in United States, on Monday 7 Feb 2022
Theobromine
CAS:83-67-0
3, 7-Dimethylxanthine, a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.
Formula:
C7H8N4O2
Purity:
99.82%
Color and Shape:
White To Yellow Crystalline Powder
Molecular weight:
180.16
Estimated delivery in United States, on Monday 7 Feb 2022
Fenspiride hydrochloride
CAS:5053-08-7
Fenspiride, an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory …
Formula:
C15H20N2O2·HCl
Purity:
99.92%
Color and Shape:
solid
Molecular weight:
296.79
Estimated delivery in United States, on Monday 7 Feb 2022
Lotamilast
CAS:947620-48-6
E6005 is a phosphodiesterase 4 (PDE-4) inhibitor (IC50: 2.8 nM) potentially for the treatment of …
Formula:
C26H24N4O5
Purity:
99.29%
Color and Shape:
solid
Molecular weight:
472.17
Estimated delivery in United States, on Monday 7 Feb 2022
Luteolin
CAS:491-70-3
Luteolin is a naturally occurring flavonoid. The flavonoids are polyphenolic compounds found as integral components …
Formula:
C15H10O6
Purity:
96.61%
Color and Shape:
solid
Molecular weight:
286.24
Estimated delivery in United States, on Monday 7 Feb 2022
IBMX
CAS:28822-58-4
IBMX is a pan-phosphodiesterase (PDE) inhibitor (IC50s: 6.5/26.3/31.7 μM for PDE3/PDE4/PDE5).
Formula:
C10H14N4O2
Purity:
98.00%
Color and Shape:
Off-White
Molecular weight:
222.24
Estimated delivery in United States, on Monday 7 Feb 2022
Apremilast
CAS:608141-41-9
Apremilast (CC-10004) is a potent and orally active PDE4 (IC50=74 nM) with anti-inflammation activities.
Formula:
C22H24N2O7S
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
460.5
Estimated delivery in United States, on Monday 7 Feb 2022
Icariin
CAS:489-32-7
Icariin is a flavonol glycoside, inhibiting PDE5 and PDE4 activities. Icariin also is a PPAR …
Formula:
C33H40O15
Purity:
98.04%
Color and Shape:
solid
Molecular weight:
676.68
Estimated delivery in United States, on Monday 7 Feb 2022
Enoximone
CAS:77671-31-9
Enoximone is a selective inhibitor of phosphodiesterase III (PDE3), with treatment of congestive heart failure.
Formula:
C12H12N2O2S
Purity:
95.52%
Color and Shape:
solid
Molecular weight:
248.3
Estimated delivery in United States, on Monday 7 Feb 2022
PF-04447943
CAS:1082744-20-4
PF-04447943 is an effective inhibitor of human recombinant PDE9A (IC50=12 nM). It has >78-fold selectivity, …
Formula:
C20H25N7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
395.46
Estimated delivery in United States, on Monday 7 Feb 2022
ATX inhibitor 5
CAS:2402772-45-4
ATX inhibitor 5 is an orally active autotaxin (ATX) inhibitor (IC50: 15.3 nM). It has …
Formula:
C22H18ClF3N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
474.87
Estimated delivery in United States, on Monday 7 Feb 2022
Deltasonamide 2 (TFA)
CAS:2235358-74-2
Deltasonamide 2 TFA is competitive, high affinity PDE inhibitor with a Kd of ~385 pM.
Formula:
C32H40ClF3N6O6S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
761.27
Estimated delivery in United States, on Monday 7 Feb 2022
BI-409306
CAS:1189767-28-9
BI-409306 is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be …
Formula:
C16H17N5O2
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
311.34
Estimated delivery in United States, on Monday 7 Feb 2022
CM-675
CAS:1872466-47-1
CM-675 is a dual inhibitor of phosphodiesterase 5 (PDE5) and class I histone deacetylases (IC50s: …
Formula:
C31H32N6O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
536.62
Estimated delivery in United States, on Monday 7 Feb 2022
MBCQ
CAS:150450-53-6
MBCQ is an inhibitor of cGMP-specific phosphodiesterase PDE5.
Formula:
C16H12ClN3O2
Molecular weight:
313.74
Estimated delivery in United States, on Monday 7 Feb 2022
Sildenafil
CAS:139755-83-2
Sildenafil is a phosphodiesterase type 5 (PDE5) inhibitor, used to treat erectile dysfunction and reduce …
Formula:
C22H30N6O4S
Purity:
99.6%
Color and Shape:
White Crystalline Powder
Molecular weight:
474.58
Estimated delivery in United States, on Monday 7 Feb 2022
Crisaborole
CAS:906673-24-3
AN-2728 is a Phosphodiesterase 4 Inhibitor.
Formula:
C14H10BNO3
Purity:
99.91%
Color and Shape:
solid
Molecular weight:
251.05
Estimated delivery in United States, on Monday 7 Feb 2022
Sildenafil citrate
CAS:171599-83-0
Sildenafil, a cyclic guanosine monophosphate (cGMP)-specific phosphodiesterase type 5 (PDE5) Inhibitor, is used extensively for …
Formula:
C28H38N6O11S
Purity:
99.57%
Color and Shape:
White Solid
Molecular weight:
666.7
Estimated delivery in United States, on Monday 7 Feb 2022
Olprinone
CAS:106730-54-5
Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and …
Formula:
C14H10N4O
Purity:
99.87%
Color and Shape:
solid
Molecular weight:
250.26
Estimated delivery in United States, on Monday 7 Feb 2022
VP3.15 dihydrobromide
CAS:1281681-33-1
VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE7- glycogen synthase kinase …
Formula:
C20H24Br2N4OS
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
528.3
Estimated delivery in United States, on Monday 7 Feb 2022
PAT-048
CAS:1359983-15-5
PAT-048 is an effective and selective autotaxin inhibitor. PAT-048 reduces dermal fibrosis in vivo. PAT-048 …
Formula:
C22H18ClF2N3O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
461.91
Estimated delivery in United States, on Monday 7 Feb 2022
Cilostazol
CAS:73963-72-1
Cilostazol is a Phosphodiesterase 3 Inhibitor. The mechanism of action of cilostazol is as a …
Formula:
C20H27N5O2
Purity:
99.86%
Color and Shape:
Off-White Solid
Molecular weight:
369.46
Estimated delivery in United States, on Monday 7 Feb 2022
TAK063
CAS:1238697-26-1
TAK-063 is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is …
Formula:
C23H17FN6O2
Purity:
99.28%
Color and Shape:
solid
Molecular weight:
428.42
Estimated delivery in United States, on Monday 7 Feb 2022
ent-Tadalafil
CAS:629652-72-8
ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS).
Formula:
C22H19N3O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
389.4
Estimated delivery in United States, on Monday 7 Feb 2022
Cilostamide
CAS:68550-75-4
Cilostamide is a selective phosphodiesterase (PDE)3A and PDE3B inhibitor(IC50 values of 27 and 50 nM, …
Formula:
C20H26N2O3
Purity:
98.00%
Color and Shape:
White To Off-White Solid
Molecular weight:
342.43
Estimated delivery in United States, on Monday 7 Feb 2022
Autotaxin-IN-1
CAS:1619971-30-0
Autotaxin-IN-1 is a potent autotaxin inhibitor, which has favorable potency (IC50=2.2 nM), PK properties, and …
Formula:
C21H23N7O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
405.45
Estimated delivery in United States, on Monday 7 Feb 2022
Deltasonamide 2 hydrochloride
Deltasonamide 2 hydrochloride is a competitive high-affinity PDE inhibitor with a Kd of approximately 385 …
Formula:
C30H40Cl2N6O4S2
Molecular weight:
683.71
Estimated delivery in United States, on Monday 7 Feb 2022
(+)-pinoresinol--D-glucoside; (+)-pinor
CAS:69251-96-3
Formula:
C26H32O11
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
520.53
Estimated delivery in United States, on Monday 7 Feb 2022
Anagrelide HCl
CAS:58579-51-4
Anagrelide Hydrochloride(BL4162A) is a drug used for the treatment of essential thrombocytosis.
Formula:
C10H7Cl2N3O·HCl
Purity:
99.77%
Color and Shape:
Off-White Powder
Molecular weight:
292.55
Estimated delivery in United States, on Monday 7 Feb 2022
Autotaxin-IN-4
CAS:2156655-86-4
Autotaxin-IN-4 is an Autotaxin inhibitor extracted from patent WO2018212534A1 (compound 51). It has the potential …
Formula:
C22H21N9O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
443.46
Estimated delivery in United States, on Monday 7 Feb 2022
Vardenafil hydrochloride
CAS:224785-91-5
Vardenafil hydrochloride is a New Phosphodiesterase Type 5(PDE5) Inhibitor, in the Treatment of Erectile Dysfunction …
Formula:
C23H33ClN6O4S
Purity:
99.76%
Color and Shape:
White To Off-White Cyrstalline Solid
Molecular weight:
525.06
Estimated delivery in United States, on Monday 7 Feb 2022
Deltasonamide 2
CAS:2088485-34-9
Deltasonamide 2 is a competitive, high affinity PDE inhibitor with a Kd of ~385 pM.
Formula:
C30H39ClN6O4S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
647.25
Estimated delivery in United States, on Monday 7 Feb 2022
YM976
CAS:191219-80-4
YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)
Formula:
C17H16ClN3O
Purity:
99.84%
Color and Shape:
solid
Molecular weight:
313.78
Estimated delivery in United States, on Monday 7 Feb 2022
Amino Tadalafil
CAS:385769-84-6
Amino tadalafil is a potent phosphodiesterase 5 (PDE5) inhibitor.
Formula:
C21H18N4O4
Purity:
99.67%
Color and Shape:
White Powder
Molecular weight:
390.39
Estimated delivery in United States, on Monday 7 Feb 2022
Vardenafil hydrochloride trihydrate
CAS:330808-88-3
Vardenafil HCl Trihydrate is a new type PDE inhibitor with IC50 of 0.7 and 180 …
Formula:
C23H32N6O4S·HCl·3H2O
Purity:
99.66%
Color and Shape:
solid
Molecular weight:
579.11
Estimated delivery in United States, on Monday 7 Feb 2022
OR-1896
CAS:220246-81-1
OR-1896 is an active long-lived Levosimendan metabolite, is a highly selective inhibitor of phosphodiesterase (PDE) …
Formula:
C13H15N3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
245.28
Estimated delivery in United States, on Monday 7 Feb 2022
K-Ras-PDE-IN-1
CAS:1841464-21-8
K-Ras-PDE-IN-1 is a potent inhibitor of competitive K-Ras-PDE.It binds to the farnesyl binding pocket of …
Formula:
C25H26FN5O2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
447.5
Estimated delivery in United States, on Monday 7 Feb 2022
Robustine
CAS:2255-50-7
Robustine is a natural product, exhibits inhibitory potency against human phosphodiesterase 5 (hPDE5A) in vitro.
Formula:
C12H9NO3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
215.2
Estimated delivery in United States, on Monday 7 Feb 2022
Zaprinast
CAS:37762-06-4
Zaprinast was an unsuccessful Clinicalal drug candidate that was a precursor to the chemically related …
Formula:
C13H13N5O2
Color and Shape:
White To Off White Powder
Molecular weight:
271.27
Estimated delivery in United States, on Monday 7 Feb 2022
Apremilast D5
CAS:1258597-47-5
Apremilast D5 (CC-10004 D5) is a deuterium-labeled Apremilast. Apremilast is an orally available inhibitor of …
Formula:
C22H19D5N2O7S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
465.53
Estimated delivery in United States, on Monday 7 Feb 2022
Mardepodect hydrochloride (898562-94-2 free base)
Mardepodect hydrochloride can cross the blood-brain barrier. Mardepodect hydrochloride is an effective and selective PDE10A …
Formula:
C25H21ClN4O
Molecular weight:
428.91
Estimated delivery in United States, on Monday 7 Feb 2022
SEP-0372814
CAS:1516895-53-6
SEP-0372814 is a potent inhibitor of PDE10.
Formula:
C21H19N7
Color and Shape:
Solid
Molecular weight:
369.42
Estimated delivery in United States, on Monday 7 Feb 2022
GSK 256066 Trifluoroacetate
CAS:1415560-64-3
GSK 256066 Trifluoroacetate is a selective and high-affinity phosphodiesterase 4 (PDE) inhibitor (IC50: 3.2 pM …
Formula:
C29H27F3N4O7S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
632.61
Estimated delivery in United States, on Monday 7 Feb 2022
PF-05180999
CAS:1394033-54-5
PF-05180999 is an inhibitor of phosphodiesterase 2A (IC50: 1.6 nM).
Formula:
C19H17F3N8
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
414.39
Estimated delivery in United States, on Monday 7 Feb 2022
HA-155
CAS:1229652-22-5
HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively …
Formula:
C24H19BFNO5S
Purity:
98.92%
Molecular weight:
463.29
Estimated delivery in United States, on Monday 7 Feb 2022
Autotaxin-IN-5
CAS:2156655-99-9
Autotaxin-IN-5 is an Autotaxin inhibitor extracted from patent WO2018212534A1 (compound 63). It has the potential …
Formula:
C30H29N9O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
547.61
Estimated delivery in United States, on Monday 7 Feb 2022
Lodenafil
CAS:139755-85-4
Lodenafil is a potent PDE5 inhibitor, with treatment of erectile dysfunction (ED)
Formula:
C23H32N6O5S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
504.6
Estimated delivery in United States, on Monday 7 Feb 2022
Mirodenafil
CAS:862189-95-5
Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.
Formula:
C26H37N5O5S
Purity:
99.85%
Color and Shape:
solid
Molecular weight:
531.67
Estimated delivery in United States, on Monday 7 Feb 2022
Bay 60-7550
CAS:439083-90-6
Bay 60-7550 is an inhibitor of PDE2(Ki: 3.8 nM).
Formula:
C27H32N4O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
476.57
Estimated delivery in United States, on Monday 7 Feb 2022
PF-2545920
CAS:1292799-56-4
PF-2545920, a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity …
Formula:
C25H20N4O
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
392.45
Estimated delivery in United States, on Monday 7 Feb 2022
GLPG1690
CAS:1628260-79-6
GLPG-1690, an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic …
Formula:
C30H33FN8O2S
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
588.71
Estimated delivery in United States, on Monday 7 Feb 2022
BAY 73-6691
CAS:794568-92-6
BAY 73-6691 is an inhibitor of brain penetrant PDE9A.
Formula:
C15H12ClF3N4O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
356.73
Estimated delivery in United States, on Monday 7 Feb 2022
K134
CAS:189362-06-9
K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, …
Formula:
C22H29N3O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
399.48
Estimated delivery in United States, on Monday 7 Feb 2022
Isoprenaline hydrochloride
CAS:51-30-9
Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
Formula:
C11H18ClNO3
Purity:
99.50%
Color and Shape:
Physical Description Odorless White Crystalline Powder Slightly Bitter Taste Aqueous
Molecular weight:
247.72
Estimated delivery in United States, on Monday 7 Feb 2022
Autotaxin modulator 1
CAS:1548743-69-6
Autotaxin modulator 1 is a new modulator of Autotaxin extracted from Patent WO 2014018881 A1.
Formula:
C28H31F6NO3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
543.54
Estimated delivery in United States, on Monday 7 Feb 2022
Anagrelide
CAS:68475-42-3
Anagrelide is a Platelet-reducing Agent. The mechanism of action of anagrelide is as a Phosphodiesterase …
Formula:
C10H7Cl2N3O
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
256.09
Estimated delivery in United States, on Monday 7 Feb 2022
ATX inhibitor 1
CAS:2225892-70-4
ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, …
Formula:
C21H23Cl2N2O6P
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
501.3
Estimated delivery in United States, on Monday 7 Feb 2022
PDE5-IN-2
CAS:2244517-61-9
PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM)
Formula:
C25H21N3O6S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
491.52
Estimated delivery in United States, on Monday 7 Feb 2022
TAK-915
CAS:1476727-50-0
TAK-915 is a potent, selective, and brain-penetrant phosphodiesterase 2A (PDE2A) inhibitor (IC50: 0.61 nM). TAK-915 …
Formula:
C19H18F4N4O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
458.36
Estimated delivery in United States, on Monday 7 Feb 2022
Homo Sildenafil
CAS:642928-07-2
Homo Sildenafil is an analog of Sildenafil, It acts as a phosphodiesterase inhibitor.
Formula:
C23H32N6O4S
Molecular weight:
488.6
Estimated delivery in United States, on Monday 7 Feb 2022
HA130
CAS:1229652-21-4
HA130 is a selective ATX (autotaxin) inhibitor.
Formula:
C24H19BFNO5S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
463.29
Estimated delivery in United States, on Monday 7 Feb 2022
PF8380
CAS:1144035-53-9
PF-8380 is an effective and orally available autotaxin inhibitor (IC50: 2.8 nM, in isolated enzyme …
Formula:
C22H21Cl2N3O5
Purity:
99.25%
Color and Shape:
solid
Molecular weight:
478.33
Estimated delivery in United States, on Monday 7 Feb 2022
Lirimilast
CAS:329306-27-6
Lirimilast is an effective, selective, and orally active phosphodiesterase-4 (PDE4) inhibitor (IC50: 49 nM). Lirimilast …
Formula:
C17H12Cl2N2O6S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
443.26
Estimated delivery in United States, on Monday 7 Feb 2022
TPN171
CAS:1229018-87-4
TPN171 is a selective and oral bioavailable phosphodiesterase type 5 (PDE5) inhibitor (IC50: 0.62 nM), …
Formula:
C24H35N5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
441.57
Estimated delivery in United States, on Monday 7 Feb 2022
PF-05085727
CAS:1415637-72-7
PF-05085727 inhibits PDE2A >4,000-fold selectivity over PDE1 and PDE3-11. PF-05085727 is an effective, selective and …
Formula:
C20H18F3N7
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
413.4
Estimated delivery in United States, on Monday 7 Feb 2022
CDC801
CAS:192819-27-5
CDC801 is a potent and orally active inhibitor of PDE4 and TNF- (IC50: 1.1 μM …
Formula:
C23H24N2O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
408.45
Estimated delivery in United States, on Monday 7 Feb 2022
TyK2-IN-2
CAS:2098466-94-3
TyK2-IN-2 is a selective inhibitor of TYK2 (IC50s: 7 nM, 0.1 μM, and 0.05 μM …
Formula:
C16H18N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
310.35
Estimated delivery in United States, on Monday 7 Feb 2022
MR-L2
CAS:2374703-19-0
MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).
Formula:
C19H16Cl3FN4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
441.71
Estimated delivery in United States, on Monday 7 Feb 2022
Proxyphylline
CAS:603-00-9
Proxyphylline is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts …
Formula:
C10H14N4O3
Purity:
99.79%
Color and Shape:
solid
Molecular weight:
238.24
Estimated delivery in United States, on Monday 7 Feb 2022
Nortadalafil
CAS:171596-36-4
Nortadalafil is demethyl Tadalafil, which is a PDE5 inhibitor, treating erectile dysfunction (ED) ; and …
Formula:
C21H16N3O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
375.38
Estimated delivery in United States, on Monday 7 Feb 2022
Milrinone
CAS:78415-72-2
Milrinone is a Phosphodiesterase 3 Inhibitor. The mechanism of action of milrinone is as a …
Formula:
C12H9N3O
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
211.22
Estimated delivery in United States, on Monday 7 Feb 2022
BRL 50481
CAS:433695-36-4
BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 …
Formula:
C9H12N2O4S
Purity:
99.88%
Color and Shape:
solid
Molecular weight:
244.27
Estimated delivery in United States, on Monday 7 Feb 2022
Autotaxin-IN-3
CAS:2156655-68-2
Autotaxin-IN-3 is an Autotaxin(ATX) inhibitor (IC50: 2.4 nM) sourced from patent WO2018212534A1 (compound 33).
Formula:
C22H21N9O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
443.46
Estimated delivery in United States, on Monday 7 Feb 2022
Irsogladine
CAS:57381-26-7
Irsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine …
Formula:
C9H7Cl2N5
Purity:
99.74%
Color and Shape:
White Or Colorless Crystal Or Crystalline Powder Odorless Slightly Bitter
Molecular weight:
256.09
Estimated delivery in United States, on Monday 7 Feb 2022
S- (+)-Rolipram
CAS:85416-73-5
S-(+)-Rolipram inhibits human monocyte cyclic AMP-specific PDE4 with IC50 of 0.75 μM, has anti-inflammatory and …
Formula:
C16H21NO3
Purity:
99.71%
Color and Shape:
solid
Molecular weight:
275.34
Estimated delivery in United States, on Monday 7 Feb 2022
ITI214
CAS:1642303-38-5
ITI214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and …
Formula:
C29H29FN7O5P
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
605.56
Estimated delivery in United States, on Monday 7 Feb 2022
PAT-505
CAS:1782070-22-7
PAT-505 is a selective, noncompetitive and orally available inhibitor of autotaxin(IC50 of 2 nM in …
Formula:
C23H18ClF2N3O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
473.92
Estimated delivery in United States, on Monday 7 Feb 2022
Zomepirac Sodium
CAS:64092-48-4
Zomepirac sodium salt is a prostaglandin synthetase inhibitor.
Formula:
C15H13ClNNaO3
Purity:
98.65%
Color and Shape:
solid
Molecular weight:
313.71
Estimated delivery in United States, on Monday 7 Feb 2022
Naproxen etemesil
CAS:385800-16-8
Naproxen is a COX-1 and COX-2 inhibitor (IC50s: 8.72 and 5.15 μM, respectively in cell …
Formula:
C17H20O5S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
336.4
Estimated delivery in United States, on Monday 7 Feb 2022
N-Methylbenzamide
CAS:613-93-4
N-Methylbenzamide is a potent phosphodiesterase 10A (PDE10A) inhibitor,with anti-cancer activity.
Formula:
C8H9NO
Purity:
98.00%
Color and Shape:
Physical Description Off-White Crystalline Solid (Ntp 1992)
Molecular weight:
135.16
Estimated delivery in United States, on Monday 7 Feb 2022
