Transferase
Transferases are a large class of enzymes that catalyze the transfer of functional groups, such as methyl, glycosyl, and phosphate groups, from one molecule to another. Inhibitors of transferases are used to study a wide range of biological processes, including signal transduction, metabolism, and gene expression. These inhibitors are essential tools in research areas such as cancer, metabolic diseases, and epigenetics, where dysregulation of transferase activity is implicated. At CymitQuimica, we offer a comprehensive selection of transferase inhibitors to support your research in enzymology, cell signaling, and disease mechanisms.
Found 35 products for "Transferase".
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Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Formula:C6H11NO2Purity:99.90%Color and Shape:SolidMolecular weight:129.16Opicapone
CAS:Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).Formula:C15H10Cl2N4O6Purity:98.17% - 99.36%Color and Shape:SolidMolecular weight:413.17β-1,4-GALT1-IN-1
β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.Formula:C29H23NO10Color and Shape:SolidMolecular weight:545.494R1-11
R1-11 is an indole-based ICMT inhibitor with an IC50 of 0.6 μM, exhibiting anticancer properties. It inhibits MDA-MB231 and PC3 cells with IC50 values of 2.2 μM and 2.0 μM, respectively.Formula:C25H37N5Molecular weight:407.3049Squalene synthase-IN-2
Squalene synthase-IN-2 (compound isomer A-(1S, 3R)-14i) is an orally active inhibitor of squalene synthase, with IC50 values of 3.4 nM for squalene synthase and 99 nM for cholesterol synthesis enzymes. Squalene synthase-IN-2 effectively reduces plasma cholesterol and triglycerides.Formula:C31H39ClN2O6Molecular weight:570.24966Sinbaglustat
CAS:Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.Formula:C11H23NO4Purity:99.97%Color and Shape:SolidMolecular weight:233.3Ref: TM-T40542
1mg69.00€1mL*10mM (DMSO)140.00€5mg156.00€10mg225.00€25mg359.00€50mg487.00€100mg648.00€200mg875.00€Histamine glutarimide
CAS:Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.Formula:C10H13N3O2Purity:99.79%Color and Shape:SolidMolecular weight:207.23L-739750 2HCl
L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.Formula:C23H41Cl2N3O6S2Purity:98.69% - 99.16%Color and Shape:SoildMolecular weight:590.62FUT8-IN-1
FUT8-IN-1 (Compound 37) is an inhibitor of α-1,6-fucosyltransferase (FUT8), with a dissociation constant (KD) of 49 nM and an IC50 around 50 µM. In the presence of FUT8, FUT8-IN-1 forms a highly active naphthoquinone imine intermediate, thereby inhibiting FUT8's enzymatic activity.Formula:C23H25ClN2OColor and Shape:SolidMolecular weight:380.91FTI-277
CAS:FTI-277, an FTase inhibitor, blocks H-Ras/K-Ras signaling and HDV infection; mimics Ras CAAX peptide.Formula:C22H29N3O3S2Purity:99.63%Color and Shape:SolidMolecular weight:447.61BAY-593
CAS:BAY-593 is an orally active GGTase-I inhibitor capable of blocking YAP1/TAZ signaling in vivo, exhibiting antitumor activity.Formula:C26H31F3N2O3Color and Shape:SolidMolecular weight:476.53Ervogastat
CAS:Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.Formula:C21H21N5O4Purity:99.97%Color and Shape:SolidMolecular weight:407.42Ref: TM-T9186
1mg123.00€5mg290.00€1mL*10mM (DMSO)301.00€10mg485.00€25mg782.00€50mg1,063.00€100mg1,431.00€Ibiglustat
CAS:Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Formula:C20H24FN3O2SPurity:97.97% - 98.81%Color and Shape:SolidMolecular weight:389.49Tipifarnib (S enantiomer)
CAS:Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Formula:C27H22Cl2N4OPurity:99.05%Color and Shape:SolidMolecular weight:489.4Ref: TM-T17102
1mg49.00€5mg102.00€1mL*10mM (DMSO)109.00€10mg163.00€25mg284.00€50mg409.00€100mg577.00€200mg778.00€PD 128042
CAS:PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formula:C23H39NO4Purity:99.79%Color and Shape:SolidMolecular weight:393.56CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Formula:C29H22ClN3O2Purity:99.86% - 99.87%Color and Shape:SolidMolecular weight:479.96Ref: TM-T38050
1mg52.00€5mg110.00€1mL*10mM (DMSO)127.00€10mg177.00€25mg301.00€50mg425.00€100mg605.00€200mg797.00€Entacapone
CAS:Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Formula:C14H15N3O5Purity:98.80% - >99.99%Color and Shape:Yellow Crystalline SolidMolecular weight:305.29Ref: TM-T2216
5mg34.00€10mg49.00€1mL*10mM (DMSO)50.00€25mg75.00€50mg90.00€100mg137.00€200mg197.00€500mg333.00€Tipifarnib
CAS:Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Formula:C27H22Cl2N4OPurity:97.1% - 99.22%Color and Shape:Off-White To Pale Beige SolidMolecular weight:489.4Nitecapone
CAS:Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Formula:C12H11NO6Purity:98.39%Color and Shape:SolidMolecular weight:265.223-O-Methyltolcapone
CAS:3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Formula:C15H13NO5Purity:98%Color and Shape:SolidMolecular weight:287.27
