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Neuroscience

Neuroscience

Neuroscience inhibitors are compounds designed to modulate the activity of specific proteins, enzymes, or receptors within the nervous system. These inhibitors are crucial for studying the molecular mechanisms underlying neural function, synaptic transmission, and neurodegenerative diseases. By targeting neurotransmitter receptors, ion channels, and signaling pathways, neuroscience inhibitors aid in the exploration of brain function and the development of therapeutic strategies for neurological disorders such as Alzheimer's, Parkinson's, and epilepsy. At CymitQuimica, we offer a comprehensive range of high-quality neuroscience inhibitors to support your research in neurobiology, neuropharmacology, and cognitive sciences.

Subcategories of "Neuroscience"

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Found 5389 products of "Neuroscience"

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  • DS2

    CAS:
    Positive allosteric modulator of δ-subunit containing GABAA receptors
    Formula:C18H12ClN3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.83
  • LY-411575 isomer 1

    CAS:
    <p>LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575.</p>
    Formula:C26H23F2N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.48
  • L-CCG-l

    CAS:
    <p>group II metabotropic glutamate receptor agonist</p>
    Formula:C6H9NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:159.14
  • Muscarine iodide

    CAS:
    <p>Muscarinic acetylcholine receptor agonist</p>
    Formula:C9H20INO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.17
  • Mavoglurant racemate

    CAS:
    <p>Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.</p>
    Formula:C19H23NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:313.39
  • MK-0343

    CAS:
    <p>MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.</p>
    Formula:C19H17F2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:397.38
  • Muscarine chloride

    CAS:
    <p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>
    Formula:C9H20ClNO2
    Color and Shape:Solid
    Molecular weight:209.71
  • BHF-177

    CAS:
    <p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>
    Formula:C19H20F3N3
    Color and Shape:Solid
    Molecular weight:347.38
  • Piclozotan

    CAS:
    <p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>
    Formula:C23H24ClN3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:409.91
  • Foliglurax monohydrochloride

    CAS:
    Foliglurax monohydrochloride, an antiparkinsonian, is a selective brain-penetrant mGluR4 PAM with an EC50 of 79 nM.
    Formula:C23H24ClN3O3S
    Color and Shape:Solid
    Molecular weight:457.97
  • ML337

    CAS:
    ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.
    Formula:C21H20FNO3
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:353.39
  • 17-PA

    CAS:
    17-PA is a GABAA receptor antagonist.
    Formula:C25H34O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.54
  • Prenylamine lactate

    CAS:
    <p>Prenylamine lactate, an ex-angina drug, depletes heart catecholamines and blocks calcium channels.</p>
    Formula:C27H33NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.56
  • LY 302148

    CAS:
    <p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>
    Formula:C19H23FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.41
  • AY1511

    CAS:
    <p>AY1511 is a low cytotoxic inhibitor of amyloid β (Aβ) aggregation [1].</p>
    Formula:C17H14O6
    Color and Shape:Solid
    Molecular weight:314.29
  • VU0400195

    CAS:
    <p>VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).</p>
    Formula:C21H16ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.82
  • WAY-361789

    CAS:
    <p>WAY-361789 is an agonist of alpha7 nicotinic acetylcholine receptor.</p>
    Formula:C22H31N5O3
    Color and Shape:Solid
    Molecular weight:413.51
  • GABAA receptor modulator-2

    CAS:
    <p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>
    Formula:C22H22FN3O5S
    Color and Shape:Solid
    Molecular weight:459.49
  • PXS-4787

    CAS:
    <p>PXS-4787 selectively inhibits LOX with IC50 values: 2 μM (Bovine), 3.2 μM (LOXL1), 0.6 μM (LOXL2), 1.4 μM (LOXL3), 0.2 μM (LOXL4).</p>
    Formula:C10H12FNO2S
    Color and Shape:Solid
    Molecular weight:229.27
  • 5-HT7 receptor ligand 1

    CAS:
    <p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>
    Formula:C21H23N7
    Color and Shape:Solid
    Molecular weight:373.45
  • UCSF678

    CAS:
    <p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>
    Formula:C15H18N2O2S
    Color and Shape:Solid
    Molecular weight:290.38
  • ATC0065

    CAS:
    <p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>
    Formula:C25H29BrF3N5O
    Color and Shape:Solid
    Molecular weight:552.43
  • Desmethyl-YM 298198

    CAS:
    mGlu1-selective antagonist
    Formula:C17H21ClN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:364.89
  • Deramciclane fumarate

    CAS:
    <p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>
    Formula:C24H35NO5
    Color and Shape:Solid
    Molecular weight:417.54
  • Talsaclidine

    CAS:
    <p>Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.</p>
    Formula:C10H15NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:165.23
  • A-85380 HCl

    CAS:
    <p>A-85380 is an agonist of nicotinic acetylcholine receptor.</p>
    Formula:C9H14Cl2N2O
    Color and Shape:Solid
    Molecular weight:237.13
  • Usmarapride

    CAS:
    <p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>
    Formula:C23H31N5O6
    Color and Shape:Solid
    Molecular weight:473.53
  • SEN-1269

    CAS:
    <p>SEN-1269 prevents amyloid-β aggregation, shields neurons, and improves memory by hindering Aβ(1-42)-induced issues.</p>
    Formula:C18H18N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.36
  • Phenglutarimid

    CAS:
    <p>Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.</p>
    Formula:C17H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.38
  • sEH/AChE-IN-1

    CAS:
    <p>Compound 12a is a dual sEH/AChE inhibitor with potential for treating Alzheimer's-related neuroinflammation and memory loss.</p>
    Formula:C29H31ClF3N5O3
    Color and Shape:Solid
    Molecular weight:590.04
  • (RS)-4-Carboxy-3-hydroxyphenylglycine

    CAS:
    <p>broad spectrum EAA agonist/antagonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17
  • Carburazepam

    CAS:
    <p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>
    Formula:C17H16ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.78
  • MAO-B ligand-1

    CAS:
    <p>MAO-B ligand-1 is a selective MAO-B inhibitor.</p>
    Formula:C19H19N5O4S
    Color and Shape:Solid
    Molecular weight:413.45
  • Ro4491533

    CAS:
    <p>Ro4491533 is a potent and selective negative allosteric modulator for group II of the metabotropic glutamate receptors (mGluR2/3).</p>
    Formula:C24H20F3N3O
    Color and Shape:Solid
    Molecular weight:423.43
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Formula:C21H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:446.33
  • BuChE-IN-3

    CAS:
    <p>BuChE-IN-3 (Compound C4) is a potent inhibitor of BuChE (IC50: 8.3 nM). buChE-IN-3 is a mild antioxidant, non-toxic, lipophilic and neuroprotective agent.</p>
    Formula:C21H21F2N3O4S
    Color and Shape:Solid
    Molecular weight:449.47
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>5-HT1A serotonin receptor agonist</p>
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29
  • Org-25935

    CAS:
    <p>Org-25935, a GlyT-1 inhibitor, is used potentially for the treatment of schizophrenia and alcohol dependence.</p>
    Formula:C21H26ClNO3
    Color and Shape:Solid
    Molecular weight:375.89
  • JNJ1930942

    CAS:
    <p>JNJ1930942 is a novel positive allosteric modulator of the α7 nicotinic acetylcholine receptor.</p>
    Formula:C16H11F4N3OS
    Color and Shape:Solid
    Molecular weight:369.34
  • Auglurant

    CAS:
    <p>Auglurant is a novel and selective mGlu5 antagonist (IC50: 11 nM (rat) and an IC50: 14 nM (human)). Auglurant has an acceptable CNS penetration.</p>
    Formula:C16H12FN5O2
    Color and Shape:Solid
    Molecular weight:325.3
  • S 14063

    CAS:
    <p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>
    Formula:C22H29Cl2N3O2S
    Color and Shape:Solid
    Molecular weight:470.45
  • ZLWH-23

    CAS:
    <p>ZLWH-23: AChE inhibitor (IC50: 0.27μM), GSK-3β (6.78μM), BChE (20.82μM), potential in Alzheimer's research.</p>
    Formula:C30H32FN5O2
    Color and Shape:Solid
    Molecular weight:513.61
  • AChE/BChE/BACE-1-IN-1

    CAS:
    <p>Compound 4k is an oral AChE, BChE, BACE-1 inhibitor with IC50s: 0.058, 0.082, 0.115 μM, crosses blood-brain barrier, and has neuroprotective effects.</p>
    Formula:C19H21F3N2O
    Color and Shape:Solid
    Molecular weight:350.38
  • AChE/MAO-IN-2


    <p>Potent AChE/MAO-B inhibitor; IC50: AChE 0.0224 μM, MAO-B 0.0412 μM, MAO-A 0.1116 μM. Antioxidant, anti-β-amyloid, for AD research.</p>
    Formula:C23H26N2O3
    Color and Shape:Solid
    Molecular weight:378.46
  • Itameline

    CAS:
    RU 47213 can be used to inhibit scopolamine-induced working memory impairment in rats.
    Formula:C14H15ClN2O3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:294.73
  • AChE/BChE/MAO-B-IN-2


    <p>AChE/BChE/MAO-B-IN-2 inhibits AChE (48.2 nM), BChE (83.9 nM), MAO-B (31.2 nM), has antioxidant activity, and aids Parkinson's research.</p>
    Formula:C25H31N3O3
    Color and Shape:Solid
    Molecular weight:421.53
  • Dual AChE-MAO B-IN-2

    CAS:
    <p>Potent Dual AChE-MAO B-IN-2 inhibits AChE (0.12 μM) &amp; MAO B (0.01 μM); promising for Alzheimer's research.</p>
    Formula:C26H25NO4
    Color and Shape:Solid
    Molecular weight:415.48
  • MMPIP

    CAS:
    <p>allosteric mGlu7-selective receptor antagonist</p>
    Formula:C19H15N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.34
  • Fonazine

    CAS:
    <p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>
    Formula:C19H25N3O2S2
    Color and Shape:Solid
    Molecular weight:391.55
  • ENS-163 phosphate

    CAS:
    <p>Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.</p>
    Formula:C11H19N2O5PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.32
  • VU0361747

    CAS:
    <p>VU0361747 is a positive allosteric modulators (PAM) of metabotropic glutamate receptor subtype 5 (mGlu5).</p>
    Formula:C19H17FN2O2
    Color and Shape:Solid
    Molecular weight:324.35
  • Rivanicline oxalate

    CAS:
    <p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>
    Formula:C12H16N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:252.27
  • Hexafluronium Bromide

    CAS:
    <p>Hexafluronium bromide enhances muscle relaxation in surgery by blocking acetylcholine receptors.</p>
    Formula:C36H42BrN2
    Color and Shape:Solid
    Molecular weight:582.649
  • TMPH hydrochloride

    CAS:
    <p>neuronal nicotinic ACh receptors (nAChRs) antagonist</p>
    Formula:C16H32ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.88
  • BACE1/2-IN-1

    CAS:
    <p>BACE1/2-IN-1 inhibits BACE1/2 with IC50s of 0.01μM/0.0053μM, has better permeability and lower Pgp efflux but reduced metabolic stability.</p>
    Formula:C21H31N5OS
    Color and Shape:Solid
    Molecular weight:401.57
  • TC 2559 difumarate

    CAS:
    partial agonist of α4β2 nicotinic acetylcholine receptor
    Formula:C12H18N2OC4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.39
  • UMB68 sodium

    CAS:
    <p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) &gt;100 microM) at GABA(A) or GABA(B) receptors.</p>
    Formula:C6H12NaO3
    Color and Shape:Solid
    Molecular weight:155.149
  • mGAT3/4-IN-1

    CAS:
    <p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>
    Formula:C26H31ClN2O2S2
    Color and Shape:Solid
    Molecular weight:503.12
  • EGIS-7625

    CAS:
    <p>EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.</p>
    Formula:C18H24Cl2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.32
  • MAO-B-IN-16

    CAS:
    <p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>
    Formula:C18H19NO3
    Color and Shape:Solid
    Molecular weight:297.35
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Formula:C26H31FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.53
  • Tridihexethyl chloride

    CAS:
    <p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>
    Formula:C21H36ClNO
    Color and Shape:Solid
    Molecular weight:353.97
  • Trimedoxime bromide

    CAS:
    <p>Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.</p>
    Formula:C15H18Br2N4O2
    Color and Shape:Solid
    Molecular weight:446.14
  • AChE/BuChE-IN-2

    CAS:
    Compound 5f, an oral AChE/BuChE inhibitor, crosses BBB; IC50: 0.72 μM (AChE), 0.16 μM (BuChE), 62.52 μM (Aβ aggregation).
    Formula:C20H18N2O2
    Color and Shape:Solid
    Molecular weight:318.37
  • DV 7028 hydrochloride

    CAS:
    <p>DV 7028 hydrochloride is a 5-HT2A receptor antagonist.</p>
    Formula:C21H26ClFN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.91
  • S20928

    CAS:
    <p>S20928 is an antagonist of melatonin receptor.</p>
    Formula:C17H19NO
    Color and Shape:Solid
    Molecular weight:253.34
  • AChE/MAO-IN-1


    <p>AChE/MAO-IN-1 is a potent inhibitor of human acetylcholinesterase (AChE), monoamine oxidase A (MAO-A), and monoamine oxidase B (MAO-B), demonstrating inhibitory</p>
    Formula:C23H26N2O3
    Color and Shape:Solid
    Molecular weight:378.46
  • LSP4-2022

    CAS:
    <p>LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.</p>
    Formula:C13H18NO8P
    Purity:100%
    Color and Shape:Solid
    Molecular weight:347.26
  • BACE2-IN-1

    CAS:
    <p>BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.</p>
    Formula:C36H38F3N3O3
    Color and Shape:Solid
    Molecular weight:617.7
  • FG-5893

    CAS:
    <p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>
    Formula:C27H29F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.53
  • NW-1772

    CAS:
    <p>NW-1772 is a highly potent and orally active inhibitor of monoamine oxidase B.</p>
    Formula:C19H20ClNO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.88
  • RU-505

    CAS:
    <p>RU-505 is an interaction inhibitor of Aβ-fibrinogen that acts by rescuing altered thrombosis and cognitive decline in Alzheimer's disease mice.</p>
    Formula:C28H32FN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.58
  • NAP-1

    CAS:
    <p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>
    Formula:C20H18ClNO2
    Color and Shape:Solid
    Molecular weight:339.82
  • SERT-IN-2


    <p>SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.</p>
    Color and Shape:Solid
  • Org 24598

    CAS:
    <p>Potent GlyT1b inhibitor, IC50 = 6.9 nM; little effect on GlyT-2, adrenoceptors, dopamine, 5HT receptors, GABA transporters.</p>
    Formula:C19H20F3NO3
    Color and Shape:Solid
    Molecular weight:367.36
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Formula:C17H24N2O
    Color and Shape:Solid
    Molecular weight:272.39
  • Dihydro Donepezil

    CAS:
    <p>Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).</p>
    Formula:C24H31NO3
    Color and Shape:Solid
    Molecular weight:381.51
  • Remeglurant

    CAS:
    <p>Remeglurant is used as a selective antagonist of the mGlu5 receptor.</p>
    Formula:C17H15BrN4O
    Color and Shape:Solid
    Molecular weight:371.23
  • LY314228

    CAS:
    <p>LY314228 is an antagonist of 5-HT2A receptor.</p>
    Formula:C20H24N4O3
    Color and Shape:Solid
    Molecular weight:368.43
  • VU0455691

    CAS:
    <p>VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.</p>
    Formula:C24H25N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.55
  • ML169

    CAS:
    <p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>
    Formula:C21H17BrFN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.34
  • Antioxidant agent-2

    CAS:
    <p>Antioxidant agent-2 (3c), BBB-permeable, selectively chelates metals; shows neuroprotection, fights liver damage in Alzheimer's research.</p>
    Formula:C23H26N2O7
    Color and Shape:Solid
    Molecular weight:442.46
  • MAO-B-IN-12

    CAS:
    <p>MAO-B-IN-12 (16c) is a potent MAO-B inhibitor with an IC50 of 1.3 μM and has neuroprotective properties.</p>
    Formula:C22H30O4
    Color and Shape:Solid
    Molecular weight:358.47
  • (R)-Oxybutynin

    CAS:
    <p>(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.</p>
    Formula:C22H31NO3
    Color and Shape:Solid
    Molecular weight:357.49
  • Caroxazone

    CAS:
    <p>Caroxazone is an antidepressant drug, monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective meanwhile.</p>
    Formula:C10H10N2O3
    Color and Shape:Solid
    Molecular weight:206.2
  • PXS-6302

    CAS:
    <p>PXS-6302: irreversible lysyl oxidase inhibitor, skin-penetrating, reduces scar collagen; IC50: 0.3-3.7 μM. May treat various fibrotic diseases.</p>
    Formula:C10H10F3NO2S
    Color and Shape:Solid
    Molecular weight:265.25
  • CP-809101

    CAS:
    CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
    Formula:C15H17ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.77
  • Bornaprine

    CAS:
    <p>Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.</p>
    Formula:C21H31NO2
    Color and Shape:Solid
    Molecular weight:329.48
  • SB 207710

    CAS:
    SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.
    Formula:C19H27IN2O4
    Color and Shape:Solid
    Molecular weight:474.33
  • Ambutonium bromide

    CAS:
    <p>Ambutonium bromide is an antagonist of acetylcholine.</p>
    Formula:C20H27BrN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.35
  • BChE-IN-7

    CAS:
    <p>BChE-IN-7 inhibits AChE/BChE selectively and reversibly; IC50 for BChE: 0.06 μM; crosses blood-brain barrier, protects neurons from Aβ toxicity.</p>
    Formula:C21H24N2O2
    Color and Shape:Solid
    Molecular weight:336.43
  • IEM 1925 dihydrobromide

    CAS:
    <p>AMPA receptor antagonist</p>
    Formula:C17H30Br2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.24
  • Ro 60-0175 fumarate

    CAS:
    <p>5-HT2 receptor agonist</p>
    Formula:C15H16ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.75
  • PHCCC(4Me)

    CAS:
    <p>THCCC, a PHCCC analog, is a dual metabotropic glutamate receptor 2/3 negative/positive allosteric modulator.</p>
    Formula:C18H16N2O3
    Color and Shape:Solid
    Molecular weight:308.33
  • Memoquin

    CAS:
    <p>Memoquin is a multi-target-directed ligand for the therapy of Alzheimer's disease.</p>
    Formula:C38H56N4O4
    Color and Shape:Solid
    Molecular weight:632.88
  • 5-HT7 agonist 2

    CAS:
    <p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>
    Formula:C23H29N3O
    Color and Shape:Solid
    Molecular weight:363.5
  • GABAA receptor agent 7

    CAS:
    <p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>
    Formula:C18H13ClN4O
    Color and Shape:Solid
    Molecular weight:336.77
  • Yhhu-3792

    CAS:
    <p>Yhhu-3792 activates Notch, boosts Hes3/Hes5, enhances NSC renewal, expands NSC pool, and may improve memory.</p>
    Formula:C24H24N4O2
    Color and Shape:Solid
    Molecular weight:400.47
  • sEH inhibitor-5

    CAS:
    <p>sEH inhibitor-5 is a potent inhibitor of sEH (soluble epoxide hydrolase) (IC50: 0.1 nM).</p>
    Formula:C27H26Cl2N6O3S
    Color and Shape:Solid
    Molecular weight:585.5
  • Zicronapine

    CAS:
    <p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>
    Formula:C22H27ClN2
    Color and Shape:Solid
    Molecular weight:354.92
  • Ethybenztropine

    CAS:
    <p>Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.</p>
    Formula:C22H27NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.46
  • Pheniprazine

    CAS:
    <p>Pheniprazine, a potent and long-acting monoamine oxidase inhibitor, shows promise for depression research.</p>
    Formula:C9H14N2
    Color and Shape:Solid
    Molecular weight:150.22
  • Anabasine hydrochloride

    CAS:
    <p>neuronal nicotinic ACh receptor partial agonist</p>
    Formula:C10H15ClN2
    Purity:98%
    Color and Shape:White To Off-White Solid
    Molecular weight:198.693
  • NPEC-caged-LY379268

    CAS:
    <p>NPEC-caged-LY379268 is a type II mGluR agonist [1].</p>
    Formula:C16H16N2O9
    Color and Shape:Solid
    Molecular weight:380.31
  • BChE-IN-11

    CAS:
    <p>BChE-IN-11: potent, selective, non-competitive BChE inhibitor; IC50=2.1μM; used in AD research.</p>
    Formula:C22H18O4
    Color and Shape:Solid
    Molecular weight:346.38
  • Nerispirdine HCl

    CAS:
    Nerispirdine enhances acetylcholine, blocks Na+ channels (IC50 11.9µM) and K(v) 1.1/1.2 channels (IC50 3.6/3.7µM).
    Formula:C17H19ClFN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.8
  • A 841720

    CAS:
    <p>Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.</p>
    Formula:C17H21N5OS
    Color and Shape:Solid
    Molecular weight:343.45
  • Aβ-IN-5

    CAS:
    <p>Aβ-IN-5 (Compound e12) is an orally active Aβ aggregation inhibitor that also inhibits AChE and BuChE with IC50 values of 21.29 μM and 1.32 μM, respectively.</p>
    Formula:C21H20N2O3
    Color and Shape:Solid
    Molecular weight:348.4
  • RO5488608

    CAS:
    <p>RO5488608 is a new type of high-efficiency mGlu2/3 NAM.</p>
    Formula:C23H17F3N2O4S
    Color and Shape:Solid
    Molecular weight:474.45
  • AC260584

    CAS:
    AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).
    Formula:C20H29FN2O2
    Color and Shape:Solid
    Molecular weight:348.45
  • LY487379 hydrochloride

    CAS:
    Positive allosteric modulator of mGlu2 receptors
    Formula:C21H20ClF3N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.91
  • Adenylyl cyclase type 2 agonist-1

    CAS:
    <p>Potent AC2 agonist with an EC50 of 90 nM, potential for respiratory disease treatment.</p>
    Formula:C27H17BrClNO5
    Color and Shape:Solid
    Molecular weight:550.78
  • Belaperidone

    CAS:
    <p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>
    Formula:C22H22FN3O2
    Color and Shape:Solid
    Molecular weight:379.43
  • RJR-2403 oxalate

    CAS:
    <p>RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.</p>
    Formula:C14H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.308
  • PF-4479745

    CAS:
    <p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>
    Formula:C17H22N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.38
  • RX 67668

    CAS:
    <p>RX 67668: Muscle relaxant, relieves fatigue; cholinesterase inhibitor (IC50: 5 μM); reverses D-tubocurarine effects.</p>
    Formula:C16H24ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:265.82
  • Bibn 140

    CAS:
    <p>Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.</p>
    Formula:C32H44N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.72
  • Eplivanserin hemifumarate

    CAS:
    <p>Eplivanserin is an inverse agonist of 5-HT2A.</p>
    Formula:C23H25FN2O6
    Color and Shape:Solid
    Molecular weight:444.45
  • MRK-623

    CAS:
    <p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>
    Formula:C20H17FN4O
    Color and Shape:Solid
    Molecular weight:348.37
  • hMAO-B-IN-2

    CAS:
    <p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>
    Formula:C18H23NO3
    Color and Shape:Solid
    Molecular weight:301.38
  • AChE/BChE-IN-4

    CAS:
    <p>AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.</p>
    Formula:C17H26N2O3
    Color and Shape:Solid
    Molecular weight:306.4
  • RS 23597-190 hydrochloride

    CAS:
    <p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>
    Formula:C16H24Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.28
  • LY 2365109 hydrochloride

    CAS:
    <p>glycine transporter 1 (GlyT1) inhibitor</p>
    Formula:C22H27NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.45
  • Ambenonium dichloride

    CAS:
    <p>AChE inhibitor</p>
    Formula:C28H42Cl3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.02
  • AChE/BChE/MAO-B-IN-4


    <p>AChE/BChE/MAO-B-IN-4 inhibits MAO-B (IC50: 0.0393 µM), AChE (IC50: 0.0458 µM), BChE (IC50: 0.075 µM), and fights AD with antioxidant action.</p>
    Formula:C26H33N3O4
    Color and Shape:Solid
    Molecular weight:451.56
  • Alaproclate (hydrochloride)

    CAS:
    <p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>
    Formula:C13H19Cl2NO2
    Color and Shape:Solid
    Molecular weight:292.2
  • 5-HT6/5-HT2A receptor ligand-2

    CAS:
    <p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>
    Formula:C20H18FN3O2
    Color and Shape:Solid
    Molecular weight:351.37
  • Brofaromine Hydrochloride

    CAS:
    <p>Brofaromine hydrochloride treats depression/anxiety, inhibits MAO-A, affects serotonin/dopamine.</p>
    Formula:C14H17BrClNO2
    Color and Shape:Solid
    Molecular weight:346.65
  • TIM-063

    CAS:
    TIM-063: ATP-competitive CaMKKα/β inhibitor, cell-permeable, Ki: 0.35/0.2 μM, IC50: 0.63/0.96 μM.
    Formula:C18H9N3O4
    Color and Shape:Solid
    Molecular weight:331.28
  • MPDC

    CAS:
    <p>MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.</p>
    Formula:C7H9NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:171.15
  • SD-6

    CAS:
    <p>SD-6, oral hAChE/hBChE inhibitor (IC50: 0.907/1.579 µM), crosses BBB, non-toxic, for Alzheimer's research.</p>
    Formula:C20H22N4OS
    Color and Shape:Solid
    Molecular weight:366.48
  • Levemopamil HCl

    CAS:
    Levemopamil HCl is used as a calcium channel blocker.
    Formula:C23H31ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.96
  • AZD 0328

    CAS:
    <p>AZD 0328 is a nicotinic receptor agonist for α7 neurons.</p>
    Formula:C13H16N2O
    Color and Shape:Solid
    Molecular weight:216.28
  • Talaglumetad hydrochloride

    CAS:
    <p>Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.</p>
    Formula:C11H17ClN2O5
    Color and Shape:Solid
    Molecular weight:292.72
  • PF-06455943

    CAS:
    <p>PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK &amp; Parkinson's research.</p>
    Formula:C17H14FN5O
    Color and Shape:Solid
    Molecular weight:323.32
  • mGluR2 modulator 2

    CAS:
    <p>mGluR2 modulator 2: potent, selective, oral, EC50 = 0.13 μM, for antipsychotic research.</p>
    Formula:C20H22FN3
    Color and Shape:Solid
    Molecular weight:323.41
  • SB 206553 hydrochloride

    CAS:
    <p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>
    Formula:C17H17ClN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:328.8
  • Ro 19-4603

    CAS:
    <p>Benzodiazepine inverse agonist</p>
    Formula:C15H17N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.38
  • AR-A 2

    CAS:
    <p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>
    Formula:C27H36N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.6
  • Befloxatone

    CAS:
    <p>Befloxatone is a potent, selective and reversible inhibitor of monoamine oxidase A.</p>
    Formula:C15H18F3NO5
    Color and Shape:Solid
    Molecular weight:349.3
  • J 104129 fumarate

    CAS:
    <p>M3 muscarinic receptor antagonist</p>
    Formula:C24H36N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.55
  • Telenzepine

    CAS:
    <p>Telenzepine is a potent and selective M1 antimuscarinic.</p>
    Formula:C19H22N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.47
  • sEH/AChE-IN-2

    CAS:
    <p>sEH/AChE-IN-2 targets sEH &amp; AChE, may reduce neuroinflammation &amp; memory loss, potential in Alzheimer's research.</p>
    Formula:C30H33ClF3N5O3
    Color and Shape:Solid
    Molecular weight:604.06
  • BChE-IN-14

    CAS:
    <p>BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).</p>
    Formula:C24H29N
    Color and Shape:Solid
    Molecular weight:331.49
  • Nitroflurbiprofen

    CAS:
    <p>Nitroflurbiprofen (Nitroxybutyl flurbiprofen) is a NO-releasing COX inhibitor and modulates the increased intrahepatic vascular tone in portal hypertensive</p>
    Formula:C19H20FNO5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:361.36
  • 2-Iodomelatonin

    CAS:
    <p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, &gt;5x selective over MT2, used to map melatonin sites in brain/tissues.</p>
    Formula:C13H15IN2O2
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:358.17
  • WAY208466 dihydrochloride

    CAS:
    <p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>
    Formula:C17H20Cl2FN3O2S
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:420.33
  • Cimetropium Bromide

    CAS:
    <p>Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.</p>
    Formula:C21H28BrNO4
    Color and Shape:Solid
    Molecular weight:438.36
  • RG-12915

    CAS:
    <p>RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).</p>
    Formula:C20H25ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.88
  • E-3620

    CAS:
    E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.
    Formula:C20H27Cl2N3O2
    Purity:98.88% - 98.88%
    Color and Shape:Solid
    Molecular weight:412.35
  • DBO-83

    CAS:
    <p>DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.</p>
    Formula:C10H15Cl3N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.61
  • SB 258585 hydrochloride

    CAS:
    SB 258585 hydrochloride is a 5-HT6 receptor antagonist.
    Formula:C18H23ClIN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.82
  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Formula:C16H13ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:364.8
  • RS-0466

    CAS:
    <p>RS-0466 is an β-amyloid-induced cytotoxicity inhibitor.</p>
    Formula:C17H17N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.35
  • Fluoroclorgyline

    CAS:
    Fluoroclorgyline is a specific inhibitor of monoamine oxidase A (MAO-A).
    Formula:C13H15ClFNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.72
  • HOCPCA

    CAS:
    <p>HOCPCA: potent, selective GHB site ligand; 27x higher affinity than GHB; crosses blood-brain barrier.</p>
    Formula:C6H8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:128.13
  • DAT 582

    CAS:
    <p>DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent</p>
    Formula:C22H28ClN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.95
  • RS 56812 hydrochloride

    CAS:
    <p>5-HT3 partial agonist</p>
    Formula:C18H22ClN3O2
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:347.84
  • Ro 04-6790 dihydrochloride

    CAS:
    <p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>
    Formula:C12H18Cl2N6O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.28
  • GSK931145

    CAS:
    <p>GSK931145 is a positron emission tomography (PET) radioligand, it is suitable for quantifying glycine transporter (GlyT1) availability in the living brain.</p>
    Formula:C23H30N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.5
  • Vesamicol

    CAS:
    Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.
    Formula:C17H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:259.39
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Formula:C7H9F2NO2
    Color and Shape:Solid
    Molecular weight:177.15
  • Altanserin hydrochloride

    CAS:
    <p>Altanserin hydrochloride is a 5-HT2A receptor antagonist.</p>
    Formula:C22H23ClFN3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.95
  • RGH 1756

    CAS:
    <p>RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.</p>
    Formula:C26H30N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.61
  • NGX-267

    CAS:
    <p>NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.</p>
    Formula:C10H18N2OS
    Color and Shape:Solid
    Molecular weight:214.33
  • LY2607540

    CAS:
    <p>LY2607540 is a metabotropic glutamate 2 potentiator with potential anxiolytic/antidepressant properties (EC(50) = 23 and 13 nM, respectively).</p>
    Formula:C24H24F3N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:475.46
  • Prifuroline

    CAS:
    <p>Prifuroline is an agent of antiarrhythmic.</p>
    Formula:C14H16N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:228.29
  • Palonosetron

    CAS:
    <p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>
    Formula:C19H24N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.41
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Formula:C30H35NO6
    Purity:97%
    Color and Shape:Solid
    Molecular weight:505.6
  • TIK-301

    CAS:
    <p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>
    Formula:C14H17ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.75
  • S 14506 hydrochloride

    CAS:
    <p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>
    Formula:C24H27ClFN3O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:443.94
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Formula:C6H11NO2
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:129.16
  • W-13 hydrochloride

    CAS:
    <p>W-13 hydrochloride (W-13 HCl) is a calmodulin antagonist.</p>
    Formula:C14H18Cl2N2O2S
    Purity:98.51%
    Color and Shape:White Powder
    Molecular weight:349.28
  • S 24795

    CAS:
    <p>S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.</p>
    Formula:C14H13BrINO
    Purity:99.934%
    Color and Shape:Solid
    Molecular weight:418.07
  • hMAO-B-IN-7

    CAS:
    <p>Compound 11n (hMAO-B-IN-7) is a potent inhibitor of human monoamine oxidase-B (hMAO-B) that can cross the blood-brain barrier (BBB). It demonstrates an IC 50 value of 0.79±0.05 μM and is useful in research related to Alzheimer's disease (AD) and Parkinson's disease (PD) [1].</p>
    Formula:C23H19FN2O5
    Color and Shape:Solid
    Molecular weight:422.41
  • BuChE-IN-6

    CAS:
    <p>BuChE-IN-6 inhibits BuChE (IC50: 0.46 μM eqBuChE, 0.51 μM hBuChE) and prevents Aβ 42 self-aggregation.</p>
    Formula:C21H26N4O2
    Color and Shape:Solid
    Molecular weight:366.46
  • SSAO inhibitor-3

    CAS:
    <p>SSAO inhibitor-3 targets human AOC1/SSAO in atherosclerosis, diabetes, obesity, CKD, and more, with IC50s of 0.1-10 μM/&lt;10 nM.</p>
    Formula:C15H23FN4O3
    Color and Shape:Solid
    Molecular weight:326.37
  • SV5

    CAS:
    <p>SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.</p>
    Formula:C21H30N2O4S2
    Color and Shape:Solid
    Molecular weight:438.6
  • 5-HT2A receptor agonist-2

    CAS:
    <p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>
    Formula:C20H21ClN2O3
    Color and Shape:Solid
    Molecular weight:372.85
  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.37
  • AChE/BuChE-IN-1

    CAS:
    <p>AChE/BuChE-IN-1: BuChE inhibitor (IC50=0.48µM), weaker AChE blocker (IC50=7.16µM), ·OH scavenger (IC50=0.1674µM), may aid in AD research.</p>
    Formula:C19H19NO4
    Color and Shape:Solid
    Molecular weight:325.36
  • Pralidoxime

    CAS:
    <p>Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.</p>
    Formula:C7H9N2O
    Color and Shape:Solid
    Molecular weight:137.16
  • (S)-VQW-765


    <p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39
  • BuChE-IN-7


    <p>BuChE-IN-7: selective hBuChe &amp; eqBuChe inhibitor, IC50s 40/80 nM, boosts cognition &amp; memory, and penetrates blood-brain barrier.</p>
    Formula:C25H34N2O2
    Color and Shape:Solid
    Molecular weight:394.55
  • MAO-B-IN-14

    CAS:
    <p>MAO-B-IN-14 (Compound 9) is a potent and selective inhibitor of monoamine oxidase-B (MAO-B) with an IC 50 of 0.95 μM and a Ki of 0.55 μM for human MAO-B.</p>
    Formula:C17H14O3S
    Color and Shape:Solid
    Molecular weight:298.36
  • AChE-IN-12

    CAS:
    <p>AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.</p>
    Formula:C33H41NO7
    Color and Shape:Solid
    Molecular weight:563.68
  • TC-2153

    CAS:
    <p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>
    Formula:C7H5ClF3NS5
    Color and Shape:Solid
    Molecular weight:355.89
  • Pimprinine

    CAS:
    <p>Pimprinine: an alkaloid, inhibits MAO, and has anticonvulsant properties.</p>
    Formula:C12H10N2O
    Color and Shape:Solid
    Molecular weight:198.22
  • (Rac)-SEP-363856

    CAS:
    <p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27
  • S-15535

    CAS:
    <p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>
    Formula:C21H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.43
  • Oxybutynin R-isomer HCl

    CAS:
    <p>Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.</p>
    Formula:C22H32ClNO3
    Color and Shape:Solid
    Molecular weight:393.95
  • UoS 12258

    CAS:
    <p>UoS 12258 is a positive allosteric modulator of AMPA receptors, used for studying cognitive impairments.</p>
    Formula:C17H19FN2O2S
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:334.41
  • F13714 fumarate

    CAS:
    <p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>
    Formula:C25H29ClF2N4O5
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:538.97
  • Aβ42-IN-2

    CAS:
    <p>Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].</p>
    Formula:C24H26N6O2
    Purity:98.09% - 99.87%
    Color and Shape:Solid
    Molecular weight:430.5
  • ONT-093

    CAS:
    <p>ONT-093 (OC-144-093) is an oral P-glycoprotein (P-gp) inhibitor with potential anti-cancer activity, used in the study of myelodysplastic syndromes.</p>
    Formula:C32H38N4O
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:494.67
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49
  • MAO-B-IN-23

    CAS:
    <p>MAO-B-IN-23, also known as Compound 11f, is a reversible and competitive monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 1.44 μM and a Ki of 0.51 μM</p>
    Formula:C19H18BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.26
  • Mazaticol

    CAS:
    <p>Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.</p>
    Formula:C21H27NO3S2
    Color and Shape:Solid
    Molecular weight:405.57
  • PD-102807

    CAS:
    <p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>
    Formula:C23H24N2O4
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:392.45
  • 5-HT7 agonist 1

    CAS:
    <p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>
    Formula:C19H20ClN3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:325.84